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Extract from the Register of European Patents

EP About this file: EP2222648

EP2222648 - PYRIMIDINE DERIVATIVES FOR THE TREATMENT OF ASTHMA, COPD, ALLERGIC RHINITIS, ALLERGIC CONJUNCTIVITIS, ATOPIC DERMATITIS, CANCER, HEPATITIS B, HEPATITIS C, HIV, HPV, BACTERIAL INFECTIONS AND DERMATOSIS [Right-click to bookmark this link]
StatusNo opposition filed within time limit
Status updated on  15.11.2013
Database last updated on 03.10.2024
Most recent event   Tooltip24.01.2014Change - lapse in a contracting state
State(s) deleted from list of lapses: CY
published on 26.02.2014  [2014/09]
Applicant(s)For all designated states
AstraZeneca AB
151 85 Södertälje / SE
For all designated states
Dainippon Sumitomo Pharma Co., Ltd.
6-8, Dosho-machi 2-chome Chuo-ku Osaka-shi
Osaka 541-8524 / JP
[2010/35]
Inventor(s)01 / BENNETT, Nicholas, J.
AstraZeneca R&D Charnwood
Bakewell Road
Loughborough, Leicestershire LE11 5RH / GB
02 / MCINALLY, Thomas
AstraZeneca R&D Charnwood
Bakewell Road
Loughborough, Leicestershire LE11 5RH / GB
03 / MOCHEL, Tobias
AstraZeneca R&D Charnwood
Bakewell Road
Loughborough, Leicestershire LE11 5RH / GB
04 / THOM, Stephen
AstraZeneca R&D Charnwood
Bakewell Road
Loughborough, Leicestershire LE11 5RH / GB
05 / TIDÉN, Anna-Karin
AstraZeneca R&D Charnwood
Bakewell Road
Loughborough Leicestershire LE11 5RH / GB
 [2013/02]
Former [2010/35]01 / BENNETT, Nicholas, J.
AstraZeneca R&D Charnwood Bakewell Road
Loughborough, Leicestershire LE11 5RH / GB
02 / MCINALLY, Thomas
AstraZeneca R&D Charnwood Bakewell Road
Loughborough, Leicestershire LE11 5RH / GB
03 / MOCHEL, Tobias
AstraZeneca R&D Charnwood Bakewell Road
Loughborough, Leicestershire LE11 5RH / GB
04 / THOM, Stephen
AstraZeneca R&D Charnwood Bakewell Road
Loughborough, Leicestershire LE11 5RH / GB
05 / TIDÉN, Anna-Karin
AstraZeneca R&D Charnwood Bakewell Road
Loughborough Leicestershire LE11 5RH / GB
Representative(s)Curran, Sally Ann, et al
AstraZeneca
Intellectual Property
Milstein Building
Granta Park
Cambridge CB21 6GH / GB
[N/P]
Former [2013/28]Curran, Sally Ann, et al
AstraZeneca Intellectual Property
Alderley Park
Macclesfield, Cheshire SK10 4TG / GB
Former [2010/38]Nelson, Michael Andrew, et al
AstraZeneca AB, Global Intellectual Property
151 85 Sodertalje / SE
Application number, filing date08851708.121.11.2008
[2010/35]
WO2008SE51334
Priority number, dateSE2007000257722.11.2007         Original published format: SE 0702577
US20070013699P14.12.2007         Original published format: US 13699 P
[2010/35]
Filing languageEN
Procedural languageEN
PublicationType: A1 Application with search report
No.:WO2009067081
Date:28.05.2009
Language:EN
[2009/22]
Type: A1 Application with search report 
No.:EP2222648
Date:01.09.2010
Language:EN
The application published by WIPO in one of the EPO official languages on 28.05.2009 takes the place of the publication of the European patent application.
[2010/35]
Type: B1 Patent specification 
No.:EP2222648
Date:09.01.2013
Language:EN
[2013/02]
Search report(s)International search report - published on:SE28.05.2009
(Supplementary) European search report - dispatched on:EP05.11.2010
ClassificationIPC:C07D239/48, A61K31/505, A61P11/00, A61P17/00, A61P27/14, A61P31/00, A61P35/00, C07D239/49, C07D401/10, C07D401/12, C07D403/10, C07D403/12, C07D417/10
[2010/35]
CPC:
C07D239/48 (EP,KR,US); A61K31/505 (KR); A61P1/16 (EP);
A61P11/00 (EP); A61P11/02 (EP); A61P11/06 (EP);
A61P17/00 (EP); A61P27/00 (EP); A61P27/14 (EP);
A61P31/00 (EP); A61P31/04 (EP); A61P31/12 (EP);
A61P31/14 (EP); A61P31/18 (EP); A61P31/20 (EP);
A61P35/00 (EP); A61P37/08 (EP); C07D239/49 (EP,KR,US);
C07D401/10 (EP,KR,US); C07D401/12 (EP,KR,US); C07D403/10 (EP,KR,US);
C07D403/12 (EP,KR,US); C07D417/10 (KR); C07D417/12 (EP,US) (-)
Designated contracting statesAT,   BE,   BG,   CH,   CY,   CZ,   DE,   DK,   EE,   ES,   FI,   FR,   GB,   GR,   HR,   HU,   IE,   IS,   IT,   LI,   LT,   LU,   LV,   MC,   MT,   NL,   NO,   PL,   PT,   RO,   SE,   SI,   SK,   TR [2010/35]
Extension statesAL22.06.2010
BA22.06.2010
MK22.06.2010
RS22.06.2010
TitleGerman:PYRIMIDINDERIVATE ZUR BEHANDLUNG VON ASTHMA, COPD, ALLERGISCHER RHINITIS, ALLERGISCHER KONJUNKTIVITIS, ATOPISCHER DERMATITIS, KREBS, HEPATITIS B, HEPATITIS C, HIV, HPV, BAKTERIELLEN INFEKTIONEN UND DERMATOSE[2010/35]
English:PYRIMIDINE DERIVATIVES FOR THE TREATMENT OF ASTHMA, COPD, ALLERGIC RHINITIS, ALLERGIC CONJUNCTIVITIS, ATOPIC DERMATITIS, CANCER, HEPATITIS B, HEPATITIS C, HIV, HPV, BACTERIAL INFECTIONS AND DERMATOSIS[2010/35]
French:DÉRIVÉS DE PYRIMIDINE POUR LE TRAITEMENT DE L'ASTHME, DE LA BRONCHO-PNEUMOPATHIE CHRONIQUE OBSTRUCTIVE (COPD), DE LA RHINITE ALLERGIQUE, DE LA CONJONCTIVITE ALLERGIQUE, DE LA DERMATITE ATOPIQUE, DU CANCER, DE L'HÉPATITE B, DE L'HÉPATITE C, DU VIH, DU VPP, DES INFECTIONS BACTÉRIENNES ET DE LA DERMATOSE[2010/35]
Entry into regional phase22.06.2010National basic fee paid 
22.06.2010Search fee paid 
22.06.2010Designation fee(s) paid 
22.06.2010Examination fee paid 
Examination procedure22.06.2010Examination requested  [2010/35]
15.07.2010Amendment by applicant (claims and/or description)
21.12.2010Despatch of a communication from the examining division (Time limit: M04)
07.04.2011Reply to a communication from the examining division
10.07.2012Communication of intention to grant the patent
26.10.2012Fee for grant paid
26.10.2012Fee for publishing/printing paid
Divisional application(s)The date of the Examining Division's first communication in respect of the earliest application for which a communication has been issued is  21.12.2010
Opposition(s)10.10.2013No opposition filed within time limit [2013/51]
Fees paidRenewal fee
30.11.2010Renewal fee patent year 03
30.11.2011Renewal fee patent year 04
30.11.2012Renewal fee patent year 05
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See the Register of the Unified Patent Court for opt-out data
Responsibility for the accuracy, completeness or quality of the data displayed under the link provided lies entirely with the Unified Patent Court.
Lapses during opposition  Tooltipdeleted
[2014/09]
Former [2013/52]CY09.01.2013
Documents cited:Search[A]US2005119273  (LIPFORD GRAYSON B [US], et al) [A] 1,17* the whole document *
International search[A]US2657206  (HITCHINGS GEORGE H, et al);
 [A]GB1375162  (STUART, A ET AL);
 [A]US4179562  (PONSFORD ROGER J [GB]);
 [A]US4912112  (SEYDEL JOACHIM [DE], et al);
 [A]US6458798  (FUJITA HITOSHI [JP], et al);
 [A]US2004214192  (HASHIDA RYOICHI [JP], et al);
 [A]  - YOSHIMOTO, M ET AL., "Correlation analysis of Baker's studies on enzyme inhibition. 2. Chymotrypsin, trypsin, thymidine phosphorylase, uridine phosphorylase, thymidylate synthetase, cytosine nucleoside deaminase, dihydrofolate reductase, malate dehydrogenase, glutamate dehydrogenase, lactate dehydrogenase, and glycera...", JOURNAL OF MEDICINAL CHEMISTRY, (1976), vol. 19, no. 1, pages 71 - 98, XP000609047

DOI:   http://dx.doi.org/10.1021/jm00223a015
 [A]  - FALCO, E.A. ET AL., "2,4-Diaminopyrimidines as antimalarials. I. 5-Aryloxyl and 5-alkoxyl derivatives.", JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, (1951), vol. 73, no. 8, pages 3753 - 3758, XP002063219

DOI:   http://dx.doi.org/10.1021/ja01152a058
The EPO accepts no responsibility for the accuracy of data originating from other authorities; in particular, it does not guarantee that it is complete, up to date or fit for specific purposes.