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Extract from the Register of European Patents

EP About this file: EP1056450

EP1056450 - FARNESYL-PROTEIN TRANSFERASE INHIBITORS [Right-click to bookmark this link]
StatusThe application is deemed to be withdrawn
Status updated on  17.01.2003
Database last updated on 17.09.2024
Most recent event   Tooltip17.01.2003Application deemed to be withdrawnpublished on 05.03.2003  [2003/10]
Applicant(s)For all designated states
International Phytochemistry Research Labs, Ltd.
Suite 107, 4870 Haygood Road
Virginia Beach, VA 23455 / US
[2000/49]
Inventor(s)01 / SHAIKENOV, Tattym, E.
ALMATY / KZ
02 / ADEKENOV, Sergazy, M.
Karaganda / KZ
[2000/49]
Representative(s)Jones, Helen M.M., et al
Gill Jennings & Every LLP The Broadgate Tower
20 Primrose Street
London EC2A 2ES / GB
[N/P]
Former [2000/49]Jones, Helen Marjorie Meredith, et al
Gill Jennings & Every, Broadgate House, 7 Eldon Street
London EC2M 7LH / GB
Application number, filing date99908471.825.02.1999
[2000/49]
WO1999US04124
Priority number, dateUS1998003030025.02.1998         Original published format: US 30300
[2000/49]
Filing languageEN
Procedural languageEN
PublicationType: A2 Application without search report
No.:WO9943314
Date:02.09.1999
[1999/35]
Type: A1 Application with search report 
No.:EP1056450
Date:06.12.2000
Language:EN
The application published by WIPO in one of the EPO official languages on 02.09.1999 takes the place of the publication of the European patent application.
[2000/49]
Search report(s)International search report - published on:US01.03.2001
(Supplementary) European search report - dispatched on:EP18.04.2001
ClassificationIPC:A61K31/34, A61K31/66, C07C53/136, C07D307/93, C07D407/02
[2000/49]
CPC:
A61K31/34 (EP,KR,US); A61K31/343 (EP,US); A61K31/365 (EP,US);
A61K31/475 (EP,US); A61K31/505 (EP,US); A61K31/5377 (EP,US);
A61K31/66 (EP,US); A61K31/675 (EP,US); A61K33/24 (EP);
A61K45/06 (EP,US); A61P35/00 (EP); A61P43/00 (EP);
C07D303/38 (EP,US); C07D307/93 (EP,US); C07D307/935 (EP,US);
C07D493/04 (EP,US); C07D493/10 (EP,US); C07F9/098 (EP,US) (-)
C-Set:
A61K31/365, A61K2300/00 (EP,US);
A61K31/475, A61K2300/00 (US,EP);
A61K31/505, A61K2300/00 (US,EP);
A61K31/675, A61K2300/00 (US,EP);
A61K33/24, A61K2300/00 (EP,US)
(-)
Designated contracting statesAT,   BE,   CH,   CY,   DE,   DK,   ES,   FI,   FR,   GB,   GR,   IE,   IT,   LI,   LU,   MC,   NL,   PT,   SE [2000/49]
Extension statesAL25.09.2000
LT25.09.2000
LV25.09.2000
MK25.09.2000
RO25.09.2000
SI25.09.2000
TitleGerman:FARNESYL-PROTEIN TRANSFERASE INHIBITOREN[2000/49]
English:FARNESYL-PROTEIN TRANSFERASE INHIBITORS[2000/49]
French:INHIBITEURS DE FARNESYL PROTEINE TRANSFERASE[2000/49]
Entry into regional phase25.09.2000National basic fee paid 
25.09.2000Search fee paid 
25.09.2000Designation fee(s) paid 
25.09.2000Examination fee paid 
Examination procedure20.09.1999Request for preliminary examination filed
International Preliminary Examining Authority: US
25.09.2000Examination requested  [2000/49]
03.09.2002Application deemed to be withdrawn, date of legal effect  [2003/10]
07.10.2002Despatch of communication that the application is deemed to be withdrawn, reason: renewal fee not paid in time  [2003/10]
Fees paidRenewal fee
15.02.2001Renewal fee patent year 03
Penalty fee
Additional fee for renewal fee
28.02.200204   M06   Not yet paid
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Responsibility for the accuracy, completeness or quality of the data displayed under the link provided lies entirely with the Unified Patent Court.
Documents cited:Search[PX]WO9848789  (PARACURE INC DOING BUSINESS AS [US]) [PX] 6-8 * page 9, lines 5,6 * * tables III,IV * * example 6 *;
 [Y]  - OVERHAND M ET AL, "Synthesis of triphosphonate analogues of farnesyl pyrophosphate. Inhibitors of squalene synthase and protein:farnesyl transferase", BIOORGANIC & MEDICINAL CHEMISTRY LETTERS,GB,OXFORD, (19970923), vol. 7, no. 18, ISSN 0960-894X, pages 2435 - 2440, XP004136459 [Y] 1-23 * formula A *

DOI:   http://dx.doi.org/10.1016/S0960-894X(97)00448-4
 [Y]  - SHAIKENOV ET AL, "Arglabine as a novel inhibitor of the farnesylation of Ras proteins", STN CAPLUS, XP002114697 [Y] 1-23 * abstract *
International search[X]  - ADEKENOV, ET AL., ""THE CHEMISTRY OF SESQUITERPENE LACTONES"", CHEMISTRY OF SESQUITERPENE LACTONES, XX, XX, XX, (19900101), pages 01 - 17 + 20, XP002919766
 [X]  - BLANCO J. G., ET AL., "A NOVEL ACTIVITY FOR A GROUP OF SESQUITERPENE LACTONES: INHIBITION OF AROMATASE.", FEBS LETTERS., ELSEVIER, AMSTERDAM., NL, NL, (19970101), vol. 409., doi:10.1016/S0014-5793(97)00560-7, ISSN 0014-5793, pages 396 - 400., XP002919765

DOI:   http://dx.doi.org/10.1016/S0014-5793(97)00560-7
The EPO accepts no responsibility for the accuracy of data originating from other authorities; in particular, it does not guarantee that it is complete, up to date or fit for specific purposes.