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Extract from the Register of European Patents

EP About this file: EP2226322

EP2226322 - IMIDAZOLE CARBONYL COMPOUND [Right-click to bookmark this link]
StatusNo opposition filed within time limit
Status updated on  27.11.2015
Database last updated on 02.11.2024
Most recent event   Tooltip20.07.2018Lapse of the patent in a contracting state
New state(s): PT		published on 22.08.2018  [2018/34]
Applicant(s)For all designated states
Daiichi Sankyo Company, Limited
3-5-1, Nihonbashi Honcho Chuo-ku
Tokyo 103-8426 / JP
[2010/36]
Inventor(s)01 / SONEDA, Tsuyoshi
c/o Daiichi Sankyo Company, Limited
1-16-13, Kitakasai
Edogawa-ku Tokyo 134-0081 / JP
02 / TAKESHITA, Hiroshi
c/o Daiichi Sankyo Company, Limited
1-16-13, Kitakasai
Edogawa-ku Tokyo 134-0081 / JP
03 / KAGOSHIMA, Yoshiko
c/o Daiichi Sankyo Company, Limited
1-16-13, Kitakasai
Edogawa-ku Tokyo 134-0081 / JP
04 / YAMAMOTO, YUKO
c/o Daiichi Sankyo Company, Limited
1-16-13, Kitakasai
Edogawa-ku Tokyo 134-0081 / JP
05 / HOSOKAWA, Takafumi
c/o Daiichi Sankyo Company, Limited
1-16-13, Kitakasai
Edogawa-ku Tokyo 134-0081 / JP
06 / KONOSU, Toshiyuki
c/o Daiichi Sankyo Company, Limited
1-16-13, Kitakasai
Edogawa-ku Tokyo 134-0081 / JP
07 / MASUDA, Nobuhisa
c/o Daiichi Sankyo Company, Limited
1-16-13, Kitakasai
Edogawa-ku Tokyo 134-0081 / JP
08 / UCHIDA, Takuya
c/o Daiichi Sankyo Company, Limited
1-16-13, Kitakasai
Edogawa-ku Tokyo 134-0081 / JP
09 / ACHIWA, Issei
c/o Daiichi Sankyo Company, Limited
1-16-13, Kitakasai
Edogawa-ku Tokyo 134-0081 / JP
10 / KUROYANAGI, Junichi
c/o Daiichi Sankyo Company, Limited
1-16-13, Kitakasai
Edogawa-ku Tokyo 134-0081 / JP
11 / FUJISAWA, Tetsunori
c/o Daiichi Sankyo Company, Limited
1-16-13, Kitakasai
Edogawa-ku Tokyo 134-0081 / JP
12 / YOKOMIZO, Aki
c/o Daiichi Sankyo Company, Limited
1-16-13, Kitakasai
Edogawa-ku Tokyo 134-0081 / JP
13 / NOGUCHI, Tetsuji
c/o Daiichi Sankyo Company, Limited
1-16-13, Kitakasai
Edogawa-ku Tokyo 134-0081 / JP
 [2015/04]
Former [2010/36]01 / SONEDA, Tsuyoshi
c/o Daiichi Sankyo Company, Limited 1-16-13, Kitakasai
Edogawa-ku Tokyo 134-0081 / JP
02 / TAKESHITA, Hiroshi
c/o Daiichi Sankyo Company, Limited 1-16-13, Kitakasai
Edogawa-ku Tokyo 134-0081 / JP
03 / KAGOSHIMA, Yoshiko
c/o Daiichi Sankyo Company, Limited 1-16-13, Kitakasai
Edogawa-ku Tokyo 134-0081 / JP
04 / YAMAMOTO, YUKO
c/o Daiichi Sankyo Company, Limited 1-16-13, Kitakasai
Edogawa-ku Tokyo 134-0081 / JP
05 / HOSOKAWA, Takafumi
c/o Daiichi Sankyo Company, Limited 1-16-13, Kitakasai
Edogawa-ku Tokyo 134-0081 / JP
06 / KONOSU, Toshiyuki
c/o Daiichi Sankyo Company, Limited 1-16-13, Kitakasai
Edogawa-ku Tokyo 134-0081 / JP
07 / MASUDA, Nobuhisa
c/o Daiichi Sankyo Company, Limited 1-16-13, Kitakasai
Edogawa-ku Tokyo 134-0081 / JP
08 / UCHIDA, Takuya
c/o Daiichi Sankyo Company, Limited 1-16-13, Kitakasai
Edogawa-ku Tokyo 134-0081 / JP
09 / ACHIWA, Issei
c/o Daiichi Sankyo Company, Limited 1-16-13, Kitakasai
Edogawa-ku Tokyo 134-0081 / JP
10 / KUROYANAGI, Junichi
c/o Daiichi Sankyo Company, Limited 1-16-13, Kitakasai
Edogawa-ku Tokyo 134-0081 / JP
11 / FUJISAWA, Tetsunori
c/o Daiichi Sankyo Company, Limited 1-16-13, Kitakasai
Edogawa-ku Tokyo 134-0081 / JP
12 / YOKOMIZO, Aki
c/o Daiichi Sankyo Company, Limited 1-16-13, Kitakasai
Edogawa-ku Tokyo 134-0081 / JP
13 / NOGUCHI, Tetsuji
c/o Daiichi Sankyo Company, Limited 1-16-13, Kitakasai
Edogawa-ku Tokyo 134-0081 / JP
Representative(s)Fairbairn, Angus Chisholm
Marks & Clerk LLP
15 Fetter Lane
London EC4A 1BW / GB
[N/P]
Former [2015/04]Fairbairn, Angus Chisholm
Marks & Clerk LLP
90 Long Acre
London
WC2E 9RA / GB
Former [2010/36]Fairbairn, Angus Chisholm
Marks & Clerk LLP 90 Long Acre London
WC2E 9RA / GB
Application number, filing date08867971.726.12.2008
[2010/36]
WO2008JP73686
Priority number, dateJP2007033769327.12.2007         Original published format: JP 2007337693
[2010/36]
Filing languageJA
Procedural languageEN
PublicationType: A1 Application with search report
No.:WO2009084614
Date:09.07.2009
Language:JA
[2009/28]
Type: A1 Application with search report 
No.:EP2226322
Date:08.09.2010
Language:EN
[2010/36]
Type: B1 Patent specification 
No.:EP2226322
Date:21.01.2015
Language:EN
[2015/04]
Search report(s)International search report - published on:JP09.07.2009
(Supplementary) European search report - dispatched on:EP11.05.2011
ClassificationIPC:C07D417/14, A61K31/4164, A61K31/4178, A61K31/422, A61K31/427, A61K31/454, A61K31/4545, A61K31/506, A61K31/538, A61P31/00, A61P31/04, C07D233/66, C07D401/12, C07D401/14, C07D403/12, C07D409/14, C07D413/12, C07D413/14, C07D417/12, C07D487/06
[2010/36]
CPC:
C07D487/04 (EP,US); A61P31/00 (EP); A61P31/04 (EP);
A61P43/00 (EP); C07D233/66 (EP,US); C07D233/90 (EP,US);
C07D401/12 (EP,US); C07D401/14 (EP,US); C07D403/12 (EP,US);
C07D409/14 (EP,US); C07D413/12 (EP,US); C07D413/14 (EP,US);
C07D417/12 (EP,US); C07D417/14 (EP,US); C07D487/06 (EP,US);
C07D487/12 (EP,US); C07D495/04 (EP,US); C07D495/16 (EP,US);
C07D498/04 (EP,US); C07D513/04 (EP,US); C07D519/00 (EP,US) (-)
Designated contracting statesAT,   BE,   BG,   CH,   CY,   CZ,   DE,   DK,   EE,   ES,   FI,   FR,   GB,   GR,   HR,   HU,   IE,   IS,   IT,   LI,   LT,   LU,   LV,   MC,   MT,   NL,   NO,   PL,   PT,   RO,   SE,   SI,   SK,   TR [2010/36]
TitleGerman:IMIDAZOL-CARBONYL-VERBINDUNG[2010/36]
English:IMIDAZOLE CARBONYL COMPOUND[2010/36]
French:COMPOSÉ CARBONYLE D'IMIDAZOLE[2010/36]
Entry into regional phase28.06.2010Translation filed 
25.06.2010National basic fee paid 
25.06.2010Search fee paid 
25.06.2010Designation fee(s) paid 
25.06.2010Examination fee paid 
Examination procedure28.06.2010Examination requested  [2010/36]
09.12.2011Amendment by applicant (claims and/or description)
07.05.2012Despatch of a communication from the examining division (Time limit: M04)
06.09.2012Reply to a communication from the examining division
22.07.2014Communication of intention to grant the patent
01.12.2014Fee for grant paid
01.12.2014Fee for publishing/printing paid
01.12.2014Receipt of the translation of the claim(s)
Divisional application(s)The date of the Examining Division's first communication in respect of the earliest application for which a communication has been issued is  07.05.2012
Opposition(s)22.10.2015No opposition filed within time limit [2015/53]
Fees paidRenewal fee
15.12.2010Renewal fee patent year 03
12.12.2011Renewal fee patent year 04
11.12.2012Renewal fee patent year 05
12.12.2013Renewal fee patent year 06
11.12.2014Renewal fee patent year 07
Opt-out from the exclusive  Tooltip
competence of the Unified
Patent Court		 See the Register of the Unified Patent Court for opt-out data
Responsibility for the accuracy, completeness or quality of the data displayed under the link provided lies entirely with the Unified Patent Court.
Lapses during opposition  TooltipHU26.12.2008
AT21.01.2015
BE21.01.2015
CY21.01.2015
CZ21.01.2015
DK21.01.2015
EE21.01.2015
FI21.01.2015
HR21.01.2015
LT21.01.2015
LV21.01.2015
MC21.01.2015
MT21.01.2015
NL21.01.2015
PL21.01.2015
PT21.01.2015
RO21.01.2015
SE21.01.2015
SI21.01.2015
SK21.01.2015
TR21.01.2015
BG21.04.2015
NO21.04.2015
GR22.04.2015
IS21.05.2015
[2018/34]
Former [2017/40]HU26.12.2008
AT21.01.2015
BE21.01.2015
CY21.01.2015
CZ21.01.2015
DK21.01.2015
EE21.01.2015
FI21.01.2015
HR21.01.2015
LT21.01.2015
LV21.01.2015
MC21.01.2015
MT21.01.2015
NL21.01.2015
PL21.01.2015
RO21.01.2015
SE21.01.2015
SI21.01.2015
SK21.01.2015
TR21.01.2015
BG21.04.2015
NO21.04.2015
GR22.04.2015
IS21.05.2015
Former [2016/33]AT21.01.2015
BE21.01.2015
CZ21.01.2015
DK21.01.2015
EE21.01.2015
FI21.01.2015
HR21.01.2015
LT21.01.2015
LV21.01.2015
MC21.01.2015
NL21.01.2015
PL21.01.2015
RO21.01.2015
SE21.01.2015
SI21.01.2015
SK21.01.2015
BG21.04.2015
NO21.04.2015
GR22.04.2015
IS21.05.2015
Former [2016/24]AT21.01.2015
BE21.01.2015
CZ21.01.2015
DK21.01.2015
EE21.01.2015
FI21.01.2015
HR21.01.2015
LT21.01.2015
LV21.01.2015
NL21.01.2015
PL21.01.2015
RO21.01.2015
SE21.01.2015
SI21.01.2015
SK21.01.2015
BG21.04.2015
NO21.04.2015
GR22.04.2015
IS21.05.2015
Former [2016/12]AT21.01.2015
CZ21.01.2015
DK21.01.2015
EE21.01.2015
FI21.01.2015
HR21.01.2015
LT21.01.2015
LV21.01.2015
NL21.01.2015
PL21.01.2015
RO21.01.2015
SE21.01.2015
SI21.01.2015
SK21.01.2015
BG21.04.2015
NO21.04.2015
GR22.04.2015
IS21.05.2015
Former [2015/49]AT21.01.2015
CZ21.01.2015
DK21.01.2015
EE21.01.2015
FI21.01.2015
HR21.01.2015
LT21.01.2015
LV21.01.2015
NL21.01.2015
PL21.01.2015
RO21.01.2015
SE21.01.2015
SK21.01.2015
BG21.04.2015
NO21.04.2015
GR22.04.2015
IS21.05.2015
Former [2015/39]AT21.01.2015
FI21.01.2015
HR21.01.2015
LT21.01.2015
LV21.01.2015
NL21.01.2015
PL21.01.2015
SE21.01.2015
BG21.04.2015
NO21.04.2015
GR22.04.2015
IS21.05.2015
Former [2015/38]AT21.01.2015
FI21.01.2015
HR21.01.2015
LT21.01.2015
PL21.01.2015
SE21.01.2015
BG21.04.2015
NO21.04.2015
GR22.04.2015
IS21.05.2015
Former [2015/37]FI21.01.2015
HR21.01.2015
LT21.01.2015
PL21.01.2015
SE21.01.2015
BG21.04.2015
NO21.04.2015
GR22.04.2015
Former [2015/36]FI21.01.2015
HR21.01.2015
LT21.01.2015
SE21.01.2015
BG21.04.2015
NO21.04.2015
Former [2015/35]LT21.01.2015
NO21.04.2015
Documents cited:Search[X]US4602095  (ZANNO PAUL R [US], et al) [X] 1,4,6,10-13 * 3-hydroxy-4-methoxyphenyl 2-imidazolecarboxylate; column 3 *;
 [X]EP0585500  (MERRELL DOW PHARMA [US]) [X] 1,4,6,10,11 * N-[3-(1-imidazoylmethyl)phenyl]-N-phenylamine; page 16 - page 17; example 11 *;
 [X]WO2006066790  (HOFFMANN LA ROCHE [CH], et al) [X] 1,4,10-13 * page 55; table 1; compound 61 *;
 [X]WO2006047277  (JANSSEN PHARMACEUTICA NV [BE], et al) [X] 1,3,4,6,9-13 * page 135 - page 147; examples 6-8, 14, 16-48, 51a-58; table 1 *;
 [X]US4179277  (BECK GUNTHER [DE], et al) [X] 1,3,4,6,9-11 * column 101 - column 103; compounds 178, 179, 185, 196, 197 *;
 [X]US5318975  (LIS RANDALL E [US]) [X] 1,3,5,7,9-13 * N-[[4-Ethyl-2-(2-ethyl-4-methyl-1H-imidazol-1-yl)]pyrimidin-5-yl]-1H-imidazol-2-carboxamide; column 7; example 4 *;
 [X]US5082847  (PASCAL JEAN-CLAUDE [FR], et al) [X] 1,3,5,7-11 * 4-imidazolylcarbonylamino-1-phenylmethylpiperidine; column 24 *;
 [X]US4772617  (ARCHIBALD JOHN L [GB], et al) [X] 1,3,5,7-11 * N-[1-(2-[1H-indol-3-yl]ethyl)4-piperidinyl]-1H-imidazole-2-carboxamide; column 11 - column 12; example 2 *;
 [X]WO2005009966  (PFIZER LTD [GB], et al) [X] 1,3,4,6,10-13 * Syn-5-fluoro-N-{4-[(4-methyl-1H-imidazole-2-carbonyl)-amino]-cyclohexyl}-2-(3- methylsulfanyl-phenoxy)-nicotinamide;; claim 9 *;
 [X]WO2005105802  (TAKEDA PHARMACEUTICAL [JP], et al) [X] 1,3,4,6,9-13 * page 198; example 129 *;
 [XP]WO2008075196  (PFIZER PROD INC [US], et al) [XP] 1,3,4,6,9-13 * page 116; example 61 *;
 [A]WO2005026149  (ASTRAZENECA AB [SE], et al) [A] 1-17 * abstract * * claims 1-26 *
 [X]  - REGEL E ET AL, "C-ACYLIERUNG VON 5 GLIEDRIGEN N-HETEROCYCLEN, I ACYLIERUNG AN C-2 VON IMIDAZOLEN UND BENZIMIDAZOLEN//C-ACYLATION OF 5-MEMBERED N-HETEROCYCLES, I. - ACYLATION AT C-2 OF IMIDAZOLES AND BENZIMIDAZOLES", JUSTUS LIEBIGS ANNALEN DER CHEMIE, VERLAG CHEMIE GMBH, WEINHEIM; DE, (19770101), doi:DOI:10.1002/JLAC.197719770115, ISSN 0075-4617, pages 145 - 158, XP009003467 [X] 1,2,4,6,9-11 * page 152 - page 155; table 6; compounds 13_1-13_19 *

DOI:   http://dx.doi.org/10.1002/jlac.197719770115
 [X]  - DIRLAM J P ET AL, JOURNAL OF ORGANIC CHEMISTRY, AMERICAN CHEMICAL SOCIETY, EASTON.; US, (19820101), vol. 47, no. 11, doi:DOI:10.1021/JO00132A045, ISSN 0022-3263, pages 2196 - 2199, XP002105948 [X] 1,3,4,6,9-11 * page 2196; compound 2 *

DOI:   http://dx.doi.org/10.1021/jo00132a045
 [X]  - PAPADOPOULOS E P, "Reactions of imidazoles with isocyanates at elevated temperature", JOURNAL OF ORGANIC CHEMISTRY, AMERICAN CHEMICAL SOCIETY, EASTON.; US, (19771125), vol. 42, no. 24, doi:DOI:10.1021/JO00444A029, ISSN 0022-3263, pages 3925 - 3929, XP002378857 [X] 1,3,4,6,9-11 * page 3925; compound 1a *

DOI:   http://dx.doi.org/10.1021/jo00444a029
International search[X]JPS52111573  (BAYER AG);
 [X]WO9500512  (JANSSEN PHARMACEUTICA NV [BE], et al);
 [X]WO9911642  (ZENECA LTD [GB], et al);
 [X]WO0132655  (ABBOTT LAB [US]);
 [X]WO02100352  (MERCK & CO INC [US], et al);
 [X]WO2004018439  (ORCHID CHEMICALS & PHARM LTD [IN], et al);
 [X]US2004209921  (BRIDGER GARY [US], et al);
 [X]WO2005003087  (ORCHID CHEMICALS & PHARM LTD [IN], et al);
 [Y]WO2005026149  (ASTRAZENECA AB [SE], et al);
 [X]WO2005105802  (TAKEDA PHARMACEUTICAL [JP], et al);
 [Y]WO2006087543  (ASTRAZENECA AB [SE], et al);
 [Y]WO2006087544  (ASTRAZENECA AB [SE], et al);
 [Y]WO2006087548  (ASTRAZENECA AB [SE], et al);
 [Y]WO2006092599  (ASTRAZENECA AB [SE], et al);
 [Y]WO2006092608  (ASTRAZENECA AB [SE], et al);
 [X]WO2007112093  (SYNTA PHARMACEUTICALS CORP [US], et al);
 [XP]WO2008051757  (IRM LLC [US], et al);
 [XP]WO2008075196  (PFIZER PROD INC [US], et al)
ExaminationUS5990109
 WO2005030128
 WO2006099379
 US2006281788
 WO2006047504
by applicantWO2005026149
 WO2006087543
 WO2006087544
 WO2006087548
 WO2006092599
 WO2006092608
 WO2007071965
The EPO accepts no responsibility for the accuracy of data originating from other authorities; in particular, it does not guarantee that it is complete, up to date or fit for specific purposes.