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Extract from the Register of European Patents

EP About this file: EP1660503

EP1660503 - NAPHTHALENE CARBOXAMIDES AND THEIR DERIVATIVES USEFUL AS NEW ANTI-ANGIOGENIC AGENTS [Right-click to bookmark this link]
StatusThe application is deemed to be withdrawn
Status updated on  31.07.2009
Database last updated on 02.11.2024
Most recent event   Tooltip31.07.2009Application deemed to be withdrawnpublished on 02.09.2009  [2009/36]
Applicant(s)For all designated states
Pfizer Inc.
235 East 42nd Street
New York, NY 10017 / US
[N/P]
Former [2006/22]For all designated states
PFIZER INC.
235 East 42nd Street
New York, N.Y. 10017 / US
Inventor(s)01 / HE, Mingying, Agouron Pharmaceuticals Inc.
A Pfizer Company, 10777 Science Center Drive
San Diego, CA 92121 / US
02 / KANIA, Robert, Steven, Agouron Pharmaceuticals Inc
A Pfizer Company, 10777 Science Center Drive
San Diego, CA 92121 / US
03 / LOU, Jihong, Agouron Pharmaceuticals Inc.
A Pfizer Company, 10777 Science Center Drive
San Diego, CA 92121 / US
04 / ZHOU, Ru, Agouron Pharmaceuticals Inc.
A Pfizer Company, 10777 Science Center Drive
San Diego, CA 92121 / US
 [2006/22]
Representative(s)Dekker, Henrike Cornelie Christine, et al
Pfizer Limited
European Patent Department
Ramsgate Road
Sandwich
Kent CT13 9NJ / GB
[N/P]
Former [2009/20]Dekker, Henrike Cornelie Christine, et al
Pfizer Limited European Patent Department Ramsgate Road Sandwich
Kent CT13 9NJ / GB
Former [2006/33]Dekker, Henrike Cornelie Christine, et al
Pfizer European Pharma Patent Department 23-25, avenue du Docteur Lannelongue
75668 Paris Cedex 14 / FR
Former [2006/22]Bridle, Andrew Barry, et al
Pfizer Limited European Patent Department, Ramsgate Road
Sandwich, Kent CT13 9NJ / GB
Application number, filing date04744300.716.08.2004
[2006/22]
WO2004IB02685
Priority number, dateUS20030499261P29.08.2003         Original published format: US 499261 P
[2006/22]
Filing languageEN
Procedural languageEN
PublicationType: A1 Application with search report
No.:WO2005021553
Date:10.03.2005
Language:EN
[2005/10]
Type: A1 Application with search report 
No.:EP1660503
Date:31.05.2006
Language:EN
The application published by WIPO in one of the EPO official languages on 10.03.2005 takes the place of the publication of the European patent application.
[2006/22]
Search report(s)International search report - published on:EP10.03.2005
ClassificationIPC:C07D495/04, C07D239/42, C07D239/34, C07D215/20, C07D213/68, A61K31/4365, A61K31/505, A61K31/47, A61P35/00
[2006/22]
CPC:
C07D239/34 (EP,US); A61P35/00 (EP); A61P43/00 (EP);
A61P9/00 (EP); C07D213/68 (EP,US); C07D215/20 (EP,US);
C07D239/42 (EP,US); C07D495/04 (EP,US) (-)
Designated contracting statesAT,   BE,   BG,   CH,   CY,   CZ,   DE,   DK,   EE,   ES,   FI,   FR,   GB,   GR,   HU,   IE,   IT,   LI,   LU,   MC,   NL,   PL,   PT,   RO,   SE,   SI,   SK,   TR [2006/22]
Extension statesALNot yet paid
HRNot yet paid
LTNot yet paid
LVNot yet paid
MKNot yet paid
TitleGerman:NAPHTHALINCARBOXAMIDE UND DERIVATE ALS NEUE ANTI-ANGIOGENE MITTEL[2006/22]
English:NAPHTHALENE CARBOXAMIDES AND THEIR DERIVATIVES USEFUL AS NEW ANTI-ANGIOGENIC AGENTS[2006/22]
French:CARBOXAMIDES DE NAPHTALENE ET LEURS DERIVES UTILES COMME NOUVEAUX AGENTS ANTI-ANGIOGENIQUES[2006/22]
Entry into regional phase29.03.2006National basic fee paid 
29.03.2006Designation fee(s) paid 
29.03.2006Examination fee paid 
Examination procedure15.09.2004Request for preliminary examination filed
International Preliminary Examining Authority: EP
29.03.2006Examination requested  [2006/22]
19.06.2006Despatch of a communication from the examining division (Time limit: M06)
10.04.2007Reply to a communication from the examining division
03.03.2009Application deemed to be withdrawn, date of legal effect  [2009/36]
07.04.2009Despatch of communication that the application is deemed to be withdrawn, reason: renewal fee not paid in time  [2009/36]
Request for further processing for:10.04.2007Request for further processing filed
10.04.2007Full payment received (date of receipt of payment)
Request granted
27.04.2007Decision despatched
Fees paidRenewal fee
07.08.2006Renewal fee patent year 03
03.08.2007Renewal fee patent year 04
Penalty fee
Additional fee for renewal fee
31.08.200805   M06   Not yet paid
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Cited inInternational search[X]DE482438  (IG FARBENINDUSTRIE AG) [X] 1 * example 3 *;
 [X]DE573723  (IG FARBENINDUSTRIE AG) [X] 1 * tables pages 2, 3 *;
 [X]US1935930  (GENERAL ANILINE WORKS INC.) [X] 1 * the whole document *;
 [X]US2003055110  (VOEGEL JOHANNES [FR], et al) [X] 1 * compound 40 *;
 [XA]WO9946268  (NOVO NORDISK AS [DK], et al) [X] 1,7-13 * page 17, line 16 - page 18, line 25 * * Formula I * * page 25, lines 20,21 * * page 29, lines 14-19 * [A] 2-6,14,15;
 [A]US4814454  (MISRA RAJ N [US]) [A] 1,7-13 * column 1, lines 1-50; examples 8,32 *
 [X]  - OIKAWA, Y., YONEMITSU, O., "Cyclization of beta-Ketosulfoxide -III. Synthesis of Naphthalene and Phenanthrene Derivatives", TETRAHEDRON, GB, (1974), vol. 30, pages 2653 - 2660, XP002303233 [X] 1 * page 2659, compound 19 *

DOI:   http://dx.doi.org/10.1016/S0040-4020(01)97425-3
 [X]  - CHATTERJEE, A., RAYCHAUDHURI, S.R., CHATTERJEE, S.K., "Eficient Synthesies of Some 1-Naphthylalkyl Ketones and Studies on their Autooxidation in Basic Medium", TETRAHEDRON, GB, (1981), vol. 37, no. 21, pages 3653 - 3660, XP002303234 [X] 1 * compound i *

DOI:   http://dx.doi.org/10.1016/S0040-4020(01)98894-5
 [X]  - CONNOR, D.T., WIACZESLAW, A. CETENKO, MULLICAN, M.D., SORENSON, R.J., UNANGST,P.C. ET AL, "Novel Benzothiophene-, Benzofuran-, and Naphthalenecarboxamidotetrazoles as Potential Antiallergy Agents", J. MED. CHEM., US, (1992), vol. 35, pages 958 - 965, XP002303235 [X] 1 * table II, compound 13v *

DOI:   http://dx.doi.org/10.1021/jm00083a023
 [X]  - SATOSHI FUJITA, MASAYOSHI MOMIYAMA, YASUMITSU KONDO, "Fluorescent Substrates for Potential Use in Enzyme-Linked Immunosorbent Assay of Membrane-Bound Nucleic Acids", ANAL. CHEM., US, (1994), vol. 66, pages 1347 - 1353, XP002303236 [X] 1 * compounds 49,50 *

DOI:   http://dx.doi.org/10.1021/ac00080a022
 [X]  - SHINJI KAWATA, SHUKUKO ASHIZAWA, MASAHIRO HIRAMA, "Synthetic Study of Kedarcidin Chromophore: Revised Structure", J. AM. CHEM. SOC., US, (1997), vol. 119, pages 12012 - 12013, XP002303237 [X] 1 * compound 3 *

DOI:   http://dx.doi.org/10.1021/ja973231n
 [X]  - MARSILJE, T.A., MILKIEWICZ, K.L., HANGAUER, D.G., "The Design, Synthesis and Activity of Non-ATP Competitive Inhibitors of pp60c-src Tyrosine Kinase. Part 1: Hydroxynaphthalene Derivatives", BIOORGANIC AND MEDICINAL CHEMISTRY LETTERS, (2000), vol. 10, pages 477 - 481, XP002303238 [X] 1,7,10 * compounds 2e-2h,2m,2n,2q-2s *

DOI:   http://dx.doi.org/10.1016/S0960-894X(00)00039-1
The EPO accepts no responsibility for the accuracy of data originating from other authorities; in particular, it does not guarantee that it is complete, up to date or fit for specific purposes.