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EP About this file: EP1144403

EP1144403 - SUBSTITUTED PYRAZOLES AS P38 KINASE INHIBITORS [Right-click to bookmark this link]
Former [2001/42]	SUBSTITUED PYRAZOLES AS P38 KINASE INHIBITORS
	[2004/32]
Status	No opposition filed within time limit Status updated on 12.08.2005 Database last updated on 31.08.2024
Most recent event Tooltip	26.09.2008	Change - representative	published on 29.10.2008 [2008/44]
Applicant(s)	For all designated states G.D. Searle LLC 575 Maryville Centre Drive St. Louis, Missouri 63141 / US
	[2004/19]
Former [2001/42]	For all designated states G.D. SEARLE & CO. P.O. Box 5110 Chicago, IL 60680-5110 / US
Inventor(s)	01 / Anantanarayan, Ashok 54 Lisk Drive Hainesville, IL 60030 / US
	02 / Clare, Michael 5154 West Brown Street Skokie, IL 60077 / US
	03 / Collins, Paul W. 2317 Carillon Drive Grayslake, IL 60030 / US
	04 / Crich, Joyce Z. 1501 G. Topp Lane Glenview, IL 60025 / US
	05 / Devraj, Rajesh 1331 Oak Borough Drive Ballwin, MO 63021 / US
	06 / Flynn, Daniel One Amgen Center Drive Thousand Oaks, CA 91320 / US
	07 / Geng, Lifeng 5300 Davis Street Skokie, IL 60077 / US
	08 / Graneto, Matthew J. 352 Hartwell Court Chesterfield, MO 63017 / US
	09 / Hanau, Cathleen E. 15551 Wendimill Drive Chesterfield, MO 63017 / US
	10 / Hanson, Gunnar J. 7410 Keystone Avenue Skokie, IL 60077 / US
	11 / Hartmann, Susan J. 613 West Essex Avenue Kirkwood, MO 63122 / US
	12 / Hepperle, Michael 1460 Keystone Court St. Charles, MO 63303 / US
	13 / Huang, He 2309 F S. Stewart Avenue Chicago, IL 60616 / US
	14 / Khanna, Ish K. 1821 S. Falcon Drive Libertyville, IL 60048 / US
	15 / Koszyk, Francis J. 11 Wildwood Drive South Prospect Heights, IL 60070 / US
	16 / Liao, Shuyuan 1536 Walters Avenue Northbrook, IL 60062 / US
	17 / Metz, Suzanne 525 Westernmill Drive Chesterfield, MO 63017 / US
	18 / Partis, Richard A. 2221 Noyes Street Evanston, IL 60201 / US
	19 / Perry, Thao D. 516 Bloom Street Red Bud, IL 62278 / US
	20 / Rao, Shashidhar N. 736 Bellerive Manor Drive St. Louis, MO 63141 / US
	21 / Selness, Shaun Raj 1875 Cedarmill Drive Chesterfield, MO 63017 / US
	22 / South, Michael S. 11671 Cheiftain Drive Chesterfield, MO 63146 / US
	23 / Stealey, Michael A. 502 Juniper Parkway Libertyville, IL 60048 / US
	24 / Talley, John Jeffrey 4701 Clifton Avenue St. Louis, MO 63109 / US
	25 / Vazquez, Michael L. 614 Castle Meadows Court Ballwin, MO 63021 / US
	26 / Weier, Richard M. 240 Hickory Court Lake Bluff, IL 60044 / US
	27 / Xu, Xiangdong 7498 Abbey Road Gurnee, IL 60031 / US
	28 / BALDUS, John E. 2340 Louisiana Avenue St. Louis, MO 63104 / US
	29 / JEROME, Kevin D. 2339 Pheasant Run Drive Maryland Heights, MO 63043 / US
	30 / NAING, Win 1198 Nooning Tree Drive Chesterfield, MO 63017 / US
	31 / WALKER, John K. 11946 Autumn Lakes Drive Maryland Heights, MO 63043 / US
	32 / YANG, Syaulan 2157 Englewood Terrace Chesterfield, MO 63017 / US
	33 / YU, Yi 1019 Castle Dr. Glenview, IL 60025 / US
	[2004/29]
Former [2004/02]	01 / Anantanarayan, Ashok 54 Lisk Drive Hainesville, IL 60030 / US
	02 / Clare, Michael 5154 West Brown Street Skokie, IL 60077 / US
	03 / Collins, Paul W. 2317 Carillon Drive Grayslake, IL 60030 / US
	04 / Crich, Joyce Z. 1501 G. Topp Lane Glenview, IL 60025 / US
	05 / Devraj, Rajesh 1331 Oak Borough Drive Ballwin, MO 63021 / US
	06 / Flynn, Daniel One Amgen Center Drive Thousand Oaks, CA 91320 / US
	07 / Geng, Lifeng 5300 Davis Street Skokie, IL 60077 / US
	08 / Graneto, Matthew J. 352 Hartwell Court Chesterfield, MO 63017 / US
	09 / Hanau, Cathleen E. 15551 Wendimill Drive Chesterfield, MO 63017 / US
	10 / Hanson, Gunnar J. 7410 Keystone Avenue Skokie, IL 60077 / US
	11 / Hartmann, Susan J. 613 West Essex Avenue Kirkwood, MO 63122 / US
	12 / Hepperle, Michael 1460 Keystone Court St. Charles, MO 63303 / US
	13 / Huang, He 2309 F S. Stewart Avenue Chicago, IL 60616 / US
	14 / Khanna, Ish K. 1821 S. Falcon Drive Libertyville, IL 60048 / US
	15 / Koszyk, Francis J. 11 Wildwood Drive South Prospect Heights, IL 60070 / US
	16 / Liao, Shuyuan 1536 Walters Avenue Northbrook, IL 60062 / US
	17 / Metz, Suzanne 525 Westernmill Drive Chesterfield, MO 63017 / US
	18 / Partis, Richard A. 2221 Noyes Street Evanston, IL 60201 / US
	19 / Perry, Thao D. 516 Bloom Street Red Bud, IL 62278 / US
	20 / Rao, Shashidhar N. 736 Bellerive Manor Drive St. Louis, MO 63141 / US
	21 / Selness, Shaun Raj 1875 Cedarmill Drive Chesterfiedl, MO 63017 / US
	22 / South, Michael S. 11671 Cheiftain Drive Chesterfield, MO 63146 / US
	23 / Stealey, Michael A. 502 Juniper Parkway Libertyville, IL 60048 / US
	24 / Talley, John Jeffrey 4701 Clifton Avenue St. Louis, MO 63109 / US
	25 / Vazquez, Michael L. 614 Castle Meadows Court Ballwin, MO 63021 / US
	26 / Weier, Richard M. 240 Hickory Court Lake Bluff, IL 60044 / US
	27 / Xu, Xiangdong 7498 Abbey Road Gurnee, IL 60031 / US
	28 / BALDUS, John E. 2340 Louisiana Avenue St. Louis, MO 63104 / US
	29 / JEROME, Kevin D. 2339 Pheasant Run Drive Maryland Heights, MO 63043 / US
	30 / NAING, Win 1198 Nooning Tree Drive Chesterfield, MO 63017 / US
	31 / WALKER, John K. 11946 Autumn Lakes Drive Maryland Heights, MO 63043 / US
	32 / YANG, Syaulan 2157 Englewood Terrace Chesterfield, MO 63017 / US
	33 / YU, Yi 1019 Castle Dr. Glenview, IL 60025 / US
Former [2003/49]	01 / Anantanarayan, Ashok 54 Lisk Drive Hainesville, IL 60030 / US
	02 / Clare, Michael 5154 West Brown Street Skokie, IL 60077 / US
	03 / Collins, Paul W. 2317 Carillon Drive Grayslake, IL 60030 / US
	04 / Crich, Joyce Z. 1501 G. Topp Lane Glenview, IL 60025 / US
	05 / Devraj, Rajesh 1331 Oak Borough Drive Ballwin, MO 63021 / US
	06 / Flynn, Daniel One Amgen Center Drive Thousand Oaks, CA 91320 / US
	07 / Geng, Lifeng 5300 Davis Street Skokie, IL 60077 / US
	08 / Graneto, Matthew J. 352 Hartwell Court Chesterfield, MO 63017 / US
	09 / Hanau, Cathleen E. 15551 Wendimill Drive Chesterfield, MO 63017 / US
	10 / Hanson, Gunnar J. 7410 Keystone Avenue Skokie, IL 60077 / US
	11 / Hartmann, Susan J. 613 West Essex Avenue Kirkwood, MO 63122 / US
	12 / Hepperle, Michael 1460 Keystone Court St. Charles, MO 63303 / US
	13 / Huang, He 2309 F S. Stewart Avenue Chicago, IL 60616 / US
	14 / Khanna, Ish K. 1821 S. Falcon Drive Libertyville, IL 60048 / US
	15 / Koszyk, Francis J. 11 Wildwood Drive South Prospect Heights, IL 60070 / US
	16 / Liao, Shuyuan 1536 Walters Avenue Northbrook, IL 60062 / US
	17 / Metz, Suzanne 525 Westernmill Drive Chesterfield, MO 63017 / US
	18 / Partis, Richard A. 2221 Noyes Street Evanston, IL 60201 / US
	19 / Perry, Thao D. 516 Bloom Street Red Bud, IL 62278 / US
	20 / Rao, Shashidhar N. 736 Bellerive Manor Drive St. Louis, MO 63141 / US
	21 / Selness, Shaun Raj 1875 Cedarmill Drive Chesterfiedl, MO 63017 / US
	22 / South, Michael S. 11671 Cheiftain Drive Chesterfield, MO 63146 / US
	23 / Stealey, Michael A. 502 Juniper Parkway Libertyville, IL 60048 / US
	24 / Talley, John Jeffrey 4701 Clifton Avenue St. Louis, MO 63109 / US
	25 / Vazquez, Michael L. 614 Castle Meadows Court Ballwin, MO 63021 / US
	26 / Weier, Richard M. 240 Hickory Court Lake Bluff, IL 60044 / US
	27 / Xu, Xiangdong 7498 Abbey Road Gurnee, IL 60031 / US
	28 / BALDUS, John E. 2340 Louisiana Avenue St. Louis, MO 63104 / US
	29 / JEROME, Kevin D. 2339 Pheasant Run Drive Maryland Heights, MO 63043 / US
	30 / NAING, Win 1198 Nooning Tree Drive Chesterfield, MO 63017 / US
	31 / WALKER, John K. 11949 Autumn Lakes Drive Maryland Heights, MO 63043 / US
	32 / YANK, Syaulan 2157 Englewood Terrace Chesterfield, MO 63017 / US
	33 / YU, Yi 1019 Castle Dr. Glenview, IL 60025 / US
Former [2003/48]	01 / Anantanarayan, Ashok 54 Lisk Drive Hainesville, IL 60030 / US
	02 / Clare, Michael 5154 West Brown Street Skokie, IL 60077 / US
	03 / Collins, Paul W. 2317 Carillon Drive Grayslake, IL 60030 / US
	04 / Crich, Joyce Z. 1501 G. Topp Lane Glenview, IL 60025 / US
	05 / Devraj, Rajesh 1331 Oak Borough Drive Ballwin, MO 63021 / US
	06 / Flynn, Daniel One Amgen Center Drive Thousand Oaks, CA 91320 / US
	07 / Geng, Lifeng 5300 Davis Street Skokie, IL 60077 / US
	08 / Graneto, Matthew J. 352 Hartwell Court Chesterfield, MO 63017 / US
	09 / Hanau, Cathleen E. 15551 Wendimill Drive Chesterfield, MO 63017 / US
	10 / Hanson, Gunnar J. 7410 Keystone Avenue Skokie, IL 60077 / US
	11 / Hartmann, Susan J. 613 West Essex Avenue Kirkwood, MO 63122 / US
	12 / Hepperle, Michael 1460 Keystone Court St. Charles, MO 63303 / US
	13 / Huang, He 2309 F S. Stewart Avenue Chicago, IL 60616 / US
	14 / Khanna, Ish K. 1821 S. Falcon Drive Libertyville, IL 60048 / US
	15 / Koszyk, Francis J. 11 Wildwood Drive South Prospect Heights, IL 60070 / US
	16 / Liao, Shuyuan 1536 Walters Avenue Northbrook, IL 60062 / US
	17 / Metz, Suzanne 525 Westernmill Drive Chesterfield, MO 63017 / US
	18 / Partis, Richard A. 2221 Noyes Street Evanston, IL 60201 / US
	19 / Perry, Thao D. 516 Bloom Street Red Bud, IL 62278 / US
	20 / Rao, Shashidhar N. 736 Bellerive Manor Drive St. Louis, MO 63141 / US
	21 / Selness, Shaun Raj 1875 Cedarmill Drive Chesterfiedl, MO 63017 / US
	22 / South, Michael S. 11671 Cheiftain Drive Chesterfield, MO 63146 / US
	23 / Stealey, Michael A. 502 Juniper Parkway Libertyville, IL 60048 / US
	24 / Talley, John Jeffrey 4701 Clifton Avenue St. Louis, MO 63109 / US
	25 / Vazquez, Michael L. 614 Castle Meadows Court Ballwin, MO 63021 / US
	26 / Weier, Richard M. 240 Hickory Court Lake Bluff, IL 60044 / US
	27 / Xu, Xiangdong 7498 Abbey Road Gurnee, IL 60031 / US
	28 / BALDUS, John E. 2340 Louisiana Avenue St. Louis, MO 63104 / US
	29 / JEROME, Kevin D. 2339 Pheasant Run Drive Maryland Heights, MO 63043 / US
	30 / NAING, Win 1198 Nooning Tree Drive Chesterfield, MO 63017 / US
	31 / WALKER, John K. 11949 Autumn Lakes Drive Maryland Heights, MO 63043 / US
	32 / YANK, Syaulan 2157 Englewood Terrace Chesterfield, MO 63017 / US
Former [2001/42]	01 / Anantanarayan, Ashok 54 Lisk Drive Hainesville, IL 60030 / US
	02 / Clare, Michael 5154 West Brown Street Skokie, IL 60077 / US
	03 / Collins, Paul W. 2317 Carillon Drive Grayslake, IL 60030 / US
	04 / Crich, Joyce Z. 1501 G. Topp Lane Glenview, IL 60025 / US
	05 / Devraj, Rajesh 1331 Oak Borough Drive Ballwin, MO 63021 / US
	06 / Flynn, Daniel One Amgen Center Drive Thousand Oaks, CA 91320 / US
	07 / Geng, Lifeng 5300 Davis Street Skokie, IL 60077 / US
	08 / Graneto, Matthew J. 352 Hartwell Court Chesterfield, MO 63017 / US
	09 / Hanau, Cathleen E. 15551 Wendimill Drive Chesterfield, MO 63017 / US
	10 / Hanson, Gunnar J. 7410 Keystone Avenue Skokie, IL 60077 / US
	11 / Hartmann, Susan J. 613 West Essex Avenue Kirkwood, MO 63122 / US
	12 / Hepperle, Michael 1460 Keystone Court St. Charles, MO 63303 / US
	13 / Huang, He 2309 F S. Stewart Avenue Chicago, IL 60616 / US
	14 / Khanna, Ish K. 1821 S. Falcon Drive Libertyville, IL 60048 / US
	15 / Koszyk, Francis J. 11 Wildwood Drive South Prospect Heights, IL 60070 / US
	16 / Liao, Shuyuan 1536 Walters Avenue Northbrook, IL 60062 / US
	17 / Metz, Suzanne 525 Westernmill Drive Chesterfield, MO 63017 / US
	18 / Partis, Richard A. 2221 Noyes Street Evanston, IL 60201 / US
	19 / Perry, Thao D. 516 Bloom Street Red Bud, IL 62278 / US
	20 / Rao, Shashidhar N. 736 Bellerive Manor Drive St. Louis, MO 63141 / US
	21 / Selness, Shaun Raj 1875 Cedarmill Drive Chesterfiedl, MO 63017 / US
	22 / South, Michael S. 11671 Cheiftain Drive Chesterfield, MO 63146 / US
	23 / Stealey, Michael A. 502 Juniper Parkway Libertyville, IL 60048 / US
	24 / Talley, John Jeffrey 4701 Clifton Avenue St. Louis, MO 63109 / US
	25 / Vasquez, Michael L. 614 Castle Meadows Court Ballwin, MO 63021 / US
	26 / Weier, Richard M. 240 Hickory Court Lake Bluff, IL 60044 / US
	27 / Xu, Xiangdong 7498 Abbey Road Gurnee, IL 60031 / US
Representative(s)	Albrecht, Thomas Kraus & Weisert Patentanwälte PartGmbB Thomas-Wimmer-Ring 15 80539 München / DE
	[N/P]
Former [2008/44]	Albrecht, Thomas Kraus & Weisert Patent- und Rechtsanwälte Thomas-Wimmer-Ring 15 80539 München / DE
Former [2001/42]	Albrecht, Thomas, Dr. Kraus & Weisert, Thomas-Wimmer-Ring 15 80539 München / DE
Application number, filing date	99965756.2	17.11.1999
	[2001/42]
	WO1999US26007
Priority number, date	US19980196623	20.11.1998 Original published format: US 196623
	[2001/42]
Filing language	EN
Procedural language	EN
Publication	Type:	A1 Application with search report
	No.:	WO0031063
	Date:	02.06.2000
	Language:	EN
	[2000/22]
	Type:	A1 Application with search report
	No.:	EP1144403
	Date:	17.10.2001
	Language:	EN
	The application published by WIPO in one of the EPO official languages on 02.06.2000 takes the place of the publication of the European patent application.
	[2001/42]
	Type:	B1 Patent specification
	No.:	EP1144403
	Date:	06.10.2004
	Language:	EN
	[2004/41]
Search report(s)	International search report - published on:	EP	02.06.2000
Classification	IPC:	C07D401/04, A61K31/415, A61K31/47, A61K31/445, A61K31/44, A61K31/50, A61K31/505, A61K31/52, C07D405/14, C07D401/14, C07D409/14, C07D403/04	[2001/42]
	CPC:	C07D409/14 (EP,US); C07D417/14 (EP,KR,US); A61P1/04 (EP); A61P11/00 (EP); A61P11/06 (EP); A61P13/12 (EP); (+) A61P19/00 (EP); A61P19/02 (EP); A61P19/06 (EP); A61P29/00 (EP); A61P29/02 (EP); A61P43/00 (EP); A61P9/00 (EP); C07D401/04 (EP,US); C07D401/14 (EP,US); C07D403/04 (EP,US); C07D405/14 (EP,US); C07D413/14 (EP,US); C07D453/02 (EP,US); C07D471/04 (EP,US); C07D473/00 (EP,US); C07D487/04 (EP,US) (-)
Designated contracting states	AT, BE, CH, CY, DE, DK, ES, FI, FR, GB, GR, IE, IT, LI, LU, MC, NL, PT, SE [2001/42]
Extension states	AL	Not yet paid
	LT	Not yet paid
	LV	Not yet paid
	MK	Not yet paid
	RO	Not yet paid
	SI	Not yet paid
Title	German:	SUBSTITUIERTE PYRAZOLE ALS P38-KINASEINHIBITOREN	[2001/42]
	English:	SUBSTITUTED PYRAZOLES AS P38 KINASE INHIBITORS	[2004/32]
	French:	PYRAZOLES SUBSTITUES UTILES COMME INHIBITEURS DE KINASE P38	[2003/51]
	Former [2001/42]	SUBSTITUED PYRAZOLES AS P38 KINASE INHIBITORS
	Former [2001/42]	PYRAZOLES SUBSITUES UTILES COMME INHIBITEURS DE KINASE P38
Miscellaneous	EPB 2001/42: Derzeit sind die WIPO-Publikationsdaten A3 nicht verfügbar.
	EPB 2001/42: WIPO A3 publication data is not currently available.
	EPB 2001/42: L'OMPI données de publication A3 ne sont pas actuellement disponibles.
Entry into regional phase	08.05.2001	National basic fee paid
	08.05.2001	Designation fee(s) paid
	08.05.2001	Examination fee paid
Examination procedure	14.06.2000	Request for preliminary examination filed International Preliminary Examining Authority: EP
	08.05.2001	Examination requested [2001/42]
	18.09.2001	Amendment by applicant (claims and/or description)
	21.01.2002	Despatch of a communication from the examining division (Time limit: M08)
	17.09.2002	Reply to a communication from the examining division
	19.12.2002	Despatch of a communication from the examining division (Time limit: M06)
	16.06.2003	Reply to a communication from the examining division
	25.11.2003	Communication of intention to grant the patent
	24.05.2004	Fee for grant paid
	24.05.2004	Fee for publishing/printing paid
Divisional application(s)	EP04023186.2 / EP1500657
Opposition(s)	07.07.2005	No opposition filed within time limit [2005/39]
Fees paid	Renewal fee
	22.11.2001	Renewal fee patent year 03
	25.11.2002	Renewal fee patent year 04
	21.11.2003	Renewal fee patent year 05
Opt-out from the exclusive Tooltip competence of the Unified Patent Court	See the Register of the Unified Patent Court for opt-out data
	Responsibility for the accuracy, completeness or quality of the data displayed under the link provided lies entirely with the Unified Patent Court.
Cited in	International search	[A]DD295374 (STERLING DRUG INC [US]) [A] 1,39,71,82,93,94,101 * page 7 - page 8; example -; claim - *;
		[A]EP0531901 (FUJISAWA PHARMACEUTICAL CO [JP]) [A] 1,39,71,82,93,94,101 * abstract * * pages 49 - 51, preparations; page 52; example 1 *;
		[A]WO9419350 (FUJISAWA PHARMACEUTICAL CO [JP], et al) [A] 1,39,71,82,93,94,101 * page 53; example 8 *;
		[A]WO9531451 (SMITHKLINE BEECHAM CORP [US], et al) [A] 1,39,71,82,93,94,101,126-140 * page 1 - page 3; claim 1 * * page 16 - page 19; example - *;
		[DX]WO9603385 (SEARLE & CO [US], et al) [DX] 1,39,71,82,93,94,101,126-140 * abstract * * page 9 - page 73 *;
		[A]EP0846687 (LILLY CO ELI [US]) [A] 1,39,71,82,93,94,101 * abstract * * page 21; table 1A * * page 23 - page 25; table 2A *;
		[A]EP0846686 (PFIZER LTD [GB], et al) [A] 1,39,71,82,93,94,101 * abstract * * page 19; example A24 *;
		[XP]WO9852937 (SEARLE & CO [US], et al) [XP] 1-160 * abstract * * page 35 - page 49; example - *;
		[XP]WO9852940 (SEARLE & CO [US], et al) [XP] 1-160 * abstract *;
		[XP]WO9852941 (SEARLE & CO [US], et al) [XP] 1-160 * abstract ** page 21 - page 24; examples 1,2 *

The EPO accepts no responsibility for the accuracy of data originating from other authorities; in particular, it does not guarantee that it is complete, up to date or fit for specific purposes.

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