EP2424366 - PYRIDO [4, 3-B]INDOLES AND METHODS OF USE [Right-click to bookmark this link] | Status | No opposition filed within time limit Status updated on 23.12.2016 Database last updated on 03.09.2024 | Most recent event Tooltip | 20.07.2018 | Lapse of the patent in a contracting state New state(s): MT | published on 22.08.2018 [2018/34] | Applicant(s) | For all designated states Medivation Technologies, Inc. 525 Market Street, 36th Floor San Francisco, CA 94105 / US | [2013/32] |
Former [2012/10] | For all designated states Medivation Technologies, Inc. 201 Spear Street, 3rd Floor San Francisco, CA 94105 / US | Inventor(s) | 01 /
JAIN, Rajendra, Parasmal E-202 Sapphire Park Park Street Phase Ii Wakad, Pune Maharashtra 411 057 / IN | 02 /
CHAKRAVARTY, Sarvajit 1888 Miramonte Avenue Mountain View CA 94040 / US | [2012/10] | Representative(s) | Sexton, Jane Helen, et al J A Kemp 14 South Square Gray's Inn London WC1R 5JJ / GB | [2016/07] |
Former [2012/10] | Sexton, Jane Helen, et al J.A. Kemp & Co. 14 South Square Gray's Inn London WC1R 5JJ / GB | Application number, filing date | 10808471.6 | 29.04.2010 | [2016/07] | WO2010US33055 | Priority number, date | US20090181259P | 26.05.2009 Original published format: US 181259 P | IN2009MUM1135 | 29.04.2009 Original published format: IN MU11352009 | [2012/10] | Filing language | EN | Procedural language | EN | Publication | Type: | A1 Application with search report | No.: | WO2011019417 | Date: | 17.02.2011 | Language: | EN | [2011/07] | Type: | A1 Application with search report | No.: | EP2424366 | Date: | 07.03.2012 | Language: | EN | The application published by WIPO in one of the EPO official languages on 17.02.2011 takes the place of the publication of the European patent application. | [2012/10] | Type: | B1 Patent specification | No.: | EP2424366 | Date: | 17.02.2016 | Language: | EN | [2016/07] | Search report(s) | International search report - published on: | US | 17.02.2011 | (Supplementary) European search report - dispatched on: | EP | 16.11.2012 | Classification | IPC: | C07D471/04, A61P25/00, A61P25/28, A61K31/437 | [2012/51] | CPC: |
C07D471/04 (EP,US);
A61P21/02 (EP);
A61P21/04 (EP);
A61P25/00 (EP);
A61P25/14 (EP);
A61P25/16 (EP);
A61P25/18 (EP);
A61P25/22 (EP);
A61P25/24 (EP);
|
Former IPC [2012/10] | A01N43/42 | Designated contracting states | AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LI, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, SE, SI, SK, SM, TR [2012/10] | Extension states | AL | Not yet paid | BA | Not yet paid | ME | Not yet paid | RS | Not yet paid | Title | German: | PYRIDO-[4,3-B-]INDOLE UND VERWENDUNGSVERFAHREN DAFÜR | [2012/10] | English: | PYRIDO [4, 3-B]INDOLES AND METHODS OF USE | [2012/10] | French: | PYRIDO[4,3-B]INDOLES ET LEURS MÉTHODES D'UTILISATION | [2012/10] | Entry into regional phase | 10.11.2011 | National basic fee paid | 10.11.2011 | Search fee paid | 10.11.2011 | Designation fee(s) paid | 10.11.2011 | Examination fee paid | Examination procedure | 10.11.2011 | Examination requested [2012/10] | 24.07.2013 | Despatch of communication that the application is deemed to be withdrawn, reason: reply to the Extended European Search Report/Written Opinion of the International Searching Authority/International Preliminary Examination Report/Supplementary international search report not received in time | 02.10.2013 | Amendment by applicant (claims and/or description) | 05.11.2013 | Despatch of a communication from the examining division (Time limit: M06) | 14.05.2014 | Reply to a communication from the examining division | 15.04.2015 | Despatch of a communication from the examining division (Time limit: M02) | 17.04.2015 | Reply to a communication from the examining division | 22.07.2015 | Communication of intention to grant the patent | 25.11.2015 | Fee for grant paid | 25.11.2015 | Fee for publishing/printing paid | 14.12.2015 | Information about intention to grant a patent | 14.12.2015 | Receipt of the translation of the claim(s) | Divisional application(s) | The date of the Examining Division's first communication in respect of the earliest application for which a communication has been issued is 05.11.2013 | Opposition(s) | 18.11.2016 | No opposition filed within time limit [2017/04] | Request for further processing for: | The application is deemed to be withdrawn due to failure to reply to the Extended European Search Report/Written Opinion of the International Searching Authority/International Preliminary Examination Report/Supplementary international search report/Supplementary European search report | 02.10.2013 | Request for further processing filed | 02.10.2013 | Full payment received (date of receipt of payment) Request granted | 14.10.2013 | Decision despatched | Fees paid | Renewal fee | 26.07.2012 | Renewal fee patent year 03 | 26.03.2013 | Renewal fee patent year 04 | 26.03.2014 | Renewal fee patent year 05 | 08.04.2015 | Renewal fee patent year 06 | Penalty fee | Additional fee for renewal fee | 30.04.2012 | 03   M06   Fee paid on   26.07.2012 |
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Responsibility for the accuracy, completeness or quality of the data displayed under the link provided lies entirely with the Unified Patent Court. | Lapses during opposition Tooltip | HU | 29.04.2010 | AT | 17.02.2016 | BE | 17.02.2016 | CY | 17.02.2016 | CZ | 17.02.2016 | DK | 17.02.2016 | EE | 17.02.2016 | ES | 17.02.2016 | FI | 17.02.2016 | HR | 17.02.2016 | IS | 17.02.2016 | IT | 17.02.2016 | LT | 17.02.2016 | LV | 17.02.2016 | MC | 17.02.2016 | MK | 17.02.2016 | NL | 17.02.2016 | PL | 17.02.2016 | RO | 17.02.2016 | SE | 17.02.2016 | SI | 17.02.2016 | SK | 17.02.2016 | SM | 17.02.2016 | TR | 17.02.2016 | IE | 29.04.2016 | LU | 29.04.2016 | CH | 30.04.2016 | LI | 30.04.2016 | MT | 30.04.2016 | FR | 02.05.2016 | BG | 17.05.2016 | GB | 17.05.2016 | NO | 17.05.2016 | GR | 18.05.2016 | PT | 17.06.2016 | DE | 01.11.2016 | [2018/32] |
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GR | 18.05.2016 | Documents cited: | Search | [E]WO2010051501 (MEDIVATION TECHNOLOGIES INC [US], et al) [E] 1-4,12,22,23 * alpha,alpha-diphenyl-[1,2,3,4-tetrahydro-2,8-dimethyl-5H-pyrido[4,3-b]indole-5]-ethanol; alpha,alpha-diphenyl-[1,2,3,4-tetrahydro-2,8-dimethyl-5H-Pyrido[4,3-b]indole-5-]ethanol hydrochloride; alpha,alpha-diphenyl-[8-chloro-1,2,3,4-tetrahydro-2-methyl-H-pyrido[4,3-b]indole-5-]ethanol; alpha,alpha-diphenyl-[8-chloro-1,2,3,4-tetrahydro-2-methyl-H-pyrido[4,3-b]indole-5-]ethanol hydrochloride; alpha-[(4-fluorophenyl)-1,2,3,4-tetrahydro-2,8-dimethyl]-alpha-[phenyl]-5H-pyrido[4,3-b]indole-5-ethanol; alpha-[(4-fluorophenyl)-1,2,3,4-tetrahydro-2,8-dimethyl]-alpha-[phenyl]-5H-pyrido[4,3-b]indole-5-ethanol 2,2,2-trifluoroacetate;;; table 3; compounds 176,465, 466 * * 8-chloro-5-[2-chloro-2- (3-methyl- pyridin-4-yl)-propyl]-2-methyl-2,3,4,5-tetrahydro-lH-pyrido[4, 3-b]indole; page 380, line 4, paragraph 0770 * * Use in therapy of cognitive disorders ;;; claim 47 * * Pharmaceutical compositions :;; claim 49 * * Mode of action is 5-HT modulation :; page 10 *; | [IP]WO2009055828 (MEDIVATION TECHNOLOGIES INC [US], et al) [IP] 1-23 * compounds 44,110,116,122,125,381-384,447,480,512 * * Use in therapy of cognitive disorders :;; claim 13 * * Mode of action is 5-HT modulation :;; claim 12 *; | [A]WO2009038764 (D2E LLC [US], et al) [A] 1-23 * Compounds of type 5-[2-(pyridinyl)ethyl]-2,3,4,5-tetrahydro-2-methyl-1H-pyrido[4,3-b]indole :; page 25 - page 27; compounds 1 - 4-08 * * use for enhancing cognitive abilities :;; claim 20 * * Mode of action is 5-HT receptor modulation :;; claim 8 *; | [E]WO2010127177 (MEDIVATION TECHNOLOGIES INC [US], et al) [E] 1 * page 47; table 1; compounds 1-1 * * page 48; table 1; compounds 1-6 *; | [IP]WO2009082268 (ALLA CHEM LLC [US], et al) [IP] 1 * compounds of :;; claims 13,14 * | International search | [Y]WO2007087425 (MEDIVATION INC [US], et al); | [Y]WO2007016353 (SQUIBB BRISTOL MYERS CO [US], et al); | [Y] - DEZI, "Modeling of 5-HT2A and 5-HT2C Receptors and of Their Complexes with Actual and Potential Antipsychotic Drugs", PHD THESIS, BARCELONA, (2007), pages 1 - 239, XP008143584 | by applicant | US6187785 | US7071206 | WO2009055828 | WO2010051501 | WO2009038764 | WO2010012177 | WO2009082268 | WO2004US41081 | WO2007US20483 | WO2006US39077 | WO2008US77090 | WO2007US20516 | WO2007US22645 | WO2007US02117 | WO2008US06667 | WO2007US24626 | WO2008US09357 | WO2007US24623 | WO2008US08121 | WO2009US32065 | WO2009US38142 | US20080259234 |