EP0995751 - Pyrazolopyrimidinone cGMP PDE5 inhibitors for the treatment of sexual dysfunction [Right-click to bookmark this link] | Status | No opposition filed within time limit Status updated on 12.05.2006 Database last updated on 16.07.2024 | Most recent event Tooltip | 20.04.2007 | Lapse of the patent in a contracting state New state(s): CY, LU | published on 23.05.2007 [2007/21] | Applicant(s) | For:AT
BE
CH
DE
DK
ES
FI
FR
GR
IE
IT
LI
LU
MC
NL
CY
PT
SE
Pfizer Inc. 235 East 42nd Street New York, NY 10017 / US | For:GB
Pfizer Limited Ramsgate Road Sandwich, Kent CT13 9NJ / GB | [N/P] |
Former [2005/26] | For:AT
BE
CH
DE
DK
ES
FI
FR
GR
IE
IT
LI
LU
MC
NL
CY
PT
SE
PFIZER INC. 235 East 42nd Street New York, N.Y. 10017 / US | ||
For:GB
Pfizer Limited Ramsgate Road Sandwich, Kent CT13 9NJ / GB | |||
Former [2000/17] | For:AT
BE
CH
DE
DK
ES
FI
FR
GR
IE
IT
LI
LU
MC
NL
CY
PT
SE
PFIZER INC. 235 East 42nd Street New York, N.Y. 10017 / US | ||
For:GB
Pfizer Limited Ramsgate Road Sandwich Kent CT13 9NJ / GB | Inventor(s) | 01 /
Bunnage, Mark Edward, Pfizer Central Research Ramsgate Road Sandwich, Kent CT13 9NJ / GB | 02 /
Street, Stephen Derek Albert, Pfizer Central Res. Ramsgate Road Sandwich, Kent CT13 9NJ / GB | 03 /
Mathias, John Paul, Pfizer Central Research Ramsgate Road Sandwich, Kent CT13 9NJ / GB | 04 /
Wood, Anthony, Pfizer Central Research Ramsgate Road Sandwich, Kent CT13 9NJ / GB | [2000/17] | Representative(s) | Edwards, Fiona Anne Pfizer Limited, UK Patents Department, Ramsgate Road Sandwich Kent CT13 9NJ / GB | [N/P] |
Former [2005/23] | Edwards, Fiona Anne Pfizer Limited, UK Patents Department, Ramsgate Road Sandwich, Kent CT13 9NJ / GB | ||
Former [2000/17] | McNeeney, Stephen Phillip Eric Potter Clarkson, Park View House, 58 The Ropewalk Nottingham NG1 5DD / GB | Application number, filing date | 99308158.7 | 15.10.1999 | [2000/17] | Priority number, date | GB19980023103 | 23.10.1998 Original published format: GB 9823103 | [2000/17] | Filing language | EN | Procedural language | EN | Publication | Type: | A2 Application without search report | No.: | EP0995751 | Date: | 26.04.2000 | Language: | EN | [2000/17] | Type: | A3 Search report | No.: | EP0995751 | Date: | 18.10.2000 | [2000/42] | Type: | B1 Patent specification | No.: | EP0995751 | Date: | 29.06.2005 | Language: | EN | [2005/26] | Search report(s) | (Supplementary) European search report - dispatched on: | EP | 30.08.2000 | Classification | IPC: | C07D487/04, A61K31/506, C07D231/14, C07D401/12, // (C07D487/04, 239:00, 213:00) | [2000/17] | CPC: |
C07D487/04 (EP,US);
A61P1/00 (EP);
A61P11/00 (EP);
A61P11/06 (EP);
A61P13/00 (EP);
A61P13/08 (EP);
A61P13/10 (EP);
A61P15/10 (EP);
A61P17/00 (EP);
A61P17/06 (EP);
A61P17/14 (EP);
A61P25/00 (EP);
A61P25/28 (EP);
A61P27/06 (EP);
A61P35/04 (EP);
A61P43/00 (EP);
A61P9/00 (EP);
A61P9/10 (EP);
A61P9/12 (EP)
(-)
| Designated contracting states | AT, BE, CH, CY, DE, DK, ES, FI, FR, GB, GR, IE, IT, LI, LU, MC, NL, PT, SE [2000/17] | Title | German: | Pyrazolopyrimidinone cGMP PDE5 Inhibitoren zur Behandlung der sexuellen Dysfunktion | [2000/17] | English: | Pyrazolopyrimidinone cGMP PDE5 inhibitors for the treatment of sexual dysfunction | [2000/17] | French: | Inhibiteurs de cGMP PDE5 de pyrazolopyrimidinone servant à traiter le dysfonctionnement sexuel | [2000/17] | Examination procedure | 03.11.2000 | Examination requested [2001/01] | 26.03.2003 | Despatch of a communication from the examining division (Time limit: M04) | 25.07.2003 | Reply to a communication from the examining division | 29.09.2004 | Date of oral proceedings | 15.10.2004 | Minutes of oral proceedings despatched | 17.12.2004 | Communication of intention to grant the patent | 27.04.2005 | Fee for grant paid | 27.04.2005 | Fee for publishing/printing paid | Opposition(s) | 30.03.2006 | No opposition filed within time limit [2006/24] | Fees paid | Renewal fee | 11.10.2001 | Renewal fee patent year 03 | 07.10.2002 | Renewal fee patent year 04 | 14.10.2003 | Renewal fee patent year 05 | 14.10.2004 | Renewal fee patent year 06 |
Opt-out from the exclusive Tooltip competence of the Unified Patent Court | See the Register of the Unified Patent Court for opt-out data | ||
Responsibility for the accuracy, completeness or quality of the data displayed under the link provided lies entirely with the Unified Patent Court. | Lapses during opposition Tooltip | AT | 29.06.2005 | BE | 29.06.2005 | CH | 29.06.2005 | FI | 29.06.2005 | LI | 29.06.2005 | NL | 29.06.2005 | DK | 29.09.2005 | GR | 29.09.2005 | SE | 29.09.2005 | CY | 15.10.2005 | LU | 31.10.2005 | MC | 31.10.2005 | PT | 07.12.2005 | [2007/21] |
Former [2006/30] | AT | 29.06.2005 | |
BE | 29.06.2005 | ||
CH | 29.06.2005 | ||
FI | 29.06.2005 | ||
LI | 29.06.2005 | ||
NL | 29.06.2005 | ||
DK | 29.09.2005 | ||
GR | 29.09.2005 | ||
SE | 29.09.2005 | ||
MC | 31.10.2005 | ||
PT | 07.12.2005 | ||
Former [2006/26] | AT | 29.06.2005 | |
BE | 29.06.2005 | ||
CH | 29.06.2005 | ||
FI | 29.06.2005 | ||
LI | 29.06.2005 | ||
NL | 29.06.2005 | ||
DK | 29.09.2005 | ||
GR | 29.09.2005 | ||
SE | 29.09.2005 | ||
PT | 07.12.2005 | ||
Former [2006/22] | AT | 29.06.2005 | |
BE | 29.06.2005 | ||
CH | 29.06.2005 | ||
FI | 29.06.2005 | ||
LI | 29.06.2005 | ||
NL | 29.06.2005 | ||
GR | 29.09.2005 | ||
SE | 29.09.2005 | ||
PT | 07.12.2005 | ||
Former [2006/14] | AT | 29.06.2005 | |
BE | 29.06.2005 | ||
CH | 29.06.2005 | ||
FI | 29.06.2005 | ||
LI | 29.06.2005 | ||
GR | 29.09.2005 | ||
SE | 29.09.2005 | ||
PT | 07.12.2005 | ||
Former [2006/13] | AT | 29.06.2005 | |
BE | 29.06.2005 | ||
FI | 29.06.2005 | ||
SE | 29.09.2005 | ||
Former [2005/52] | FI | 29.06.2005 | |
SE | 29.09.2005 | ||
Former [2005/50] | SE | 29.09.2005 | Documents cited: | Search | [YX]JPH08253484 ; | [XDY]WO9307149 (PFIZER LTD [GB], et al) [XD] 1-16 * see examples 2 and 10 *; column W * [Y] 19,20; | [Y]WO9400453 (PFIZER LTD [GB], et al) [Y] 1-16,19,20 * column W *; | [Y]WO9428902 (PFIZER LTD [GB], et al) [Y] 1-16,19,20 * column W *; | [YX]EP0636626 (GLAXO LAB SA [FR]) [Y] 1-16,19,20 * see page 7, formula II *; column W * [X] 17,18; | [XDY]WO9616657 (PFIZER LTD [GB], et al) [XD] 1-16 * see page 9, 5th ex. *; column W * [Y] 19,20; | [Y]WO9628448 (SANOFI WINTHROP INC [US]) [Y] 1-16 * column W *; | [Y]WO9628429 (SANOFI WINTHROP INC [US]) [Y] 1-16 * column W *; | [Y]EP0812845 (PFIZER LTD [GB], et al) [Y] 17,18 * see page 5 ,scheme, ex. (II) *; column W *; | [PX]WO9849166 (PFIZER LTD [GB], et al) [PX] 1-16,19,20,17,18 * see page 11, cpd. (VI); page 13, cpds. (IXA), (IXB) *; column W *; | [E]WO9954333 (PFIZER [US], et al) [E] 1-20* column W *; | [Y] - DUMAITRE B ET AL, "SYNTHESIS AND CYCLIC GMP PHOSPHODIESTERASE INHIBITORY ACTIVITY OF A SERIES OF 6-PHENYLPYRAZOLO- 3,4-DIHYDRO-PYRIMIDONES", JOURNAL OF MEDICINAL CHEMISTRY,US,AMERICAN CHEMICAL SOCIETY. WASHINGTON, (19960101), vol. 39, no. 8, ISSN 0022-2623, pages 1635 - 1644, XP002024856 [Y] 1-16 * column W * DOI: http://dx.doi.org/10.1021/jm950812j | [YX] - PATENT ABSTRACTS OF JAPAN, (19970228), vol. 1997, no. 02, & JP08253484 A 19961001 (TAISHO PHARMACEUT CO LTD) [Y] 1-16 * abstract * [X] 17,18 | [Y] - TERRETT N K ET AL, "Sildenafil (VIAGRA), a potent and selective inhibitor of type 5 CGMP phosphodiesterase with utility for the treatment of male erectile dysfunction", BIOORGANIC & MEDICINAL CHEMISTRY LETTERS,GB,OXFORD, (19960806), vol. 6, no. 15, ISSN 0960-894X, pages 1819 - 1824, XP004135609 [Y] 1-16,19,20,17,18 * see p.1823,, ex. 5 *; column W * DOI: http://dx.doi.org/10.1016/0960-894X(96)00323-X |