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Extract from the Register of European Patents

EP About this file: EP1383786

EP1383786 - ANTI-INFLAMMATORY 17.BETA.-CARBOTHIOATE ESTER DERIVATIVES OF ANDROSTANE WITH A CYCLIC ESTER GROUP IN POSITION 17.ALPHA [Right-click to bookmark this link]
StatusNo opposition filed within time limit
Status updated on  21.08.2009
Database last updated on 16.11.2024
Most recent event   Tooltip27.09.2013Lapse of the patent in a contracting state
New state(s): TR		published on 30.10.2013  [2013/44]
Applicant(s)For all designated states
GLAXO GROUP LIMITED
Glaxo Wellcome House, Berkeley Avenue
Greenford, Middlesex UB6 0NN / GB
[N/P]
Former [2008/42]For all designated states
GLAXO GROUP LIMITED
Glaxo Wellcome House, Berkeley Avenue
Greenford, Middlesex UB6 ONN / GB
Former [2004/05]For all designated states
GLAXO GROUP LIMITED
Glaxo Wellcome House Berkeley Avenue
Greenford, Middlesex UB6 ONN / GB
Inventor(s)01 / BIGGADIKE, Keith
Gunnels Wood Road
Stevenage, Hertforshire SG1 2NY / GB
02 / JONES, Paul
Gunnels Wood Road
Stevenage, Hertforshire SG1 2NY / GB
03 / PAYNE, Jeremy John
Gunnels Wood Road
Stevenage, Hertforshire SG1 2NY / GB
 [2004/05]
Representative(s)Pritchard, Judith, et al
GlaxoSmithKline
Global Patents (CN925.1)
980 Great West Road
Brentford, Middlesex TW8 9GS / GB
[N/P]
Former [2009/40]Pritchard, Judith, et al
GlaxoSmithKline Corporate Intellectual Property (CN925.1) 980 Great West Road Brentford, Middlesex
TW8 9GS / GB
Former [2004/05]Pritchard, Judith, et al
GlaxoSmithKline, 980 Great West Road
Brentford, Middlesex TW8 9GS / GB
Application number, filing date02722463.330.04.2002
[2004/05]
WO2002GB01971
Priority number, dateGB2001001057830.04.2001         Original published format: GB 0110578
GB2001002798822.11.2001         Original published format: GB 0127988
GB2002000244202.02.2002         Original published format: GB 0202442
GB2002000263705.02.2002         Original published format: GB 0202637
[2004/05]
Filing languageEN
Procedural languageEN
PublicationType: A1 Application with search report
No.:WO02088167
Date:07.11.2002
Language:EN
[2002/45]
Type: A1 Application with search report 
No.:EP1383786
Date:28.01.2004
Language:EN
The application published by WIPO in one of the EPO official languages on 07.11.2002 takes the place of the publication of the European patent application.
[2004/05]
Type: B1 Patent specification 
No.:EP1383786
Date:15.10.2008
Language:EN
[2008/42]
Search report(s)International search report - published on:EP07.11.2002
ClassificationIPC:C07J31/00, A61K31/56, A61P5/44, A61P11/06, A61P17/00
[2004/05]
CPC:
C07J31/006 (EP,US); C07J31/00 (KR); A61P1/04 (EP);
A61P11/00 (EP); A61P11/02 (EP); A61P11/06 (EP);
A61P17/00 (EP); A61P17/04 (EP); A61P17/06 (EP);
A61P19/02 (EP); A61P27/14 (EP); A61P27/16 (EP);
A61P29/00 (EP); A61P37/08 (EP); A61P43/00 (EP);
A61P5/00 (EP); A61P5/44 (EP) (-)
Designated contracting statesAT,   BE,   CH,   CY,   DE,   DK,   ES,   FI,   FR,   GB,   GR,   IE,   IT,   LI,   LU,   MC,   NL,   PT,   SE,   TR [2004/05]
Extension statesALNot yet paid
LTNot yet paid
LVNot yet paid
MKNot yet paid
RONot yet paid
SI25.11.2003
TitleGerman:ANTIPHLOGISTISCHE 7.BETA.-CARBOTHIOATE ESTERDERIVATE VON ANDROSTAN MIT EINER 17.ALPHA.-ZYKLISCHEN ESTERGRUPPE[2004/05]
English:ANTI-INFLAMMATORY 17.BETA.-CARBOTHIOATE ESTER DERIVATIVES OF ANDROSTANE WITH A CYCLIC ESTER GROUP IN POSITION 17.ALPHA[2004/05]
French:DERIVES ANTI-INFLAMMATOIRES D'ANDROSTANE 17.BETA.-CARBOTHIOATE ESTER AVEC UN GROUPE CYCLIQUE EN POSITION 17.ALPHA[2004/05]
Entry into regional phase25.11.2003National basic fee paid 
25.11.2003Designation fee(s) paid 
25.11.2003Examination fee paid 
Examination procedure06.11.2002Request for preliminary examination filed
International Preliminary Examining Authority: EP
25.11.2003Amendment by applicant (claims and/or description)
25.11.2003Examination requested  [2004/05]
29.11.2007Communication of intention to grant the patent
20.03.2008Fee for grant paid
20.03.2008Fee for publishing/printing paid
Divisional application(s)EP08157256.2  / EP2039700
Opposition(s)16.07.2009No opposition filed within time limit [2009/39]
Fees paidRenewal fee
06.04.2004Renewal fee patent year 03
04.04.2005Renewal fee patent year 04
27.03.2006Renewal fee patent year 05
10.04.2007Renewal fee patent year 06
18.03.2008Renewal fee patent year 07
Opt-out from the exclusive  Tooltip
competence of the Unified
Patent Court		 See the Register of the Unified Patent Court for opt-out data
Responsibility for the accuracy, completeness or quality of the data displayed under the link provided lies entirely with the Unified Patent Court.
Lapses during opposition  TooltipTR15.10.2008
AT30.04.2009
CH30.04.2009
CY30.04.2009
DK30.04.2009
FI30.04.2009
IE30.04.2009
LI30.04.2009
LU30.04.2009
MC30.04.2009
SE01.05.2009
[2013/44]
Former [2011/31]AT30.04.2009
CH30.04.2009
CY30.04.2009
DK30.04.2009
FI30.04.2009
IE30.04.2009
LI30.04.2009
LU30.04.2009
MC30.04.2009
SE01.05.2009
Former [2011/21]AT30.04.2009
CH30.04.2009
CY30.04.2009
DK30.04.2009
FI30.04.2009
IE30.04.2009
LI30.04.2009
LU30.04.2009
MC30.04.2009
Former [2010/37]AT30.04.2009
CH30.04.2009
CY30.04.2009
DK30.04.2009
FI30.04.2009
IE30.04.2009
LI30.04.2009
MC30.04.2009
Former [2010/21]CH30.04.2009
CY30.04.2009
DK30.04.2009
FI30.04.2009
IE30.04.2009
LI30.04.2009
MC30.04.2009
Former [2010/20]CH30.04.2009
CY30.04.2009
DK30.04.2009
FI30.04.2009
IE30.04.2009
LI30.04.2009
Former [2010/16]CH30.04.2009
CY30.04.2009
FI30.04.2009
LI30.04.2009
Former [2010/09]CH30.04.2009
FI30.04.2009
LI30.04.2009
Former [2010/08]CH30.04.2009
LI30.04.2009
Cited inInternational search[Y]US3312590  (JOSEPH ELKS, et al) [Y] 1-26 * column 1, lines 15-27; example 8 *;
 [Y]US3557162  (LENS JAN, et al) [Y] 1-26 * page 3, lines 44-50; example VI *;
 [Y]US3639434  (OXLEY PETER, et al) [Y] 1-26 * column 1, lines 49-57; examples 1,19 *;
 [Y]US3891631  (PHILLIPPS GORDON HANLEY, et al) [Y] 1-26 * column 1, lines 6-14 * * column 5, line 10 *;
 [Y]US4113680  (KAMANO YOSHIAKI, et al) [Y] 1-26 * page 2, lines 34-38,51-56; examples 7,24,73,83,104G,108C,113,141,156,194,219 *;
 [Y]BE889563  (OTSUKA PHARMA CO LTD) [Y] 1-26 * page 2, paragraph 2 * * page 64, paragraph 3 - page 65, paragraph 1 * * page 66, paragraph 1 * * page 99 *;
 [Y]US4335121  (PHILLIPPS GORDON H, et al) [Y] 1-26 * column 32, lines 52-65; examples 9,10,14,30 * * column 33, lines 12-16 *;
 [PY]WO0200679  (NOVARTIS AG [CH], et al) [PY] 1-26* page 7, paragraph L - page 8, paragraph L; examples 8,9,12,14,24,32,34; claim 1 *;
 [Y]  - PHILLIPPS G H ET AL, "SYNTHESIS AND STRUCTURE-ACTIVITY RELATIONSHIPS IN A SERIES OF ANTIINFLAMMATORY CORTICOSTEROID ANALOGUES, HALOMETHYL ANDROSTANE- 17BETA-CARBOTHIOATES AND-17BETA-CARBOSELENOATES", JOURNAL OF MEDICINAL CHEMISTRY, AMERICAN CHEMICAL SOCIETY. WASHINGTON, US, (19941001), vol. 37, no. 22, ISSN 0022-2623, pages 3717 - 3729, XP002025925 [Y] 1-26 * page 3722; example 13F; table 3 *

DOI:   http://dx.doi.org/10.1021/jm00048a008
 [Y]  - ISOGAI M ET AL, "BINDING AFFINITIES OF MOMETASONE FUROATE AND RELATED COMPOUNDS INCLUDING ITS METABOLITES FOR THE GLUCOCORTICOID RECEPTOR OF RAT SKIN TISSUE", JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY, ELSEVIER SCIENCE LTD., OXFORD, GB, (1993), vol. 44, no. 2, ISSN 0960-0760, pages 141 - 145, XP001040943 [Y] 1-26 * page 143; example XI * * page 144; table 1 *

DOI:   http://dx.doi.org/10.1016/0960-0760(93)90021-N
 [Y]  - UENO H ET AL, "Synthesis and evaluation of antiinflammatory activities of a series of corticosteroid 17.alpha.-esters containing a functional group", JOURNAL OF MEDICINAL CHEMISTRY, AMERICAN CHEMICAL SOCIETY. WASHINGTON, US, (19910801), vol. 34, no. 8, ISSN 0022-2623, pages 2468 - 2473, XP002086576 [Y] 1-26 * page 2470; example 13I; table II * * page 2471, column 1, paragraph 1 *

DOI:   http://dx.doi.org/10.1021/jm00112a023
The EPO accepts no responsibility for the accuracy of data originating from other authorities; in particular, it does not guarantee that it is complete, up to date or fit for specific purposes.