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Extract from the Register of European Patents

EP About this file: EP1569646

EP1569646 - PIPERIDINE DERIVATIVES AS CCR5 ANTAGONISTS [Right-click to bookmark this link]
StatusThe application is deemed to be withdrawn
Status updated on  17.09.2010
Database last updated on 24.08.2024
Most recent event   Tooltip17.09.2010Application deemed to be withdrawnpublished on 20.10.2010  [2010/42]
Applicant(s)For all designated states
GlaxoSmithKline LLC
One Franklin Plaza
200 North 16th Street
Philadelphia, PA 19102 / US
[N/P]
Former [2010/09]For all designated states
GlaxoSmithKline LLC
One Franklin Plaza 200 North 16th Street
Philadelphia, PA 19102 / US
Former [2005/36]For all designated states
SMITHKLINE BEECHAM CORPORATION
One Franklin Plaza
Philadelphia, PA 19102 / US
Inventor(s)01 / KAZMIERSKI, Wieslaw Mieczyslaw
GlaxoSmithKline, Five Moore Drive, PO Box 13398
Research Triangle Par, NC 27709 / US
02 / AQUINO, Christopher Joseph
GlaxoSmithKline, Five Moore Drive, PO Box 13398
Research Triangle Park, NC 27709 / US
03 / BIFULCO, Neil
GlaxoSmithKline, Five Moore Drive, PO Box 13398
Research Triangle Park, NC 27709 / US
04 / BOROS, Eric Eugene
GlaxoSmithKline, Five Moore Drive, PO Box 13398
Research Triangle Park, NC 27709 / US
05 / CHAUDER, Brian Andrew
GlaxoSmithKline, Five Moore Drive, PO Box 13398
Research Triangle Park, NC 27709 / US
06 / CHONG, Pek Yoke
GlaxoSmithKline, Five Moore Drive, PO Box 13398
Research Triangle Park, NC 27709 / US
07 / DUAN, Maosheng
GlaxoSmithKline, Five Moore Drive, PO Box 13398
Research Triangle Park, NC 27709 / US
08 / DEANDA, JR. Felix
GlaxoSmithKline, Five Moore Drive, PO Box 13398
Research Triangle Park, NC 27709 / US
09 / KOBLE, Cecilia Suarez
GlaxoSmithKline, Five Moore Drive, PO Box 13398
Research Triangle Park, NC 27709 / US
10 / MCLEAN, Ed Williams
GlaxoSmithKline, Five Moore Drive, PO Box 13398
Research Triangle Park, NC 27709 / US
11 / PECKHAM, Jennifer Poole
GlaxoSmithKline, Five Moore Drive, PO Box 13398
Research Triangle Park, NC 27709 / US
12 / PERKINS, Angilique C.
GlaxoSmithKline, Five Moore Drive, PO Box 13398
Research Triangle Park, NC 027709 / US
13 / THOMPSON, James Benjamin
GlaxoSmithKline, Five Moore Drive, PO Box 13398
Research Triangle Park, NC 27709 / US
14 / VANDERWALL, Dana
GlaxoSmithKline, Five Moore Drive, O Box 13398
Research Triangle Park, NC 27709 / US
 [2005/36]
Representative(s)Gladwin, Amanda Rachel
GlaxoSmithKline
Global Patents (CN925.1)
980 Great West Road
Brentford, Middlesex TW8 9GS / GB
[N/P]
Former [2005/36]Gladwin, Amanda Rachel
GlaxoSmithKline, Corporate Intellectual Property, CN925.1, 980 Great West Road Brentford
Middlesex TW8 9GS / GB
Application number, filing date03813419.312.12.2003
[2005/36]
WO2003US39644
Priority number, dateUS20020433634P13.12.2002         Original published format: US 433634 P
[2005/36]
Filing languageEN
Procedural languageEN
PublicationType: A2 Application without search report
No.:WO2004054974
Date:01.07.2004
Language:EN
[2004/27]
Type: A2 Application without search report 
No.:EP1569646
Date:07.09.2005
Language:EN
The application published by WIPO in one of the EPO official languages on 01.07.2004 takes the place of the publication of the European patent application.
[2005/36]
Search report(s)International search report - published on:EP02.09.2004
ClassificationIPC:A61K31/46, A61K31/445, C07D451/04, A61P31/18
[2005/36]
CPC:
C07D451/04 (EP,KR,US); A61K31/46 (KR); A61P31/12 (EP);
A61P31/18 (EP)
Designated contracting statesAT,   BE,   BG,   CH,   CY,   CZ,   DE,   DK,   EE,   ES,   FI,   FR,   GB,   GR,   HU,   IE,   IT,   LI,   LU,   MC,   NL,   PT,   RO,   SE,   SI,   SK,   TR [2005/36]
Extension statesALNot yet paid
LT06.06.2005
LV06.06.2005
MKNot yet paid
TitleGerman:PIPERIDINDERVIATEALS CCR5-ANTAGONISTEN[2005/36]
English:PIPERIDINE DERIVATIVES AS CCR5 ANTAGONISTS[2005/36]
French:ANTAGONISTES DE CCR5 UTILES COMME AGENTS THERAPEUTIQUES[2005/36]
Entry into regional phase06.06.2005National basic fee paid 
06.06.2005Designation fee(s) paid 
06.06.2005Examination fee paid 
Examination procedure09.06.2004Request for preliminary examination filed
International Preliminary Examining Authority: EP
06.06.2005Examination requested  [2005/36]
11.11.2008Despatch of a communication from the examining division (Time limit: M06)
11.05.2009Reply to a communication from the examining division
12.10.2009Despatch of a communication from the examining division (Time limit: M06)
23.04.2010Application deemed to be withdrawn, date of legal effect  [2010/42]
01.06.2010Despatch of communication that the application is deemed to be withdrawn, reason: reply to the communication from the examining division not received in time  [2010/42]
Fees paidRenewal fee
05.12.2005Renewal fee patent year 03
05.12.2006Renewal fee patent year 04
05.12.2007Renewal fee patent year 05
08.12.2008Renewal fee patent year 06
07.12.2009Renewal fee patent year 07
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Cited inInternational search[Y]WO9904794  (MERCK & CO INC [US], et al) [Y] 1-61 * page 103, line 12 - line 17; claims 1,15,18,20 *;
 [Y]WO0038680  (PFIZER LTD [GB], et al) [Y] 1-61 * page 27, line 10; claims 1,2,5-20 *;
 [A]WO02079190  (SMITHKLINE BEECHAM PLC [GB], et al) [A] 1-61 * page 12, line 1 - line 3; claim 1; table 1 *;
 [X]WO9825605  (MERCK & CO INC [US], et al) [X] 1-61 * page 61, line 5 - line 11; claims 1,11 * * page 16 - page 34 *;
 [X]US5340822  (EMONDS-ALT XAVIER [FR], et al) [X] 1-23,25-28,52-54,59,60 * column 1, line 11 - line 24; examples 22-24; claim 1 *;
 [X]BE601228  (JANSSEN PAUL ADRIAAN JAN) [X] 1-23,25-28,54 * page 2, line 23 - line 27; claim 1 * * page 9, line 10 - page 28, line 10 *;
 [X]US2773870  (BILL ELPERN) [X] 1-23,25-28,54 * column 1, line 20 - line 61 * * examples *;
 [X]US3539580  (HERMANS HUBERT KAREL FRANS, et al) [X] 1-23,25-28,54 * column 1, line 13 - line 15; claims 1,5-7 * * table *;
 [X]US3334106  (BIEL JOHN H) [X] 1-23,25-28,54 * the whole document *;
 [X]US2248018  (OTTO EISLEB) [X] 1,25-28,54 * column 1, line 52 - line 55; examples 3,4; claim 6 *;
 [X]WO9825604  (MERCK & CO INC [US], et al) [X] 1,7-12,20,25-61 * page 30, line 26 - line 30 * * page 34, line 1 - line 22 * * page 55 - page 85; claim 1 *;
 [X]JP2002348288
 [X]  - REHSE K ET AL, "Platelet aggregation inhibiting and anticoagulant effects of oligoamines, 1: N-(4-piperidinyl)methanamines", ARCHIV DER PHARMAZIE, VCH VERLAGSGESELLSCHAFT MBH, WEINHEIM, DE, (1986), vol. 319, no. 319, ISSN 0365-6233, pages 505 - 515, XP001085385 [X] 1,25-28,52-54,59,60 * the whole document *

DOI:   http://dx.doi.org/10.1002/ardp.19863190606
 [X]  - STEVENTON ET AL, "4,4-disubstituted Piperidine High-Affinity NK1 Antagonists: Structure-Activity Relationships and in Vivo Activity", JOURNAL OF MEDICINAL CHEMISTRY, AMERICAN CHEMICAL SOCIETY, US, (1998), vol. 41, no. 23, ISSN 0022-2623, pages 4623 - 4622, XP002173109 [X] 1,25-28,54 * the whole document *

DOI:   http://dx.doi.org/10.1021/jm980376b
 [X]  - DATABASE WPI, 0, Derwent World Patents Index, vol. 2003, no. 35, Database accession no. 2003-367209, XP002283279 & JP2002348288 A 20021204 (ONO PHARM CO LTD) [X] 1,7-12,20,25-61 * abstract *
The EPO accepts no responsibility for the accuracy of data originating from other authorities; in particular, it does not guarantee that it is complete, up to date or fit for specific purposes.