Extract from the Register of European Patents

EP Citations: EP2257529

Cited inInternational search
Type:Patent literature
Publication No.:DE2051013  [X]
 (SANDOZ AG (BASEL)) [X] 1-7 * page 4; compound VI * * page 32; example 10a *;
Type:Patent literature
Publication No.:GB2073185  [X]
 (STERLING DRUG INC) [X] 1-4 * page 1; compound I * * page 10; compounds F11-F41 *;
Type:Patent literature
Publication No.:WO9743267  [X]
 (KING S COLLEGE LONDON [GB], et al) [X] 1-7 * page 5; compound II * * page 9; example 1 * * page 10; examples 2-7; table coupling *;
Type:Patent literature
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Type:Patent literature
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 (SUGEN INC [US], et al) [X] 1-4 * page 220; compounds II-93 *;
Type:Patent literature
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 (BIOFOCUS DISCOVERY LTD [GB], et al) [X] 1-4 * page 105; compound 15 *;
Type:Patent literature
Publication No.:US2006030583  [X]
 (ARNOLD WILLIAM D [US], et al) [X] 1-7 * page 108, method 44; ; page 107, paragraph 369; page 109, paragraph 376; table 29, relating to method 44 *;
Type:Patent literature
Publication No.:WO2006021881  [X]
 (PFIZER [US], et al) [X] 1-3 * claims 1,22-24 *;
Type:Patent literature
Publication No.:WO2006021886  [X]
 (PFIZER [US], et al) [X] 1-3,9-10 * claims 1,14,15 *;
Type:Patent literature
Publication No.:WO2006051270  [X]
 (ASTRAZENECA AB [SE], et al) [X] 1-4,9-13 * claims 1,19 * * pages 78-79 * * page 149, line 22; example 88 *;
Type:Patent literature
Publication No.:WO2007095588  [X]
 (NOVARTIS AG [CH], et al) [X] 1-2,9-13 * claims 20,49,61 * * table 1; compounds 145,184,261 * * page 149; table 1; compound 6 *;
Type:Patent literature
Publication No.:WO2008012326  [A]
 (NOVARTIS AG [CH], et al) [A] 1-13 * page 76; compounds 73-A *;
Type:Patent literature
Publication No.:WO2008038955  [XP]
 (CHONG KUN DANG PHARM CORP [KR], et al) [XP] 1-7,9-13 * claims 1,18,19 * * page 17; table 6; compounds 421,426 *;
Type:Patent literature
Publication No.:WO2008053157  [XP]
 (CHROMA THERAPEUTICS LTD [GB], et al) [XP] 1-4,9-13 * claims 1,18-21 * * page 53; table 2 *;
Type:Patent literature
Publication No.:WO2008094992  [XP]
 (VERTEX PHARMA [US], et al) [XP] 1-7,9-13 * claims 1,96,99,101 * * pages 118-121 *;
Type:Non-patent literature
Publication information:[X]  - KEENAN, MARTINE ET AL, "Highly efficient and flexible total synthesis of coelenterazine", CHEMICAL COMMUNICATIONS (CAMBRIDGE) , (3), 323-324 CODEN: CHCOFS; ISSN: 1359-7345, (1997), XP000652586 [X] 1-7 * page 323; figure 1; compound 6 *
DOI: http://dx.doi.org/10.1039/a607460j
Type:Non-patent literature
Publication information:[X]  - JONES, KEITH ET AL, "A Suzuki coupling approach to pyrazines related to coelenterazine", SYNLETT , (6), 509-510 CODEN: SYNLES; ISSN: 0936-5214, (1996), XP002485380 [X] 1-7 * page 510; compounds 7A-F *
DOI: http://dx.doi.org/10.1055/s-1996-5489
Type:Non-patent literature
Publication information:[A]  - TERANISHI K ET AL, "SYNTHESIS AND CHEMILUMINESCENCE OF COELENTERAZINE (OPLOPHORUS LUCIFERIN) ANALOGUES", BULLETIN OF THE CHEMICAL SOCIETY OF JAPAN, CHEMICAL SOCIETY OF JAPAN, TOKYO, JP, (19901101), vol. 63, no. 11, ISSN 0009-2673, pages 3132 - 3140, XP002037163 [A] 1-7 * page 3133; compound 47 *
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Publication information:[X]  - SATO N, "STUDIES ON PYRAZINES. THE SYNTHESIS OF 2-HYDROXY-6-PHENYLPYRAZINE AND ITS DERIVATIVES", JOURNAL OF HETEROCYCLIC CHEMISTRY, HETEROCORPORATION. PROVO, (19780601), vol. 15, no. 4, ISSN 0022-152X, pages 665 - 670, XP002049109 [X] 1-4 * page 665; figure III; compound 12 *
DOI: http://dx.doi.org/10.1002/jhet.5570150428
Type:Non-patent literature
Publication information:[X]  - WATANABE T ET AL, "A CONVENIENT SYNTHESIS OF METHYLAMINO AND DIMETHYLAMINO SUBSTITUTED AROMATIC COMPOUNDS", SYNTHESIS, GEORG THIEME VERLAG, STUTTGART, DE, (19800101), vol. 1, ISSN 0039-7881, pages 39 - 41, XP000919036 [X] 1-4 * page 40; table 1; compounds 4(3B), 5(3B) *
DOI: http://dx.doi.org/10.1055/s-1980-28915
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Publication information:[X]  - HAGEN V ET AL, "POTENTIAL CARDIOTONIC AGENTS: PART 14. SYNTHESIS AND POSITIVE INOTROPIC ACTIVITIES OF 2-MORPHOLINO-5-(4-PYRIDINYL)PYRIDINES//POTENT IELLE KARDIOTONIKA. 14. MITTEILUNG: SYNTHESE UND POSITIV INOTROPE WIRKUNGEN IN VITRO VON 2-MORPHOLINO-5-(PYRID-4-YL)PYRIDIN-DERIVATEN", PHARMAZIE, DIE, GOVI VERLAG, ESCHBORN, DE, (19920101), vol. 47, no. 10, ISSN 0031-7144, pages 767 - 769, XP001247557 [X] 1-3,9-10 * page 768; compounds 12, 13 *
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Publication information:   - STOYANOVA, S.; BULGARELLI-LEVA, G.; KIRSCH, C.; HANCK, T.; KLINGER, R.; WETZKER, R.; WYMANN, M.P., "Lipid- and protein kinase activities of G protein-coupled PI 3-kinase g: structure-activity analysis and interactions with wortmannin", BIOCHEM. J., (1997), pages 324 - 489
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