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Extract from the Register of European Patents

EP About this file: EP2516392

EP2516392 - SUBSTITUTED BENZAMIDE DERIVATIVES [Right-click to bookmark this link]
StatusThe application is deemed to be withdrawn
Status updated on  16.06.2017
Database last updated on 03.09.2024
FormerExamination is in progress
Status updated on  04.11.2016
Most recent event   Tooltip16.06.2017Application deemed to be withdrawnpublished on 19.07.2017  [2017/29]
Applicant(s)For all designated states
F. Hoffmann-La Roche AG
Grenzacherstrasse 124
4070 Basel / CH
[N/P]
Former [2012/44]For all designated states
F.Hoffmann-La Roche AG
Grenzacherstrasse 124
4070 Basel / CH
Inventor(s)01 / GROEBKE ZBINDEN, Katrin
Laubibergstrasse 61
CH-4410 Liestal / CH
02 / NORCROSS, Roger
Rheinfelderstrasse 2
CH-4305 Olsberg / CH
03 / PFLIEGER, Philippe
1 rue du Vignoble
F-68130 Schwoben / FR
 [2012/44]
Representative(s)Poppe, Regina
F.Hoffmann-La Roche AG
Patent Department
Grenzacherstrasse 124
4070 Basel / CH
[N/P]
Former [2012/44]Poppe, Regina
F.Hoffmann-La Roche AG Patent Department Grenzacherstrasse 124
4070 Basel / CH
Application number, filing date10793256.817.12.2010
WO2010EP70045
Priority number, dateEP2009018050422.12.2009         Original published format: EP 09180504
[2012/44]
Filing languageEN
Procedural languageEN
PublicationType: A1 Application with search report
No.:WO2011076678
Date:30.06.2011
Language:EN
[2011/26]
Type: A1 Application with search report 
No.:EP2516392
Date:31.10.2012
Language:EN
The application published by WIPO in one of the EPO official languages on 30.06.2011 takes the place of the publication of the European patent application.
[2012/44]
Search report(s)International search report - published on:EP30.06.2011
ClassificationIPC:C07D207/09, C07D207/10, C07D207/12, C07D211/26, C07D241/04, C07D265/30, C07D401/04, C07D401/12, C07D413/12, C07D413/14, C07D417/12, C07D417/14, A61K31/4025, A61K31/4523, A61K31/5355
[2012/44]
CPC:
C07D207/09 (EP,CN,US); C07D207/06 (KR); C07D413/14 (EP,CN,US);
A61K31/4025 (KR); A61K9/2018 (EP,US); A61P25/00 (EP);
A61P25/06 (EP); A61P25/08 (EP); A61P25/16 (EP);
A61P25/18 (EP); A61P25/20 (EP); A61P25/22 (EP);
A61P25/24 (EP); A61P25/28 (EP); A61P25/30 (EP);
A61P25/36 (EP); A61P3/00 (EP); A61P3/04 (EP);
A61P3/06 (EP); A61P3/10 (EP); A61P9/00 (EP);
A61P9/12 (EP); C07D207/10 (EP,CN,US); C07D207/12 (EP,CN,US);
C07D211/26 (EP,CN,US); C07D241/04 (EP,CN,US); C07D263/32 (EP,US);
C07D265/30 (EP,CN,US); C07D267/08 (EP,CN,US); C07D267/10 (EP,US);
C07D295/135 (EP,CN,US); C07D401/04 (EP,CN,US); C07D401/12 (EP,CN,KR,US);
C07D401/14 (EP,US); C07D403/12 (EP,US); C07D413/12 (EP,CN,US);
C07D417/12 (EP,CN,US); C07D417/14 (EP,CN,US); C07D495/04 (EP,US) (-)
Designated contracting statesAL,   AT,   BE,   BG,   CH,   CY,   CZ,   DE,   DK,   EE,   ES,   FI,   FR,   GB,   GR,   HR,   HU,   IE,   IS,   IT,   LI,   LT,   LU,   LV,   MC,   MK,   MT,   NL,   NO,   PL,   PT,   RO,   RS,   SE,   SI,   SK,   SM,   TR [2012/44]
TitleGerman:SUBSTITUIERTE BENZAMIDDERIVATE[2012/44]
English:SUBSTITUTED BENZAMIDE DERIVATIVES[2012/44]
French:DÉRIVÉS DE BENZAMIDE SUBSTITUÉS[2012/44]
Entry into regional phase23.07.2012National basic fee paid 
23.07.2012Designation fee(s) paid 
23.07.2012Examination fee paid 
Examination procedure19.08.2011Request for preliminary examination filed
International Preliminary Examining Authority: EP
23.07.2012Examination requested  [2012/44]
22.04.2014Despatch of a communication from the examining division (Time limit: M04)
18.07.2014Reply to a communication from the examining division
31.03.2015Despatch of a communication from the examining division (Time limit: M04)
20.05.2015Reply to a communication from the examining division
22.10.2015Despatch of a communication from the examining division (Time limit: M04)
07.01.2016Reply to a communication from the examining division
02.08.2016Despatch of a communication from the examining division (Time limit: M06)
14.02.2017Application deemed to be withdrawn, date of legal effect  [2017/29]
13.03.2017Despatch of communication that the application is deemed to be withdrawn, reason: reply to the communication from the examining division not received in time  [2017/29]
Divisional application(s)EP17151744.4  / EP3187490
The date of the Examining Division's first communication in respect of the earliest application for which a communication has been issued is  22.04.2014
Fees paidRenewal fee
07.12.2012Renewal fee patent year 03
06.12.2013Renewal fee patent year 04
05.12.2014Renewal fee patent year 05
07.12.2015Renewal fee patent year 06
08.12.2016Renewal fee patent year 07
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Cited inInternational search[X]DE2123246  ((BADI ) BADISCHE ANILIN & SODA FAB AG) [X] 1,10,15,21 * page 8; examples 20-23, 25 *;
 [X]US4636504  (ROSSY PHILLIP A [US], et al) [X] 1,12,15,16,18,21 * 6-{p-[3-(4-Phenyl-1-piperidino)-propionylamino]-phenyl}-5-methyl-4,5-dihydropyridazinone;; claim 7 *;
 [X]US6184242  (BLEY KEITH ROGER [US], et al) [X] 1,4,14,15,21 * 2,2,2-trifluoro-N-[4-(piperidin-4-ylmethyl)-phenyl]acetamide; column 58, line 15 - line 16 *;
 [X]US6444686  (KO SOO S [US], et al) [X] 1,2,15,16,18,21 * N-(2,5-Difluorophenyl)-N'-[[3-[[4-(phenylmethyl)-1-piperidinyl]methyl]phenyl]methyl]-urea; column 129; example 220 *;
 [X]WO2004039764  (BOEHRINGER INGELHEIM PHARMA [DE], et al) [X] 1,2,8,15-21 * abstract * * page 128 - page 129; example 31 * * page 161; example 137 * * page 185; example 169 *;
 [X]US2004157849  (LEE CHIH-HUNG [US], et al) [X] 1,10,15,16,18,21 * N-[4-(1-azepanyl)benzyl]-2-(5-isoquinolinyl)propanamide;; claim 55 *;
 [X]WO2006077425  (ASTEX THERAPEUTICS LTD [GB], et al) [X] 1,4,15,16,18,21 * page 202 - page 203; example 230 * * page 4 - page 5 *;
 [X]WO2007017728  (ORCHID RES LAB LTD [IN], et al) [X] 1,6,15,16,18,21 * page 31; compounds 50, 51 *;
 [X]WO2007064818  (TEVA PHARMA [IL], et al) [X] 1,6,15,21 * 4-(4-morpholinyl)-N-benzyloxycarbonylaniline; page 12 *;
 [A]US2009036420  (GALLEY GUIDO [DE], et al) [A] 1-21 * abstract * * claim 1 ** page 2, paragraph [0006] - paragraph [0026] *;
 [X]  - PERNER R J ET AL, "In vitro Structure-Activity Relationship and in vivo Characterization of 1-(Aryl)-3-(4-(amino)benzyl)urea transient Receptor Potential Vanilloid 1 Antagonists", JOURNAL OF MEDICINAL CHEMISTRY, AMERICAN CHEMICAL SOCIETY, WASHINGTON, US, vol. 50, no. 15, doi:DOI:10.1021/JM070276I, ISSN 0022-2623, (20070101), pages 3651 - 3660, (20070621), XP002591492 [X] 1,2,14-16,18,21 * page 3654; table 1; compounds 30-37, 39, 41 * * Scheme 1; page 3652 *

DOI:   http://dx.doi.org/10.1021/JM070276I
ExaminationUS4735959
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 US2007099919
 WO2008054702
 EP2009005
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 EP2401275
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