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Extract from the Register of European Patents

EP About this file: EP2665722

EP2665722 - PROCESS FOR THE PREPARATION OF DIOL SULFONES [Right-click to bookmark this link]
StatusNo opposition filed within time limit
Status updated on  23.06.2017
Database last updated on 02.11.2024
Most recent event   Tooltip10.07.2020Lapse of the patent in a contracting state
New state(s): IS		published on 12.08.2020  [2020/33]
Applicant(s)For all designated states
DSM Sinochem Pharmaceuticals Netherlands B.V.
P.O.Box 245
Alexander Fleminglaan 1
2613 AX Delft / NL
[2013/48]
Inventor(s)01 / DE LANGE, Ben
P.O.Box 4
NL-6100 AA Echt / NL
02 / RIEBEL, Peter, Hans
P.O.Box 4
NL-6100 AA Echt / NL
03 / WOLBERG, Michael
P.O.Box 4
NL-6100 AA Echt / NL
04 / HEEMSKERK, Dennis
P.O.Box 4
NL-6100 AA Echt / NL
05 / MINK, Daniel
P.O.Box 4
NL-6100 AA Echt / NL
 [2013/48]
Representative(s)van Dam, Vincent, et al
Octrooibureau Vriesendorp & Gaade B.V.
Koninginnegracht 19
2514 AB Den Haag / NL
[N/P]
Former [2013/48]De Vroom, Erik
DSM Intellectual Property
P.O. Box 4
6100 AA Echt / NL
Application number, filing date12701093.213.01.2012
[2016/33]
WO2012EP50468
Priority number, dateEP2011015128018.01.2011         Original published format: EP 11151280
[2013/48]
Filing languageEN
Procedural languageEN
PublicationType: A1 Application with search report
No.:WO2012098048
Date:26.07.2012
Language:EN
[2012/30]
Type: A1 Application with search report 
No.:EP2665722
Date:27.11.2013
Language:EN
The application published by WIPO in one of the EPO official languages on 26.07.2012 takes the place of the publication of the European patent application.
[2013/48]
Type: B1 Patent specification 
No.:EP2665722
Date:17.08.2016
Language:EN
[2016/33]
Search report(s)International search report - published on:EP26.07.2012
ClassificationIPC:C07D405/12, C07D417/12, C07D413/12, C07D419/12
[2016/08]
CPC:
C07D417/12 (EP,US); C07D405/12 (EP,US); C07D413/12 (EP,US);
C07D419/12 (EP,US)
Former IPC [2013/48]C07D413/12, C07D419/12
Designated contracting statesAL,   AT,   BE,   BG,   CH,   CY,   CZ,   DE,   DK,   EE,   ES,   FI,   FR,   GB,   GR,   HR,   HU,   IE,   IS,   IT,   LI,   LT,   LU,   LV,   MC,   MK,   MT,   NL,   NO,   PL,   PT,   RO,   RS,   SE,   SI,   SK,   SM,   TR [2013/48]
Extension statesBANot yet paid
MENot yet paid
TitleGerman:VERFAHREN ZUR HERSTELLUNG VON DIOLSULFONEN[2013/48]
English:PROCESS FOR THE PREPARATION OF DIOL SULFONES[2013/48]
French:PROCÉDÉ POUR LA PRÉPARATION DE SULFONES DE DIOL[2013/48]
Entry into regional phase12.07.2013National basic fee paid 
12.07.2013Designation fee(s) paid 
12.07.2013Examination fee paid 
Examination procedure12.07.2013Examination requested  [2013/48]
27.02.2014Amendment by applicant (claims and/or description)
24.03.2014Observations by third parties
28.05.2014Despatch of a communication from the examining division (Time limit: M06)
13.11.2014Reply to a communication from the examining division
11.03.2015Despatch of a communication from the examining division (Time limit: M04)
14.04.2015Reply to a communication from the examining division
29.09.2015Despatch of a communication from the examining division (Time limit: M02)
20.11.2015Reply to a communication from the examining division
16.03.2016Communication of intention to grant the patent
23.06.2016Fee for grant paid
23.06.2016Fee for publishing/printing paid
23.06.2016Receipt of the translation of the claim(s)
Divisional application(s)The date of the Examining Division's first communication in respect of the earliest application for which a communication has been issued is  28.05.2014
Opposition(s)18.05.2017No opposition filed within time limit [2017/30]
Fees paidRenewal fee
21.01.2014Renewal fee patent year 03
13.01.2015Renewal fee patent year 04
11.01.2016Renewal fee patent year 05
Opt-out from the exclusive  Tooltip
competence of the Unified
Patent Court		 See the Register of the Unified Patent Court for opt-out data
Responsibility for the accuracy, completeness or quality of the data displayed under the link provided lies entirely with the Unified Patent Court.
Lapses during opposition  TooltipAL17.08.2016
AT17.08.2016
BE17.08.2016
CY17.08.2016
CZ17.08.2016
DK17.08.2016
EE17.08.2016
FI17.08.2016
HR17.08.2016
IT17.08.2016
LT17.08.2016
LV17.08.2016
MC17.08.2016
MK17.08.2016
NL17.08.2016
RO17.08.2016
RS17.08.2016
SE17.08.2016
SK17.08.2016
SM17.08.2016
TR17.08.2016
BG17.11.2016
NO17.11.2016
GR18.11.2016
IS17.12.2016
PT19.12.2016
IE13.01.2017
LU13.01.2017
CH31.01.2017
LI31.01.2017
[2020/33]
Former [2020/15]AL17.08.2016
AT17.08.2016
BE17.08.2016
CY17.08.2016
CZ17.08.2016
DK17.08.2016
EE17.08.2016
FI17.08.2016
HR17.08.2016
IT17.08.2016
LT17.08.2016
LV17.08.2016
MC17.08.2016
MK17.08.2016
NL17.08.2016
RO17.08.2016
RS17.08.2016
SE17.08.2016
SK17.08.2016
SM17.08.2016
TR17.08.2016
BG17.11.2016
NO17.11.2016
GR18.11.2016
PT19.12.2016
IE13.01.2017
LU13.01.2017
CH31.01.2017
LI31.01.2017
Former [2019/51]AL17.08.2016
AT17.08.2016
BE17.08.2016
CY17.08.2016
CZ17.08.2016
DK17.08.2016
EE17.08.2016
FI17.08.2016
HR17.08.2016
IT17.08.2016
LT17.08.2016
LV17.08.2016
MC17.08.2016
MK17.08.2016
NL17.08.2016
RO17.08.2016
RS17.08.2016
SE17.08.2016
SK17.08.2016
SM17.08.2016
BG17.11.2016
NO17.11.2016
GR18.11.2016
PT19.12.2016
IE13.01.2017
LU13.01.2017
CH31.01.2017
LI31.01.2017
Former [2019/46]AL17.08.2016
AT17.08.2016
BE17.08.2016
CY17.08.2016
CZ17.08.2016
DK17.08.2016
EE17.08.2016
FI17.08.2016
HR17.08.2016
IT17.08.2016
LT17.08.2016
LV17.08.2016
MC17.08.2016
NL17.08.2016
RO17.08.2016
RS17.08.2016
SE17.08.2016
SK17.08.2016
SM17.08.2016
BG17.11.2016
NO17.11.2016
GR18.11.2016
PT19.12.2016
IE13.01.2017
LU13.01.2017
CH31.01.2017
LI31.01.2017
Former [2018/46]AL17.08.2016
AT17.08.2016
BE17.08.2016
CZ17.08.2016
DK17.08.2016
EE17.08.2016
FI17.08.2016
HR17.08.2016
IT17.08.2016
LT17.08.2016
LV17.08.2016
MC17.08.2016
NL17.08.2016
RO17.08.2016
RS17.08.2016
SE17.08.2016
SK17.08.2016
SM17.08.2016
BG17.11.2016
NO17.11.2016
GR18.11.2016
PT19.12.2016
IE13.01.2017
LU13.01.2017
CH31.01.2017
LI31.01.2017
Former [2018/13]AT17.08.2016
BE17.08.2016
CZ17.08.2016
DK17.08.2016
EE17.08.2016
FI17.08.2016
HR17.08.2016
IT17.08.2016
LT17.08.2016
LV17.08.2016
MC17.08.2016
NL17.08.2016
RO17.08.2016
RS17.08.2016
SE17.08.2016
SK17.08.2016
SM17.08.2016
BG17.11.2016
NO17.11.2016
GR18.11.2016
PT19.12.2016
IE13.01.2017
LU13.01.2017
CH31.01.2017
LI31.01.2017
Former [2017/51]AT17.08.2016
BE17.08.2016
CZ17.08.2016
DK17.08.2016
EE17.08.2016
FI17.08.2016
HR17.08.2016
IT17.08.2016
LT17.08.2016
LV17.08.2016
MC17.08.2016
NL17.08.2016
RO17.08.2016
RS17.08.2016
SE17.08.2016
SK17.08.2016
SM17.08.2016
BG17.11.2016
NO17.11.2016
GR18.11.2016
PT19.12.2016
LU13.01.2017
CH31.01.2017
LI31.01.2017
Former [2017/47]AT17.08.2016
BE17.08.2016
CZ17.08.2016
DK17.08.2016
EE17.08.2016
FI17.08.2016
HR17.08.2016
IT17.08.2016
LT17.08.2016
LV17.08.2016
MC17.08.2016
NL17.08.2016
RO17.08.2016
RS17.08.2016
SE17.08.2016
SK17.08.2016
SM17.08.2016
BG17.11.2016
NO17.11.2016
GR18.11.2016
PT19.12.2016
Former [2017/32]AT17.08.2016
BE17.08.2016
CZ17.08.2016
DK17.08.2016
EE17.08.2016
FI17.08.2016
HR17.08.2016
IT17.08.2016
LT17.08.2016
LV17.08.2016
NL17.08.2016
RO17.08.2016
RS17.08.2016
SE17.08.2016
SK17.08.2016
SM17.08.2016
BG17.11.2016
NO17.11.2016
GR18.11.2016
PT19.12.2016
Former [2017/13]AT17.08.2016
FI17.08.2016
HR17.08.2016
IT17.08.2016
LT17.08.2016
LV17.08.2016
NL17.08.2016
RS17.08.2016
SE17.08.2016
NO17.11.2016
GR18.11.2016
PT19.12.2016
Former [2017/11]AT17.08.2016
FI17.08.2016
HR17.08.2016
IT17.08.2016
LT17.08.2016
NL17.08.2016
RS17.08.2016
SE17.08.2016
NO17.11.2016
GR18.11.2016
PT19.12.2016
Former [2017/10]FI17.08.2016
HR17.08.2016
IT17.08.2016
LT17.08.2016
NL17.08.2016
RS17.08.2016
SE17.08.2016
NO17.11.2016
Former [2017/09]FI17.08.2016
IT17.08.2016
LT17.08.2016
NL17.08.2016
NO17.11.2016
Former [2017/07]LT17.08.2016
Cited inInternational search[AD]WO02098854  (SQUIBB BRISTOL MYERS CO [US], et al) [AD] 1-10 * process of example 1, compounds B, C;; claims 1,4 *;
 [AD]WO0196311  (SQUIBB BRISTOL MYERS CO [US], et al) [AD] 1-10 * scheme 6;;; example 36 *
 [XAI]  - JORDI MUÑOZ-MURIEDAS ET AL, "Hydrophobic Molecular Similarity from MST Fractional Contributions to the Octanol/water Partition Coefficient", JOURNAL OF COMPUTER-AIDED MOLECULAR DESIGN, KLUWER ACADEMIC PUBLISHERS, DO, (20050601), vol. 19, no. 6, ISSN 1573-4951, pages 401 - 419, XP019248184 [X] 9 * table 1, compound 4 * [A] 1-8 [I] 10
 [XAI]  - HARRIS N V ET AL, "ACYL-COA:CHOLESTEROL O-ACYL TRANSFERASE (ACAT) INHIBITORS. 1. 2-(ALKYLTHIO)-4,5-DIPHENYL-1H-IMIDAZOLES AS POTENT INHIBITORS OF CAT", JOURNAL OF MEDICINAL CHEMISTRY, AMERICAN CHEMICAL SOCIETY, WASHINGTON, US, (19920101), vol. 35, doi:DOI:10.1021/JM00101A016, ISSN 0022-2623, pages 4384 - 4392, XP002027356 [X] 9 * table III, compound 48 * [A] 1-8 [I] 10

DOI:   http://dx.doi.org/10.1021/jm00101a016
ExaminationEP0414206
 WO2010086438
    - UEDA I ET AL, "Synthesis and Pharmacological properties of N-[3-{3(1-piperidinylmethyl)phenoxy}propyl]-2-(2-hydroxyethylthio)acetamide and related compounds as antiulcer agents", CHEMICAL AND PHARMACEUTICAL BULLETIN, PHARMACEUTICAL SOCIETY OF JAPAN, JP, (19901101), vol. 38, no. 1, ISSN 0009-2363, pages 3035 - 3041, XP002555584
    - UEDA I ET AL, Synthesis and Pharmacological properties of N-[3-{3(1-piperidinylmethyl)phenoxy}propyl]-2-(2-hydroxyethylthio)acetamide and related compounds as antiulcer agents, CHEMICAL AND PHARMACEUTICAL BULLETIN, PHARMACEUTICAL SOCIETY OF JAPAN, JP, PAGE(S) 3035 - 3041, (19901101), ISSN 0009-2363, XP002555584
by applicantWO02098854
 WO0196311
 EP1024139
 WO2010140765
 WO0206266
 WO03004459
 US6844437
 WO2007000121
    - P.R. BLAKEMORE, J. CHEM. SOC., PERKIN TRANS., (2002), vol. 1, page 2563
    - HOUBEN-WEYL, METHODEN DER ORGANISCHEN CHEMIE, (1960), vol. V/4, page 700
    - M. E. JUNG ET AL., J. ORG. CHEM., (1998), vol. 63, pages 347 - 355
    - D. G. BOURKE ET AL., AUST. J. CHEM., (1996), vol. 49, pages 425 - 434
    - W. E. WILLY ET AL., BULL. CHEM. SOC. JAPAN, (1976), vol. 49, pages 1989 - 1995
    - S. D. RYCHNOVSKY ET AL., J. ORG. CHEM., (1992), vol. 57, pages 1559 - 1563
    - M. KABEYA ET AL., TETRAHEDRON, (1997), vol. 53, pages 9777 - 9788
otherWO02098854
 WO2010086438
 WO2010140765
    - UEDA I. ET AL, "SYNTHESIS AND PHARMACOLOGICAL PROPERTIES OF N-[3-{3(1-PIPERIDINYLMETHYL)PHENOXY}PROPYL]-2-(2-HYDROXYETHYLTHIO)ACETAMIDE AND RELATED COMPOUNDS AS ANTIULCER AGENTS", CHEMICAL AND PHARMACEUTICAL BULLETIN, (19901101), vol. 38, no. 1, pages 3035 - 3041, XP002555584
The EPO accepts no responsibility for the accuracy of data originating from other authorities; in particular, it does not guarantee that it is complete, up to date or fit for specific purposes.