EP1442024 - AMINOBENZAMIDE DERIVATIVES AS GLYCOGEN SYNTHASE KINASE 3$g(b) INHIBITORS [Right-click to bookmark this link] | Status | No opposition filed within time limit Status updated on 20.09.2013 Database last updated on 18.11.2024 | Most recent event Tooltip | 20.09.2013 | No opposition filed within time limit | published on 23.10.2013 [2013/43] | 20.09.2013 | Change - no opposition filed | published on 23.10.2013 [2013/43] | Applicant(s) | For all designated states Janssen Pharmaceutica NV Turnhoutseweg 30 2340 Beerse / BE | [2008/12] |
Former [2004/32] | For all designated states JANSSEN PHARMACEUTICA N.V. Turnhoutsebaan 30 2340 Beerse / BE | Inventor(s) | 01 /
FREYNE, Eddy J. E., Janssen Pharmaceutica N.V. Turnhoutseweg 30 B-2340 Beerse / BE | 02 /
BUIJNSTERS, Peter J. J. A., Janssen Pharmaceutica N.V. Turnhoutseweg 30 B-2340 Beerse / BE | 03 /
WILLEMS, Marc, Janssen Pharmaceutica N.V. Turnhoutseweg 30 B-2340 Beerse / BE | 04 /
EMBRECHTS, Werner C. J., Janssen Pharmaceutica N.V. Turnhoutseweg 30 B-2340 Beerse / BE | 05 /
JANSSEN, Paul A. J. (deceased) / BE | 06 /
LEWI, Paulus Joannes, Janssen Pharmaceutica N.V. Turnhoutseweg 30 B-2340 Beerse / BE | 07 /
HEERES, Jan, Janssen Pharmaceutica N.V. Turnhoutseweg 30 B-2340 Beerse / BE | 08 /
DE JONGE, Marc R., Janssen Pharmaceutica N.V. Turnhoutseweg 30 B-2340 Beerse / BE | 09 /
KOYMANS, Lucien M. H., Janssen Pharmaceutica N.V. Turnhoutseweg 30 B-2340 Beerse / BE | 10 /
DAEYAERT, Frederik F. D., Janssen Pharmaceutica N.V. Turnhoutseweg 30 B-2340 Beerse / BE | 11 /
KUKLA, Michael J. 1551 Oak Hollow Drive Maple Glen, PA 19002 / US | 12 /
GEERTS, Hugo A. G. 686 Westwind Drive Berwyn, PA 19312 / US | 13 /
NUYDENS, Rony M., Janssen Pharmaceutica N.V. Turnhoutseweg 30 B-2340 Beerse / BE | 14 /
MERCKEN, Marc H., Janssen Pharmaceutica N.V. Turnhoutseweg 30 B-2340 Beerse / BE | 15 /
LUDOVICI, Donald W., Janssen Pharmaceutica Inc. 1125 Trenton-Harbourton Road Titusville, NJ 08560 / US | 16 /
JANSSEN, Jasmine, Josee, Werner Zinkvalstraat 5 B-2360 Aartselaar / BE | 17 /
JANSSEN, Maroussia, Godelieve, Frank Dreve du Carmel 17 B-1410 Waterloo / BE | 18 /
JANSSEN, Paul, Peter, Maria Grotesteenweg-Zuid 4 B-9052 Zwijnaarde / BE | 19 /
ARTS, Theodora, Joanna, Francisca Antwerpsesteenweg 20 B-2350 Vosselaar / BE | 20 /
JANSSEN, Herwig, Josephus, Margareta Koekoeksdreef 47 B-2970 Schide / BE | [2008/07] |
Former [2004/32] | 01 /
FREYNE, Eddy J. E., Janssen Pharma. N.V. Turnhoutseweg 30 B-2340 Beerse / BE | ||
02 /
BUIJNSTERS, Peter J. J. A., Janssen Pharma. N.V. Turnhoutseweg 30 B-2340 Beerse / BE | |||
03 /
WILLEMS, Marc, Janssen Pharma. N.V. Turnhoutseweg 30 B-2340 Beerse / BE | |||
04 /
EMBRECHTS, Werner C. J., Janssen Pharma. N.V. Turnhoutseweg 30 B-2340 Beerse / BE | |||
05 /
JANSSEN, Paul A. J. (deceased) / BE | |||
06 /
LEWI, Paulus Joannes, Janssen Pharma. N.V. Turnhoutseweg 30 B-2340 Beerse / BE | |||
07 /
HEERES, Jan, Janssen Pharma. N.V. Turnhoutseweg 30 B-2340 Beerse / BE | |||
08 /
DE JONGE, Marc R., Janssen Pharma. N.V. Turnhoutseweg 30 B-2340 Beerse / BE | |||
09 /
KOYMANS, Lucien M. H., Janssen Pharma. N.V. Turnhoutseweg 30 B-2340 Beerse / BE | |||
10 /
DAEYAERT, Frederik F. D., Janssen Pharma. N.V. Turnhoutseweg 30 B-2340 Beerse / BE | |||
11 /
KUKLA, Michael J. 1551 Oak Hollow Drive Maple Glen, PA 19002 / US | |||
12 /
GEERTS, Hugo A. G. 686 Westwind Drive Berwyn, PA 19312 / US | |||
13 /
NUYDENS, Rony M., Janssen Pharma. N.V. Turnhoutseweg 30 B-2340 Beerse / BE | |||
14 /
MERCKEN, Marc H., Janssen Pharma. N.V. Turnhoutseweg 30 B-2340 Beerse / BE | |||
15 /
LUDOVICI, Donald W., Janssen Pharma. Inc. 1125 Trenton-Harbourton Road Titusville, NJ 08560 / US | |||
16 /
JANSSEN, Jasmine, Josee, Werner Zinkvalstraat 5 B-2360 Aartselaar / BE | |||
17 /
JANSSEN, Maroussia, Godelieve, Frank Dreve du Carmel 17 B-1410 Waterloo / BE | |||
18 /
JANSSEN, Paul, Peter, Maria Grotesteenweg-Zuid 4 B-9052 Zwijnaarde / BE | |||
19 /
ARTS, Theodora, Joanna, Francisca Antwerpsesteenweg 20 B-2350 Vosselaar / BE | |||
20 /
JANSSEN, Herwig, Josephus, Margareta Koekoeksdreef 47 B-2970 Schide / BE | Application number, filing date | 02802307.5 | 29.10.2002 | [2004/32] | WO2002EP12079 | Priority number, date | EP20010204192 | 01.11.2001 Original published format: EP 01204192 | [2004/32] | Filing language | EN | Procedural language | EN | Publication | Type: | A1 Application with search report | No.: | WO03037877 | Date: | 08.05.2003 | Language: | EN | [2003/19] | Type: | A1 Application with search report | No.: | EP1442024 | Date: | 04.08.2004 | Language: | EN | The application published by WIPO in one of the EPO official languages on 08.05.2003 takes the place of the publication of the European patent application. | [2004/32] | Type: | B1 Patent specification | No.: | EP1442024 | Date: | 19.03.2008 | Language: | EN | [2008/12] | Search report(s) | International search report - published on: | EP | 08.05.2003 | Classification | IPC: | C07D239/30, C07D239/46, C07D239/48, C07D403/10, A61K31/506, A61P3/10, A61P25/28 | [2004/32] | CPC: |
C07D239/42 (EP,US);
C07D239/46 (KR);
A61K31/506 (EP,US);
A61P17/00 (EP);
A61P21/04 (EP);
A61P25/00 (EP);
A61P25/04 (EP);
A61P25/16 (EP);
A61P25/18 (EP);
A61P25/24 (EP);
A61P25/28 (EP);
A61P29/00 (EP);
A61P3/10 (EP);
A61P35/00 (EP);
A61P43/00 (EP);
A61P7/00 (EP);
C07D239/47 (EP,US);
C07D239/48 (EP,US);
| Designated contracting states | AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, IE, IT, LI, LU, MC, NL, PT, SE, SK, TR [2004/32] | Extension states | AL | 01.06.2004 | LT | 01.06.2004 | LV | 01.06.2004 | MK | 01.06.2004 | RO | 01.06.2004 | SI | 01.06.2004 | Title | German: | AMINOBENZAMIDDERIVATE ALS INHIBITOREN DER GLYCOGENSYNTHASEKINASE-3- | [2004/32] | English: | AMINOBENZAMIDE DERIVATIVES AS GLYCOGEN SYNTHASE KINASE 3$g(b) INHIBITORS | [2004/32] | French: | DERIVES D'AMINOBENZAMIDE UTILES COMME INHIBITEURS DE LA GLYCOGENE SYNTHASE KINASE 3$G(B) | [2004/32] | Entry into regional phase | 01.06.2004 | National basic fee paid | 01.06.2004 | Designation fee(s) paid | 01.06.2004 | Examination fee paid | Examination procedure | 10.04.2003 | Request for preliminary examination filed International Preliminary Examining Authority: EP | 01.06.2004 | Examination requested [2004/32] | 05.11.2004 | Despatch of a communication from the examining division (Time limit: M06) | 04.05.2005 | Reply to a communication from the examining division | 29.03.2006 | Despatch of a communication from the examining division (Time limit: M04) | 28.07.2006 | Reply to a communication from the examining division | 10.09.2007 | Communication of intention to grant the patent | 07.01.2008 | Fee for grant paid | 07.01.2008 | Fee for publishing/printing paid | Opposition(s) | 22.12.2008 | No opposition filed within time limit [2009/09] | 22.12.2008 | No opposition filed within time limit [2013/43] | Fees paid | Renewal fee | 02.11.2004 | Renewal fee patent year 03 | 31.10.2005 | Renewal fee patent year 04 | 31.10.2006 | Renewal fee patent year 05 | 31.10.2007 | Renewal fee patent year 06 |
Opt-out from the exclusive Tooltip competence of the Unified Patent Court | See the Register of the Unified Patent Court for opt-out data | ||
Responsibility for the accuracy, completeness or quality of the data displayed under the link provided lies entirely with the Unified Patent Court. | Lapses during opposition Tooltip | CY | 19.03.2008 | CZ | 19.03.2008 | EE | 19.03.2008 | SK | 19.03.2008 | BG | 19.06.2008 | MC | 31.10.2008 | [2009/42] |
Former [2009/25] | CZ | 19.03.2008 | |
EE | 19.03.2008 | ||
SK | 19.03.2008 | ||
BG | 19.06.2008 | ||
MC | 31.10.2008 | ||
Former [2009/23] | CZ | 19.03.2008 | |
EE | 19.03.2008 | ||
SK | 19.03.2008 | ||
BG | 19.06.2008 | ||
Former [2009/22] | CZ | 19.03.2008 | |
EE | 19.03.2008 | ||
SK | 19.03.2008 | ||
Former [2008/50] | CZ | 19.03.2008 | |
SK | 19.03.2008 | Cited in | International search | [DA]EP0162204 (GRIMME LANDMASCHF FRANZ [DE]) [DA] 1 * R1 is phenyl substituted by CONH2;; claim 1 *; | [DX]EP0233461 (AMERICAN CYANAMID CO [US]) [DX] 1 * R2 is phenyl substituted by CONH(CH2)nNRR;; example 266; claim 1 *; | [DX]EP0337943 (CIBA GEIGY AG [CH]) [DX] 1 * Compounds (II);; example 2.687; claim 7 *; | [DA]WO9118887 (SMITHKLINE BEECHAM INTERCREDIT [NL]) [DA] 1 * claim 1 *; | [DX]US5516775 (ZIMMERMANN JUERG [CH], et al) [DX] 1 * example F; claim 1 *; | [DX]EP0945443 (JANSSEN PHARMACEUTICA NV [BE]) [DX] 1 * Page 8, lines 31 and 40. *; | [X]WO9965897 (CHIRON CORP [US], et al) [X] 1-14 * Compounds where one of R5 and R7 is hydrogen and the other is aryl amino whereby the aryl group can be phenyl substituted by (alkyl)aminocarbonyl.;; claims 1,18 *; | [X]US6048866 (HUTCHINGS MARTIN CLIVE [GB], et al) [X] 1 * R1 is ((di)alkyl)carbamoyl.;; claim 1 *; | [A]WO0078731 (CELLTECH CHIROSCIENCE LTD [GB], et al) [A] 1* claim 7 *; | [X]WO0164655 (ASTRAZENECA AB [SE], et al) [X] 1 * page 37; examples 21-30,60-98,105-107,109-113,115,117-119 *; | [A] - ZIMMERMANN J ET AL, "Potent and selective inhibitors of the Abl-kinase: phenylamino-pyrimidine (PAP) derivatives", BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, OXFORD, GB, (19970121), vol. 7, no. 2, ISSN 0960-894X, pages 187 - 192, XP004135990 [A] 1 * example 13 * DOI: http://dx.doi.org/10.1016/S0960-894X(96)00601-4 |