blank Quick help
blank Maintenance news

Scheduled maintenance

Regular maintenance outages:
between 05.00 and 05.15 hrs CET (Monday to Sunday).

Other outages
Availability
Register Forum

2022.02.11

More...
blank News flashes

News flashes

New version of the European Patent Register - SPC information for Unitary Patents.

2024-03-06

More...
blank Related links

Extract from the Register of European Patents

EP About this file: EP1227084

EP1227084 - DRUG DISCHARGE PUMP INHIBITORS [Right-click to bookmark this link]
StatusNo opposition filed within time limit
Status updated on  20.10.2006
Database last updated on 15.07.2024
Most recent event   Tooltip05.12.2008Lapse of the patent in a contracting state
New state(s): CY
published on 07.01.2009  [2009/02]
Applicant(s)For all designated states
Trine Pharmaceuticals, Inc.
78 Fourth Avenue
Waltham, MA 02451 / US
For all designated states
DAIICHI PHARMACEUTICAL CO., LTD.
14-10, Nihonbashi 3-chome Chuo-ku
Tokyo 103-8234 / JP
[N/P]
Former [2005/50]For all designated states
Trine Pharmaceuticals, Inc.
78 Fourth Avenue
Waltham, MA 02451 / US
For all designated states
DAIICHI PHARMACEUTICAL CO., LTD.
14-10, Nihonbashi 3-chome Chuo-ku
Tokyo 103-8234 / JP
Former [2005/42]For all designated states
Trine Pharmaceuticals Inc.
78 Fourth Avenue
Waltham, MA 02451 / US
For all designated states
DAIICHI PHARMACEUTICAL CO., LTD.
14-10, Nihonbashi 3-chome
Chuo-ku, Tokyo 103-8234 / JP
Former [2002/35]For all designated states
Essential Therapeutics, Inc.
1365 Main Street
Waltham, MA 02451 / US
For all designated states
DAIICHI PHARMACEUTICAL CO., LTD.
14-10, Nihonbashi 3-chome
Chuo-ku, Tokyo 103-8234 / JP
Former [2002/31]For all designated states
Microcide Pharmaceuticals, Inc.
850 Maude Avenue
Mountainview, CA 94043 / US
For all designated states
DAIICHI PHARMACEUTICAL CO., LTD.
14-10, Nihonbashi 3-chome
Chuo-ku, Tokyo 103-8234 / JP
Inventor(s)01 / LEGER, Roger
202, Upper Edison
Saint-Lambert, Quebec J4R 2V8 / CA
02 / WATKINS, William, John
626, Oneida Drive
Sunnyvale, CA 94087 / US
03 / ZHANG, Jason, Zhijia
770, Crane Avenue
Foster City, CA 94404 / US
04 / RENAU, Thomas, Eric
900, Pepper Tree Lane 224
Santa Clara, CA 95051 / US
05 / LEE, Ving, Jack
1335, Carvo Court
Los Altos, CA 94024 / US
06 / OHTA, Toshiharu, Daiichi Pharmaceutical Co., Ltd.
Tokyo R & D Center, 16-13, Kita-kasai 1-chome
Edogawa-ku, Tokyo 134-8630 / JP
07 / NAKAYAMA, Kiyoshi, Daiichi Pharmaceutical Co., Ltd
Tokyo R & D Center, 16-13, Kita-kasai 1-chome
Edogawa-ku, Tokyo 134-8630 / JP
08 / ISHIDA, Yohhei, Daiichi Pharmaceutical Co., Ltd.
Tokyo R & D Center, 16-13, Kita-kasai 1-chome
Edogawa-ku, Tokyo 134-8630 / JP
09 / OHTSUKA, Masami, Daiichi Pharmaceutical Co., Ltd.
Tokyo R & D Center, 16-13, Kita-kasai 1-chome
Edogawa-ku, Tokyo 134-8630 / JP
10 / KAWATO, Haruko, Daiichi Pharmaceutical Co., Ltd.
Tokyo R & D Center, 16-13, Kita-kasai 1-chome
Edogawa-ku, Tokyo 134-8630 / JP
 [2002/31]
Representative(s)polypatent
Patentanwälte
An den Gärten 7
51491 Overath / DE
[N/P]
Former [2002/31]Sternagel, Fleischer, Godemeyer & Partner Patentanwälte
An den Gärten 7
51491 Overath / DE
Application number, filing date00970155.827.10.2000
[2002/31]
WO2000JP07565
Priority number, dateUS1999042846628.10.1999         Original published format: US 428466
JP2000032671326.10.2000         Original published format: JP 2000326713
[2002/31]
Filing languageJA
Procedural languageEN
PublicationType: A1 Application with search report
No.:WO0130757
Date:03.05.2001
Language:EN
[2001/18]
Type: A1 Application with search report 
No.:EP1227084
Date:31.07.2002
Language:EN
The application published by WIPO in one of the EPO official languages on 03.05.2001 takes the place of the publication of the European patent application.
[2002/31]
Type: B1 Patent specification 
No.:EP1227084
Date:14.12.2005
Language:EN
[2005/50]
Search report(s)International search report - published on:JP03.05.2001
(Supplementary) European search report - dispatched on:EP07.07.2003
ClassificationIPC:C07D213/30, C07D277/26, C07D277/28, C07D277/32, C07D277/44, C07D215/14, C07D215/56, C07D307/52, C07D513/04, C07D263/56, A61K31/425, A61K31/44
[2003/18]
CPC:
G01N33/6803 (EP); A61K31/4738 (EP,KR); A61K31/341 (EP);
A61K31/41 (EP); A61K31/421 (EP); A61K31/423 (EP);
A61K31/425 (EP); A61K31/426 (EP); A61K31/427 (EP);
A61K31/433 (EP); A61K31/437 (EP); A61K31/4375 (EP);
A61K31/44 (EP); A61K31/4439 (EP); A61K31/47 (EP);
A61K31/4709 (EP); A61K31/502 (EP); A61K31/517 (EP);
A61K31/519 (EP); A61K31/5383 (EP); A61P31/04 (EP);
C07D213/30 (EP); C07D215/14 (EP); C07D215/56 (EP);
C07D263/56 (EP); C07D277/24 (EP); C07D277/28 (EP);
C07D285/08 (EP); C07D307/52 (EP); C07D409/12 (EP);
C07D417/04 (EP); C07D417/06 (EP); C07D417/10 (EP);
C07D417/12 (EP); C07D417/14 (EP); C07D471/04 (EP);
C07D513/04 (EP); C12Q1/18 (EP); C07K2299/00 (EP);
G01N2500/04 (EP) (-)
Former IPC [2002/31]C07D213/30, C07D277/26, C07D277/28, C07D277/32, C07D277/44, C07D215/14, C07D215/56, C07D307/52, C07D513/04, C07D263/56, C07D417/04
Designated contracting statesAT,   BE,   CH,   CY,   DE,   DK,   ES,   FI,   FR,   GB,   GR,   IE,   IT,   LI,   LU,   MC,   NL,   PT,   SE [2002/31]
Extension statesALNot yet paid
LTNot yet paid
LVNot yet paid
MKNot yet paid
RONot yet paid
SINot yet paid
TitleGerman:PUMPENINHIBITOREN ZUR FREISETZUNG VON MEDIKAMENTEN[2002/31]
English:DRUG DISCHARGE PUMP INHIBITORS[2002/31]
French:INHIBITEURS DE LA POMPE PAR LIBERATION DE MEDICAMENTS[2002/31]
Entry into regional phase19.04.2002Translation filed 
19.04.2002National basic fee paid 
19.04.2002Search fee paid 
19.04.2002Designation fee(s) paid 
19.04.2002Examination fee paid 
Examination procedure27.10.2000Request for preliminary examination filed
International Preliminary Examining Authority: JP
19.04.2002Examination requested  [2002/31]
25.09.2003Despatch of a communication from the examining division (Time limit: M06)
01.04.2004Reply to a communication from the examining division
30.12.2004Despatch of a communication from the examining division (Time limit: M04)
05.04.2005Reply to a communication from the examining division
29.04.2005Communication of intention to grant the patent
05.09.2005Fee for grant paid
05.09.2005Fee for publishing/printing paid
Divisional application(s)EP05019514.8  / EP1652839
Opposition(s)15.09.2006No opposition filed within time limit [2006/47]
Fees paidRenewal fee
15.10.2002Renewal fee patent year 03
14.10.2003Renewal fee patent year 04
14.10.2004Renewal fee patent year 05
12.10.2005Renewal fee patent year 06
Opt-out from the exclusive  Tooltip
competence of the Unified
Patent Court
See the Register of the Unified Patent Court for opt-out data
Responsibility for the accuracy, completeness or quality of the data displayed under the link provided lies entirely with the Unified Patent Court.
Lapses during opposition  TooltipAT14.12.2005
CY14.12.2005
FI14.12.2005
DK14.03.2006
GR14.03.2006
ES25.03.2006
PT15.05.2006
[2009/02]
Former [2007/50]AT14.12.2005
FI14.12.2005
DK14.03.2006
GR14.03.2006
ES25.03.2006
PT15.05.2006
Former [2007/35]AT14.12.2005
FI14.12.2005
IT14.12.2005
DK14.03.2006
GR14.03.2006
ES25.03.2006
PT15.05.2006
Former [2006/51]AT14.12.2005
FI14.12.2005
DK14.03.2006
GR14.03.2006
ES25.03.2006
PT15.05.2006
Former [2006/48]AT14.12.2005
FI14.12.2005
GR14.03.2006
ES25.03.2006
PT15.05.2006
Former [2006/38]AT14.12.2005
FI14.12.2005
GR14.03.2006
ES25.03.2006
Former [2006/34]AT14.12.2005
FI14.12.2005
ES25.03.2006
Former [2006/23]FI14.12.2005
Documents cited:Search[X]JPH03207789  ;
 [X]JPH02219892  ;
 [X]JPH0543878  ;
 [X]JPH09323971  ;
 [X]JPH10310578  ;
 [X]US3907808  (LESHER GEORGE Y, et al) [X] 1-10 * claim - *;
 [X]US4013647  (SELLSTEDT JOHN H, et al) [X] 1-10 * example 4; claim 3 *;
 [A]US4404207  (STERN RICHARD M [US]) [A] 1-10 * claim - *;
 [X]DE3417840  (CIBA GEIGY AG [CH]) [X] 1-8 * example 20 *;
 [X]US4665079  (CULBERTSON TOWNLEY P [US], et al) [X] 1-10 * column 11 - column 16; example -; claims 1-4 *;
 [X]EP0279239  (CIBA GEIGY AG [CH]) [X] 1-10 * page 2, line 1 - line 24; example 3.097; claim -; table 3 *;
 [X]EP0513974  (MERCK & CO INC [US]) [X] 1-10 * page 128 - page 129; example E; claim 1 *;
 [X]EP0513387  (OTSUKA PHARMA CO LTD [JP]) [X] 1-10 * example 1; claim -; tables 8-10 *;
 [X]EP0594861  (KASHIMA OIL [JP]) [X] 1-8 * example 8 *;
 [A]WO9633285  (MICROCIDE PHARMACEUTICALS INC [US], et al) [A] 1-10 * claims 52-79 *;
 [X]WO9802430  (PFIZER PHARMA [JP], et al) [X] 1-10 * example 63; claim - *;
 [A]WO9937667  (MICROCIDE PHARMACEUTICALS INC [US], et al) [A] 1-10* page 63 - page 84 *
 [X]  - PATENT ABSTRACTS OF JAPAN, (19911204), vol. 015, no. 478, Database accession no. (C - 0891), & JP03207789 A 19910911 (DAINIPPON INK & CHEM INC;OTHERS: 01) [X] 1-8 * abstract * * page 719 *
 [X]  - PATENT ABSTRACTS OF JAPAN, (19901119), vol. 014, no. 526, Database accession no. (C - 0779), & JP02219892 A 19900903 (DAINIPPON INK & CHEM INC;OTHERS: 01) [X] 1-8 * abstract * * page 847 - page 850 *
 [X]  - PATENT ABSTRACTS OF JAPAN, (19930630), vol. 017, no. 345, Database accession no. (C - 1077), & JP05043878 A 19930223 (DAINIPPON INK & CHEM INC) [X] 1-8 * abstract * * page 647 *
 [X]  - PATENT ABSTRACTS OF JAPAN, (19980331), vol. 1998, no. 04, & JP09323971 A 19971216 (SANKYO CO LTD) [X] 1-10 * abstract * * page 10, paragraph L - page 19 *
 [X]  - PATENT ABSTRACTS OF JAPAN, (19990226), vol. 1999, no. 02, & JP10310578 A 19981124 (YOSHITOMI PHARMACEUT IND LTD) [X] 1-10 * abstract * * example 13; claim - *
International search[X]FR1458066  (BOEHRINGER & SOEHNE GMBH);
 [X]JPS442219B  ;
 [X]JPS4413952B  ;
 [X]GB1305820  ;
 [X]US3870712  (HOLMES RICHARD E);
 [X]US4891428  (NORDHOFF ERHARD [DE], et al);
 [X]WO9322312  (STANFORD RES INST INT [US]);
 [X]WO9322315  (STANFORD RES INST INT [US]);
 [X]WO9602507  (ABBOTT LAB [US]);
 [X]WO9633285  (MICROCIDE PHARMACEUTICALS INC [US], et al);
 [X]WO9703967  (RHONE POULENC RORER LTD [GB], et al);
 [X]EP0786457  (YAMANOUCHI PHARMA CO LTD [JP]);
 [X]WO9817625  (DAIICHI SEIYAKU CO [JP], et al);
 [X]WO9857957  (NISSAN CHEMICAL IND LTD [JP], et al);
 [X]WO9936442  (GRAIN PROCESSING CORP [US], et al);
 [X]US5936977  (CHURCHILL JONATHAN F [GB], et al);
 [X]WO9950304  (RHODIA ACETOW AKTIENGESELLSCHA [DE], et al);
 [X]  - NISHIGAKI S. ET AL., "Synthesis of 1-substituted 1,4-dihydro-7-(2-(5-nitro-2-furyl)vinyl)-4-oxo-1,8-naphthyridine derivatives. I.", CHEM. PHARM. BULL., (1969), vol. 17, no. 9, pages 1827 - 1831, XP002944105
 [Y]  - LI X.-A., LIVERMORE D.M., NIKAIDO H., "Role of efflux pumps(s) in intrinsic resistance of pseudomonas aeruginosa: Resistance to tetracycline, chloramphenicol and norfloxacin", ANTIMICROB. CHEMTH., (1994), vol. 38, no. 8, pages 1732 - 1734, XP002944106
 [Y]  - GREENE J. ET AL., "Chemical function queries for 3D database search", J. CHEM. INF. COMPUT. SCI., (1994), no. 34, pages 1297 - 1308, XP002944107

DOI:   http://dx.doi.org/10.1021/ci00022a012
 [X]  - CHUPP J.P., MOLYNEAUX J.M., "Derivation of fluorine-containing pyridinedicarboxylates. III. Regioselective anion chemistry at the 2- and 4-position", J. HETEROCYCL. CHEM., (1989), vol. 26, no. 6, pages 1771 - 1780, XP002944108
 [X]  - DEJOHN D. ET AL., "Functionalization of substituted 2(1H)- and 4(1H)-pyridones. III. The preparation of substituted 6-vinyl-1,2-dihydro-2-oxo- and 1,4-dihydro-4-oxo-3-pyridinecarboxylic acids through the chemistry of pyridone dianions", J. HETEROCYCL. CHEM., (1983), vol. 20, no. 5, pages 1295 - 1302, XP002944109

DOI:   http://dx.doi.org/10.1002/jhet.5570200529
 [X]  - ROZENBLIT A. ET AL., "Computer-aided prediction and study of biological properties of nitrofurylvinyl(polyenyl)quinolines", CHEMICAL ABSTRACTS, (1991), vol. 115, Database accession no. 105447
    [ ] - KHIM.-FARM. ZH., (1991), vol. 25, no. 5, pages 55 - 58 [ ] * Registry Nos. 5774-31-2, 59666-11-4, 73263-92-0 *
 [X]  - SUKHOVA N.M. ET AL., "Search for new drugs in a series of furan derivatives", CHEMICAL ABSTRACTS, (1980), vol. 92, Database accession no. 157718
    [ ] - KONF. KHIM. TEKHNOL. FURANOVYKH SOEDIN., (TEZISY DOKL.), 3RD, (1978), pages 97 - 98 [ ] * Registry Nos. 5774-31-2, 26170-82-1, 73263-92-0 *
 [X]  - LIPKIN A.E., BESPALOVA ZH. P., "Synthesis based on 2-methyl-4-quinolinecarboxylic acid", CHEMICAL ABSTRACTS, (1970), vol. 72, Database accession no. 111193
    [ ] - KHIM.-FARM. ZH., (1970), vol. 4, no. 1, pages 24 - 26 [ ] * Registry Nos. 5774-31-2, 26170-82-1, 26170-84-3, 26280-17-1 *
 [X]  - FUJITA AKIO ET AL., "Nitrofuran derivatives. VI. Synthesis of 2-(2-(5-nitro-2-furyl)vinyl)pyridinemethanol and 2-(2-(5-nitro-2-furyl)vinyl)pyridinecarboxylic acid derivatives", CHEMICAL ABSTRACTS, (1967), vol. 66, Database accession no. 75885
    [ ] - YAKUGAKU ZASSHI, (1966), vol. 86, no. 11, pages 1014 - 1021 [ ] * Registry Nos. 1030-71-3, 1030-72-4 *
 [X]  - CHEMICAL ABSTRACTS, (1988), vol. 108, Database accession no. 142146
    [ ] - INORG. CHEM., (1988), vol. 27, no. 7, pages 1167 - 1173
 [X]  - CHEMICAL ABSTRACTS, (1987), vol. 106, Database accession no. 196227
    [ ] - TAP CHI HOA HOC, (1985), vol. 23, no. 5, pages 9 - 11
 [X]  - CHEMICAL ABSTRACTS, (1985), vol. 103, Database accession no. 87754
    [ ] - YIYAO GONGYE, (1985), vol. 16, no. 2, pages 66 - 68, 91
 [X]  - CHEMICAL ABSTRACTS, (1984), vol. 100, Database accession no. 138915
    [ ] - KHIM. GETEROTSIKL. SOEDIN., (1983), no. 11, pages 1521 - 1523
 [X]  - CHEMICAL ABSTRACTS, (1980), vol. 92, Database accession no. 128023
    [ ] - KHIM. GETEROTSIKL. SOEDIN., (1979), no. 9, pages 1194 - 1200
 [X]  - CHEMICAL ABSTRACTS, (1978), vol. 89, Database accession no. 109013
    [ ] - TEZISY DOKL. - RESP. KONF. MOLODYKH UCH.-KHIM., 2ND, AKAD. NAUK EST. SSR, INST. KHIM.: TALLINN, USSR, (1977), vol. 1, pages 14 - 15
 [X]  - CHEMICAL ABSTRACTS, (1973), vol. 78, Database accession no. 97460
    [ ] - J. HETEROCYCL. CHEM., (1972), vol. 9, no. 6, pages 1203 - 1207
The EPO accepts no responsibility for the accuracy of data originating from other authorities; in particular, it does not guarantee that it is complete, up to date or fit for specific purposes.