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Extract from the Register of European Patents

EP About this file: EP1917252

EP1917252 - PYRAZINE DERIVATIVES AND USE AS PI3K INHIBITORS [Right-click to bookmark this link]
StatusNo opposition filed within time limit
Status updated on  07.11.2014
Database last updated on 24.08.2024
Most recent event   Tooltip15.07.2016Lapse of the patent in a contracting state
New state(s): TR		published on 17.08.2016  [2016/33]
Applicant(s)For all designated states
Merck Serono SA
Centre Industriel
1267 Coinsins, Vaud / CH
[2009/25]
Former [2008/19]For all designated states
LABORATOIRES SERONO S.A.
Centre Industriel
1267 Coinsins / CH
Inventor(s)01 / GAILLARD, Pascale
Domaine de la Prasle
243, route du Fer à Cheval
Bat C2
F-74160 Collonges Sous Salève / FR
02 / QUATTROPANI, Anna
2, route de Chene
CH-1207 Geneva / CH
03 / POMEL, Vincent
228, chemin du Bois des Presses
F-74570 Groisy / FR
04 / RUECKLE, Thomas
rue Daubin 4
CH-1203 Geneva / CH
05 / KLICIC, Jasna
19, rue des Délices
CH-1203 Geneva / CH
06 / CHURCH, Dennis
Chemin des Vignes 4
CH-1291 Commugny / CH
 [2014/01]
Former [2008/19]01 / GAILLARD, Pascale
Domaine de la Prasle 243, route du Fer à Cheval Bat C2
F-74160 Collonges Sous Salève / FR
02 / QUATTROPANI, Anna
2, route de Chene
CH-1207 Geneva / CH
03 / POMEL, Vincent
228, chemin du Bois des Presses
F-74570 Groisy / FR
04 / RUECKLE, Thomas
rue Daubin 4
CH-1203 Geneva / CH
05 / KLICIC, Jasna
19, rue des Délices
CH-1203 Geneva / CH
06 / CHURCH, Dennis
Chemin des Vignes 4
CH-1291 Commugny / CH
Representative(s)Merck Serono S.A. Intellectual Property
Zone Industrielle de l'Ouriettaz
1170 Aubonne / CH
[N/P]
Former [2014/01]Merck Serono S.A. Intellectual Property
Centre Industriel
1267 Coinsins / CH
Former [2008/19]Merck Serono International S.A. Intellectual Property
Intellectual Property Department 9, chemin des Mines
1202 Geneva / CH
Application number, filing date06793019.825.08.2006
[2008/19]
WO2006EP65688
Priority number, dateEP2005010783826.08.2005         Original published format: EP 05107838
US20050711873P26.08.2005         Original published format: US 711873 P
[2008/19]
Filing languageEN
Procedural languageEN
PublicationType: A1 Application with search report
No.:WO2007023186
Date:01.03.2007
Language:EN
[2007/09]
Type: A1 Application with search report 
No.:EP1917252
Date:07.05.2008
Language:EN
The application published by WIPO in one of the EPO official languages on 01.03.2007 takes the place of the publication of the European patent application.
[2008/19]
Type: B1 Patent specification 
No.:EP1917252
Date:01.01.2014
Language:EN
[2014/01]
Search report(s)International search report - published on:EP01.03.2007
ClassificationIPC:C07D241/44, C07D401/12, C07D403/12, C07D405/12, C07D409/12, C07D417/12, A61K31/498, A61P35/00
[2008/19]
CPC:
C07D241/44 (EP,KR,US); A61K31/498 (KR); A61P1/00 (EP);
A61P1/04 (EP); A61P1/18 (EP); A61P11/00 (EP);
A61P11/06 (EP); A61P13/12 (EP); A61P15/00 (EP);
A61P15/08 (EP); A61P17/06 (EP); A61P19/02 (EP);
A61P19/04 (EP); A61P21/00 (EP); A61P25/00 (EP);
A61P25/14 (EP); A61P25/28 (EP); A61P29/00 (EP);
A61P31/04 (EP); A61P31/12 (EP); A61P35/00 (EP);
A61P35/04 (EP); A61P37/00 (EP); A61P37/06 (EP);
A61P37/08 (EP); A61P43/00 (EP); A61P7/00 (EP);
A61P7/02 (EP); A61P7/06 (EP); A61P9/00 (EP);
A61P9/04 (EP); A61P9/08 (EP); A61P9/10 (EP);
A61P9/12 (EP); C07D401/12 (EP,US); C07D403/12 (EP,US);
C07D405/12 (EP,KR,US); C07D407/12 (EP,US); C07D409/12 (EP,US);
C07D413/12 (EP,US); C07D417/12 (EP,US); C07D471/04 (EP,US) (-)
Designated contracting statesAT,   BE,   BG,   CH,   CY,   CZ,   DE,   DK,   EE,   ES,   FI,   FR,   GB,   GR,   HU,   IE,   IS,   IT,   LI,   LT,   LU,   LV,   MC,   NL,   PL,   PT,   RO,   SE,   SI,   SK,   TR [2008/19]
Extension statesAL01.02.2008
BA01.02.2008
HR01.02.2008
MK01.02.2008
RS01.02.2008
TitleGerman:PYRAZINDERIVATE UND VERWENDUNG ALS PI3K-HEMMER[2008/19]
English:PYRAZINE DERIVATIVES AND USE AS PI3K INHIBITORS[2008/19]
French:DÉRIVÉS DE PYRAZINE ET LEUR UTILISATION EN TANT QU'INHIBITEURS DE PI3K[2013/28]
Former [2008/19]DERIVE DE PYRAZINE ET LEUR UTILISATION EN TANT QU'INHIBITEURS DE PI3K
Entry into regional phase01.02.2008National basic fee paid 
01.02.2008Designation fee(s) paid 
01.02.2008Examination fee paid 
Examination procedure01.02.2008Examination requested  [2008/19]
27.11.2008Despatch of a communication from the examining division (Time limit: M04)
27.03.2009Reply to a communication from the examining division
12.01.2010Despatch of a communication from the examining division (Time limit: M06)
16.07.2010Reply to a communication from the examining division
01.03.2011Despatch of a communication from the examining division (Time limit: M04)
07.07.2011Reply to a communication from the examining division
30.12.2011Despatch of a communication from the examining division (Time limit: M06)
03.07.2012Reply to a communication from the examining division
11.09.2012Despatch of a communication from the examining division (Time limit: M04)
21.12.2012Reply to a communication from the examining division
06.08.2013Communication of intention to grant the patent
18.11.2013Fee for grant paid
18.11.2013Fee for publishing/printing paid
Divisional application(s)EP10184144.3  / EP2351745
The date of the Examining Division's first communication in respect of the earliest application for which a communication has been issued is  27.11.2008
Opposition(s)02.10.2014No opposition filed within time limit [2014/50]
Fees paidRenewal fee
01.02.2008Renewal fee patent year 03
12.08.2009Renewal fee patent year 04
17.08.2010Renewal fee patent year 05
11.08.2011Renewal fee patent year 06
10.08.2012Renewal fee patent year 07
19.08.2013Renewal fee patent year 08
Opt-out from the exclusive  Tooltip
competence of the Unified
Patent Court		 See the Register of the Unified Patent Court for opt-out data
Responsibility for the accuracy, completeness or quality of the data displayed under the link provided lies entirely with the Unified Patent Court.
Lapses during opposition  TooltipHU25.08.2006
AT01.01.2014
BE01.01.2014
BG01.01.2014
CY01.01.2014
CZ01.01.2014
DK01.01.2014
EE01.01.2014
FI01.01.2014
LT01.01.2014
LV01.01.2014
MC01.01.2014
NL01.01.2014
PL01.01.2014
RO01.01.2014
SE01.01.2014
SI01.01.2014
SK01.01.2014
TR01.01.2014
GR02.04.2014
IS01.05.2014
PT02.05.2014
IE25.08.2014
LU25.08.2014
[2016/33]
Former [2016/32]HU25.08.2006
AT01.01.2014
BE01.01.2014
BG01.01.2014
CY01.01.2014
CZ01.01.2014
DK01.01.2014
EE01.01.2014
FI01.01.2014
LT01.01.2014
LV01.01.2014
MC01.01.2014
NL01.01.2014
PL01.01.2014
RO01.01.2014
SE01.01.2014
SI01.01.2014
SK01.01.2014
GR02.04.2014
IS01.05.2014
PT02.05.2014
IE25.08.2014
LU25.08.2014
Former [2016/28]AT01.01.2014
BE01.01.2014
BG01.01.2014
CY01.01.2014
CZ01.01.2014
DK01.01.2014
EE01.01.2014
FI01.01.2014
LT01.01.2014
LV01.01.2014
MC01.01.2014
NL01.01.2014
PL01.01.2014
RO01.01.2014
SE01.01.2014
SI01.01.2014
SK01.01.2014
GR02.04.2014
IS01.05.2014
PT02.05.2014
IE25.08.2014
LU25.08.2014
Former [2016/25]AT01.01.2014
BE01.01.2014
BG01.01.2014
CY01.01.2014
CZ01.01.2014
DK01.01.2014
EE01.01.2014
FI01.01.2014
LT01.01.2014
LV01.01.2014
MC01.01.2014
NL01.01.2014
PL01.01.2014
RO01.01.2014
SE01.01.2014
SI01.01.2014
SK01.01.2014
IS01.05.2014
PT02.05.2014
IE25.08.2014
LU25.08.2014
Former [2015/37]AT01.01.2014
BE01.01.2014
CY01.01.2014
CZ01.01.2014
DK01.01.2014
EE01.01.2014
FI01.01.2014
LT01.01.2014
LV01.01.2014
MC01.01.2014
NL01.01.2014
PL01.01.2014
RO01.01.2014
SE01.01.2014
SI01.01.2014
SK01.01.2014
IS01.05.2014
PT02.05.2014
IE25.08.2014
LU25.08.2014
Former [2015/24]AT01.01.2014
BE01.01.2014
CY01.01.2014
CZ01.01.2014
DK01.01.2014
EE01.01.2014
FI01.01.2014
LT01.01.2014
LV01.01.2014
MC01.01.2014
NL01.01.2014
PL01.01.2014
RO01.01.2014
SE01.01.2014
SI01.01.2014
SK01.01.2014
IS01.05.2014
PT02.05.2014
LU25.08.2014
Former [2015/19]AT01.01.2014
BE01.01.2014
CY01.01.2014
CZ01.01.2014
DK01.01.2014
EE01.01.2014
FI01.01.2014
LT01.01.2014
LV01.01.2014
MC01.01.2014
NL01.01.2014
PL01.01.2014
RO01.01.2014
SE01.01.2014
SK01.01.2014
IS01.05.2014
PT02.05.2014
LU25.08.2014
Former [2015/18]AT01.01.2014
BE01.01.2014
CY01.01.2014
CZ01.01.2014
DK01.01.2014
EE01.01.2014
FI01.01.2014
LT01.01.2014
LV01.01.2014
MC01.01.2014
NL01.01.2014
PL01.01.2014
RO01.01.2014
SE01.01.2014
SK01.01.2014
IS01.05.2014
PT02.05.2014
Former [2014/50]AT01.01.2014
BE01.01.2014
CY01.01.2014
CZ01.01.2014
DK01.01.2014
EE01.01.2014
FI01.01.2014
LT01.01.2014
LV01.01.2014
NL01.01.2014
PL01.01.2014
RO01.01.2014
SE01.01.2014
SK01.01.2014
IS01.05.2014
PT02.05.2014
Former [2014/49]AT01.01.2014
BE01.01.2014
CY01.01.2014
CZ01.01.2014
DK01.01.2014
EE01.01.2014
FI01.01.2014
LT01.01.2014
LV01.01.2014
NL01.01.2014
RO01.01.2014
SE01.01.2014
IS01.05.2014
PT02.05.2014
Former [2014/48]AT01.01.2014
BE01.01.2014
CY01.01.2014
CZ01.01.2014
DK01.01.2014
EE01.01.2014
FI01.01.2014
LT01.01.2014
LV01.01.2014
NL01.01.2014
SE01.01.2014
IS01.05.2014
PT02.05.2014
Former [2014/41]AT01.01.2014
BE01.01.2014
CY01.01.2014
FI01.01.2014
LT01.01.2014
LV01.01.2014
NL01.01.2014
SE01.01.2014
IS01.05.2014
PT02.05.2014
Former [2014/39]AT01.01.2014
CY01.01.2014
FI01.01.2014
LT01.01.2014
NL01.01.2014
SE01.01.2014
IS01.05.2014
PT02.05.2014
Former [2014/37]AT01.01.2014
CY01.01.2014
FI01.01.2014
LT01.01.2014
SE01.01.2014
IS01.05.2014
PT02.05.2014
Former [2014/36]LT01.01.2014
IS01.05.2014
Cited inInternational search[AD]WO03035075  (ICOS CORP [US]) [AD] 1-28 * page 1, line 16 - line 19; claim 1 *;
 [X]  - CHEMCATS, CHEMICAL ABSTRACTS SERVICE, COLUMBUS, OHIO, US, (20050703), XP002408368 [X] 2,3,5,8,9,2,3,5,8,9 * Order Numbers: STT-00188957 *
 [X]  - Ambinter Stock Screening Collection, 50 AVENUE DE VERSAILLES, 75016 PARIS, FRANCE, AMBINTER SARL, (20050703) [X] 2,3,5,8,9
The EPO accepts no responsibility for the accuracy of data originating from other authorities; in particular, it does not guarantee that it is complete, up to date or fit for specific purposes.