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Extract from the Register of European Patents

EP About this file: EP1701932

EP1701932 - TOLTERODINE, COMPOSITIONS AND USES THEREOF, AND PREPARATION OF THE SAME [Right-click to bookmark this link]
StatusNo opposition filed within time limit
Status updated on  24.05.2013
Database last updated on 02.11.2024
Most recent event   Tooltip18.07.2014Lapse of the patent in a contracting state
New state(s): HU		published on 20.08.2014  [2014/34]
Applicant(s)For all designated states
Cipla Ltd.
289, Bellasis Road, Mumbai Central Mumbai 400 008
Maharashtra / IN
[2012/29]
Former [2006/38]For all designated states
Cipla Ltd.
289, Belasis Road, Mumbai Central Mumbai 400 008
Maharashtra / IN
Inventor(s)01 / KANKAN, Rajendra, Narayanrao
A-3/5, NBD Society, NSS Road, Ghatkopar(West)
Mumbai 400 084, Maharashtra / IN
02 / RAO, Dharmaraj, Ramachandra
4/403 Garden Enclave, Pokhran Road 2, Thane West
Mumbai 400 601, Maharashtra / IN
 [2006/38]
Representative(s)Curtis, Philip Anthony, et al
A.A. Thornton & Co.
10 Old Bailey
London EC4M 7NG / GB
[N/P]
Former [2012/29]Curtis, Philip Anthony, et al
A.A. Thornton & Co.
235 High Holborn
London
WC1V 7LE / GB
Former [2006/38]Curtis, Philip Anthony, et al
A.A. Thornton & Co., 235 High Holborn
London WC1V 7LE / GB
Application number, filing date04820622.123.12.2004
[2006/38]
WO2004GB05420
Priority number, dateGB2003003005624.12.2003         Original published format: GB 0330056
GB2004002330020.10.2004         Original published format: GB 0423300
[2006/38]
Filing languageEN
Procedural languageEN
PublicationType: A1 Application with search report
No.:WO2005061432
Date:07.07.2005
Language:EN
[2005/27]
Type: A1 Application with search report 
No.:EP1701932
Date:20.09.2006
Language:EN
The application published by WIPO in one of the EPO official languages on 07.07.2005 takes the place of the publication of the European patent application.
[2006/38]
Type: B1 Patent specification 
No.:EP1701932
Date:18.07.2012
Language:EN
[2012/29]
Search report(s)International search report - published on:EP07.07.2005
ClassificationIPC:C07C215/54, C07C213/00, C07C43/23, C07C39/12, A61K31/137
[2006/38]
CPC:
C07C213/00 (EP,US); C07C39/12 (KR); A61P13/02 (EP);
A61P25/02 (EP); C07C215/54 (EP,KR,US); C07C43/23 (KR)
Designated contracting statesAT,   BE,   BG,   CH,   CY,   CZ,   DE,   DK,   EE,   ES,   FI,   FR,   GB,   GR,   HU,   IE,   IS,   IT,   LI,   LT,   LU,   MC,   NL,   PL,   PT,   RO,   SE,   SI,   SK,   TR [2006/38]
TitleGerman:TOLTERODIN, ZUSAMMENSETZUNGEN UND ANWENDUNGEN DAVON, UND HERSTELLUNG DAVON[2006/38]
English:TOLTERODINE, COMPOSITIONS AND USES THEREOF, AND PREPARATION OF THE SAME[2006/38]
French:TOLTERODINE, COMPOSITIONS ET LEURS UTILISATIONS, ET PREPARATIONS DESDITES COMPOSITIONS[2006/38]
Entry into regional phase17.07.2006National basic fee paid 
17.07.2006Designation fee(s) paid 
17.07.2006Examination fee paid 
Examination procedure24.10.2005Request for preliminary examination filed
International Preliminary Examining Authority: EP
17.07.2006Examination requested  [2006/38]
01.08.2006Amendment by applicant (claims and/or description)
06.03.2009Despatch of a communication from the examining division (Time limit: M04)
08.07.2009Reply to a communication from the examining division
15.03.2012Communication of intention to grant the patent
01.06.2012Fee for grant paid
01.06.2012Fee for publishing/printing paid
Divisional application(s)The date of the Examining Division's first communication in respect of the earliest application for which a communication has been issued is  06.03.2009
Opposition(s)19.04.2013No opposition filed within time limit [2013/26]
Fees paidRenewal fee
13.12.2006Renewal fee patent year 03
12.12.2007Renewal fee patent year 04
15.12.2008Renewal fee patent year 05
11.12.2009Renewal fee patent year 06
15.12.2010Renewal fee patent year 07
12.12.2011Renewal fee patent year 08
Opt-out from the exclusive  Tooltip
competence of the Unified
Patent Court		 See the Register of the Unified Patent Court for opt-out data
Responsibility for the accuracy, completeness or quality of the data displayed under the link provided lies entirely with the Unified Patent Court.
Lapses during opposition  TooltipHU23.12.2004
AT18.07.2012
BE18.07.2012
CY18.07.2012
CZ18.07.2012
DK18.07.2012
EE18.07.2012
FI18.07.2012
IT18.07.2012
LT18.07.2012
NL18.07.2012
PL18.07.2012
RO18.07.2012
SE18.07.2012
SI18.07.2012
SK18.07.2012
BG18.10.2012
GR19.10.2012
ES29.10.2012
IS18.11.2012
PT19.11.2012
IE23.12.2012
LU23.12.2012
CH31.12.2012
LI31.12.2012
MC31.12.2012
[2014/34]
Former [2014/27]AT18.07.2012
BE18.07.2012
CY18.07.2012
CZ18.07.2012
DK18.07.2012
EE18.07.2012
FI18.07.2012
IT18.07.2012
LT18.07.2012
NL18.07.2012
PL18.07.2012
RO18.07.2012
SE18.07.2012
SI18.07.2012
SK18.07.2012
BG18.10.2012
GR19.10.2012
ES29.10.2012
IS18.11.2012
PT19.11.2012
IE23.12.2012
LU23.12.2012
CH31.12.2012
LI31.12.2012
MC31.12.2012
Former [2013/48]AT18.07.2012
BE18.07.2012
CY18.07.2012
CZ18.07.2012
DK18.07.2012
EE18.07.2012
FI18.07.2012
IT18.07.2012
LT18.07.2012
NL18.07.2012
PL18.07.2012
RO18.07.2012
SE18.07.2012
SI18.07.2012
SK18.07.2012
BG18.10.2012
GR19.10.2012
ES29.10.2012
IS18.11.2012
PT19.11.2012
IE23.12.2012
CH31.12.2012
LI31.12.2012
MC31.12.2012
Former [2013/47]AT18.07.2012
BE18.07.2012
CY18.07.2012
CZ18.07.2012
DK18.07.2012
EE18.07.2012
FI18.07.2012
IT18.07.2012
LT18.07.2012
NL18.07.2012
PL18.07.2012
RO18.07.2012
SE18.07.2012
SI18.07.2012
SK18.07.2012
BG18.10.2012
GR19.10.2012
ES29.10.2012
IS18.11.2012
PT19.11.2012
IE23.12.2012
MC31.12.2012
Former [2013/34]AT18.07.2012
BE18.07.2012
CY18.07.2012
CZ18.07.2012
DK18.07.2012
EE18.07.2012
FI18.07.2012
IT18.07.2012
LT18.07.2012
NL18.07.2012
PL18.07.2012
RO18.07.2012
SE18.07.2012
SI18.07.2012
SK18.07.2012
BG18.10.2012
GR19.10.2012
ES29.10.2012
IS18.11.2012
PT19.11.2012
MC31.12.2012
Former [2013/33]AT18.07.2012
BE18.07.2012
CY18.07.2012
CZ18.07.2012
DK18.07.2012
EE18.07.2012
FI18.07.2012
IT18.07.2012
LT18.07.2012
NL18.07.2012
PL18.07.2012
RO18.07.2012
SE18.07.2012
SI18.07.2012
SK18.07.2012
GR19.10.2012
ES29.10.2012
IS18.11.2012
PT19.11.2012
MC31.12.2012
Former [2013/23]AT18.07.2012
BE18.07.2012
CY18.07.2012
CZ18.07.2012
DK18.07.2012
EE18.07.2012
FI18.07.2012
IT18.07.2012
LT18.07.2012
NL18.07.2012
PL18.07.2012
RO18.07.2012
SE18.07.2012
SI18.07.2012
SK18.07.2012
GR19.10.2012
ES29.10.2012
IS18.11.2012
PT19.11.2012
Former [2013/22]AT18.07.2012
BE18.07.2012
CY18.07.2012
CZ18.07.2012
DK18.07.2012
EE18.07.2012
FI18.07.2012
LT18.07.2012
NL18.07.2012
PL18.07.2012
SE18.07.2012
SI18.07.2012
GR19.10.2012
ES29.10.2012
IS18.11.2012
PT19.11.2012
Former [2013/21]AT18.07.2012
BE18.07.2012
CY18.07.2012
DK18.07.2012
FI18.07.2012
LT18.07.2012
NL18.07.2012
PL18.07.2012
SE18.07.2012
SI18.07.2012
GR19.10.2012
IS18.11.2012
PT19.11.2012
Former [2013/15]AT18.07.2012
BE18.07.2012
CY18.07.2012
FI18.07.2012
LT18.07.2012
NL18.07.2012
PL18.07.2012
SE18.07.2012
SI18.07.2012
GR19.10.2012
IS18.11.2012
PT19.11.2012
Former [2013/13]AT18.07.2012
BE18.07.2012
CY18.07.2012
FI18.07.2012
LT18.07.2012
PL18.07.2012
SE18.07.2012
SI18.07.2012
GR19.10.2012
IS18.11.2012
PT19.11.2012
Former [2013/12]AT18.07.2012
BE18.07.2012
CY18.07.2012
FI18.07.2012
LT18.07.2012
PL18.07.2012
SE18.07.2012
SI18.07.2012
GR19.10.2012
IS18.11.2012
Former [2013/11]AT18.07.2012
BE18.07.2012
CY18.07.2012
FI18.07.2012
LT18.07.2012
PL18.07.2012
SI18.07.2012
GR19.10.2012
IS18.11.2012
Former [2013/10]AT18.07.2012
BE18.07.2012
CY18.07.2012
FI18.07.2012
LT18.07.2012
IS18.11.2012
Former [2013/09]AT18.07.2012
BE18.07.2012
FI18.07.2012
LT18.07.2012
Former [2013/08]AT18.07.2012
BE18.07.2012
LT18.07.2012
Former [2013/07]AT18.07.2012
Cited inInternational search[XDY]US5382600  (JOENSSON NILS A [SE], et al) [XD] 1-33 * column 2, line 35 * * column 3, line 20 - line 21 * * column 3, line 58 - line 60 * * column 4, line 65 - line 66 * * column 5, line 1 * * column 5, line 18 - line 21 * * column 5, line 30 - line 46 * * column 8, line 4 - line 6 * * examples 3a,4b,5d,9g,22; compounds 4,4A,4B * [Y] 1-3,5,13,15-24,26,27,29-33;
 [X]US5922914  (GAGE JAMES R [US], et al) [X] 1-33 * column 4, line 57; examples 3,4 *;
 [X]WO03035599  (UPJOHN CO [US], et al) [X] 1-33 * example 1 *;
 [X]US2003199582  (HAWLEY MICHAEL [US], et al) [X] 1-33 * example 1 *;
 [Y]  - KEESE R ET AL, "Crystallisation", FUNDAMENTALS OF PREPARATIVE ORGANIC CHEMISTRY, (1982), pages 18 - 20, XP002310738 [Y] 1-3,13,24,29-33 * the whole document *
 [Y]  - T. W. GREENE & P. G. M. WUTS, Protective Groups in Organic Synthesis, JOHN WILEY & SONS, (1991), XP002327043 [Y] 5 * page 145 - page 149 *
 [Y]  - ANDERSSON P G ET AL, "ASYMMETRIC TOTAL SYNTHESIS OF (+)-TOLTERODINE, A NEW MUSCARINIC RECEPTOR ANTAGONIST, VIA COPPER-ASSISTED ASYMMETRIC CONJUGATE ADDITION OF ARYL GRIGNARD REAGENTS TO 3-PHENYL-PROP-2-ENOYL-OXAZOLIDINONES", JOURNAL OF ORGANIC CHEMISTRY, AMERICAN CHEMICAL SOCIETY. EASTON, US, (1998), vol. 63, no. 22, ISSN 0022-3263, pages 8067 - 8070, XP001037685 [Y] 15-23,26,27 * compound 11 *

DOI:   http://dx.doi.org/10.1021/jo981259r
The EPO accepts no responsibility for the accuracy of data originating from other authorities; in particular, it does not guarantee that it is complete, up to date or fit for specific purposes.