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Extract from the Register of European Patents

EP About this file: EP2106396

EP2106396 - CHEMICAL COMPOUNDS 637: PYRIDOPYRIMIDINEDIONES AS PDE4 INHIBITORS [Right-click to bookmark this link]
StatusNo opposition filed within time limit
Status updated on  31.07.2015
Database last updated on 20.09.2024
Most recent event   Tooltip13.10.2017Lapse of the patent in a contracting state
New state(s): BG, HU, TR		published on 15.11.2017  [2017/46]
Applicant(s)For all designated states
Alcon Research, Ltd.
6201 South Freeway
Fort Worth, TX 76134-2099 / US
[2013/50]
Former [2009/41]For all designated states
AstraZeneca AB
151 85 Södertälje / SE
Inventor(s)01 / BONNERT, Roger, Victor
AstraZeneca R & D Charnwood
Bakewell Road
Loughborough Leicestershire LE11 5RH / GB
02 / BURKAMP, Frank
AstraZeneca R & D Charnwood
Bakewell Road
Loughborough Leicestershire LE11 5RH / GB
03 / COX, Rhona, Jane
AstraZeneca R & D Charnwood
Bakewell Road
Loughborough Leicestershire LE11 5RH / GB
04 / DE SOUSA, Simon
AstraZeneca R & D Charnwood
Bakewell Road
Loughborough Leicestershire LE11 5RH / GB
05 / DICKINSON, Mark
AstraZeneca R & D Charnwood
Bakewell Road
Loughborough Leicestershire LE11 5RH / GB
06 / HUNT, Simon, Fraser
AstraZeneca R & D Charnwood
Bakewell Road
Loughborough Leicestershire LE11 5RH / GB
07 / MEGHANI, Premji
AstraZeneca R & D Charnwood
Bakewell Road
Loughborough Leicestershire LE11 5RH / GB
08 / PIMM, Austen
AstraZeneca R & D Charnwood
Bakewell Road
Loughborough Leicestershire LE11 5RH / GB
09 / SANGANEE, Hitesh, Jayantilal
AstraZeneca R & D Charnwood
Bakewell Road
Loughborough Leicestershire LE11 5RH / GB
 [2014/39]
Former [2009/41]01 / BONNERT, Roger, Victor
AstraZeneca R & D Charnwood Bakewell Road
Loughborough Leicestershire LE11 5RH / GB
02 / BURKAMP, Frank
AstraZeneca R & D Charnwood Bakewell Road
Loughborough Leicestershire LE11 5RH / GB
03 / COX, Rhona, Jane
AstraZeneca R & D Charnwood Bakewell Road
Loughborough Leicestershire LE11 5RH / GB
04 / DE SOUSA, Simon
AstraZeneca R & D Charnwood Bakewell Road
Loughborough Leicestershire LE11 5RH / GB
05 / DICKINSON, Mark
AstraZeneca R & D Charnwood Bakewell Road
Loughborough Leicestershire LE11 5RH / GB
06 / HUNT, Simon, Fraser
AstraZeneca R & D Charnwood Bakewell Road
Loughborough Leicestershire LE11 5RH / GB
07 / MEGHANI, Premji
AstraZeneca R & D Charnwood Bakewell Road
Loughborough Leicestershire LE11 5RH / GB
08 / PIMM, Austen
AstraZeneca R & D Charnwood Bakewell Road
Loughborough Leicestershire LE11 5RH / GB
09 / SANGANEE, Hitesh, Jayantilal
AstraZeneca R & D Charnwood Bakewell Road
Loughborough Leicestershire LE11 5RH / GB
Representative(s)Teipel, Stephan
Lederer & Keller
Patentanwälte Partnerschaft mbB
Unsöldstrasse 2
80538 München / DE
[2014/39]
Former [2013/50]Teipel, Stephan
Lederer & Keller Patentanwälte Unsöldstrasse 2
80538 München / DE
Application number, filing date08700158.210.01.2008
[2009/41]
WO2008GB00061
Priority number, dateUS20070884454P11.01.2007         Original published format: US 884454 P
US20070941749P04.06.2007         Original published format: US 941749 P
US20070952047P26.07.2007         Original published format: US 952047 P
[2009/41]
Filing languageEN
Procedural languageEN
PublicationType: A2 Application without search report
No.:WO2008084223
Date:17.07.2008
Language:EN
[2008/29]
Type: A2 Application without search report 
No.:EP2106396
Date:07.10.2009
Language:EN
The application published by WIPO in one of the EPO official languages on 17.07.2008 takes the place of the publication of the European patent application.
[2009/41]
Type: B1 Patent specification 
No.:EP2106396
Date:24.09.2014
Language:EN
[2014/39]
Search report(s)International search report - published on:EP02.10.2008
ClassificationIPC:C07D213/80, C07D401/12, C07D471/04, C07D471/08, C07D519/00, A61K31/519, A61P11/06
[2009/41]
CPC:
C07D519/00 (EP,KR,US); C07D471/04 (EP,KR,US); A61K31/519 (KR);
A61P1/00 (EP); A61P1/02 (EP); A61P1/04 (EP);
A61P1/12 (EP); A61P1/16 (EP); A61P1/18 (EP);
A61P11/00 (EP); A61P11/02 (EP); A61P11/06 (EP);
A61P11/08 (EP); A61P11/14 (EP); A61P11/16 (EP);
A61P13/08 (EP); A61P13/10 (EP); A61P13/12 (EP);
A61P15/00 (EP); A61P15/02 (EP); A61P15/08 (EP);
A61P15/10 (EP); A61P17/00 (EP); A61P17/06 (EP);
A61P17/14 (EP); A61P19/02 (EP); A61P19/04 (EP);
A61P19/06 (EP); A61P19/08 (EP); A61P19/10 (EP);
A61P21/04 (EP); A61P25/00 (EP); A61P25/04 (EP);
A61P25/06 (EP); A61P25/24 (EP); A61P25/28 (EP);
A61P27/02 (EP); A61P27/14 (EP); A61P29/00 (EP);
A61P3/10 (EP); A61P31/00 (EP); A61P31/04 (EP);
A61P31/10 (EP); A61P31/12 (EP); A61P31/14 (EP);
A61P31/16 (EP); A61P35/00 (EP); A61P35/02 (EP);
A61P37/00 (EP); A61P37/02 (EP); A61P37/06 (EP);
A61P37/08 (EP); A61P43/00 (EP); A61P7/00 (EP);
A61P7/02 (EP); A61P9/00 (EP); A61P9/10 (EP);
A61P9/12 (EP); C07D213/80 (EP,US); C07D401/12 (EP,US);
C07D471/08 (EP,US) (-)
Designated contracting statesAT,   BE,   BG,   CH,   CY,   CZ,   DE,   DK,   EE,   ES,   FI,   FR,   GB,   GR,   HR,   HU,   IE,   IS,   IT,   LI,   LT,   LU,   LV,   MC,   MT,   NL,   NO,   PL,   PT,   RO,   SE,   SI,   SK,   TR [2009/41]
Extension statesAL11.08.2009
BA11.08.2009
MK11.08.2009
RS11.08.2009
TitleGerman:CHEMISCHE VERBINDUNGEN 637: PYRIDOPYRIMIDINDIONE ALS PDE4-INHIBITOREN[2009/41]
English:CHEMICAL COMPOUNDS 637: PYRIDOPYRIMIDINEDIONES AS PDE4 INHIBITORS[2009/41]
French:COMPOSÉS CHIMIQUES 637: PYRIDOPYRIMIDINEDIONES COMME INHIBITEURS PDE4[2009/41]
Entry into regional phase11.08.2009National basic fee paid 
11.08.2009Designation fee(s) paid 
11.08.2009Examination fee paid 
Examination procedure11.08.2009Examination requested  [2009/41]
21.08.2012Despatch of a communication from the examining division (Time limit: M06)
21.02.2013Reply to a communication from the examining division
05.08.2013Despatch of a communication from the examining division (Time limit: M02)
14.10.2013Reply to a communication from the examining division
10.04.2014Communication of intention to grant the patent
05.08.2014Fee for grant paid
05.08.2014Fee for publishing/printing paid
05.08.2014Receipt of the translation of the claim(s)
Divisional application(s)The date of the Examining Division's first communication in respect of the earliest application for which a communication has been issued is  21.08.2012
Opposition(s)25.06.2015No opposition filed within time limit [2015/36]
Fees paidRenewal fee
01.02.2010Renewal fee patent year 03
31.01.2011Renewal fee patent year 04
31.01.2012Renewal fee patent year 05
31.01.2013Renewal fee patent year 06
21.01.2014Renewal fee patent year 07
Opt-out from the exclusive  Tooltip
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Patent Court		 See the Register of the Unified Patent Court for opt-out data
Responsibility for the accuracy, completeness or quality of the data displayed under the link provided lies entirely with the Unified Patent Court.
Lapses during opposition  TooltipHU10.01.2008
AT24.09.2014
BG24.09.2014
CY24.09.2014
CZ24.09.2014
DK24.09.2014
EE24.09.2014
ES24.09.2014
FI24.09.2014
HR24.09.2014
IT24.09.2014
LT24.09.2014
LV24.09.2014
MC24.09.2014
MT24.09.2014
NL24.09.2014
PL24.09.2014
RO24.09.2014
SE24.09.2014
SI24.09.2014
SK24.09.2014
TR24.09.2014
NO24.12.2014
GR25.12.2014
GB10.01.2015
IE10.01.2015
LU10.01.2015
IS24.01.2015
PT26.01.2015
BE31.01.2015
CH31.01.2015
LI31.01.2015
FR02.02.2015
[2017/39]
Former [2017/03]AT24.09.2014
CY24.09.2014
CZ24.09.2014
DK24.09.2014
EE24.09.2014
ES24.09.2014
FI24.09.2014
HR24.09.2014
IT24.09.2014
LT24.09.2014
LV24.09.2014
MC24.09.2014
MT24.09.2014
NL24.09.2014
PL24.09.2014
RO24.09.2014
SE24.09.2014
SI24.09.2014
SK24.09.2014
NO24.12.2014
GR25.12.2014
GB10.01.2015
IE10.01.2015
LU10.01.2015
IS24.01.2015
PT26.01.2015
BE31.01.2015
CH31.01.2015
LI31.01.2015
FR02.02.2015
Former [2016/12]AT24.09.2014
CY24.09.2014
CZ24.09.2014
DK24.09.2014
EE24.09.2014
ES24.09.2014
FI24.09.2014
HR24.09.2014
IT24.09.2014
LT24.09.2014
LV24.09.2014
MC24.09.2014
NL24.09.2014
PL24.09.2014
RO24.09.2014
SE24.09.2014
SI24.09.2014
SK24.09.2014
NO24.12.2014
GR25.12.2014
GB10.01.2015
IE10.01.2015
LU10.01.2015
IS24.01.2015
PT26.01.2015
BE31.01.2015
CH31.01.2015
LI31.01.2015
FR02.02.2015
Former [2016/07]AT24.09.2014
CY24.09.2014
CZ24.09.2014
DK24.09.2014
EE24.09.2014
ES24.09.2014
FI24.09.2014
HR24.09.2014
IT24.09.2014
LT24.09.2014
LV24.09.2014
MC24.09.2014
NL24.09.2014
PL24.09.2014
RO24.09.2014
SE24.09.2014
SK24.09.2014
NO24.12.2014
GR25.12.2014
GB10.01.2015
IE10.01.2015
LU10.01.2015
IS24.01.2015
PT26.01.2015
BE31.01.2015
CH31.01.2015
LI31.01.2015
FR02.02.2015
Former [2015/51]AT24.09.2014
CY24.09.2014
CZ24.09.2014
DK24.09.2014
EE24.09.2014
ES24.09.2014
FI24.09.2014
HR24.09.2014
IT24.09.2014
LT24.09.2014
LV24.09.2014
MC24.09.2014
NL24.09.2014
PL24.09.2014
RO24.09.2014
SE24.09.2014
SK24.09.2014
NO24.12.2014
GR25.12.2014
GB10.01.2015
LU10.01.2015
IS24.01.2015
PT26.01.2015
BE31.01.2015
CH31.01.2015
LI31.01.2015
FR02.02.2015
Former [2015/48]AT24.09.2014
CY24.09.2014
CZ24.09.2014
DK24.09.2014
EE24.09.2014
ES24.09.2014
FI24.09.2014
HR24.09.2014
IT24.09.2014
LT24.09.2014
LV24.09.2014
MC24.09.2014
NL24.09.2014
PL24.09.2014
RO24.09.2014
SE24.09.2014
SK24.09.2014
NO24.12.2014
GR25.12.2014
GB10.01.2015
LU10.01.2015
IS24.01.2015
PT26.01.2015
BE31.01.2015
CH31.01.2015
LI31.01.2015
Former [2015/47]AT24.09.2014
CY24.09.2014
CZ24.09.2014
DK24.09.2014
EE24.09.2014
ES24.09.2014
FI24.09.2014
HR24.09.2014
IT24.09.2014
LT24.09.2014
LV24.09.2014
MC24.09.2014
NL24.09.2014
PL24.09.2014
RO24.09.2014
SE24.09.2014
SK24.09.2014
NO24.12.2014
GR25.12.2014
LU10.01.2015
IS24.01.2015
PT26.01.2015
BE31.01.2015
CH31.01.2015
LI31.01.2015
Former [2015/43]AT24.09.2014
CY24.09.2014
CZ24.09.2014
DK24.09.2014
EE24.09.2014
ES24.09.2014
FI24.09.2014
HR24.09.2014
IT24.09.2014
LT24.09.2014
LV24.09.2014
MC24.09.2014
NL24.09.2014
PL24.09.2014
RO24.09.2014
SE24.09.2014
SK24.09.2014
NO24.12.2014
GR25.12.2014
LU10.01.2015
IS24.01.2015
PT26.01.2015
BE31.01.2015
Former [2015/39]AT24.09.2014
CY24.09.2014
CZ24.09.2014
DK24.09.2014
EE24.09.2014
ES24.09.2014
FI24.09.2014
HR24.09.2014
IT24.09.2014
LT24.09.2014
LV24.09.2014
NL24.09.2014
PL24.09.2014
RO24.09.2014
SE24.09.2014
SK24.09.2014
NO24.12.2014
GR25.12.2014
LU10.01.2015
IS24.01.2015
PT26.01.2015
BE31.01.2015
Former [2015/37]AT24.09.2014
CY24.09.2014
CZ24.09.2014
DK24.09.2014
EE24.09.2014
ES24.09.2014
FI24.09.2014
HR24.09.2014
IT24.09.2014
LT24.09.2014
LV24.09.2014
NL24.09.2014
PL24.09.2014
RO24.09.2014
SE24.09.2014
SK24.09.2014
NO24.12.2014
GR25.12.2014
IS24.01.2015
PT26.01.2015
BE31.01.2015
Former [2015/34]AT24.09.2014
CY24.09.2014
CZ24.09.2014
DK24.09.2014
EE24.09.2014
ES24.09.2014
FI24.09.2014
HR24.09.2014
LT24.09.2014
LV24.09.2014
NL24.09.2014
PL24.09.2014
RO24.09.2014
SE24.09.2014
SK24.09.2014
NO24.12.2014
GR25.12.2014
IS24.01.2015
PT26.01.2015
BE31.01.2015
Former [2015/30]AT24.09.2014
CY24.09.2014
CZ24.09.2014
EE24.09.2014
ES24.09.2014
FI24.09.2014
HR24.09.2014
LT24.09.2014
LV24.09.2014
NL24.09.2014
PL24.09.2014
RO24.09.2014
SE24.09.2014
SK24.09.2014
NO24.12.2014
GR25.12.2014
IS24.01.2015
PT26.01.2015
BE31.01.2015
Former [2015/25]AT24.09.2014
CY24.09.2014
CZ24.09.2014
EE24.09.2014
ES24.09.2014
FI24.09.2014
HR24.09.2014
LT24.09.2014
LV24.09.2014
NL24.09.2014
PL24.09.2014
RO24.09.2014
SE24.09.2014
SK24.09.2014
NO24.12.2014
GR25.12.2014
IS24.01.2015
PT26.01.2015
Former [2015/24]CY24.09.2014
CZ24.09.2014
EE24.09.2014
ES24.09.2014
FI24.09.2014
HR24.09.2014
LT24.09.2014
LV24.09.2014
NL24.09.2014
PL24.09.2014
RO24.09.2014
SE24.09.2014
SK24.09.2014
NO24.12.2014
GR25.12.2014
IS24.01.2015
PT26.01.2015
Former [2015/23]CY24.09.2014
CZ24.09.2014
EE24.09.2014
ES24.09.2014
FI24.09.2014
HR24.09.2014
LT24.09.2014
LV24.09.2014
NL24.09.2014
RO24.09.2014
SE24.09.2014
SK24.09.2014
NO24.12.2014
GR25.12.2014
IS24.01.2015
PT26.01.2015
Former [2015/22]CY24.09.2014
FI24.09.2014
HR24.09.2014
LT24.09.2014
LV24.09.2014
NL24.09.2014
RO24.09.2014
SE24.09.2014
NO24.12.2014
GR25.12.2014
PT26.01.2015
Former [2015/16]CY24.09.2014
FI24.09.2014
HR24.09.2014
LT24.09.2014
LV24.09.2014
NL24.09.2014
SE24.09.2014
NO24.12.2014
GR25.12.2014
Former [2015/12]CY24.09.2014
FI24.09.2014
HR24.09.2014
LT24.09.2014
LV24.09.2014
SE24.09.2014
NO24.12.2014
GR25.12.2014
Former [2015/11]CY24.09.2014
FI24.09.2014
LT24.09.2014
SE24.09.2014
NO24.12.2014
GR25.12.2014
Former [2015/10]FI24.09.2014
LT24.09.2014
SE24.09.2014
NO24.12.2014
Former [2015/09]FI24.09.2014
LT24.09.2014
SE24.09.2014
Former [2015/08]LT24.09.2014
Cited inInternational search[X]DE2257203  (YAMANOUCHI PHARMA CO LTD) [X] 17 * Claim 1; examples 20, 23. *;
 [X]US3838156  (BRUNDAGE R, et al) [X] 17 * Example 2. *;
 [DA]WO9319068  (SYNTEX INC [US]) [DA] 1-17 * Abstract; claims; examples. *;
 [X]WO2005086656  (BAYER PHARMACEUTICALS CORP [US], et al) [X] 17* Claim 1; examples, e.g. nos. 1, 8-9, 17-18, 28-36. *;
 [PX]WO2007004958  (ASTRAZENECA AB [SE], et al) [PX] 1-17 * Abstract; claims; examples. *;
 [PX]WO2007108750  (ASTRAZENECA AB [SE], et al) [PX] 1-17 * Abstract; claims; examples. *;
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DOI:   http://dx.doi.org/10.1021/jm00106a024
 [XA]  - BEILSTEIN, BEILSTEIN INSTITUTE FOR ORGANIC CHEMISTRY, FRANKFURT-MAIN, DE, Database accession no. 388408 (BRN), XP002477479 [X] 17 * The whole document, e.g. reactions 2 of 4 and 3 of 4. * [A] 1-16
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