blank Quick help
blank Maintenance news

Scheduled maintenance

Regular maintenance outages:
between 05.00 and 05.15 hrs CET (Monday to Sunday).

Other outages
Availability
Register Forum

2022.02.11

More...
blank News flashes

News Flashes

New version of the European Patent Register – SPC proceedings information in the Unitary Patent Register.

2024-07-24

More...
blank Related links

Extract from the Register of European Patents

EP About this file: EP1542994

EP1542994 - NOVEL OXAZOLE COMPOUNDS AS TRANSFORMING GROWTH FACTOR (TGF) INHIBITOR [Right-click to bookmark this link]
Former [2005/25]NOVEL TRIAZOLE AND OXAZOLE COMPOUNDS AS TRANSFORMING GROWTH FACTOR (TGF) INHIBITOR
[2008/45]
StatusNo opposition filed within time limit
Status updated on  05.03.2010
Database last updated on 31.08.2024
Most recent event   Tooltip07.10.2011Lapse of the patent in a contracting state
New state(s): CY, TR
published on 09.11.2011  [2011/45]
Applicant(s)For all designated states
Pfizer Products Inc.
Eastern Point Road
Groton, CT 06340 / US
[2009/18]
Former [2005/25]For all designated states
Pfizer Products Inc.
Eastern Point Road
Groton, Connecticut 06340 / US
Inventor(s)01 / BLUMBERG, Laura, Cook
5 Division Street, Waterford
Connecticut 06385 / US
02 / MUNCHHOF, Michael, John
266 West Road, Salem
Connecticut 06420 / US
 [2005/25]
Representative(s)Pringot, Thomas, et al
ATTENTION: ADDRESS INACTIVE - USE ASS-NR - CDR / FR
[N/P]
Former [2009/21]Pringot, Thomas, et al
Pfizer Limited European Patent Department Ramsgate Road
Sandwich, Kent CT13 9NJ / GB
Former [2009/20]Pringot, Thomas, et al
Pfizer Limited European Patent Department Ramsgate Road
Sandwich, Kent CT13 9NJ / FR
Former [2006/16]Pringot, Thomas, et al
Pfizer European Pharma Patent Dept. 23/25 Avenue du Docteur Lannelongue
F-75668 Paris Cedex 14 / FR
Former [2005/25]Tesch, Rudolf, Dr., et al
c/o Pfizer GmbH, Arzneimittelwerk Gödecke Mooswaldallee 1
79090 Freiburg / DE
Application number, filing date03797426.808.09.2003
[2005/25]
WO2003IB03823
Priority number, dateUS20020412120P18.09.2002         Original published format: US 412120 P
US20030471265P16.05.2003         Original published format: US 471265 P
US20030484581P02.07.2003         Original published format: US 484581 P
[2005/25]
Filing languageEN
Procedural languageEN
PublicationType: A1 Application with search report
No.:WO2004026863
Date:01.04.2004
Language:EN
[2004/14]
Type: A1 Application with search report 
No.:EP1542994
Date:22.06.2005
Language:EN
The application published by WIPO in one of the EPO official languages on 01.04.2004 takes the place of the publication of the European patent application.
[2005/25]
Type: B1 Patent specification 
No.:EP1542994
Date:29.04.2009
Language:EN
[2009/18]
Search report(s)International search report - published on:EP01.04.2004
ClassificationIPC:C07D413/14, C07D417/14, C07D419/14, C07D413/04, C07D417/04, A61P35/00
[2005/25]
CPC:
C07D413/14 (EP,KR,US); A61P1/16 (EP); A61P11/00 (EP);
A61P13/12 (EP); A61P17/00 (EP); A61P17/02 (EP);
A61P3/10 (EP); A61P35/00 (EP); A61P43/00 (EP);
A61P9/10 (EP); C07D417/14 (EP,KR,US) (-)
Designated contracting statesAT,   BE,   BG,   CH,   CY,   CZ,   DE,   DK,   EE,   ES,   FI,   FR,   GB,   GR,   HU,   IE,   IT,   LI,   LU,   MC,   NL,   PT,   RO,   SE,   SI,   SK,   TR [2009/18]
Former [2005/25]AT,  BE,  BG,  CH,  CY,  CZ,  DE,  DK,  EE,  ES,  FI,  FR,  GB,  GR,  HU,  IE,  IT,  LI,  LU,  MC,  NL,  PT,  RO,  SE,  SI,  SK,  TR 
Extension statesAL18.04.2005
LT18.04.2005
LV18.04.2005
MK18.04.2005
TitleGerman:NEUE OXAZOLVERBINDUNGEN ALS INHIBITOREN DES TRANSFORMING GROWTH FACTOR (TGF)[2008/45]
English:NOVEL OXAZOLE COMPOUNDS AS TRANSFORMING GROWTH FACTOR (TGF) INHIBITOR[2008/45]
French:NOUVEAUX DERIVES D'OXAZOLE COMME INHIBITEURS DU FACTEUR DE CROISSANCE TRANSFORMANT[2008/45]
Former [2005/25]NEUE TRIAZOL- UND OXAZOLVERBINDUNGEN ALS INHIBITOREN DES TRANSFORMING GROWTH FACTOR (TGF)
Former [2005/25]NOVEL TRIAZOLE AND OXAZOLE COMPOUNDS AS TRANSFORMING GROWTH FACTOR (TGF) INHIBITOR
Former [2005/25]NOUVEAUX COMPOSES DE TRIAZOLE ET D'OXAZOLE, INHIBITEURS DU FACTEUR DE CROISSANCE TRANSFORMANT
Entry into regional phase18.04.2005National basic fee paid 
18.04.2005Designation fee(s) paid 
18.04.2005Examination fee paid 
Examination procedure06.10.2003Request for preliminary examination filed
International Preliminary Examining Authority: EP
12.03.2005Amendment by applicant (claims and/or description)
18.04.2005Examination requested  [2005/25]
30.01.2006Despatch of a communication from the examining division (Time limit: M06)
13.09.2006Despatch of communication that the application is deemed to be withdrawn, reason: reply to the communication from the examining division not received in time
08.11.2006Reply to a communication from the examining division
25.10.2007Despatch of a communication from the examining division (Time limit: M04)
27.11.2007Reply to a communication from the examining division
09.12.2008Communication of intention to grant the patent
16.03.2009Fee for grant paid
16.03.2009Fee for publishing/printing paid
Opposition(s)01.02.2010No opposition filed within time limit [2010/14]
Request for further processing for:08.11.2006Request for further processing filed
08.11.2006Full payment received (date of receipt of payment)
Request granted
21.11.2006Decision despatched
Fees paidRenewal fee
05.09.2005Renewal fee patent year 03
08.09.2006Renewal fee patent year 04
05.09.2007Renewal fee patent year 05
30.09.2008Renewal fee patent year 06
Opt-out from the exclusive  Tooltip
competence of the Unified
Patent Court
See the Register of the Unified Patent Court for opt-out data
Responsibility for the accuracy, completeness or quality of the data displayed under the link provided lies entirely with the Unified Patent Court.
Lapses during opposition  TooltipAT29.04.2009
BE29.04.2009
CY29.04.2009
CZ29.04.2009
DK29.04.2009
EE29.04.2009
FI29.04.2009
NL29.04.2009
RO29.04.2009
SI29.04.2009
SK29.04.2009
TR29.04.2009
BG29.07.2009
SE29.07.2009
GR30.07.2009
PT29.08.2009
LU08.09.2009
CH30.09.2009
LI30.09.2009
MC30.09.2009
HU30.10.2009
[2011/44]
Former [2011/31]AT29.04.2009
BE29.04.2009
CZ29.04.2009
DK29.04.2009
EE29.04.2009
FI29.04.2009
NL29.04.2009
RO29.04.2009
SI29.04.2009
SK29.04.2009
BG29.07.2009
SE29.07.2009
GR30.07.2009
PT29.08.2009
LU08.09.2009
CH30.09.2009
LI30.09.2009
MC30.09.2009
HU30.10.2009
Former [2011/21]AT29.04.2009
BE29.04.2009
CZ29.04.2009
DK29.04.2009
EE29.04.2009
FI29.04.2009
NL29.04.2009
RO29.04.2009
SI29.04.2009
SK29.04.2009
BG29.07.2009
SE29.07.2009
GR30.07.2009
PT29.08.2009
LU08.09.2009
CH30.09.2009
LI30.09.2009
MC30.09.2009
Former [2010/46]AT29.04.2009
BE29.04.2009
CZ29.04.2009
DK29.04.2009
EE29.04.2009
FI29.04.2009
NL29.04.2009
RO29.04.2009
SI29.04.2009
SK29.04.2009
BG29.07.2009
SE29.07.2009
GR30.07.2009
PT29.08.2009
CH30.09.2009
LI30.09.2009
MC30.09.2009
Former [2010/20]AT29.04.2009
BE29.04.2009
CZ29.04.2009
DK29.04.2009
EE29.04.2009
FI29.04.2009
NL29.04.2009
RO29.04.2009
SI29.04.2009
SK29.04.2009
BG29.07.2009
SE29.07.2009
PT29.08.2009
MC30.09.2009
Former [2010/18]AT29.04.2009
BE29.04.2009
CZ29.04.2009
DK29.04.2009
EE29.04.2009
FI29.04.2009
NL29.04.2009
RO29.04.2009
SI29.04.2009
SK29.04.2009
BG29.07.2009
SE29.07.2009
PT29.08.2009
Former [2010/10]AT29.04.2009
BE29.04.2009
CZ29.04.2009
DK29.04.2009
EE29.04.2009
FI29.04.2009
NL29.04.2009
RO29.04.2009
SI29.04.2009
SK29.04.2009
SE29.07.2009
PT29.08.2009
Former [2010/09]AT29.04.2009
CZ29.04.2009
DK29.04.2009
EE29.04.2009
FI29.04.2009
NL29.04.2009
RO29.04.2009
SI29.04.2009
SE29.07.2009
PT29.08.2009
Former [2010/08]AT29.04.2009
DK29.04.2009
EE29.04.2009
FI29.04.2009
NL29.04.2009
SI29.04.2009
SE29.07.2009
PT29.08.2009
Former [2009/51]AT29.04.2009
FI29.04.2009
NL29.04.2009
SI29.04.2009
SE29.07.2009
PT29.08.2009
Former [2009/50]AT29.04.2009
FI29.04.2009
NL29.04.2009
PT29.08.2009
Cited inInternational search[X]WO0240476  (SMITHKLINE BEECHAM CORP [US], et al) [X] 1-12 * see claim 1 and examples on pages 12-20 *;
 [X]  - YANG, QIANG ET AL, "The reaction of heteroaryl-substituted heterocyclic ketene aminals with 2,3,4,6-tetra-O-acetyl-.beta.-D-glucopyranosyl azide", HETEROATOM CHEMISTRY (2002), 13(3), 242-247, XP009022047 [X] 1-10 * see compound 6c-8c and 12c-14c *

DOI:   http://dx.doi.org/10.1002/hc.10023
 [X]  - LIU, BO ET AL, "The reaction of aroyl-substituted heterocyclic ketene aminals with aryl azides", HETEROATOM CHEMISTRY (2000), 11(6), 387-391, XP009022048 [X] 1-10 * see compounds 4c and 5c *

DOI:   http://dx.doi.org/10.1002/1098-1071(2000)11:6<387::AID-HC5>3.0.CO;2-H
The EPO accepts no responsibility for the accuracy of data originating from other authorities; in particular, it does not guarantee that it is complete, up to date or fit for specific purposes.