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Extract from the Register of European Patents

EP About this file: EP1412354

EP1412354 - DERIVATIVES OF TRIAZOLYL-IMIDAZOPYRIDINE AND OF THE TRIAZOLYLPURINES USEFUL AS LIGANDS OF THE ADENOSINE A 2a? RECEPTOR AND THEIR USE AS MEDICAMENTS [Right-click to bookmark this link]
StatusNo opposition filed within time limit
Status updated on  16.03.2007
Database last updated on 12.11.2024
Most recent event   Tooltip05.10.2007Change - lapse in a contracting state
State(s) deleted from list of lapses: IT
published on 07.11.2007  [2007/45]
Applicant(s)For all designated states
SIGMA-TAU Industrie Farmaceutiche Riunite S.p.A.
Viale Shakespeare, 47
00144 Roma / IT
[2006/19]
Former [2004/18]For all designated states
SIGMA-TAU Industrie Farmaceutiche Riunite S.p.A.
Viale Shakespeare, 47
00144 Roma / IT
Inventor(s)01 / TARZIA, Giorgio, Sigma-Tau Ind. Farm. Riu. SpA
Via Pontina Km. 30,400
I-00040 Pomezia / IT
02 / PIERSANTI, Giovanni, Sigma-Tau Ind. Farm. Riu. SpA
Via Pontina Km. 30,400
I-00040 Pomezia / IT
03 / MINETTI, Patrizia, Sigma-Tau Ind. Farm. Riu. SpA
Via Pontina Km. 30,400
I-00040 Pomezia / IT
04 / DI CESARE, Maria A., Sigma-Tau Ind. Farm. Riu. SpA
Via Pontina Km. 30,400
I-00040 Pomezia / IT
05 / GALLO, Grazia, Sigma-Tau Ind. Farm. Riu. SpA
Via Pontina Km. 30,400
I-00040 Pomezia / IT
06 / GIORGI, Fabrizio, Sigma-Tau Ind. Farm. Riu. SpA
Via Pontina Km. 30,400
I-00040 Pomezia / IT
07 / GIORGI, Luca, Sigma-Tau Ind. Farm. Riu. SpA
Via Pontina Km. 30,400
I-00040 Pomezia / IT
 [2004/18]
Representative(s)Spadaro, Marco
Cavattoni-Raimondi
Viale dei Parioli 160
00197 Roma / IT
[N/P]
Former [2004/18]Spadaro, Marco
Cavattoni-Raimondi Viale dei Parioli 160
00197 Roma / IT
Application number, filing date02760555.925.07.2002
[2004/18]
WO2002IT00489
Priority number, dateIT2001RM0046531.07.2001         Original published format: IT RM20010465
[2004/18]
Filing languageEN
Procedural languageEN
PublicationType: A1 Application with search report
No.:WO03011864
Date:13.02.2003
Language:EN
[2003/07]
Type: A1 Application with search report 
No.:EP1412354
Date:28.04.2004
Language:EN
The application published by WIPO in one of the EPO official languages on 13.02.2003 takes the place of the publication of the European patent application.
[2004/18]
Type: B1 Patent specification 
No.:EP1412354
Date:10.05.2006
Language:EN
[2006/19]
Search report(s)International search report - published on:EP13.02.2003
ClassificationIPC:C07D473/34, C07D471/04, A61K31/435, A61K31/52, A61P25/00, A61P25/28, A61P25/16
[2004/18]
CPC:
C07D471/04 (EP,US); C07D473/34 (EP,KR,US); A61K31/198 (EP,US);
A61K31/435 (EP,US); A61K31/52 (EP,US); A61P13/12 (EP);
A61P25/00 (EP); A61P25/14 (EP); A61P25/16 (EP);
A61P25/28 (EP); A61P43/00 (EP); A61P9/10 (EP) (-)
C-Set:
A61K31/198, A61K2300/00 (EP,US);
A61K31/435, A61K2300/00 (US,EP);
A61K31/52, A61K2300/00 (US,EP)
Designated contracting statesAT,   BE,   BG,   CH,   CY,   CZ,   DE,   DK,   EE,   ES,   FI,   FR,   GB,   GR,   IE,   IT,   LI,   LU,   MC,   NL,   PT,   SE,   SK,   TR [2004/18]
Extension statesALNot yet paid
LTNot yet paid
LVNot yet paid
MKNot yet paid
RONot yet paid
SINot yet paid
TitleGerman:DERIVATE VON TRIAZOLYL-IMIDAZOPYRIDINE UND VON TRIAZOLYLPURINE ALS LIGANDE DES ADENOSINE A2A REZEPTOREN UND IHRE VERWENDUNG ALS MEDICAMENTE[2004/18]
English:DERIVATIVES OF TRIAZOLYL-IMIDAZOPYRIDINE AND OF THE TRIAZOLYLPURINES USEFUL AS LIGANDS OF THE ADENOSINE A 2a? RECEPTOR AND THEIR USE AS MEDICAMENTS[2004/18]
French:DERIVES DE TRIAZOLYL-IMIDAZOPYRIDINE ET DE TRIAZOLYLPURINES UTILISES EN TANT QUE LIGANDS DU RECEPTEUR DE L'ADENOSINE A2A ET LEUR UTILISATION EN TANT QUE MEDICAMENTS[2004/18]
Entry into regional phase20.01.2004National basic fee paid 
20.01.2004Designation fee(s) paid 
20.01.2004Examination fee paid 
Examination procedure23.01.2003Request for preliminary examination filed
International Preliminary Examining Authority: EP
20.01.2004Examination requested  [2004/18]
21.07.2004Despatch of a communication from the examining division (Time limit: M04)
15.11.2004Reply to a communication from the examining division
08.06.2005Despatch of communication that the application is deemed to be withdrawn, reason: fee for grant / fee for printing not paid in time
16.06.2005Request for decision received: Application is deemed to be withdrawn
20.07.2005Fee for grant paid
20.07.2005Fee for publishing/printing paid
11.10.2005Communication of intention to grant the patent
11.10.2005Result of request for decision (Application is deemed to be withdrawn): Request accepted
Opposition(s)13.02.2007No opposition filed within time limit [2007/16]
Fees paidRenewal fee
21.06.2004Renewal fee patent year 03
17.06.2005Renewal fee patent year 04
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Patent Court
See the Register of the Unified Patent Court for opt-out data
Responsibility for the accuracy, completeness or quality of the data displayed under the link provided lies entirely with the Unified Patent Court.
Lapses during opposition  Tooltipdeleted
[2007/45]
Former [2007/39]IT10.05.2006
Cited inInternational search[A]WO9009178  (WHITBY RESEARCH INC [US]) [A] 1-31 * page 3 - page 6; example - *;
 [A]WO9606845  (DISCOVERY THERAPEUTICS INC [US]) [A] 1-31 * example - *;
 [A]EP1054012  (EISAI CO LTD [JP]) [A] 1-31 * claim - *;
 [AD]WO0102409  (VERNALIS RES LTD [GB], et al) [AD] 1-31 * example - *;
 [AD]  - YACOUBI ET AL., "SCH 58261 and ZM 241385 differentially prevent the motor effects of CGS 21680 in mice: evidence for a functional "atypical" adenosine A2a receptor", EUROPEAN JOURNAL OF PHARMACOLOGY, (2000), vol. 401, pages 63 - 77, XP002221553 [AD] 1-31 * the whole document *

DOI:   http://dx.doi.org/10.1016/S0014-2999(00)00399-X
 [A]  - CAMAIONI E ET AL, "NEW SUBSTITUTED 9-ALKYLPURINES AS ADENOSINE RECEPTOR LIGANDS", BIOORGANIC & MEDICINAL CHEMISTRY, ELSEVIER SCIENCE LTD, GB, (1998), vol. 6, no. 5, ISSN 0968-0896, pages 523 - 533, XP002926121 [A] 1-31 * page 524 - page 525; tables 1,2 *

DOI:   http://dx.doi.org/10.1016/S0968-0896(98)00007-8
 [AD]  - ONGINI E ET AL, "Pharmacology of Adenosine A2A Receptors", TRENDS IN PHARMACOLOGICAL SCIENCES, ELSEVIER TRENDS JOURNAL, CAMBRIDGE, GB, (199610), vol. 17, no. 10, ISSN 0165-6147, pages 364 - 372, XP002123410 [AD] 1-31 * page 370 *

DOI:   http://dx.doi.org/10.1016/S0165-6147(96)10045-6
The EPO accepts no responsibility for the accuracy of data originating from other authorities; in particular, it does not guarantee that it is complete, up to date or fit for specific purposes.