EP1412354 - DERIVATIVES OF TRIAZOLYL-IMIDAZOPYRIDINE AND OF THE TRIAZOLYLPURINES USEFUL AS LIGANDS OF THE ADENOSINE A 2a? RECEPTOR AND THEIR USE AS MEDICAMENTS [Right-click to bookmark this link] | Status | No opposition filed within time limit Status updated on 16.03.2007 Database last updated on 12.11.2024 | Most recent event Tooltip | 05.10.2007 | Change - lapse in a contracting state State(s) deleted from list of lapses: IT | published on 07.11.2007 [2007/45] | Applicant(s) | For all designated states SIGMA-TAU Industrie Farmaceutiche Riunite S.p.A. Viale Shakespeare, 47 00144 Roma / IT | [2006/19] |
Former [2004/18] | For all designated states SIGMA-TAU Industrie Farmaceutiche Riunite S.p.A. Viale Shakespeare, 47 00144 Roma / IT | Inventor(s) | 01 /
TARZIA, Giorgio, Sigma-Tau Ind. Farm. Riu. SpA Via Pontina Km. 30,400 I-00040 Pomezia / IT | 02 /
PIERSANTI, Giovanni, Sigma-Tau Ind. Farm. Riu. SpA Via Pontina Km. 30,400 I-00040 Pomezia / IT | 03 /
MINETTI, Patrizia, Sigma-Tau Ind. Farm. Riu. SpA Via Pontina Km. 30,400 I-00040 Pomezia / IT | 04 /
DI CESARE, Maria A., Sigma-Tau Ind. Farm. Riu. SpA Via Pontina Km. 30,400 I-00040 Pomezia / IT | 05 /
GALLO, Grazia, Sigma-Tau Ind. Farm. Riu. SpA Via Pontina Km. 30,400 I-00040 Pomezia / IT | 06 /
GIORGI, Fabrizio, Sigma-Tau Ind. Farm. Riu. SpA Via Pontina Km. 30,400 I-00040 Pomezia / IT | 07 /
GIORGI, Luca, Sigma-Tau Ind. Farm. Riu. SpA Via Pontina Km. 30,400 I-00040 Pomezia / IT | [2004/18] | Representative(s) | Spadaro, Marco Cavattoni-Raimondi Viale dei Parioli 160 00197 Roma / IT | [N/P] |
Former [2004/18] | Spadaro, Marco Cavattoni-Raimondi Viale dei Parioli 160 00197 Roma / IT | Application number, filing date | 02760555.9 | 25.07.2002 | [2004/18] | WO2002IT00489 | Priority number, date | IT2001RM00465 | 31.07.2001 Original published format: IT RM20010465 | [2004/18] | Filing language | EN | Procedural language | EN | Publication | Type: | A1 Application with search report | No.: | WO03011864 | Date: | 13.02.2003 | Language: | EN | [2003/07] | Type: | A1 Application with search report | No.: | EP1412354 | Date: | 28.04.2004 | Language: | EN | The application published by WIPO in one of the EPO official languages on 13.02.2003 takes the place of the publication of the European patent application. | [2004/18] | Type: | B1 Patent specification | No.: | EP1412354 | Date: | 10.05.2006 | Language: | EN | [2006/19] | Search report(s) | International search report - published on: | EP | 13.02.2003 | Classification | IPC: | C07D473/34, C07D471/04, A61K31/435, A61K31/52, A61P25/00, A61P25/28, A61P25/16 | [2004/18] | CPC: |
C07D471/04 (EP,US);
C07D473/34 (EP,KR,US);
A61K31/198 (EP,US);
A61K31/435 (EP,US);
A61K31/52 (EP,US);
A61P13/12 (EP);
A61P25/00 (EP);
A61P25/14 (EP);
A61P25/16 (EP);
| C-Set: |
A61K31/198, A61K2300/00 (EP,US);
A61K31/435, A61K2300/00 (US,EP);
A61K31/52, A61K2300/00 (US,EP)
| Designated contracting states | AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, IE, IT, LI, LU, MC, NL, PT, SE, SK, TR [2004/18] | Extension states | AL | Not yet paid | LT | Not yet paid | LV | Not yet paid | MK | Not yet paid | RO | Not yet paid | SI | Not yet paid | Title | German: | DERIVATE VON TRIAZOLYL-IMIDAZOPYRIDINE UND VON TRIAZOLYLPURINE ALS LIGANDE DES ADENOSINE A2A REZEPTOREN UND IHRE VERWENDUNG ALS MEDICAMENTE | [2004/18] | English: | DERIVATIVES OF TRIAZOLYL-IMIDAZOPYRIDINE AND OF THE TRIAZOLYLPURINES USEFUL AS LIGANDS OF THE ADENOSINE A 2a? RECEPTOR AND THEIR USE AS MEDICAMENTS | [2004/18] | French: | DERIVES DE TRIAZOLYL-IMIDAZOPYRIDINE ET DE TRIAZOLYLPURINES UTILISES EN TANT QUE LIGANDS DU RECEPTEUR DE L'ADENOSINE A2A ET LEUR UTILISATION EN TANT QUE MEDICAMENTS | [2004/18] | Entry into regional phase | 20.01.2004 | National basic fee paid | 20.01.2004 | Designation fee(s) paid | 20.01.2004 | Examination fee paid | Examination procedure | 23.01.2003 | Request for preliminary examination filed International Preliminary Examining Authority: EP | 20.01.2004 | Examination requested [2004/18] | 21.07.2004 | Despatch of a communication from the examining division (Time limit: M04) | 15.11.2004 | Reply to a communication from the examining division | 08.06.2005 | Despatch of communication that the application is deemed to be withdrawn, reason: fee for grant / fee for printing not paid in time | 16.06.2005 | Request for decision received: Application is deemed to be withdrawn | 20.07.2005 | Fee for grant paid | 20.07.2005 | Fee for publishing/printing paid | 11.10.2005 | Communication of intention to grant the patent | 11.10.2005 | Result of request for decision (Application is deemed to be withdrawn): Request accepted | Opposition(s) | 13.02.2007 | No opposition filed within time limit [2007/16] | Fees paid | Renewal fee | 21.06.2004 | Renewal fee patent year 03 | 17.06.2005 | Renewal fee patent year 04 |
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Responsibility for the accuracy, completeness or quality of the data displayed under the link provided lies entirely with the Unified Patent Court. | Lapses during opposition Tooltip | deleted | [2007/45] |
Former [2007/39] | IT | 10.05.2006 | Cited in | International search | [A]WO9009178 (WHITBY RESEARCH INC [US]) [A] 1-31 * page 3 - page 6; example - *; | [A]WO9606845 (DISCOVERY THERAPEUTICS INC [US]) [A] 1-31 * example - *; | [A]EP1054012 (EISAI CO LTD [JP]) [A] 1-31 * claim - *; | [AD]WO0102409 (VERNALIS RES LTD [GB], et al) [AD] 1-31 * example - *; | [AD] - YACOUBI ET AL., "SCH 58261 and ZM 241385 differentially prevent the motor effects of CGS 21680 in mice: evidence for a functional "atypical" adenosine A2a receptor", EUROPEAN JOURNAL OF PHARMACOLOGY, (2000), vol. 401, pages 63 - 77, XP002221553 [AD] 1-31 * the whole document * DOI: http://dx.doi.org/10.1016/S0014-2999(00)00399-X | [A] - CAMAIONI E ET AL, "NEW SUBSTITUTED 9-ALKYLPURINES AS ADENOSINE RECEPTOR LIGANDS", BIOORGANIC & MEDICINAL CHEMISTRY, ELSEVIER SCIENCE LTD, GB, (1998), vol. 6, no. 5, ISSN 0968-0896, pages 523 - 533, XP002926121 [A] 1-31 * page 524 - page 525; tables 1,2 * DOI: http://dx.doi.org/10.1016/S0968-0896(98)00007-8 | [AD] - ONGINI E ET AL, "Pharmacology of Adenosine A2A Receptors", TRENDS IN PHARMACOLOGICAL SCIENCES, ELSEVIER TRENDS JOURNAL, CAMBRIDGE, GB, (199610), vol. 17, no. 10, ISSN 0165-6147, pages 364 - 372, XP002123410 [AD] 1-31 * page 370 * DOI: http://dx.doi.org/10.1016/S0165-6147(96)10045-6 |