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Extract from the Register of European Patents

EP About this file: EP1854806

EP1854806 - Thioglycosides as pharmaceutically active agents [Right-click to bookmark this link]
StatusThe application is deemed to be withdrawn
Status updated on  24.10.2008
Database last updated on 20.12.2024
Most recent event   Tooltip24.10.2008Application deemed to be withdrawnpublished on 26.11.2008  [2008/48]
Applicant(s)For all designated states
Max-Planck-Gesellschaft zur Förderung der Wissenschaften e.V.
Hofgartenstrasse 8
80539 München / DE
[N/P]
Former [2007/46]For all designated states
MPG Max-Planck-Gesellschaft zur Förderung der Wissenschaften e.V.
Hofgartenstrasse 8
80539 München / DE
Inventor(s)01 / Castaneda, Francisco
Potthöferei 1
44388 Dortmund / DE
02 / Kinne, Rolf K-H.
Otto-Hahn-Strasse 11
44227 Dortmund / DE
03 / Boland, Wilhelm
Care-Orff-Str. 21
07743 Jena / DE
04 / Burse, Antje
Helmboldstrasse 3
07749 Jena / DE
 [2007/46]
Representative(s)Arth, Hans-Lothar, et al
ABK Patent Attorneys
Jasminweg 9
14052 Berlin / DE
[N/P]
Former [2008/23]Arth, Hans-Lothar, et al
ABK Patent Attorneys Jasminweg 9
14052 Berlin / DE
Former [2007/46]Arth, Hans-Lothar
Arth, Bucher & Kollegen, Am Klopferspitz 19 (IZB)
82152 Martinsried / DE
Application number, filing date06009058.602.05.2006
[2007/46]
Filing languageEN
Procedural languageEN
PublicationType: A1 Application with search report 
No.:EP1854806
Date:14.11.2007
Language:EN
[2007/46]
Search report(s)(Supplementary) European search report - dispatched on:EP02.08.2006
ClassificationIPC:C07H15/203
[2007/46]
CPC:
C07H15/203 (EP); A61P3/10 (EP); C07H15/14 (EP)
Designated contracting states(deleted) [2008/30]
Former [2007/46]AT,  BE,  BG,  CH,  CY,  CZ,  DE,  DK,  EE,  ES,  FI,  FR,  GB,  GR,  HU,  IE,  IS,  IT,  LI,  LT,  LU,  LV,  MC,  NL,  PL,  PT,  RO,  SE,  SI,  SK,  TR 
TitleGerman:Thioglycoside als pharmaceutisch aktive Verbindungen[2007/46]
English:Thioglycosides as pharmaceutically active agents[2007/46]
French:Thioglycosides en tant que composés pharmaceutiques[2007/46]
Examination procedure15.05.2008Application deemed to be withdrawn, date of legal effect  [2008/48]
30.06.2008Despatch of communication that the application is deemed to be withdrawn, reason: examination fee not paid in time  [2008/48]
Fees paidPenalty fee
Additional fee for renewal fee
31.05.200803   M06   Not yet paid
Opt-out from the exclusive  Tooltip
competence of the Unified
Patent Court		 See the Register of the Unified Patent Court for opt-out data
Responsibility for the accuracy, completeness or quality of the data displayed under the link provided lies entirely with the Unified Patent Court.
Documents cited:Search[Y]EP1268502  (SQUIBB BRISTOL MYERS CO [US]) [Y] 1-13 * claim 1 *;
 [Y]EP1528066  (TAISHO PHARMA CO LTD [JP]) [Y] 1-13 * claim 1 *;
 [X]WO2005118609  (CALIFORNIA INST OF TECHN [US], et al) [X] 1,2 * page 22; compound 1 *;
 [X]  - NOBUKO IINO, KAZUDO YOSHIDA, "An Improved Method for the Synthesis of p-Aminophenyl 1-Thio-beta-D-glycosides", CARBOHYDRATE RESEARCH, (1976), vol. 51, pages 223 - 228, XP002388261 [X] 1-3 * the whole document *
 [X]  - CHEN M-Y ET AL, "Chemoselective deprotection of acid labile primary hydroxyl protecting groups under CBr4-photoirradiation conditions", TETRAHEDRON, ELSEVIER SCIENCE PUBLISHERS, AMSTERDAM, NL, (20041206), vol. 60, no. 50, ISSN 0040-4020, pages 11465 - 11475, XP004628607 [X] 1-3 * compounds 37,47 *

DOI:   http://dx.doi.org/10.1016/j.tet.2004.09.095
 [X]  - A. LIONEL CLINGMAN, NELSON K. RICHTMYER, "Aryl Thioglycopyranosides, Aryl Glycopyranosyl Sulfones, and the novel Oxidation-Acetylation of Aryl 1-Thio-beta-D-glucopyranosides to 6-O-Acetyl-beta-D-glucopyranosyl Aryl Sulfones", JOURNAL OF ORGANIC CHEMISTRY, (1964), vol. 29, pages 1782 - 1787, XP002388262 [X] 1-3 * compounds IV, X, XVII, XX *

DOI:   http://dx.doi.org/10.1021/jo01030a028
 [X]  - EDNA M. MONTGOMERY ET AL., "Attempts to find new antimalarials. VIII. Phenyl beta-D-glucothiosides, Diphenyl Disulfides, Phenyl Thiocyanates, and related compounds", JOURNAL OF ORGANIC CHEMISTRY, (1946), vol. 11, pages 301 - 305, XP002388263 [X] 1,2 * the whole document *

DOI:   http://dx.doi.org/10.1021/jo01173a015
 [X]  - M. H. BENN ET AL., "Cytotoxic Compounds. Part I. p-(N,N-Di-2'-chloroethyl- and p-(NN-Di-2'-bromoethyl-amino)thiophenol", JOURNAL OF THE CHEMICAL SOCIETY, (1958), pages 2800 - 2810, XP009068829 [X] 1,2 * compound XII *

DOI:   http://dx.doi.org/10.1039/jr9580002800
 [X]  - A. M. CREIGHTON ET AL., "Cytotoxic Compounds. Part III. Some Derivatives of p-(NN-Di2-chloroethyl- and of p-(NN-Di-2-bromoethyl-amino)thiophenol", JOURNAL OF THE CHEMICAL SOCIETY, (1961), pages 2375 - 2381, XP009068827 [X] 1,2 * compound XI *

DOI:   http://dx.doi.org/10.1039/jr9610002375
 [X]  - ANTONIIO VARGAS-BERENGUEL ET AL., "Synthesis of Glycosyltyrosine Building Blocks for Solid-Phase Glycopeptide Assembly: Use of Aryl tert-Butyl Ethers as Glycosyl Acceptors in Aromatic Glycosylation", JOURNAL OF THE CHEMICAL SOCIETY PERKIN TRANSACTIONS I, (1994), no. 22, pages 3287 - 3294, XP009068831 [X] 1,2 * compound 13 *

DOI:   http://dx.doi.org/10.1039/p19940003287
 [X]  - M. YDE, C. K. DE BRUYNE, "Synthesis of para-substituted phenyl 1-thio-beta-D-galactopyranosides", CARBOHYDRATE RESEARCH, (1973), vol. 26, pages 227 - 229, XP002388264 [X] 1,3 * table II *
 [X]  - RAMESH H. SHAH, OM P. BAHL, "Glycosidases. Ligands for Affinity Chromatography: I. Synthesis of 1,2-trans p-Aminophenyl 1-Thio-D-glycopyranosides", CARBOHYDRATE RESEARCH, (1974), vol. 32, pages 15 - 23, XP002388265 [X] 1,3 * compounds 7,8 *
 [X]  - PHILIPPE L. DURETTE, TSUNG Y. SHEN, "Insulin-like, and Insulin-antagonistic, Carbohydrate Derivatives. The Synthesis of Aryl and Aralkyl D-Mannopyranosides and 1-Thio-D-Mannopyranosides", CARBOHYDRATE RESEARCH, (1980), vol. 81, pages 261 - 274, XP002388266 [X] 1 * compound 10 *

DOI:   http://dx.doi.org/10.1016/S0008-6215(00)85657-8
 [Y]  - TAKASHI MIZUMA ET AL., "Transport and Recognition of Aminopeptidase-Resistant Cellobiose-Coupled Tyrosylglycylglycine by Intestinal Na+/Glucose Cotransporter (SGLT1): Recognition of Sugar Conjugates by SGLT1 is much less restricted than Transport", BIOLOGICAL AND PHARMACEUTICAL BULLETIN, (1999), vol. 22, no. 8, pages 876 - 879, XP001246888 [Y] 1-13 * the whole document *
 [Y]  - ANTHONY L HANDLON, "Sodium glucose co-transporter 2 (SGLT2) inhibitors as potential antidiabetic agents", EXPERT OPINION ON THERAPEUTIC PATENTS, (2005), vol. 15, no. 11, pages 1531 - 1540, XP002388315 [Y] 1-13 * the whole document *

DOI:   http://dx.doi.org/10.1517/13543776.15.11.1531
 [X]  - T. V. POCHECHUEVA ET AL., "Uncharged P-selectin blockers", GLYCOCONJUGATE JOURNAL, (2004), vol. 20, pages 91 - 97, XP009069091 [X] 1,4,13 * table 2 *

DOI:   http://dx.doi.org/10.1023/B:GLYC.0000018583.63140.91
The EPO accepts no responsibility for the accuracy of data originating from other authorities; in particular, it does not guarantee that it is complete, up to date or fit for specific purposes.