EP1144403 - SUBSTITUTED PYRAZOLES AS P38 KINASE INHIBITORS [Right-click to bookmark this link] | |||
Former [2001/42] | SUBSTITUED PYRAZOLES AS P38 KINASE INHIBITORS | ||
[2004/32] | Status | No opposition filed within time limit Status updated on 12.08.2005 Database last updated on 31.08.2024 | Most recent event Tooltip | 26.09.2008 | Change - representative | published on 29.10.2008 [2008/44] | Applicant(s) | For all designated states G.D. Searle LLC 575 Maryville Centre Drive St. Louis, Missouri 63141 / US | [2004/19] |
Former [2001/42] | For all designated states G.D. SEARLE & CO. P.O. Box 5110 Chicago, IL 60680-5110 / US | Inventor(s) | 01 /
Anantanarayan, Ashok 54 Lisk Drive Hainesville, IL 60030 / US | 02 /
Clare, Michael 5154 West Brown Street Skokie, IL 60077 / US | 03 /
Collins, Paul W. 2317 Carillon Drive Grayslake, IL 60030 / US | 04 /
Crich, Joyce Z. 1501 G. Topp Lane Glenview, IL 60025 / US | 05 /
Devraj, Rajesh 1331 Oak Borough Drive Ballwin, MO 63021 / US | 06 /
Flynn, Daniel One Amgen Center Drive Thousand Oaks, CA 91320 / US | 07 /
Geng, Lifeng 5300 Davis Street Skokie, IL 60077 / US | 08 /
Graneto, Matthew J. 352 Hartwell Court Chesterfield, MO 63017 / US | 09 /
Hanau, Cathleen E. 15551 Wendimill Drive Chesterfield, MO 63017 / US | 10 /
Hanson, Gunnar J. 7410 Keystone Avenue Skokie, IL 60077 / US | 11 /
Hartmann, Susan J. 613 West Essex Avenue Kirkwood, MO 63122 / US | 12 /
Hepperle, Michael 1460 Keystone Court St. Charles, MO 63303 / US | 13 /
Huang, He 2309 F S. Stewart Avenue Chicago, IL 60616 / US | 14 /
Khanna, Ish K. 1821 S. Falcon Drive Libertyville, IL 60048 / US | 15 /
Koszyk, Francis J. 11 Wildwood Drive South Prospect Heights, IL 60070 / US | 16 /
Liao, Shuyuan 1536 Walters Avenue Northbrook, IL 60062 / US | 17 /
Metz, Suzanne 525 Westernmill Drive Chesterfield, MO 63017 / US | 18 /
Partis, Richard A. 2221 Noyes Street Evanston, IL 60201 / US | 19 /
Perry, Thao D. 516 Bloom Street Red Bud, IL 62278 / US | 20 /
Rao, Shashidhar N. 736 Bellerive Manor Drive St. Louis, MO 63141 / US | 21 /
Selness, Shaun Raj 1875 Cedarmill Drive Chesterfield, MO 63017 / US | 22 /
South, Michael S. 11671 Cheiftain Drive Chesterfield, MO 63146 / US | 23 /
Stealey, Michael A. 502 Juniper Parkway Libertyville, IL 60048 / US | 24 /
Talley, John Jeffrey 4701 Clifton Avenue St. Louis, MO 63109 / US | 25 /
Vazquez, Michael L. 614 Castle Meadows Court Ballwin, MO 63021 / US | 26 /
Weier, Richard M. 240 Hickory Court Lake Bluff, IL 60044 / US | 27 /
Xu, Xiangdong 7498 Abbey Road Gurnee, IL 60031 / US | 28 /
BALDUS, John E. 2340 Louisiana Avenue St. Louis, MO 63104 / US | 29 /
JEROME, Kevin D. 2339 Pheasant Run Drive Maryland Heights, MO 63043 / US | 30 /
NAING, Win 1198 Nooning Tree Drive Chesterfield, MO 63017 / US | 31 /
WALKER, John K. 11946 Autumn Lakes Drive Maryland Heights, MO 63043 / US | 32 /
YANG, Syaulan 2157 Englewood Terrace Chesterfield, MO 63017 / US | 33 /
YU, Yi 1019 Castle Dr. Glenview, IL 60025 / US | [2004/29] |
Former [2004/02] | 01 /
Anantanarayan, Ashok 54 Lisk Drive Hainesville, IL 60030 / US | ||
02 /
Clare, Michael 5154 West Brown Street Skokie, IL 60077 / US | |||
03 /
Collins, Paul W. 2317 Carillon Drive Grayslake, IL 60030 / US | |||
04 /
Crich, Joyce Z. 1501 G. Topp Lane Glenview, IL 60025 / US | |||
05 /
Devraj, Rajesh 1331 Oak Borough Drive Ballwin, MO 63021 / US | |||
06 /
Flynn, Daniel One Amgen Center Drive Thousand Oaks, CA 91320 / US | |||
07 /
Geng, Lifeng 5300 Davis Street Skokie, IL 60077 / US | |||
08 /
Graneto, Matthew J. 352 Hartwell Court Chesterfield, MO 63017 / US | |||
09 /
Hanau, Cathleen E. 15551 Wendimill Drive Chesterfield, MO 63017 / US | |||
10 /
Hanson, Gunnar J. 7410 Keystone Avenue Skokie, IL 60077 / US | |||
11 /
Hartmann, Susan J. 613 West Essex Avenue Kirkwood, MO 63122 / US | |||
12 /
Hepperle, Michael 1460 Keystone Court St. Charles, MO 63303 / US | |||
13 /
Huang, He 2309 F S. Stewart Avenue Chicago, IL 60616 / US | |||
14 /
Khanna, Ish K. 1821 S. Falcon Drive Libertyville, IL 60048 / US | |||
15 /
Koszyk, Francis J. 11 Wildwood Drive South Prospect Heights, IL 60070 / US | |||
16 /
Liao, Shuyuan 1536 Walters Avenue Northbrook, IL 60062 / US | |||
17 /
Metz, Suzanne 525 Westernmill Drive Chesterfield, MO 63017 / US | |||
18 /
Partis, Richard A. 2221 Noyes Street Evanston, IL 60201 / US | |||
19 /
Perry, Thao D. 516 Bloom Street Red Bud, IL 62278 / US | |||
20 /
Rao, Shashidhar N. 736 Bellerive Manor Drive St. Louis, MO 63141 / US | |||
21 /
Selness, Shaun Raj 1875 Cedarmill Drive Chesterfiedl, MO 63017 / US | |||
22 /
South, Michael S. 11671 Cheiftain Drive Chesterfield, MO 63146 / US | |||
23 /
Stealey, Michael A. 502 Juniper Parkway Libertyville, IL 60048 / US | |||
24 /
Talley, John Jeffrey 4701 Clifton Avenue St. Louis, MO 63109 / US | |||
25 /
Vazquez, Michael L. 614 Castle Meadows Court Ballwin, MO 63021 / US | |||
26 /
Weier, Richard M. 240 Hickory Court Lake Bluff, IL 60044 / US | |||
27 /
Xu, Xiangdong 7498 Abbey Road Gurnee, IL 60031 / US | |||
28 /
BALDUS, John E. 2340 Louisiana Avenue St. Louis, MO 63104 / US | |||
29 /
JEROME, Kevin D. 2339 Pheasant Run Drive Maryland Heights, MO 63043 / US | |||
30 /
NAING, Win 1198 Nooning Tree Drive Chesterfield, MO 63017 / US | |||
31 /
WALKER, John K. 11946 Autumn Lakes Drive Maryland Heights, MO 63043 / US | |||
32 /
YANG, Syaulan 2157 Englewood Terrace Chesterfield, MO 63017 / US | |||
33 /
YU, Yi 1019 Castle Dr. Glenview, IL 60025 / US | |||
Former [2003/49] | 01 /
Anantanarayan, Ashok 54 Lisk Drive Hainesville, IL 60030 / US | ||
02 /
Clare, Michael 5154 West Brown Street Skokie, IL 60077 / US | |||
03 /
Collins, Paul W. 2317 Carillon Drive Grayslake, IL 60030 / US | |||
04 /
Crich, Joyce Z. 1501 G. Topp Lane Glenview, IL 60025 / US | |||
05 /
Devraj, Rajesh 1331 Oak Borough Drive Ballwin, MO 63021 / US | |||
06 /
Flynn, Daniel One Amgen Center Drive Thousand Oaks, CA 91320 / US | |||
07 /
Geng, Lifeng 5300 Davis Street Skokie, IL 60077 / US | |||
08 /
Graneto, Matthew J. 352 Hartwell Court Chesterfield, MO 63017 / US | |||
09 /
Hanau, Cathleen E. 15551 Wendimill Drive Chesterfield, MO 63017 / US | |||
10 /
Hanson, Gunnar J. 7410 Keystone Avenue Skokie, IL 60077 / US | |||
11 /
Hartmann, Susan J. 613 West Essex Avenue Kirkwood, MO 63122 / US | |||
12 /
Hepperle, Michael 1460 Keystone Court St. Charles, MO 63303 / US | |||
13 /
Huang, He 2309 F S. Stewart Avenue Chicago, IL 60616 / US | |||
14 /
Khanna, Ish K. 1821 S. Falcon Drive Libertyville, IL 60048 / US | |||
15 /
Koszyk, Francis J. 11 Wildwood Drive South Prospect Heights, IL 60070 / US | |||
16 /
Liao, Shuyuan 1536 Walters Avenue Northbrook, IL 60062 / US | |||
17 /
Metz, Suzanne 525 Westernmill Drive Chesterfield, MO 63017 / US | |||
18 /
Partis, Richard A. 2221 Noyes Street Evanston, IL 60201 / US | |||
19 /
Perry, Thao D. 516 Bloom Street Red Bud, IL 62278 / US | |||
20 /
Rao, Shashidhar N. 736 Bellerive Manor Drive St. Louis, MO 63141 / US | |||
21 /
Selness, Shaun Raj 1875 Cedarmill Drive Chesterfiedl, MO 63017 / US | |||
22 /
South, Michael S. 11671 Cheiftain Drive Chesterfield, MO 63146 / US | |||
23 /
Stealey, Michael A. 502 Juniper Parkway Libertyville, IL 60048 / US | |||
24 /
Talley, John Jeffrey 4701 Clifton Avenue St. Louis, MO 63109 / US | |||
25 /
Vazquez, Michael L. 614 Castle Meadows Court Ballwin, MO 63021 / US | |||
26 /
Weier, Richard M. 240 Hickory Court Lake Bluff, IL 60044 / US | |||
27 /
Xu, Xiangdong 7498 Abbey Road Gurnee, IL 60031 / US | |||
28 /
BALDUS, John E. 2340 Louisiana Avenue St. Louis, MO 63104 / US | |||
29 /
JEROME, Kevin D. 2339 Pheasant Run Drive Maryland Heights, MO 63043 / US | |||
30 /
NAING, Win 1198 Nooning Tree Drive Chesterfield, MO 63017 / US | |||
31 /
WALKER, John K. 11949 Autumn Lakes Drive Maryland Heights, MO 63043 / US | |||
32 /
YANK, Syaulan 2157 Englewood Terrace Chesterfield, MO 63017 / US | |||
33 /
YU, Yi 1019 Castle Dr. Glenview, IL 60025 / US | |||
Former [2003/48] | 01 /
Anantanarayan, Ashok 54 Lisk Drive Hainesville, IL 60030 / US | ||
02 /
Clare, Michael 5154 West Brown Street Skokie, IL 60077 / US | |||
03 /
Collins, Paul W. 2317 Carillon Drive Grayslake, IL 60030 / US | |||
04 /
Crich, Joyce Z. 1501 G. Topp Lane Glenview, IL 60025 / US | |||
05 /
Devraj, Rajesh 1331 Oak Borough Drive Ballwin, MO 63021 / US | |||
06 /
Flynn, Daniel One Amgen Center Drive Thousand Oaks, CA 91320 / US | |||
07 /
Geng, Lifeng 5300 Davis Street Skokie, IL 60077 / US | |||
08 /
Graneto, Matthew J. 352 Hartwell Court Chesterfield, MO 63017 / US | |||
09 /
Hanau, Cathleen E. 15551 Wendimill Drive Chesterfield, MO 63017 / US | |||
10 /
Hanson, Gunnar J. 7410 Keystone Avenue Skokie, IL 60077 / US | |||
11 /
Hartmann, Susan J. 613 West Essex Avenue Kirkwood, MO 63122 / US | |||
12 /
Hepperle, Michael 1460 Keystone Court St. Charles, MO 63303 / US | |||
13 /
Huang, He 2309 F S. Stewart Avenue Chicago, IL 60616 / US | |||
14 /
Khanna, Ish K. 1821 S. Falcon Drive Libertyville, IL 60048 / US | |||
15 /
Koszyk, Francis J. 11 Wildwood Drive South Prospect Heights, IL 60070 / US | |||
16 /
Liao, Shuyuan 1536 Walters Avenue Northbrook, IL 60062 / US | |||
17 /
Metz, Suzanne 525 Westernmill Drive Chesterfield, MO 63017 / US | |||
18 /
Partis, Richard A. 2221 Noyes Street Evanston, IL 60201 / US | |||
19 /
Perry, Thao D. 516 Bloom Street Red Bud, IL 62278 / US | |||
20 /
Rao, Shashidhar N. 736 Bellerive Manor Drive St. Louis, MO 63141 / US | |||
21 /
Selness, Shaun Raj 1875 Cedarmill Drive Chesterfiedl, MO 63017 / US | |||
22 /
South, Michael S. 11671 Cheiftain Drive Chesterfield, MO 63146 / US | |||
23 /
Stealey, Michael A. 502 Juniper Parkway Libertyville, IL 60048 / US | |||
24 /
Talley, John Jeffrey 4701 Clifton Avenue St. Louis, MO 63109 / US | |||
25 /
Vazquez, Michael L. 614 Castle Meadows Court Ballwin, MO 63021 / US | |||
26 /
Weier, Richard M. 240 Hickory Court Lake Bluff, IL 60044 / US | |||
27 /
Xu, Xiangdong 7498 Abbey Road Gurnee, IL 60031 / US | |||
28 /
BALDUS, John E. 2340 Louisiana Avenue St. Louis, MO 63104 / US | |||
29 /
JEROME, Kevin D. 2339 Pheasant Run Drive Maryland Heights, MO 63043 / US | |||
30 /
NAING, Win 1198 Nooning Tree Drive Chesterfield, MO 63017 / US | |||
31 /
WALKER, John K. 11949 Autumn Lakes Drive Maryland Heights, MO 63043 / US | |||
32 /
YANK, Syaulan 2157 Englewood Terrace Chesterfield, MO 63017 / US | |||
Former [2001/42] | 01 /
Anantanarayan, Ashok 54 Lisk Drive Hainesville, IL 60030 / US | ||
02 /
Clare, Michael 5154 West Brown Street Skokie, IL 60077 / US | |||
03 /
Collins, Paul W. 2317 Carillon Drive Grayslake, IL 60030 / US | |||
04 /
Crich, Joyce Z. 1501 G. Topp Lane Glenview, IL 60025 / US | |||
05 /
Devraj, Rajesh 1331 Oak Borough Drive Ballwin, MO 63021 / US | |||
06 /
Flynn, Daniel One Amgen Center Drive Thousand Oaks, CA 91320 / US | |||
07 /
Geng, Lifeng 5300 Davis Street Skokie, IL 60077 / US | |||
08 /
Graneto, Matthew J. 352 Hartwell Court Chesterfield, MO 63017 / US | |||
09 /
Hanau, Cathleen E. 15551 Wendimill Drive Chesterfield, MO 63017 / US | |||
10 /
Hanson, Gunnar J. 7410 Keystone Avenue Skokie, IL 60077 / US | |||
11 /
Hartmann, Susan J. 613 West Essex Avenue Kirkwood, MO 63122 / US | |||
12 /
Hepperle, Michael 1460 Keystone Court St. Charles, MO 63303 / US | |||
13 /
Huang, He 2309 F S. Stewart Avenue Chicago, IL 60616 / US | |||
14 /
Khanna, Ish K. 1821 S. Falcon Drive Libertyville, IL 60048 / US | |||
15 /
Koszyk, Francis J. 11 Wildwood Drive South Prospect Heights, IL 60070 / US | |||
16 /
Liao, Shuyuan 1536 Walters Avenue Northbrook, IL 60062 / US | |||
17 /
Metz, Suzanne 525 Westernmill Drive Chesterfield, MO 63017 / US | |||
18 /
Partis, Richard A. 2221 Noyes Street Evanston, IL 60201 / US | |||
19 /
Perry, Thao D. 516 Bloom Street Red Bud, IL 62278 / US | |||
20 /
Rao, Shashidhar N. 736 Bellerive Manor Drive St. Louis, MO 63141 / US | |||
21 /
Selness, Shaun Raj 1875 Cedarmill Drive Chesterfiedl, MO 63017 / US | |||
22 /
South, Michael S. 11671 Cheiftain Drive Chesterfield, MO 63146 / US | |||
23 /
Stealey, Michael A. 502 Juniper Parkway Libertyville, IL 60048 / US | |||
24 /
Talley, John Jeffrey 4701 Clifton Avenue St. Louis, MO 63109 / US | |||
25 /
Vasquez, Michael L. 614 Castle Meadows Court Ballwin, MO 63021 / US | |||
26 /
Weier, Richard M. 240 Hickory Court Lake Bluff, IL 60044 / US | |||
27 /
Xu, Xiangdong 7498 Abbey Road Gurnee, IL 60031 / US | Representative(s) | Albrecht, Thomas Kraus & Weisert Patentanwälte PartGmbB Thomas-Wimmer-Ring 15 80539 München / DE | [N/P] |
Former [2008/44] | Albrecht, Thomas Kraus & Weisert Patent- und Rechtsanwälte Thomas-Wimmer-Ring 15 80539 München / DE | ||
Former [2001/42] | Albrecht, Thomas, Dr. Kraus & Weisert, Thomas-Wimmer-Ring 15 80539 München / DE | Application number, filing date | 99965756.2 | 17.11.1999 | [2001/42] | WO1999US26007 | Priority number, date | US19980196623 | 20.11.1998 Original published format: US 196623 | [2001/42] | Filing language | EN | Procedural language | EN | Publication | Type: | A1 Application with search report | No.: | WO0031063 | Date: | 02.06.2000 | Language: | EN | [2000/22] | Type: | A1 Application with search report | No.: | EP1144403 | Date: | 17.10.2001 | Language: | EN | The application published by WIPO in one of the EPO official languages on 02.06.2000 takes the place of the publication of the European patent application. | [2001/42] | Type: | B1 Patent specification | No.: | EP1144403 | Date: | 06.10.2004 | Language: | EN | [2004/41] | Search report(s) | International search report - published on: | EP | 02.06.2000 | Classification | IPC: | C07D401/04, A61K31/415, A61K31/47, A61K31/445, A61K31/44, A61K31/50, A61K31/505, A61K31/52, C07D405/14, C07D401/14, C07D409/14, C07D403/04 | [2001/42] | CPC: |
C07D409/14 (EP,US);
C07D417/14 (EP,KR,US);
A61P1/04 (EP);
A61P11/00 (EP);
A61P11/06 (EP);
A61P13/12 (EP);
A61P19/00 (EP);
A61P19/02 (EP);
A61P19/06 (EP);
A61P29/00 (EP);
A61P29/02 (EP);
A61P43/00 (EP);
A61P9/00 (EP);
C07D401/04 (EP,US);
C07D401/14 (EP,US);
C07D403/04 (EP,US);
C07D405/14 (EP,US);
C07D413/14 (EP,US);
C07D453/02 (EP,US);
C07D471/04 (EP,US);
C07D473/00 (EP,US);
C07D487/04 (EP,US)
(-)
| Designated contracting states | AT, BE, CH, CY, DE, DK, ES, FI, FR, GB, GR, IE, IT, LI, LU, MC, NL, PT, SE [2001/42] | Extension states | AL | Not yet paid | LT | Not yet paid | LV | Not yet paid | MK | Not yet paid | RO | Not yet paid | SI | Not yet paid | Title | German: | SUBSTITUIERTE PYRAZOLE ALS P38-KINASEINHIBITOREN | [2001/42] | English: | SUBSTITUTED PYRAZOLES AS P38 KINASE INHIBITORS | [2004/32] | French: | PYRAZOLES SUBSTITUES UTILES COMME INHIBITEURS DE KINASE P38 | [2003/51] |
Former [2001/42] | SUBSTITUED PYRAZOLES AS P38 KINASE INHIBITORS | ||
Former [2001/42] | PYRAZOLES SUBSITUES UTILES COMME INHIBITEURS DE KINASE P38 | Miscellaneous | EPB 2001/42: Derzeit sind die WIPO-Publikationsdaten A3 nicht verfügbar. | EPB 2001/42: WIPO A3 publication data is not currently available. | EPB 2001/42: L'OMPI données de publication A3 ne sont pas actuellement disponibles. | Entry into regional phase | 08.05.2001 | National basic fee paid | 08.05.2001 | Designation fee(s) paid | 08.05.2001 | Examination fee paid | Examination procedure | 14.06.2000 | Request for preliminary examination filed International Preliminary Examining Authority: EP | 08.05.2001 | Examination requested [2001/42] | 18.09.2001 | Amendment by applicant (claims and/or description) | 21.01.2002 | Despatch of a communication from the examining division (Time limit: M08) | 17.09.2002 | Reply to a communication from the examining division | 19.12.2002 | Despatch of a communication from the examining division (Time limit: M06) | 16.06.2003 | Reply to a communication from the examining division | 25.11.2003 | Communication of intention to grant the patent | 24.05.2004 | Fee for grant paid | 24.05.2004 | Fee for publishing/printing paid | Divisional application(s) | EP04023186.2 / EP1500657 | Opposition(s) | 07.07.2005 | No opposition filed within time limit [2005/39] | Fees paid | Renewal fee | 22.11.2001 | Renewal fee patent year 03 | 25.11.2002 | Renewal fee patent year 04 | 21.11.2003 | Renewal fee patent year 05 |
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Responsibility for the accuracy, completeness or quality of the data displayed under the link provided lies entirely with the Unified Patent Court. | Cited in | International search | [A]DD295374 (STERLING DRUG INC [US]) [A] 1,39,71,82,93,94,101 * page 7 - page 8; example -; claim - *; | [A]EP0531901 (FUJISAWA PHARMACEUTICAL CO [JP]) [A] 1,39,71,82,93,94,101 * abstract * * pages 49 - 51, preparations; page 52; example 1 *; | [A]WO9419350 (FUJISAWA PHARMACEUTICAL CO [JP], et al) [A] 1,39,71,82,93,94,101 * page 53; example 8 *; | [A]WO9531451 (SMITHKLINE BEECHAM CORP [US], et al) [A] 1,39,71,82,93,94,101,126-140 * page 1 - page 3; claim 1 * * page 16 - page 19; example - *; | [DX]WO9603385 (SEARLE & CO [US], et al) [DX] 1,39,71,82,93,94,101,126-140 * abstract * * page 9 - page 73 *; | [A]EP0846687 (LILLY CO ELI [US]) [A] 1,39,71,82,93,94,101 * abstract * * page 21; table 1A * * page 23 - page 25; table 2A *; | [A]EP0846686 (PFIZER LTD [GB], et al) [A] 1,39,71,82,93,94,101 * abstract * * page 19; example A24 *; | [XP]WO9852937 (SEARLE & CO [US], et al) [XP] 1-160 * abstract * * page 35 - page 49; example - *; | [XP]WO9852940 (SEARLE & CO [US], et al) [XP] 1-160 * abstract *; | [XP]WO9852941 (SEARLE & CO [US], et al) [XP] 1-160 * abstract ** page 21 - page 24; examples 1,2 * |