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Extract from the Register of European Patents

EP About this file: EP2459537

EP2459537 - METHOD AND SUBSTANCES FOR PREPARATION OF N-SUBSTITUTED PYRIDINIUM COMPOUNDS [Right-click to bookmark this link]
StatusNo opposition filed within time limit
Status updated on  23.10.2015
Database last updated on 28.06.2024
Most recent event   Tooltip12.10.2018Lapse of the patent in a contracting state
New state(s): AL		published on 14.11.2018  [2018/46]
Applicant(s)For:DE 
Roche Diagnostics GmbH
Sandhofer Strasse 116
68305 Mannheim / DE
For:AL  AT  BE  BG  CH  CY  CZ  DK  EE  ES  FI  FR  GB  GR  HR  HU  IE  IS  IT  LI  LT  LU  LV  MC  MK  MT  NL  NO  PL  PT  RO  SE  SI  SK  SM  TR 
F. Hoffmann-La Roche AG
Grenzacherstrasse 124
4070 Basel / CH
[N/P]
Former [2012/23]For:DE 
Roche Diagnostics GmbH
Sandhofer Strasse 116
68305 Mannheim / DE
For:AL  AT  BE  BG  CH  CY  CZ  DK  EE  ES  FI  FR  GB  GR  HR  HU  IE  IS  IT  LI  LT  LU  LV  MC  MK  MT  NL  NO  PL  PT  RO  SE  SI  SK  SM  TR 
F.Hoffmann-La Roche AG
Grenzacherstrasse 124
4070 Basel / CH
Inventor(s)01 / HEINDL, Dieter
Magnolienweg 7
81377 München / DE
02 / MAERZ, Heribert
Sternstrasse 6
82396 Paehl / DE
03 / SCHMIDT, Axel
Ludwig-Behr-Strasse 14
82327 Tutzing / DE
 [2014/50]
Former [2012/23]01 / HEINDL, Dieter
Sternstrasse 4
82396 Paehl / DE
02 / MAERZ, Heribert
Sternstrasse 6
82396 Paehl / DE
03 / SCHMIDT, Axel
Ludwig-Behr-Strasse 14
82327 Tutzing / DE
Representative(s)Burger, Alexander, et al
Roche Diagnostics GmbH
Patentabteilung
Nonnenwald 2
82377 Penzberg / DE
[N/P]
Former [2012/23]Burger, Alexander, et al
Roche Diagnostics GmbH Patent Department (LPP.....6164) P.O.Box 11 52
82372 Penzberg / DE
Application number, filing date10740156.423.07.2010
WO2010EP04522
Priority number, dateEP2009016645527.07.2009         Original published format: EP 09166455
[2012/23]
Filing languageEN
Procedural languageEN
PublicationType: A2 Application without search report
No.:WO2011012269
Date:03.02.2011
Language:EN
[2011/05]
Type: A2 Application without search report 
No.:EP2459537
Date:06.06.2012
Language:EN
The application published by WIPO in one of the EPO official languages on 03.02.2011 takes the place of the publication of the European patent application.
[2012/23]
Type: B1 Patent specification 
No.:EP2459537
Date:17.12.2014
Language:EN
[2014/51]
Search report(s)International search report - published on:EP11.08.2011
ClassificationIPC:C07D213/82, C07D401/04, C07D473/16
[2012/23]
CPC:
C07D401/04 (EP,US); C07D213/82 (EP,US); C07D473/16 (EP,US)
Designated contracting statesAL,   AT,   BE,   BG,   CH,   CY,   CZ,   DE,   DK,   EE,   ES,   FI,   FR,   GB,   GR,   HR,   HU,   IE,   IS,   IT,   LI,   LT,   LU,   LV,   MC,   MK,   MT,   NL,   NO,   PL,   PT,   RO,   SE,   SI,   SK,   SM,   TR [2012/23]
Extension statesBANot yet paid
MENot yet paid
RSNot yet paid
TitleGerman:VERFAHREN UND SUBSTANZEN ZUR HERSTELLUNG VON N-SUBSTITUIERTEN PYRIDINIUMVERBINDUNGEN[2014/32]
English:METHOD AND SUBSTANCES FOR PREPARATION OF N-SUBSTITUTED PYRIDINIUM COMPOUNDS[2012/23]
French:PROCÉDÉS ET SUBSTANCES POUR LA PRÉPARATION DE COMPOSÉS DE PYRIDINIUM N-SUBSTITUÉS[2014/32]
Former [2012/23]VERFAHREN UND STOFFE ZUR HERSTELLUNG VON N-SUBSTITUIERTEN PYRIDINVERBINDUNGEN
Former [2012/23]PROCÉDÉS ET SUBSTANCES POUR LA PRÉPARATION DE COMPOSÉS DE PYRIDINIUM N-SUBSTITUÉS
Entry into regional phase27.02.2012National basic fee paid 
27.02.2012Designation fee(s) paid 
27.02.2012Examination fee paid 
Examination procedure27.02.2012Examination requested  [2012/23]
07.07.2014Communication of intention to grant the patent
03.11.2014Fee for grant paid
03.11.2014Fee for publishing/printing paid
03.11.2014Receipt of the translation of the claim(s)
Divisional application(s)The date of the Examining Division's first communication in respect of the earliest application for which a communication has been issued is  07.07.2014
Opposition(s)18.09.2015No opposition filed within time limit [2015/48]
Fees paidRenewal fee
10.07.2012Renewal fee patent year 03
08.07.2013Renewal fee patent year 04
08.07.2014Renewal fee patent year 05
Opt-out from the exclusive  Tooltip
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Patent Court		 See the Register of the Unified Patent Court for opt-out data
Responsibility for the accuracy, completeness or quality of the data displayed under the link provided lies entirely with the Unified Patent Court.
Lapses during opposition  TooltipHU23.07.2010
AL17.12.2014
BE17.12.2014
BG17.12.2014
CY17.12.2014
CZ17.12.2014
DK17.12.2014
EE17.12.2014
FI17.12.2014
HR17.12.2014
LT17.12.2014
LV17.12.2014
MC17.12.2014
MK17.12.2014
MT17.12.2014
NL17.12.2014
PL17.12.2014
PT17.12.2014
RO17.12.2014
SE17.12.2014
SI17.12.2014
SK17.12.2014
SM17.12.2014
TR17.12.2014
NO17.03.2015
GR18.03.2015
IS17.04.2015
IE23.07.2015
LU23.07.2015
[2018/46]
Former [2018/37]HU23.07.2010
BE17.12.2014
BG17.12.2014
CY17.12.2014
CZ17.12.2014
DK17.12.2014
EE17.12.2014
FI17.12.2014
HR17.12.2014
LT17.12.2014
LV17.12.2014
MC17.12.2014
MK17.12.2014
MT17.12.2014
NL17.12.2014
PL17.12.2014
PT17.12.2014
RO17.12.2014
SE17.12.2014
SI17.12.2014
SK17.12.2014
SM17.12.2014
TR17.12.2014
NO17.03.2015
GR18.03.2015
IS17.04.2015
IE23.07.2015
LU23.07.2015
Former [2018/30]HU23.07.2010
BE17.12.2014
BG17.12.2014
CY17.12.2014
CZ17.12.2014
DK17.12.2014
EE17.12.2014
FI17.12.2014
HR17.12.2014
LT17.12.2014
LV17.12.2014
MC17.12.2014
MK17.12.2014
MT17.12.2014
NL17.12.2014
PL17.12.2014
RO17.12.2014
SE17.12.2014
SI17.12.2014
SK17.12.2014
SM17.12.2014
TR17.12.2014
NO17.03.2015
GR18.03.2015
IS17.04.2015
IE23.07.2015
LU23.07.2015
Former [2017/38]HU23.07.2010
BE17.12.2014
BG17.12.2014
CY17.12.2014
CZ17.12.2014
DK17.12.2014
EE17.12.2014
FI17.12.2014
HR17.12.2014
LT17.12.2014
LV17.12.2014
MC17.12.2014
MT17.12.2014
NL17.12.2014
PL17.12.2014
RO17.12.2014
SE17.12.2014
SI17.12.2014
SK17.12.2014
SM17.12.2014
TR17.12.2014
NO17.03.2015
GR18.03.2015
IS17.04.2015
IE23.07.2015
LU23.07.2015
Former [2017/21]BE17.12.2014
CZ17.12.2014
DK17.12.2014
EE17.12.2014
FI17.12.2014
HR17.12.2014
LT17.12.2014
LV17.12.2014
MC17.12.2014
MT17.12.2014
NL17.12.2014
PL17.12.2014
RO17.12.2014
SE17.12.2014
SI17.12.2014
SK17.12.2014
NO17.03.2015
GR18.03.2015
IS17.04.2015
IE23.07.2015
LU23.07.2015
Former [2016/33]BE17.12.2014
CZ17.12.2014
DK17.12.2014
EE17.12.2014
FI17.12.2014
HR17.12.2014
LT17.12.2014
LV17.12.2014
MC17.12.2014
NL17.12.2014
PL17.12.2014
RO17.12.2014
SE17.12.2014
SI17.12.2014
SK17.12.2014
NO17.03.2015
GR18.03.2015
IS17.04.2015
IE23.07.2015
LU23.07.2015
Former [2016/24]BE17.12.2014
CZ17.12.2014
DK17.12.2014
EE17.12.2014
FI17.12.2014
HR17.12.2014
LT17.12.2014
LV17.12.2014
MC17.12.2014
NL17.12.2014
PL17.12.2014
RO17.12.2014
SE17.12.2014
SI17.12.2014
SK17.12.2014
NO17.03.2015
GR18.03.2015
IS17.04.2015
LU23.07.2015
Former [2016/15]CZ17.12.2014
DK17.12.2014
EE17.12.2014
FI17.12.2014
HR17.12.2014
LT17.12.2014
LV17.12.2014
MC17.12.2014
NL17.12.2014
PL17.12.2014
RO17.12.2014
SE17.12.2014
SI17.12.2014
SK17.12.2014
NO17.03.2015
GR18.03.2015
IS17.04.2015
LU23.07.2015
Former [2016/13]CZ17.12.2014
DK17.12.2014
EE17.12.2014
FI17.12.2014
HR17.12.2014
LT17.12.2014
LV17.12.2014
MC17.12.2014
NL17.12.2014
PL17.12.2014
RO17.12.2014
SE17.12.2014
SI17.12.2014
SK17.12.2014
NO17.03.2015
GR18.03.2015
IS17.04.2015
Former [2016/12]CZ17.12.2014
DK17.12.2014
EE17.12.2014
FI17.12.2014
HR17.12.2014
LT17.12.2014
LV17.12.2014
NL17.12.2014
PL17.12.2014
RO17.12.2014
SE17.12.2014
SI17.12.2014
SK17.12.2014
NO17.03.2015
GR18.03.2015
IS17.04.2015
Former [2015/50]CZ17.12.2014
DK17.12.2014
EE17.12.2014
FI17.12.2014
HR17.12.2014
LT17.12.2014
LV17.12.2014
NL17.12.2014
PL17.12.2014
RO17.12.2014
SE17.12.2014
SK17.12.2014
NO17.03.2015
GR18.03.2015
IS17.04.2015
Former [2015/38]CZ17.12.2014
EE17.12.2014
FI17.12.2014
HR17.12.2014
LT17.12.2014
LV17.12.2014
NL17.12.2014
PL17.12.2014
RO17.12.2014
SE17.12.2014
SK17.12.2014
NO17.03.2015
GR18.03.2015
IS17.04.2015
Former [2015/37]CZ17.12.2014
EE17.12.2014
FI17.12.2014
HR17.12.2014
LT17.12.2014
LV17.12.2014
NL17.12.2014
PL17.12.2014
RO17.12.2014
SE17.12.2014
SK17.12.2014
NO17.03.2015
GR18.03.2015
Former [2015/36]CZ17.12.2014
EE17.12.2014
FI17.12.2014
HR17.12.2014
LT17.12.2014
LV17.12.2014
NL17.12.2014
RO17.12.2014
SE17.12.2014
NO17.03.2015
GR18.03.2015
Former [2015/35]EE17.12.2014
FI17.12.2014
HR17.12.2014
LT17.12.2014
LV17.12.2014
NL17.12.2014
SE17.12.2014
NO17.03.2015
GR18.03.2015
Former [2015/29]FI17.12.2014
HR17.12.2014
LT17.12.2014
LV17.12.2014
NL17.12.2014
SE17.12.2014
NO17.03.2015
GR18.03.2015
Former [2015/24]FI17.12.2014
HR17.12.2014
LT17.12.2014
LV17.12.2014
SE17.12.2014
NO17.03.2015
GR18.03.2015
Former [2015/23]FI17.12.2014
LT17.12.2014
NO17.03.2015
Former [2015/21]LT17.12.2014
NO17.03.2015
Former [2015/20]LT17.12.2014
Cited inInternational search[AD]WO2007012494  (HOFFMANN LA ROCHE [CH], et al) [AD] 1,7,8,10,11 * example VII; figure 1 *;
 [A]  - N.R. CULLUM ET AL, J. CHEM. SOC., PERKIN TRANS. 2, (1996), pages 1559 - 1563, XP008113043 [A] 1 * the whole document *
 [A]  - D. WERNER ET AL, ARCHIV DER PHARMAZIE (WEINHEIM, GERMANY), (1974), vol. 307, no. 4, pages 301 - 308, XP002549392 [A] 12 * page 302, compound 8 *

DOI:   http://dx.doi.org/10.1002/ardp.19743070411
by applicantWO2007012494
 DE102006035020
 US4411995
 WO2008022966
 EP2023418
 US2009128882
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    - LIU, Y. ET AL., ORGANIC LETTERS, (2008), vol. 10, pages 765 - 768
The EPO accepts no responsibility for the accuracy of data originating from other authorities; in particular, it does not guarantee that it is complete, up to date or fit for specific purposes.