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EP0946587
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EP About this file: EP0946587
| EP0946587 - NEW AMIDE COMPOUNDS [Right-click to bookmark this link] | Status | The application is deemed to be withdrawn Status updated on 20.02.2004 Database last updated on 12.07.2024 | Most recent event Tooltip | 20.02.2004 | Application deemed to be withdrawn | published on 07.04.2004 [2004/15] | Applicant(s) | For all designated states FUJISAWA PHARMACEUTICAL CO., LTD. 4-7, Doshomachi 3-chome Chuo-ku Osaka-shi Osaka 541-8514 / JP | [N/P] |
| Former [1999/40] | For all designated states FUJISAWA PHARMACEUTICAL CO., LTD. 4-7, Doshomachi 3-chome Chuo-ku Osaka-shi Osaka 541-8514 / JP | Inventor(s) | 01 /
YATABE, Takumi deceased / JP | 02 /
ITOH, Yoshikuni 2-49-12, Himuro-cho Takatsuki-shi Osaka 569-11 / JP | 03 /
INOUE, Takayuki 4-15-2-2-201, Matsushiro,Tsukuba-shi Ibaraki 305 / JP | 04 /
HAMASHIMA, Hitoshi 3-25-4-202, Matsushiro,Tsukuba-shi Ibaraki 305 / JP | 05 /
SHIMA, Ichiro 5-25-105, Gosyogaoka,Moriya-cho Kitasouma-gun, Ibaraki 302-01 / JP | 06 /
OHNE, Kazuhiko 1-16-15-A102, Ninomiya,Tsukuba-shi Ibaraki 305 / JP | 07 /
YOSHIHARA, Kousei 2-4-38-405, Manabe,Tsuchiura-shi Ibaraki 300 / JP | 08 /
OKU, Teruo 8-2, Midorigaoka,Tsukuba-shi Ibaraki 305 / JP | [2000/06] |
| Former [1999/40] | 01 /
YATABE, Takumi +di / JP | ||
| 02 /
ITOH, Yoshikuni 2-49-12, Himuro-cho Takatsuki-shi Osaka 569-11 / JP | |||
| 03 /
INOUE, Takayuki 4-15-2-2-201, Matsushiro,Tsukuba-shi Ibaraki 305 / JP | |||
| 04 /
HAMASHIMA, Hitoshi 3-25-4-202, Matsushiro,Tsukuba-shi Ibaraki 305 / JP | |||
| 05 /
SHIMA, Ichiro 5-25-105, Gosyogaoka,Moriya-cho Kitasouma-gun, Ibaraki 302-01 / JP | |||
| 06 /
OHNE, Kazuhiko 1-16-15-A102, Ninomiya,Tsukuba-shi Ibaraki 305 / JP | |||
| 07 /
YOSHIHARA, Kousei 2-4-38-405, Manabe,Tsuchiura-shi Ibaraki 300 / JP | |||
| 08 /
OKU, Teruo 8-2, Midorigaoka,Tsukuba-shi Ibaraki 305 / JP | Representative(s) | Gille Hrabal Partnerschaftsgesellschaft mbB Patentanwälte Brucknerstraße 20 40593 Düsseldorf / DE | [N/P] |
| Former [1999/40] | Türk, Gille, Hrabal Patentanwälte - European Patent Attorneys, Brucknerstrasse 20 40593 Düsseldorf / DE | Application number, filing date | 97912529.1 | 20.11.1997 | [1999/40] | WO1997JP04243 | Priority number, date | AU1996PO04219 | 16.12.1996 Original published format: AU PO421996 | AU1997PO05929 | 01.04.1997 Original published format: AU PO592997 | AU1997PO09030 | 09.09.1997 Original published format: AU PO903097 | [1999/40] | Filing language | EN | Procedural language | EN | Publication | Type: | A2 Application without search report | No.: | WO9827108 | Date: | 25.06.1998 | Language: | EN | [1998/25] | Type: | A2 Application without search report | No.: | EP0946587 | Date: | 06.10.1999 | Language: | EN | The application published by WIPO in one of the EPO official languages on 25.06.1998 takes the place of the publication of the European patent application. | [1999/40] | Search report(s) | International search report - published on: | EP | 30.07.1998 | Classification | IPC: | C07D401/14, A61K31/415, A61K31/40, C07D401/12, C07D401/06, C07D233/54, C07D403/12, C07D521/00, C07D405/12, C07D403/14, C07D409/12, C07D413/12, C07D417/12 | [2000/06] | CPC: |
C07D233/64 (EP);
A61P1/04 (EP);
A61P1/16 (EP);
A61P11/00 (EP);
A61P11/06 (EP);
A61P13/12 (EP);
A61P17/00 (EP);
A61P19/02 (EP);
A61P19/06 (EP);
A61P19/10 (EP);
A61P25/00 (EP);
A61P25/04 (EP);
A61P25/28 (EP);
A61P27/00 (EP);
A61P29/00 (EP);
A61P3/10 (EP);
A61P35/04 (EP);
A61P43/00 (EP);
A61P9/00 (EP);
A61P9/10 (EP);
C07D231/12 (EP);
C07D233/56 (EP);
C07D233/90 (EP);
C07D249/08 (EP);
C07D401/06 (EP);
C07D401/12 (EP);
C07D401/14 (EP);
C07D403/12 (EP);
C07D403/14 (EP);
C07D405/12 (EP);
C07D405/14 (EP);
C07D409/12 (EP);
C07D413/12 (EP);
C07D417/12 (EP)
(-)
|
| Former IPC [1999/40] | C07K5/00, C07D403/00, C07D401/00 | Designated contracting states | AT, BE, CH, DE, DK, ES, FI, FR, GB, GR, IE, IT, LI, LU, MC, NL, PT, SE [1999/40] | Title | German: | AMINDVERBINDUNGEN UND IHRE VERWENDUNG ALS INHIBITOREN DER BITRIC-OXID-SYNTHASE | [1999/40] | English: | NEW AMIDE COMPOUNDS | [1999/40] | French: | NOUVEAUX COMPOSES AMIDE | [1999/40] | Entry into regional phase | 02.07.1999 | National basic fee paid | 02.07.1999 | Designation fee(s) paid | 02.07.1999 | Examination fee paid | Examination procedure | 09.06.1998 | Request for preliminary examination filed International Preliminary Examining Authority: EP | 02.07.1999 | Examination requested [1999/43] | 27.03.2003 | Despatch of a communication from the examining division (Time limit: M06) | 07.10.2003 | Application deemed to be withdrawn, date of legal effect [2004/15] | 10.11.2003 | Despatch of communication that the application is deemed to be withdrawn, reason: reply to the communication from the examining division not received in time [2004/15] | Fees paid | Renewal fee | 12.11.1999 | Renewal fee patent year 03 | 13.11.2000 | Renewal fee patent year 04 | 14.11.2001 | Renewal fee patent year 05 | 13.11.2002 | Renewal fee patent year 06 | 01.12.2003 | Renewal fee patent year 07 |
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| Responsibility for the accuracy, completeness or quality of the data displayed under the link provided lies entirely with the Unified Patent Court. | Cited in | International search | [X]EP0491525 (LILLY CO ELI [US]) [X] 1,4 * page 31 - page 32; examples 39,40 * * page 34 - page 35; example 44 *; | [Y]WO9616981 (FUJISAWA PHARMACEUTICAL CO [JP], et al) [Y] 1-5,7-9 * page 689 - page 692; claim 1 *; | [X] - LI G ET AL, "Synthesis of a Directly Connected Thiazole-Oxazole Ring System Present in Microcin B17", J. ORG. CHEM., (19960126), vol. 61, no. 2, pages 778 - 780, XP002057303 [X] 1,4 * see page 778; scheme 1, the compounds no. 4 and 5 * DOI: http://dx.doi.org/10.1021/jo951023c | [X] - HAMADA Y ET AL, "New methods and reagents in organic synthesis. 67. A general synthesis of derivatives of optically pure 2-(1-aminoalkyl)thiazole-4 -carboxylic acids", J. ORG. CHEM., (19870403), vol. 52, no. 7, pages 1252 - 1255, XP002057304 [X] 1,4 * see page 1252, scheme I, the compounds no. 6e-6h; and page 1255, paragraphs 3-5 * DOI: http://dx.doi.org/10.1021/jo00383a014 | [X] - PETTIT G R ET AL, "Antineoplastic agents. 109. Structural biochemistry. 24. Synthesis of the cyclo-[(gly)Thz-(R)- and (S)-(gln)Thz-L-Val-L-Leu-L -Pro] isomers of dolastatin 3", J. ORG. CHEM., (19850726), vol. 50, no. 15, pages 2654 - 2659, XP002057305 [X] 1,4 * see page 2655; the last but one compound of scheme II * DOI: http://dx.doi.org/10.1021/jo00215a012 | [X] - GERBERT U ET AL, "Model reactions for enzymic catalysis. IV. Structure-activity relationship of new transaminators with imidazole, thiazole, and benzimidazole skeletons", JUSTUS LIEBIGS ANN. CHEM., (1974), no. 4, pages 644 - 654, XP002057306 [X] 1,4 * page 652, paragraph 3 - paragraph 4 * DOI: http://dx.doi.org/10.1002/jlac.197419740409 | [X] - SETO Y ET AL, "Unusual amino acids and their peptides. V. Synthesis and the absolute configuration of.beta.-(2-thiazolyl)-.beta.-alanine present in bottromycin", BULL. CHEM. SOC. JAP., (197401), vol. 47, no. 1, pages 151 - 155, XP002057307 [X] 1,4 * page 153, column 2, line 30 - line 32 * | [X] - CROSS D F W ET AL, "Peptides. Part XIV. Thiazoleamino-acids, Degradation Products of Thiostrepton.", JOURNAL OF THE CHEMICAL SOCIETY., LETCHWORTH GB, (196304), pages 2143 - 2150, XP002057308 [X] 1,4 * page 2148, paragraph 7 * * page 2149, paragraph 7 * * page 2149, paragraph 11 * DOI: http://dx.doi.org/10.1039/jr9630002143 | [X] - PYL T ET AL, "Zur Darstellung von 7-Benzoylamino-pyrrolo[2.1-b]thiazolen", JUSTUS LIEBIGS ANNALEN DER CHEMIE., WEINHEIM DE, (1964), vol. 676, pages 141 - 150, XP002057309 [X] 1,2,4 * page 144, paragraph L * DOI: http://dx.doi.org/10.1002/jlac.19646760118 | [X] - PYL T ET AL, "Zur Kenntnis der Imidazo[5.1-b]thiazole", JUSTUS LIEBIGS ANNALEN DER CHEMIE., WEINHEIM DE, (1964), vol. 679, pages 144 - 150, XP002057310 [X] 1,4 * see page 145; the compounds no. Va and Vb * DOI: http://dx.doi.org/10.1002/jlac.19646790120 | [X] - CROSSFIRE, Beilstein Informationssysteme GmbH, XP002057315 [X] 1,4 * see BRN = 1025985 * | [ ] - REV. ROUM. CHIM., (1965), vol. 10, pages 617 - 620 | [X] - CROSSFIRE, Beilstein Informationssysteme GmbH, XP002057316 [X] 1,2,4 * see BRN = 859380 * | [ ] - STUD. UNIV. BABES-BOLYAI CHEM., (1960), vol. 1, page 155 | [X] - CROSSFIRE, Beilstein Informationssysteme GmbH, XP002057317 [X] 1,4 * see BRN = 259370 * | [ ] - AM. CHEM. J., (1912), vol. 47, pages 234 - 236 | [X] - HEINISCH G ET AL, "2-Dialkylaminoacylaminoimidazoles as potential local anesthetics.", CHEMICAL ABSTRACTS, (19740819), vol. 81, no. 7, Database accession no. 37511r, page 385, column 1, XP002057314 [X] 1,4 * see abstract; and Chemical Abstracts, CHEMICAL SUBSTANCES, 9th Collective Index, vol. 76-85, 1972-1976, page 3018CS: the compound with the RN [17496-81-0], * * page 3021CS: the compound with the RN [52737-56-1], and page 3028CS: the compound with the RN [52737-58-3] * | [ ] - SCI. PHARM., (1974), vol. 42, no. 1, pages 19 - 33 | [X] - MOFFETT R B ET AL, "Antiulcer Agents. p-Aminobenzamido Aromatic Compounds", JOURNAL OF MEDICINAL CHEMISTRY., WASHINGTON US, (197110), vol. 14, no. 10, pages 963 - 968, XP002057311 [X] 1,4 * see page 966; table II, the compounds no. 52 and 53 * DOI: http://dx.doi.org/10.1021/jm00292a019 | [X] - CROSSFIRE, Beilstein Informationssysteme GmbH, XP002057318 [X] 1,4 * see BRN = 838703 * | [ ] - TETRAHEDRON., OXFORD GB, (1974), vol. 30, pages 3859 - 3864 | [X] - NAIR V ET AL, "Regioselective [4+2] and [2+2] Cycloadditions of 1-Azirines to Heterocumulenes. Formation and Rearrangements of the Cycloadducts", JOURNAL OF ORGANIC CHEMISTRY., EASTON US, (19741213), vol. 39, no. 25, pages 3763 - 3767, XP002057312 [X] 1-4 * see page 3764, column 2, the compound no. 12; and page 3766, column 2, the last paragraph, and page 3767, column 1, paragraphs 4-5 * DOI: http://dx.doi.org/10.1021/jo00939a034 | [X] - LIEBSCHER J ET AL, "Formylation Products of Thioamides; Part 12. Synthesis of Thiazoles by the Reaction of S-Alkylated Thioamides or Thioureas with Acid Derivatives", SYNTHESIS., STUTTGART DE, (198504), no. 4, pages 414 - 417, XP002057313 [X] 1,2,4 * see page 415, column 1, the compound no. 11; and page 417, table 2, the compounds no. 11c and 11d * DOI: http://dx.doi.org/10.1055/s-1985-31224 | [X] - CROSSFIRE, Beilstein Informationssysteme GmbH, XP002057319 [X] 1,4 * see BRN = 1121645 * | [ ] - ARCH. PHARM., (1979), vol. 312, pages 198 - 205 | [X] - CROSSFIRE, Beilstein Informationssysteme GmbH, XP002057320 [X] 1,2,4 * see BRN = 920461 * | [ ] - CHEM. HETEROCYCL. COMPD. (ENGL. TRANSL.), (1970), vol. 6, pages 486 - 488 | [X] - CROSSFIRE, Beilstein Informationssysteme GmbH, XP002057321 [X] 1,2,4 * see BRN = 301310 * | [ ] - CHEM. PHARM. BULL., (1969), vol. 17, page 2381 | [X] - CROSSFIRE, Beilstein Informationssysteme GmbH, XP002057322 [X] 1,2,4 * see BRN = 216640 * | [ ] - SYNTH. COMMUN., (1988), vol. 18, no. 7, pages 651 - 658 | [X] - CROSSFIRE, Beilstein Informationssysteme GmbH, XP002057323 [X] 1,2,4 * see BRN = 299571 * | [ ] - UKR. KHIM. ZH. (RUSS. ED.), (1955), vol. 21, pages 726 - 729 | [Y] - GORDON T D ET AL, "Synthetic Approaches to the 'Azole' Peptide Mimetics", TETRAHEDRON LETTERS., OXFORD GB, (19930319), vol. 34, no. 12, pages 1901 - 1904, XP002038851 [Y] 1-5,7-9 * page 1901, paragraph 1 * DOI: http://dx.doi.org/10.1016/S0040-4039(00)91958-0 |