EP1620422 - PHENYL SUBSTITUTED CARBOXYLIC ACIDS AS INHIBITORS OF PROTEIN TYROSINE PHOSPHATASE-1B [Right-click to bookmark this link] | Status | The application is deemed to be withdrawn Status updated on 02.04.2010 Database last updated on 18.11.2024 | Most recent event Tooltip | 02.04.2010 | Application deemed to be withdrawn | published on 05.05.2010 [2010/18] | Applicant(s) | For all designated states The Institutes for Pharmaceutical Discovery, LLC 23 Business Park Drive Branford, CT 06405 / US | [2006/05] | Inventor(s) | 01 /
WHITEHOUSE, Darren 40 Fishing Brook Road Westbrook, CT 06498 / US | 02 /
HU, Shaojing 900 Mix Avenue, Unit 121 Hamden, CT 06514 / US | 03 /
FANG, Haiquan 304 County Road Madison, CT 06443 / US | 04 /
VAN ZANDT, Michael 91 Golden Hill Drive Guilford, CT 06437 / US | [2006/05] | Representative(s) | Adam, Holger Kraus & Weisert Patentanwälte PartGmbB Thomas-Wimmer-Ring 15 80539 München / DE | [N/P] |
Former [2006/05] | Adam, Holger Kraus & Weisert, Patent- und Rechtsanwälte, Thomas-Wimmer-Ring 15 80539 München / DE | Application number, filing date | 04751193.6 | 30.04.2004 | [2006/05] | WO2004US13701 | Priority number, date | US20030466868P | 30.04.2003 Original published format: US 466868 P | [2006/05] | Filing language | EN | Procedural language | EN | Publication | Type: | A2 Application without search report | No.: | WO2004099170 | Date: | 18.11.2004 | Language: | EN | [2004/47] | Type: | A2 Application without search report | No.: | EP1620422 | Date: | 01.02.2006 | Language: | EN | The application published by WIPO in one of the EPO official languages on 18.11.2004 takes the place of the publication of the European patent application. | [2006/05] | Search report(s) | International search report - published on: | EP | 15.09.2005 | Classification | IPC: | C07D307/91 | [2006/05] | CPC: |
C07D307/79 (EP,KR,US);
A61P25/00 (EP);
A61P3/00 (EP);
A61P3/04 (EP);
A61P3/10 (EP);
A61P35/00 (EP);
A61P37/02 (EP);
A61P43/00 (EP);
A61P9/00 (EP);
C07C311/19 (EP,US);
C07C311/29 (EP,US);
C07D209/08 (EP,US);
C07D307/80 (EP,KR,US);
C07D307/81 (EP,US);
C07D307/91 (EP,KR,US);
C07D401/04 (EP,US)
(-)
| Designated contracting states | AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HU, IE, IT, LI, LU, MC, NL, PL, PT, RO, SE, SI, SK, TR [2006/05] | Extension states | AL | 02.11.2005 | HR | 02.11.2005 | LT | 02.11.2005 | LV | 02.11.2005 | MK | 02.11.2005 | Title | German: | PHENYL SUBSTITUIERTE CARBONSÄUREN ALS HEMMER DER PROTEIN-TYROSINPHOSPHATASE-1B | [2006/05] | English: | PHENYL SUBSTITUTED CARBOXYLIC ACIDS AS INHIBITORS OF PROTEIN TYROSINE PHOSPHATASE-1B | [2006/05] | French: | ACIDES CARBOXYLIQUES SUBSTITUES PAR PHENYLE COMME INHIBITEURS DE PROTEINE TYROSINE-PHOSPHATASE-1B | [2006/05] | Entry into regional phase | 02.11.2005 | National basic fee paid | 02.11.2005 | Designation fee(s) paid | 02.11.2005 | Examination fee paid | Examination procedure | 02.11.2005 | Examination requested [2006/05] | 16.01.2008 | Despatch of a communication from the examining division (Time limit: M06) | 18.07.2008 | Reply to a communication from the examining division | 03.11.2009 | Application deemed to be withdrawn, date of legal effect [2010/18] | 07.12.2009 | Despatch of communication that the application is deemed to be withdrawn, reason: renewal fee not paid in time [2010/18] | Fees paid | Renewal fee | 26.04.2006 | Renewal fee patent year 03 | 27.04.2007 | Renewal fee patent year 04 | 25.04.2008 | Renewal fee patent year 05 | Penalty fee | Additional fee for renewal fee | 30.04.2009 | 06   M06   Not yet paid |
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Responsibility for the accuracy, completeness or quality of the data displayed under the link provided lies entirely with the Unified Patent Court. | Cited in | International search | [X]JPS59141540 (CHISSO CORP) [X] 1-4,6-8,10-17,41-45 * Compounds 3 and 4 and the precursors thereof *; | [X]EP0561639 (LILLY CO ELI [US]) [X] 1-4,6-8,10-17,41-45 * page 26; table 16 * * page 28; table 17 *; | [X]EP0744407 (LILLY CO ELI [US]) [X] 1-4,6-8,10-17,41-45 * Page 12, Preparation 3; Page 16, Preparation 12 *; | [X]WO0050375 (CLARIANT GMBH [DE], et al) [X] 1-4,6-8,10-17,41-45 * examples 5,13; claim 1 *; | [PX]JP2003238551 (FUJI PHOTO FILM CO LTD) [PX] 1-57* the whole document *; | [X] - MALAMAS M S ET AL, "Novel Benzofuran and Benzothiophene Biphenyls as Inhibitors of Protein Tyrosine Phosphatase 1B with Antihyperglycemic Properties", JOURNAL OF MEDICINAL CHEMISTRY, AMERICAN CHEMICAL SOCIETY. WASHINGTON, US, (2000), vol. 43, ISSN 0022-2623, pages 1293 - 1310, XP002216395 [X] 1-57 * the whole document * DOI: http://dx.doi.org/10.1021/jm990560c | [X] - SADASHIVA, B. K. ET AL, "A convenient method for the preparation of 4-n-alkyl-4''-cyano-p-terphenyl", CAPLUS, CHEMICAL ABSTRACTS SERVICE, COLUMBUS, OHIO, US, Database accession no. 1977:502050, URL: STN, XP002301745 [X] 1-4,6-8,10-17,41-45 * compounds 63809-04-1, 63809-05-2 * | [X] - DEBONO M. ET AL., "Semisynthetic Chemical Modification of the Antifungal Lipopeptide Echinocandin B (ECB): Structure-Activity Studies of the Lipophilic and Geometric Parameters of Polyarylated Acyl Analogs of ECB", JOURNAL OF MEDICINAL CHEMISTRY, (1995), vol. 38, no. 17, pages 3271 - 3281, XP000608473 [X] 1-4,6-8,10-17,41-45 * page 3279; compounds 14AA,14BB * DOI: http://dx.doi.org/10.1021/jm00017a012 | [X] - HIMMEL, HANS-JOERG ET AL, "Fabrication of a Carboxyl-Terminated Organic Surface with Self-Assembly of Functionalized Terphenylthiols: The Importance of Hydrogen Bond Formation", JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, (1998), vol. 120, no. 46, pages 12069 - 12074, XP002301744 [X] 1-4,6-8,10-17,41-45 * Page 12070, two intermediates in the preparation of 4'Carboxyterphenyl-4-methanethiol * DOI: http://dx.doi.org/10.1021/ja981872s | [X] - CONN M. M. ET AL., "Template Effects in New Self-Replicating Molecules", ANGEW. CHEM. INT. ED. ENGL., (1994), vol. 33, pages 1577 - 1579, XP002301796 [X] 1,7 * compounds 3,5 * DOI: http://dx.doi.org/10.1002/anie.199415771 |