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Extract from the Register of European Patents

EP About this file: EP2203412

EP2203412 - MONOACYLGLYCEROL LIPASE INHIBITORS FOR MODULATION OF CANNABINOID ACTIVITY [Right-click to bookmark this link]
StatusThe application has been withdrawn
Status updated on  15.06.2012
Database last updated on 25.09.2024
Most recent event   Tooltip15.06.2012Withdrawal of applicationpublished on 18.07.2012  [2012/29]
Applicant(s)For all designated states
NORTHEASTERN UNIVERSITY
360 Huntington Avenue
Boston, MA 02115-5000 / US
[2010/27]
Inventor(s)01 / MAKRIYANNIS, Alexandros
16 Stearns Road
Watertown MA 02472 / US
02 / NIKAS, Spyridon, P.
4 Dolores Avenue Apt. 12
Waltham, MA 02452 / US
03 / ALAPAFUJA, Shakiru, O.
47 Homer Avenue Apt. 5-3
Cambridge, MA 02138 / US
04 / SHUKLA, Vidyanand, G.
105 West 4th Street Apt. 4A
South Boston, MA 02127 / US
 [2010/46]
Former [2010/27]01 / MAKRIYANNIS, Alexandros
16 Stearns Road
Watertown MA 02472 / US
02 / NIKAS, Spyridon, P.
5 Dolores Avenue
Waltham MA 02452 / US
03 / ALAPAFUJA, Shakiru, O.
132 S. Common Street Apt. 105
Lynn MA 01962 / US
04 / SHUKLA, Vidyanand, G.
5 Dolores Avenue
Waltham MA 02452 / US
Representative(s)Atkinson, Jonathan David Mark
HGF Limited
1 City Walk
Leeds LS11 9DX / GB
[N/P]
Former [2012/03]Atkinson, Jonathan David Mark
Harrison Goddard Foote Belgrave Hall Belgrave Street
Leeds LS2 8DD / GB
Former [2010/27]Grund, Martin, et al
GRUND Intellectual Property Group Postfach 44 05 16
80754 München / DE
Application number, filing date08840122.916.10.2008
[2010/27]
WO2008US80214
Priority number, dateUS20070999127P16.10.2007         Original published format: US 999127 P
[2010/27]
Filing languageEN
Procedural languageEN
PublicationType: A1 Application with search report
No.:WO2009052319
Date:23.04.2009
Language:EN
[2009/17]
Type: A1 Application with search report 
No.:EP2203412
Date:07.07.2010
Language:EN
The application published by WIPO in one of the EPO official languages on 23.04.2009 takes the place of the publication of the European patent application.
[2010/27]
Search report(s)International search report - published on:US23.04.2009
(Supplementary) European search report - dispatched on:EP13.12.2011
ClassificationIPC:C07C309/82, C07C323/43, C07C37/50, C07C271/28, C07D211/16, A61K31/00, C07C37/62
[2012/02]
CPC:
C07C271/28 (EP,US); A61K31/00 (EP,US); A61P1/12 (EP);
A61P15/08 (EP); A61P19/02 (EP); A61P19/10 (EP);
A61P25/00 (EP); A61P25/02 (EP); A61P25/04 (EP);
A61P25/08 (EP); A61P25/16 (EP); A61P25/18 (EP);
A61P25/22 (EP); A61P25/24 (EP); A61P25/28 (EP);
A61P29/00 (EP); A61P3/00 (EP); A61P35/00 (EP);
A61P9/12 (EP); C07C271/38 (EP,US); C07C309/82 (EP,US);
C07C323/43 (EP,US); C07C37/055 (EP,US); C07C37/62 (EP,US);
C07C45/41 (EP,US); C07C45/44 (EP,US); C07C45/45 (EP,US);
C07C45/673 (EP,US); C07C45/68 (EP,US); C07C49/255 (EP,US);
C07C49/84 (EP,US); C07D211/16 (EP,US); C07D213/61 (EP,US);
C07D271/10 (EP,US); C07D275/03 (EP,US); C07D275/06 (EP,US);
C07D317/54 (EP,US); C07F9/5442 (EP,US); C07C2603/74 (EP,US) (-)
C-Set:
C07C37/055, C07C39/11 (US,EP);
C07C37/055, C07C39/24 (EP,US);
C07C37/62, C07C39/24 (EP,US);
C07C45/41, C07C47/277 (US,EP);
C07C45/44, C07C47/575 (US,EP);
C07C45/45, C07C49/233 (US,EP);
C07C45/45, C07C49/255 (US,EP);
C07C45/673, C07C49/83 (EP,US);
C07C45/673, C07C49/84 (EP,US);
C07C45/68, C07C49/84 (EP,US)
(-)
Former IPC [2010/27]C07C231/00
Designated contracting statesAT,   BE,   BG,   CH,   CY,   CZ,   DE,   DK,   EE,   ES,   FI,   FR,   GB,   GR,   HR,   HU,   IE,   IS,   IT,   LI,   LT,   LU,   LV,   MC,   MT,   NL,   NO,   PL,   PT,   RO,   SE,   SI,   SK,   TR [2010/27]
TitleGerman:MONOACYLGLYCEROLLIPASEHEMMER ZUR MODULATION DER CANNABINOIDAKTIVITÄT[2010/27]
English:MONOACYLGLYCEROL LIPASE INHIBITORS FOR MODULATION OF CANNABINOID ACTIVITY[2010/27]
French:INHIBITEURS DE LA MONOACYLGLYCÉROL LIPASE DE MODULATION DE L'ACTIVITÉ CANNABINOÏDE[2010/27]
Entry into regional phase14.04.2010National basic fee paid 
14.04.2010Search fee paid 
14.04.2010Designation fee(s) paid 
14.04.2010Examination fee paid 
Examination procedure14.04.2010Examination requested  [2010/27]
17.05.2010Amendment by applicant (claims and/or description)
07.06.2012Application withdrawn by applicant  [2012/29]
Fees paidRenewal fee
25.10.2010Renewal fee patent year 03
25.10.2011Renewal fee patent year 04
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Documents cited:Search[XP]WO2008013963  (UNIV CONNECTICUT [US], et al) [XP] 1-11 * page 43; claim -; compound 18 *;
 [XI]  - DAVID A KARANIAN ET AL, "Dual Modulation of Endocannabinoid Transport and Fatty Acid Amide Hydrolase Protects against Excitotoxicity", JOURNAL OF THE HISTORY OF THE NEUROSCIENCES, SWETS AND ZEITLINGER, LISSE, NL, (20050824), vol. 25, no. 34, doi:10.1523/JNEUROSCI.2347-05.2005, ISSN 0964-704X, pages 7813 - 7820, XP008103385 [X] 1-10 * page 1195, column L, paragraph 2 * [I] 11

DOI:   http://dx.doi.org/10.1523/JNEUROSCI.2347-05.2005
 [XI]  - M STEFFENS ET AL, "Cannabinoid CB 1 receptor-mediated modulation of evoked dopamine release and of adenylyl cyclase activity in the human neocortex", BRITISH JOURNAL OF PHARMACOLOGY, (20040401), vol. 141, no. 7, doi:10.1038/sj.bjp.0705706, ISSN 0007-1188, pages 1193 - 1203, XP055003419 [X] 1-10 * the whole document * [I] 11

DOI:   http://dx.doi.org/10.1038/sj.bjp.0705706
International search[X]WO2006116773  (UNIV CALIFORNIA [US], et al);
 [X]WO2006044617  (SCRIPPS RESEARCH INST [US], et al);
 [X]WO9013549  (STERLING DRUG INC [US]);
 [X]WO9745407  (UNIV CONNECTICUT [US]);
 [Y]US7109216  (KRUSE CORNELIS G [NL], et al);
 [Y]WO2007046550  (TANABE SEIYAKU CO [JP], et al);
 [Y]  - KOUTEK ET AL., "Inhibitors of Arachidonoyl Ethanolamide Hydrolysis", THE JOURNAL OF BIOLOGICAL CHEMISTRY, (19940916), vol. 269, no. 37, page 22938, XP008132715
The EPO accepts no responsibility for the accuracy of data originating from other authorities; in particular, it does not guarantee that it is complete, up to date or fit for specific purposes.