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Extract from the Register of European Patents

EP About this file: EP0885199

EP0885199 - KAPPA AGONIST COMPOUNDS AND PHARMACEUTICAL FORMULATIONS THEREOF [Right-click to bookmark this link]
Status	The application is deemed to be withdrawn Status updated on 23.03.2007 Database last updated on 26.06.2024
Most recent event Tooltip	23.03.2007	Application deemed to be withdrawn	published on 25.04.2007 [2007/17]
Applicant(s)	For all designated states Adolor Corporation 395 Phoenixville Pike Malvern, PA 19355 / US
	[1998/52]
Inventor(s)	01 / KRUSE, Lawrence, I. 646 Clinton Avenue Haddonfield, NJ 08033-0117 / US
	02 / CHANG, An-Chih A-178 Westridge Gardens Phoenixville, PA 19460 / US
	03 / DEHAVEN-HUDKINS, Diane, L. 430 South Saddlebrook Circle Chester Springs, PA 19425 / US
	04 / FARRAR, John, J. 1066 Bodine Road Chester Springs, PA 19425 / US
	05 / GAUL, Forrest 1787 Fairview Road Glen Moore, PA 19343 / US
	06 / MARELLA, Michael, Anthony 32 Carriage Lane Exton, PA 19341 / US
	07 / MAYCOCK, Alan, L. 1908 Standiford Drive Malvern, PA 19355 / US
	08 / ZHANG, Wei, Yuan 154 Hunsicker Drive Collegeville, PA 19426 / US
	[1998/52]
Representative(s)	Melzer, Wolfgang, et al Mitscherlich PartmbB Patent- und Rechtsanwälte Postfach 33 06 09 80066 München / DE
	[N/P]
Former [1998/52]	Melzer, Wolfgang, Dipl.-Ing., et al Patentanwälte Mitscherlich & Partner, Sonnenstrasse 33 80331 München / DE
Application number, filing date	97914850.9	01.03.1997
	[1998/52]
	WO1997US03353
Priority number, date	US19960612680	08.03.1996 Original published format: US 612680
	US19970796078	05.02.1997 Original published format: US 796078
	[1999/50]
Former [1998/52]	US19960612680	08.03.1996
Filing language	EN
Procedural language	EN
Publication	Type:	A1 Application with search report
	No.:	WO9732857
	Date:	12.09.1997
	Language:	EN
	[1997/39]
	Type:	A1 Application with search report
	No.:	EP0885199
	Date:	23.12.1998
	Language:	EN
	The application published by WIPO in one of the EPO official languages on 12.09.1997 takes the place of the publication of the European patent application.
	[1998/52]
Search report(s)	International search report - published on:	US	12.09.1997
	(Supplementary) European search report - dispatched on:	EP	17.10.2000
Classification	IPC:	C07D241/04, C07D403/06, A61K31/495, C07F9/40, C07D295/12, C07F9/24, C07D207/12, C07D403/12, C07D401/12	[2000/46]
	CPC:	C07D295/073 (EP,KR,US); C07D241/04 (EP,KR,US); A61K31/404 (EP,KR,US); A61K31/4439 (EP,KR,US); A61P25/04 (EP); C07D207/06 (KR); (+) C07D209/32 (KR); C07D209/42 (EP,KR,US); C07D213/56 (EP,KR,US); C07D401/06 (KR); C07D401/12 (KR); C07D403/12 (KR) (-)
	Former IPC [2000/11]	C07D241/04, C07D403/06, A61K31/495, C07F9/40
	Former IPC [1998/52]	C07D241/04, C07D403/06, A61K31/495
Designated contracting states	AT, BE, CH, DE, DK, ES, FI, FR, GB, GR, IE, IT, LI, NL, PT, SE [1998/52]
Title	German:	KAPPA AGONIST-VERBINDUNGEN UND PHARMAZEUTISCHE ZUBEREITUNGEN DAVON	[1998/52]
	English:	KAPPA AGONIST COMPOUNDS AND PHARMACEUTICAL FORMULATIONS THEREOF	[1998/52]
	French:	COMPOSES AGONISTES DU KAPPA ET LEURS PREPARATIONS PHARMACEUTIQUES	[1998/52]
Entry into regional phase	07.09.1998	National basic fee paid
	07.09.1998	Search fee paid
	07.09.1998	Designation fee(s) paid
	07.09.1998	Examination fee paid
Examination procedure	26.09.1997	Request for preliminary examination filed International Preliminary Examining Authority: US
	07.09.1998	Examination requested [1998/52]
	29.04.2002	Despatch of a communication from the examining division (Time limit: M06)
	02.10.2002	Reply to a communication from the examining division
	18.02.2005	Despatch of a communication from the examining division (Time limit: M06)
	26.08.2005	Reply to a communication from the examining division
	03.10.2006	Application deemed to be withdrawn, date of legal effect [2007/17]
	10.11.2006	Despatch of communication that the application is deemed to be withdrawn, reason: renewal fee not paid in time [2007/17]
Fees paid	Renewal fee
	30.03.1999	Renewal fee patent year 03
	30.03.2000	Renewal fee patent year 04
	27.03.2001	Renewal fee patent year 05
	13.03.2002	Renewal fee patent year 06
	11.03.2003	Renewal fee patent year 07
	15.03.2004	Renewal fee patent year 08
	14.03.2005	Renewal fee patent year 09
	Penalty fee
	Additional fee for renewal fee
	31.03.2006	10 M06 Not yet paid
Opt-out from the exclusive Tooltip competence of the Unified Patent Court	See the Register of the Unified Patent Court for opt-out data
	Responsibility for the accuracy, completeness or quality of the data displayed under the link provided lies entirely with the Unified Patent Court.
Documents cited:	Search	[DX]US4145435 (SZMUSZKOVICZ JACOB) [DX] 46,48,49,51 * column 3, line 42 - column 4, line 35 * * column 27 - column 36; example - * * column 3, line 6 - line 15 *;
		[X]US4360531 (MCMILLAN MOSES W, et al) [X] 46,49 * column 2, line 57 - column 3, line 55 * * column 2, line 3 - line 9 *;
		[DA]US4438130 (KAPLAN LESTER J [US]) [DA] 47 * column 3, line 7 - line 64 * * column 2, line 18 - line 29 *;
		[X]EP0108602 (UPJOHN CO [US]) [X] 46 * page 43; claim 1 * * page 30, line 3 - line 4 * * page 30, line 33 - line 34 * * page 1, line 1 - line 3 *;
		[X]EP0254545 (ICI PLC [GB]) [X] 31-36 * page 26 - page 27; claim 1 * * page 6, line 34 - line 35 * * page 6, line 49 * * page 10; the compound no. 28 *;
		[XY]EP0260555 (DU PONT [US]) [X] 18,21 * page 29 - page 30; claim 1 * * page 27, line 56 - line 57 * * page 29 - page 30; claim 1 * * page 11 - page 13; example 1 * [Y] 16-21;
		[X]EP0261842 (ZAMBELETTI SPA L [IT]) [X] 31-36 * page 23; claim 1 * * pages 19-20; table I, the examples no. 8, 10, 12 and 14 * * page 2, line 8 - line 10 *;
		[Y]EP0325406 (ICI PLC [GB]) [Y] 16-21 * page 2, line 20 - line 27 * * page 14; claim 1 * * page 7 - page 8; example 1 *;
		[X]EP0329563 (ROUSSEL UCLAF [FR]) [X] 18,21 * page 19 - page 20; claim 1 * * page 9, line 11 - line 13 *;
		[X]EP0343900 (GLAXO GROUP LTD [GB]) [X] 2,3,5,6,8,9,11,12,14,15 * page 22; claim 1 * * page 3, line 2 - line 3 *;
		[X]EP0356247 (SANKYO CO [JP]) [X] 3,6,9,12,15 * page 30; claim 1 * * page 10; table . *;
		[X]EP0374054 (ROUSSEL UCLAF [FR]) [X] 18,21 * page 20 - page 21; claim 1 * * page 9, line 29 - line 30 *;
		[X]EP0398720 (GLAXO GROUP LTD [GB]) [X] 3,6,9,12,15 * page 20 - page 21; claim 1 * * page 2, line 2 - line 3 *;
		[X]EP0483580 (MERCK PATENT GMBH [DE]) [X] 31-36 * page 14; claim 1 * * page 8, line 27 * * page 2, line 43 - line 56 *;
		[X]EP0569802 (MERCK PATENT GMBH [DE]) [X] 33,36 * page 15 - page 16; claim 1 * * page 7, line 40 * * page 3, line 19 - line 20 *;
		[X]US5475019 (PRIVETTE THOMAS H [US], et al) [X] 46,48,52,54 * column 1, line 51 - column 2, line 36 *;
		[E]WO9720831 (UNIV MINNESOTA [US]) [E] 31 * page 32; claim 1 * * page 20 - page 24; examples X,XI,XIII,XIV *;
		[X] - WEERAWARNA S A, "Isothiocyanate-Substituted kappa-Selective Opioid Receptor Ligands Derived from N-Methyl-N-[(1S)-1-phenyl-2-(1-pyrrolidinyl)ethyl]phenylacetamide", JOURNAL OF MEDICINAL CHEMISTRY., AMERICAN CHEMICAL SOCIETY. WASHINGTON., US, (19940902), vol. 37, no. 18, ISSN 0022-2623, pages 2856 - 2864, XP002148135 [X] 33 * page 2857; scheme 1, see, the compounds no. 11-14 and 19-22 * DOI: http://dx.doi.org/10.1021/jm00044a006
		[X] - DE COSTA B R ET AL, "Synthesis of an affinity ligand ('UPHIT') for in vivo acylation of the kappa-opioid receptor", FEBS LETTERS., ELSEVIER SCIENCE PUBLISHERS, AMSTERDAM., NL, (198906), vol. 249, no. 2, ISSN 0014-5793, pages 178 - 182, XP000940483 [X] 46,48 * page 180, column 1, paragraph 3 - column 2, paragraph 2 * DOI: http://dx.doi.org/10.1016/0014-5793(89)80619-2
		[A] - SCOPES D I C, "Selective non-peptide kappa opioid receptor agonists", EXPERT OPINION ON INVESTIGATIONAL DRUGS,GB,ASHLEY PUBLICATIONS LTD., LONDON, vol. 3, no. 4, ISSN 1354-3784, page 369-376, XP000196256 [A] 1-60 * see the whole document; in particular, page 370, column 1, fifth paragraph - column 2, first paragraph *
		[A] - GIARDINA G ET AL, "Central and peripheral analgesic agents: chemical strategies for limiting brain penetration in kappa-opioid agonists belonging to different chemical classes", FARMACO,IT,SOCIETA CHIMICA ITALIANA, PAVIA, (1995), vol. 50, no. 6, ISSN 0014-827X, pages 405 - 418, XP000910055 [A] 1-3,16-18,31-33,46-48 * see the whole document; in particular, page 406, column 2, third paragraph - page 407, column 1, second paragraph *
	International search	[A]US4212878 (LEDNICER DANIEL [US], et al)

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