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Extract from the Register of European Patents

EP About this file: EP2509933

EP2509933 - KINETIC RESOLUTION [Right-click to bookmark this link]
StatusNo opposition filed within time limit
Status updated on  24.02.2017
Database last updated on 04.11.2024
Most recent event   Tooltip12.10.2018Lapse of the patent in a contracting state
New state(s): AL		published on 14.11.2018  [2018/46]
Applicant(s)For all designated states
The Provost, Fellows, Foundation Scholars, & the other members of Board, of the College of the Holy & Undiv. Trinity of Queen
College Green
Dublin 2 / IE
[2012/42]
Inventor(s)01 / CONNON, Stephen Joseph
11 Foxborough Park
Lucan
Dublin / IE
02 / PESCHIULLI, Aldo
Via Gallipoli 35
Racale
Lecce / IT
03 / PROCURANTI, Barbara
Viale Monzone 121-bis
Marina di Carrara / IT
 [2012/42]
Representative(s)Tomkins & Co
5 Dartmouth Road
Dublin 6 / IE
[N/P]
Former [2012/48]Lane, Cathal Michael, et al
Tomkins & Co. 5 Dartmouth Road
Dublin 6 / IE
Former [2012/42]McCooey, Seamus, et al
Tomkins & Co
5 Dartmouth Road
Dublin 6 / IE
Application number, filing date10787133.707.12.2010
[2016/16]
WO2010EP69097
Priority number, dateEP2009017856509.12.2009         Original published format: EP 09178565
[2012/42]
Filing languageEN
Procedural languageEN
PublicationType: A1 Application with search report
No.:WO2011070028
Date:16.06.2011
Language:EN
[2011/24]
Type: A1 Application with search report 
No.:EP2509933
Date:17.10.2012
Language:EN
The application published by WIPO in one of the EPO official languages on 16.06.2011 takes the place of the publication of the European patent application.
[2012/42]
Type: B1 Patent specification 
No.:EP2509933
Date:20.04.2016
Language:EN
[2016/16]
Search report(s)International search report - published on:EP16.06.2011
ClassificationIPC:C07B57/00, C07C227/32, C07C229/08, C07C231/18, C07C233/05, C07C319/02, C07C319/12, C07C319/28, C07C321/10, C07C323/07, C07C323/16, C07C327/22, C07C327/28, C07D453/04
[2015/40]
CPC:
C07C327/22 (EP,US); C07B57/00 (EP,US); C07C227/32 (EP,US);
C07C231/18 (EP,US); C07C233/05 (EP,US); C07C319/02 (EP,US);
C07C319/12 (EP,US); C07C319/28 (EP,US); C07C321/18 (EP,US);
C07C327/28 (EP,US); C07C51/083 (US); C07D453/04 (EP,US);
C07B2200/07 (EP,US) (-)
C-Set:
C07C227/32, C07C229/08 (US,EP);
C07C231/18, C07C233/05 (US,EP);
C07C319/02, C07C321/10 (US,EP);
C07C319/02, C07C323/07 (EP,US);
C07C319/02, C07C323/16 (EP,US);
C07C319/28, C07C321/10 (EP,US);
C07C319/28, C07C323/07 (EP,US);
C07C319/28, C07C323/16 (EP,US);
C07C321/18, C07C233/05 (US)
(-)
Former IPC [2012/42]C07B53/00, C07B57/00, C07C227/32, C07C229/08, C07C231/18, C07C233/05, C07C319/02, C07C319/12, C07C321/10, C07C323/07, C07C323/16, C07C327/22, C07C327/28, C07D453/04
Designated contracting statesAL,   AT,   BE,   BG,   CH,   CY,   CZ,   DE,   DK,   EE,   ES,   FI,   FR,   GB,   GR,   HR,   HU,   IE,   IS,   IT,   LI,   LT,   LU,   LV,   MC,   MK,   MT,   NL,   NO,   PL,   PT,   RO,   RS,   SE,   SI,   SK,   SM,   TR [2012/42]
Extension statesBANot yet paid
MENot yet paid
TitleGerman:KINETISCHE AUFLÖSUNG[2012/42]
English:KINETIC RESOLUTION[2012/42]
French:RÉSOLUTION CINÉTIQUE[2012/42]
Entry into regional phase18.06.2012National basic fee paid 
18.06.2012Designation fee(s) paid 
18.06.2012Examination fee paid 
Examination procedure18.06.2012Amendment by applicant (claims and/or description)
18.06.2012Examination requested  [2012/42]
28.06.2013Despatch of a communication from the examining division (Time limit: M04)
13.09.2013Reply to a communication from the examining division
02.02.2015Despatch of a communication from the examining division (Time limit: M04)
28.05.2015Reply to a communication from the examining division
02.10.2015Communication of intention to grant the patent
09.02.2016Fee for grant paid
09.02.2016Fee for publishing/printing paid
29.02.2016Information about intention to grant a patent
29.02.2016Receipt of the translation of the claim(s)
Divisional application(s)The date of the Examining Division's first communication in respect of the earliest application for which a communication has been issued is  28.06.2013
Opposition(s)23.01.2017No opposition filed within time limit [2017/13]
Fees paidRenewal fee
06.12.2012Renewal fee patent year 03
05.06.2014Renewal fee patent year 04
18.02.2015Renewal fee patent year 05
09.12.2015Renewal fee patent year 06
Penalty fee
Additional fee for renewal fee
31.12.201304   M06   Fee paid on   05.06.2014
31.12.201405   M06   Fee paid on   18.02.2015
Opt-out from the exclusive  Tooltip
competence of the Unified
Patent Court		 See the Register of the Unified Patent Court for opt-out data
Responsibility for the accuracy, completeness or quality of the data displayed under the link provided lies entirely with the Unified Patent Court.
Lapses during opposition  TooltipHU07.12.2010
AL20.04.2016
AT20.04.2016
BE20.04.2016
BG20.04.2016
CY20.04.2016
CZ20.04.2016
DK20.04.2016
EE20.04.2016
ES20.04.2016
FI20.04.2016
HR20.04.2016
IS20.04.2016
IT20.04.2016
LT20.04.2016
LV20.04.2016
MC20.04.2016
MK20.04.2016
NL20.04.2016
PL20.04.2016
RO20.04.2016
RS20.04.2016
SE20.04.2016
SI20.04.2016
SK20.04.2016
SM20.04.2016
TR20.04.2016
NO20.07.2016
GR21.07.2016
PT22.08.2016
IE07.12.2016
LU07.12.2016
MT07.12.2016
CH31.12.2016
LI31.12.2016
[2018/46]
Former [2018/43]HU07.12.2010
AT20.04.2016
BE20.04.2016
BG20.04.2016
CY20.04.2016
CZ20.04.2016
DK20.04.2016
EE20.04.2016
ES20.04.2016
FI20.04.2016
HR20.04.2016
IS20.04.2016
IT20.04.2016
LT20.04.2016
LV20.04.2016
MC20.04.2016
MK20.04.2016
NL20.04.2016
PL20.04.2016
RO20.04.2016
RS20.04.2016
SE20.04.2016
SI20.04.2016
SK20.04.2016
SM20.04.2016
TR20.04.2016
NO20.07.2016
GR21.07.2016
PT22.08.2016
IE07.12.2016
LU07.12.2016
MT07.12.2016
CH31.12.2016
LI31.12.2016
Former [2018/38]HU07.12.2010
AT20.04.2016
BE20.04.2016
BG20.04.2016
CY20.04.2016
CZ20.04.2016
DK20.04.2016
EE20.04.2016
ES20.04.2016
FI20.04.2016
HR20.04.2016
IS20.04.2016
IT20.04.2016
LT20.04.2016
LV20.04.2016
MC20.04.2016
MK20.04.2016
NL20.04.2016
PL20.04.2016
RO20.04.2016
RS20.04.2016
SE20.04.2016
SI20.04.2016
SK20.04.2016
SM20.04.2016
TR20.04.2016
NO20.07.2016
GR21.07.2016
PT22.08.2016
IE07.12.2016
LU07.12.2016
CH31.12.2016
LI31.12.2016
Former [2018/30]HU07.12.2010
AT20.04.2016
BE20.04.2016
CY20.04.2016
CZ20.04.2016
DK20.04.2016
EE20.04.2016
ES20.04.2016
FI20.04.2016
HR20.04.2016
IS20.04.2016
IT20.04.2016
LT20.04.2016
LV20.04.2016
MC20.04.2016
MK20.04.2016
NL20.04.2016
PL20.04.2016
RO20.04.2016
RS20.04.2016
SE20.04.2016
SI20.04.2016
SK20.04.2016
SM20.04.2016
TR20.04.2016
NO20.07.2016
GR21.07.2016
PT22.08.2016
IE07.12.2016
LU07.12.2016
CH31.12.2016
LI31.12.2016
Former [2018/29]HU07.12.2010
AT20.04.2016
BE20.04.2016
CY20.04.2016
CZ20.04.2016
DK20.04.2016
EE20.04.2016
ES20.04.2016
FI20.04.2016
HR20.04.2016
IT20.04.2016
LT20.04.2016
LV20.04.2016
MC20.04.2016
MK20.04.2016
NL20.04.2016
PL20.04.2016
RO20.04.2016
RS20.04.2016
SE20.04.2016
SI20.04.2016
SK20.04.2016
SM20.04.2016
TR20.04.2016
NO20.07.2016
GR21.07.2016
PT22.08.2016
IE07.12.2016
LU07.12.2016
CH31.12.2016
LI31.12.2016
Former [2018/28]HU07.12.2010
AT20.04.2016
BE20.04.2016
CY20.04.2016
CZ20.04.2016
DK20.04.2016
EE20.04.2016
ES20.04.2016
FI20.04.2016
HR20.04.2016
IT20.04.2016
LT20.04.2016
LV20.04.2016
MC20.04.2016
MK20.04.2016
NL20.04.2016
PL20.04.2016
RO20.04.2016
RS20.04.2016
SE20.04.2016
SI20.04.2016
SK20.04.2016
SM20.04.2016
NO20.07.2016
GR21.07.2016
PT22.08.2016
IE07.12.2016
LU07.12.2016
CH31.12.2016
LI31.12.2016
Former [2017/49]AT20.04.2016
BE20.04.2016
CZ20.04.2016
DK20.04.2016
EE20.04.2016
ES20.04.2016
FI20.04.2016
HR20.04.2016
IT20.04.2016
LT20.04.2016
LV20.04.2016
MC20.04.2016
NL20.04.2016
PL20.04.2016
RO20.04.2016
RS20.04.2016
SE20.04.2016
SI20.04.2016
SK20.04.2016
SM20.04.2016
NO20.07.2016
GR21.07.2016
PT22.08.2016
IE07.12.2016
LU07.12.2016
CH31.12.2016
LI31.12.2016
Former [2017/47]AT20.04.2016
BE20.04.2016
CZ20.04.2016
DK20.04.2016
EE20.04.2016
ES20.04.2016
FI20.04.2016
HR20.04.2016
IT20.04.2016
LT20.04.2016
LV20.04.2016
MC20.04.2016
NL20.04.2016
PL20.04.2016
RO20.04.2016
RS20.04.2016
SE20.04.2016
SI20.04.2016
SK20.04.2016
SM20.04.2016
NO20.07.2016
GR21.07.2016
PT22.08.2016
Former [2017/37]AT20.04.2016
BE20.04.2016
CZ20.04.2016
DK20.04.2016
EE20.04.2016
ES20.04.2016
FI20.04.2016
HR20.04.2016
IT20.04.2016
LT20.04.2016
LV20.04.2016
NL20.04.2016
PL20.04.2016
RO20.04.2016
RS20.04.2016
SE20.04.2016
SI20.04.2016
SK20.04.2016
SM20.04.2016
NO20.07.2016
GR21.07.2016
PT22.08.2016
Former [2017/11]AT20.04.2016
BE20.04.2016
CZ20.04.2016
DK20.04.2016
EE20.04.2016
ES20.04.2016
FI20.04.2016
HR20.04.2016
IT20.04.2016
LT20.04.2016
LV20.04.2016
NL20.04.2016
PL20.04.2016
RO20.04.2016
RS20.04.2016
SE20.04.2016
SK20.04.2016
SM20.04.2016
NO20.07.2016
GR21.07.2016
PT22.08.2016
Former [2017/10]AT20.04.2016
BE20.04.2016
CZ20.04.2016
DK20.04.2016
EE20.04.2016
ES20.04.2016
FI20.04.2016
HR20.04.2016
IT20.04.2016
LT20.04.2016
LV20.04.2016
NL20.04.2016
PL20.04.2016
RO20.04.2016
RS20.04.2016
SE20.04.2016
SK20.04.2016
NO20.07.2016
GR21.07.2016
PT22.08.2016
Former [2017/09]AT20.04.2016
BE20.04.2016
CZ20.04.2016
DK20.04.2016
EE20.04.2016
ES20.04.2016
FI20.04.2016
HR20.04.2016
IT20.04.2016
LT20.04.2016
LV20.04.2016
NL20.04.2016
PL20.04.2016
RO20.04.2016
RS20.04.2016
SE20.04.2016
NO20.07.2016
GR21.07.2016
PT22.08.2016
Former [2017/07]AT20.04.2016
BE20.04.2016
DK20.04.2016
ES20.04.2016
FI20.04.2016
HR20.04.2016
IT20.04.2016
LT20.04.2016
LV20.04.2016
NL20.04.2016
PL20.04.2016
RS20.04.2016
SE20.04.2016
NO20.07.2016
GR21.07.2016
PT22.08.2016
Former [2017/03]AT20.04.2016
BE20.04.2016
ES20.04.2016
FI20.04.2016
HR20.04.2016
IT20.04.2016
LT20.04.2016
LV20.04.2016
NL20.04.2016
PL20.04.2016
RS20.04.2016
SE20.04.2016
NO20.07.2016
GR21.07.2016
PT22.08.2016
Former [2016/52]AT20.04.2016
ES20.04.2016
FI20.04.2016
HR20.04.2016
LT20.04.2016
LV20.04.2016
NL20.04.2016
PL20.04.2016
RS20.04.2016
SE20.04.2016
NO20.07.2016
GR21.07.2016
PT22.08.2016
Former [2016/51]AT20.04.2016
ES20.04.2016
FI20.04.2016
HR20.04.2016
LT20.04.2016
LV20.04.2016
NL20.04.2016
PL20.04.2016
RS20.04.2016
NO20.07.2016
GR21.07.2016
PT22.08.2016
Former [2016/50]AT20.04.2016
ES20.04.2016
FI20.04.2016
HR20.04.2016
LT20.04.2016
LV20.04.2016
NL20.04.2016
PL20.04.2016
RS20.04.2016
NO20.07.2016
Former [2016/49]FI20.04.2016
LT20.04.2016
NL20.04.2016
PL20.04.2016
NO20.07.2016
Former [2016/46]LT20.04.2016
NO20.07.2016
Cited inInternational search[AD]WO2009050216  (DSM IP ASSETS BV [NL], et al) [AD] 1-15 * claims 1, 10, 12 *;
 [IA]  - T. HONJO, ET AL., "Highly enantioselective catalytic thiolysis of prochiral cyclic dicarboxylic anhydrides utilizing a bifunctional chiral sulphonamide", ANGEWANDTE CHEMIE, INTERNATIONAL EDITION, Wiley-VCH Verlag, Weinhem, DE, (20050904), vol. 44, no. 36, doi:10.1002/anie.200501408, ISSN 1433-7851, pages 5838 - 5841, XP002591780 [I] 13-15 * tables 1, 2 * [A] 1-12

DOI:   http://dx.doi.org/10.1002/anie.200501408
 [IA]  - A. PESCHIULLI, ET AL., "Organocatalytic asymmetric addition of alcohols and thiols to activated electrophiles: efficient dynamic kinetic resolution and desymmetrisation protocols", JOURNAL OF ORGANIC CHEMISTRY, American Chemical Society, Washington, DC, US, vol. 73, no. 16, doi:10.1021/jo801158g, ISSN 0022-3263, (20080723), pages 6409 - 6412, (20080723), XP002540122 [I] 13-15 * page 6411, column r, lines 9-16 * [A] 1-12

DOI:   http://dx.doi.org/10.1021/jo801158g
 [A]  - A.B. CHAVAN, ET AL., "An efficient process of racemisation of 3-(carbamoylmethyl)-5-methylhexanoic acid: a pregabalin intermediate", ORGANIC PROCESS RESEARCH AND DEVELOPMENT, American Chemical Society, Washington, DC, US, (20090518), vol. 13, no. 4, doi:10.1021/op900064x, ISSN 1083-6160, pages 812 - 814, XP002592726 [A] 9,10 * scheme 1 *

DOI:   http://dx.doi.org/10.1021/OP900064X
Examination   - A. PESCHIULLI, ET AL., "Synergistic organocatalysis in the kinetic resolution of secondary thiols with concomitant desymmetrisation of an anhydride", NATURE CHEMISTRY, Nature Publishng Group, GB, (20100501), vol. 2, no. 5, doi:10.1038/nchem.584, ISSN 1755-4330, pages 380 - 384, XP008124429

DOI:   http://dx.doi.org/10.1038/nchem.584
    - A. PESCHIULLI, ET AL., "Kinetic Resolution of Thiols", SYNFACTS, (20100622), vol. 2010, no. 07, doi:10.1055/s-0029-1220116, ISSN 1861-1958, pages 0825 - 0825, XP055158171

DOI:   http://dx.doi.org/10.1055/s-0029-1220116
by applicantWO2009050216
    - KAGAN, H. B.; FIAUD, J. C., "Kinetic resolution", TOP. STEREOCHEM., (1988), vol. 18, pages 249 - 330
    - IRWIN, A. J.; JONES, J. B., "Asymmetric syntheses via enantiotopically selective horse liver alcohol dehydrogenase catalyzed oxidations of diols containing a prochiral center", J. AM. CHEM. SOC., (1977), vol. 99, pages 556 - 561
The EPO accepts no responsibility for the accuracy of data originating from other authorities; in particular, it does not guarantee that it is complete, up to date or fit for specific purposes.