| EP1964839 - Quinazoline derivatives as kinase inhibitors [Right-click to bookmark this link] | Status | The application has been refused Status updated on 02.09.2011 Database last updated on 11.04.2026 | Most recent event Tooltip | 02.09.2011 | Refusal of application | published on 05.10.2011 [2011/40] | Applicant(s) | For all designated states MILLENNIUM PHARMACEUTICALS, INC. 256 East Grand Avenue South San Francisco, CA 94080 / US | For all designated states KYOWA HAKKO KOGYO CO., LTD. 6-1, Ohtemachi 1-chome Chiyoda-ku Tokyo 100-8185 / JP | [2008/36] | Inventor(s) | 01 /
Pandey, Anjali 4506 Amiens Avenue Fremont, CA 94555 / US | 02 /
Scarborough, Carroll (in Trust of Bob Scarborough) 22 Greenbier Court Half Moon Bay, CA 94019 / US | 03 /
Matsuno, Kenji 1-6-1, Ohtemachi, 1-chome Tokyo 100-8185 / JP | 04 /
Ichimura, Michio 1-6-1, Ohtemachi, 1-chome Tokyo 100-8185 / JP | 05 /
Nomoto, Yuji 1-6-1, Ohtemachi, 1-chome Tokyo 100-8185 / JP | 06 /
Ide, Shinichi 1-6-1, Ohtemachi, 1-chome Tokyo 100-8185 / JP | 07 /
Tsukuda, Eiji 1-6-1, Ohtemachi, 1-chome Tokyo 100-8185 / JP | 08 /
Irie, Junko 1-6-1, Ohtemachi, 1-chome Tokyo 100-8185 / JP | 09 /
Oda, Shoji 1-6-1, Ohtemachie, 1-chome Tokyo 100-8185 / JP | [2008/50] |
| Former [2008/36] | 01 /
Pandey, Anjali 256 E. Grand Avenue South San Francisco, CA 94080 / US | ||
| 02 /
Scarborough, Robert, M. 256 E. Grand Avenue South San Franciso, CA 94080 / US | |||
| 03 /
Matsuno, Kenji 1-6-1, Ohtemachi, 1-chome Tokyo 100-8185 / JP | |||
| 04 /
Ichimura, Michio 1-6-1, Ohtemachi, 1-chome Tokyo 100-8185 / JP | |||
| 05 /
Nomoto, Yuji 1-6-1, Ohtemachi, 1-chome Tokyo 100-8185 / JP | |||
| 06 /
Ide, Shinichi 1-6-1, Ohtemachi, 1-chome Tokyo 100-8185 / JP | |||
| 07 /
Tsukuda, Eiji 1-6-1, Ohtemachi, 1-chome Tokyo 100-8185 / JP | |||
| 08 /
Irie, Junko 1-6-1, Ohtemachi, 1-chome Tokyo 100-8185 / JP | |||
| 09 /
Oda, Shoji 1-6-1, Ohtemachie, 1-chome Tokyo 100-8185 / JP | Representative(s) | Wombwell, Francis, et al Forresters 15, Hamilton Square Birkenhead Merseyside CH41 6BR / GB | [N/P] |
| Former [2008/36] | Wombwell, Francis, et al Potts, Kerr & Co. 15, Hamilton Square Birkenhead Merseyside CH41 6BR / GB | Application number, filing date | 08075237.1 | 17.08.2001 | [2008/36] | Priority number, date | US20000226122P | 18.08.2000 Original published format: US 226122 P | [2008/36] | Filing language | EN | Procedural language | EN | Publication | Type: | A2 Application without search report | No.: | EP1964839 | Date: | 03.09.2008 | Language: | EN | [2008/36] | Type: | A3 Search report | No.: | EP1964839 | Date: | 05.11.2008 | [2008/45] | Search report(s) | (Supplementary) European search report - dispatched on: | EP | 02.10.2008 | Classification | IPC: | C07D403/12, C07D239/94, C07D401/12, A61P35/00, A61K31/517 | [2008/36] | CPC: |
C07D239/94 (EP,US);
C07D401/14 (KR);
A61K31/517 (EP,US);
A61P13/12 (EP);
A61P35/00 (EP);
A61P43/00 (EP);
A61P9/00 (EP);
A61P9/02 (EP);
A61P9/08 (EP);
| Designated contracting states | AT, BE, CH, CY, DE, DK, ES, FI, FR, GB, GR, IE, IT, LI, LU, MC, NL, PT, SE, TR [2008/36] | Title | German: | Quinazolinderivate als Kinasehemmer | [2008/36] | English: | Quinazoline derivatives as kinase inhibitors | [2008/36] | French: | Dérivés de quinazoline en tant qu'inhibiteurs de la kinase | [2008/36] | Examination procedure | 02.04.2009 | Examination requested [2009/21] | 11.05.2009 | Despatch of a communication from the examining division (Time limit: M06) | 23.11.2009 | Reply to a communication from the examining division | 04.05.2011 | Date of oral proceedings | 16.05.2011 | Minutes of oral proceedings despatched | 18.05.2011 | Despatch of communication that the application is refused, reason: substantive examination [2011/40] | 28.05.2011 | Application refused, date of legal effect [2011/40] | Parent application(s) Tooltip | EP01964612.4 / EP1315715 | Divisional application(s) | EP10182322.7 / EP2277877 | The date of the Examining Division's first communication in respect of the earliest application for which a communication has been issued (EP20010964612) is 08.12.2003 | Fees paid | Renewal fee | 31.03.2008 | Renewal fee patent year 03 | 31.03.2008 | Renewal fee patent year 04 | 31.03.2008 | Renewal fee patent year 05 | 31.03.2008 | Renewal fee patent year 06 | 31.03.2008 | Renewal fee patent year 07 | 31.03.2008 | Renewal fee patent year 08 | 25.08.2009 | Renewal fee patent year 09 | 25.08.2010 | Renewal fee patent year 10 |
| Opt-out from the exclusive Tooltip competence of the Unified Patent Court | See the Register of the Unified Patent Court for opt-out data | ||
| Responsibility for the accuracy, completeness or quality of the data displayed under the link provided lies entirely with the Unified Patent Court. | Documents cited: | Search | [XD] EP0882717 (KYOWA HAKKO KOGYO KK et al.) | [PA] EP1067123 (KYOWA HAKKO KOGYO KK et al.) | [PA] WO9951582 (KYOWA HAKKO KOGYO KK et al.) | by applicant | ZA6706512 | JPH05208911 | WO9609294 | WO9220642 | JPH0687834 | WO9814431 | CELL, vol. 46, 1986, pages 155 - 169 | SCIENCE, vol. 253, 1991, pages 1129 - 1132 | NIPPON RINSHO, JAPANESE J. OF CLINICAL MEDICINE, vol. 50, 1992, pages 3038 - 3045 | NEPHROL DIAL TRANSPLANT, vol. 10, 1995, pages 787 - 795 | KIDNEY INTERNATIONAL, vol. 43, no. 39, 1993, pages 86 - 89 | JOURNAL OF RHEUMATOLOGY, vol. 21, 1994, pages 1507 - 1511 | SCANDINAVIAN JOURNAL OF IMMUNOLOGY, vol. 27, 1988, pages 285 - 294 | PHARMACOLOGY BIOCHEMISTRY AND BEHAVIOR, vol. 53, 1996, pages 87 - 97 | EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, vol. 31, 1996, pages 417 - 425 | INDIAN JOURNAL OF CHEMISTRY, vol. 26B, 1987, pages 550 - 555 | CANCER RESEARCH, vol. 54, 1994, pages 6106 | KANAZAWA, ABSTRACTS OF THE 16TH ANNUAL MEETING OF THE PHARMACEUTICAL SOCIETY OF JAPAN, vol. 2, 1996, pages 275 | T. W. GREENE: "Protective Groups in Organic Synthesis", 1981, JOHN WILEY & SONS INC. | R. C. LAROCK, COMPREHENSIVE ORGANIC TRANSFORMATIONS, 1989 | J. IMMUNOL. METHODS, vol. 142, 1991, pages 257 - 265 | IKEDA ET AL., ANNUAL REPORT OF TOLCYO METROPOLITAN RESEARCH LABORATORIES P. H., vol. 36, 1985, pages 277 | MORIYAMA ET AL., HINYO KIYO, vol. 40, 1994, pages 565 | KLOMPMALCERS ET AL., ANALYTICAL BIOCHEMISTRY, vol. 153, 1986, pages 80 | MIESEL ET AL., INFLAMMATION, vol. 17, 1993, pages 595 | TRACEY ET AL., JOURNAL OF PHARMACOLOGY & EXPERIMENTAL THERAPEUTICS, vol. 272, 1995, pages 1011 |