EP2675790 - SUBSTITUTED 1, 2, 3, 4-TETRAHYDROQUINOLIN-7-YL CARBAMATES AS ACETYLCHOLINESTERASE INHIBITORS FOR TREATMENT OF ALZHEIMER'S DISEASE [Right-click to bookmark this link] | Status | No opposition filed within time limit Status updated on 23.09.2016 Database last updated on 20.12.2024 | Most recent event Tooltip | 12.10.2018 | Lapse of the patent in a contracting state New state(s): AL | published on 14.11.2018 [2018/46] | Applicant(s) | For all designated states Council of Scientific & Industrial Research Anusandhan Bhawan Rafi Marg New Delhi 110 001 / IN | [2013/52] | Inventor(s) | 01 /
ROY, Kuldeep Kumar Central Drug Research Institute Chattar Manzil Palace Post Box No.173 Lucknow - 226001 / IN | 02 /
TOTA, Santoshkumar Central Drug Research Institute Chattar Manzil Palace Post Box No.173 Lucknow - 226001 / IN | 03 /
NATH, Chandishwar Central Drug Research Institute Chattar Manzil Palace Post Box No.173 Lucknow - 226001 / IN | 04 /
SHUKLA, Rakesh Central Drug Research Institute Chattar Manzil Palace Post Box No.173 Lucknow - 226001 / IN | 05 /
SAXENA, Anil Kumar Central Drug Research Institute Chattar Manzil Palace Post Box No.173 Lucknow - 226001 / IN | [2013/52] | Representative(s) | Fairbairn, Angus Chisholm, et al Marks & Clerk LLP 15 Fetter Lane London EC4A 1BW / GB | [N/P] |
Former [2015/47] | Robertson, James Alexander Marks & Clerk LLP 90 Long Acre London WC2E 9RA / GB | ||
Former [2013/52] | Robertson, James Alexander Marks & Clerk LLP 90 Long Acre London WC2E 9RA / GB | Application number, filing date | 12706943.3 | 24.01.2012 | [2015/47] | WO2012IN00053 | Priority number, date | IN2011DEL0363 | 14.02.2011 Original published format: IN DE03632011 | [2013/52] | Filing language | EN | Procedural language | EN | Publication | Type: | A1 Application with search report | No.: | WO2012111021 | Date: | 23.08.2012 | Language: | EN | [2012/34] | Type: | A1 Application with search report | No.: | EP2675790 | Date: | 25.12.2013 | Language: | EN | The application published by WIPO in one of the EPO official languages on 23.08.2012 takes the place of the publication of the European patent application. | [2013/52] | Type: | B1 Patent specification | No.: | EP2675790 | Date: | 18.11.2015 | Language: | EN | [2015/47] | Search report(s) | International search report - published on: | EP | 23.08.2012 | Classification | IPC: | C07D215/20, A61K31/47, A61P25/00 | [2013/52] | CPC: |
C07D215/20 (EP,US);
A61P25/00 (EP)
| Designated contracting states | AL, AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LI, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, RS, SE, SI, SK, SM, TR [2013/52] | Extension states | BA | Not yet paid | ME | Not yet paid | Title | German: | SUBSTITUIERTE 1,2,3,4-TETRAHYDROCHINOLIN-7-YL CARBAMATE VERWENDBAR ALS ACETYLCHOLINESTERASE INHIBOTOREN ZUR BEHANDLUNG DER ALZHEIMER ERKRANKUNG | [2015/19] | English: | SUBSTITUTED 1, 2, 3, 4-TETRAHYDROQUINOLIN-7-YL CARBAMATES AS ACETYLCHOLINESTERASE INHIBITORS FOR TREATMENT OF ALZHEIMER'S DISEASE | [2013/52] | French: | CARBAMATES DE 1,2,3,6-TETRAHYDROQUINOLEINES SUBSTITUÉS POUR LE TRAITEMENT DE LA MALADIE D'ALZHEIMER | [2015/19] |
Former [2013/52] | SUBSTITUIERTE 1, 2, 3, 4-TETRAHYDROCHINOLIN-7-YL CARBAMATE ALS ACETYLCHOLINESTERASEINHIBITOREN ZUR BEHANDLUNG VON MORBUS ALZHEIMER | ||
Former [2013/52] | 1,2,3,4-TÉTRAHYDROQUINOLÉIN-7-YLCARBAMATES SUBSTITUÉS EN TANT QU'INHIBITEURS D'ACÉTYLCHOLINESTÉRASE DANS LE TRAITEMENT DE LA MALADIE D'ALZHEIMER | Entry into regional phase | 12.08.2013 | National basic fee paid | 12.08.2013 | Designation fee(s) paid | 12.08.2013 | Examination fee paid | Examination procedure | 13.12.2012 | Request for preliminary examination filed International Preliminary Examining Authority: EP | 12.08.2013 | Examination requested [2013/52] | 28.03.2014 | Amendment by applicant (claims and/or description) | 31.10.2014 | Despatch of a communication from the examining division (Time limit: M04) | 10.03.2015 | Reply to a communication from the examining division | 20.05.2015 | Communication of intention to grant the patent | 30.09.2015 | Fee for grant paid | 30.09.2015 | Fee for publishing/printing paid | 30.09.2015 | Receipt of the translation of the claim(s) | Divisional application(s) | The date of the Examining Division's first communication in respect of the earliest application for which a communication has been issued is 31.10.2014 | Opposition(s) | 19.08.2016 | No opposition filed within time limit [2016/43] | Fees paid | Renewal fee | 24.01.2014 | Renewal fee patent year 03 | 20.01.2015 | Renewal fee patent year 04 |
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Responsibility for the accuracy, completeness or quality of the data displayed under the link provided lies entirely with the Unified Patent Court. | Lapses during opposition Tooltip | HU | 24.01.2012 | AL | 18.11.2015 | AT | 18.11.2015 | BE | 18.11.2015 | BG | 18.11.2015 | CY | 18.11.2015 | CZ | 18.11.2015 | DK | 18.11.2015 | EE | 18.11.2015 | ES | 18.11.2015 | FI | 18.11.2015 | HR | 18.11.2015 | IT | 18.11.2015 | LT | 18.11.2015 | LV | 18.11.2015 | MC | 18.11.2015 | MK | 18.11.2015 | NL | 18.11.2015 | PL | 18.11.2015 | RO | 18.11.2015 | RS | 18.11.2015 | SE | 18.11.2015 | SI | 18.11.2015 | SK | 18.11.2015 | SM | 18.11.2015 | TR | 18.11.2015 | IE | 24.01.2016 | LU | 24.01.2016 | CH | 31.01.2016 | LI | 31.01.2016 | MT | 31.01.2016 | NO | 18.02.2016 | GR | 19.02.2016 | IS | 18.03.2016 | PT | 18.03.2016 | [2018/46] |
Former [2018/38] | HU | 24.01.2012 | |
AT | 18.11.2015 | ||
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BG | 18.11.2015 | ||
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CZ | 18.11.2015 | ||
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IE | 24.01.2016 | ||
LU | 24.01.2016 | ||
CH | 31.01.2016 | ||
LI | 31.01.2016 | ||
MT | 31.01.2016 | ||
NO | 18.02.2016 | ||
GR | 19.02.2016 | ||
IS | 18.03.2016 | ||
PT | 18.03.2016 | ||
Former [2018/31] | HU | 24.01.2012 | |
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CZ | 18.11.2015 | ||
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EE | 18.11.2015 | ||
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SK | 18.11.2015 | ||
SM | 18.11.2015 | ||
TR | 18.11.2015 | ||
IE | 24.01.2016 | ||
LU | 24.01.2016 | ||
CH | 31.01.2016 | ||
LI | 31.01.2016 | ||
MT | 31.01.2016 | ||
NO | 18.02.2016 | ||
GR | 19.02.2016 | ||
IS | 18.03.2016 | ||
PT | 18.03.2016 | ||
Former [2018/29] | HU | 24.01.2012 | |
AT | 18.11.2015 | ||
BE | 18.11.2015 | ||
CY | 18.11.2015 | ||
CZ | 18.11.2015 | ||
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EE | 18.11.2015 | ||
ES | 18.11.2015 | ||
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RS | 18.11.2015 | ||
SE | 18.11.2015 | ||
SI | 18.11.2015 | ||
SK | 18.11.2015 | ||
SM | 18.11.2015 | ||
TR | 18.11.2015 | ||
IE | 24.01.2016 | ||
LU | 24.01.2016 | ||
CH | 31.01.2016 | ||
LI | 31.01.2016 | ||
NO | 18.02.2016 | ||
GR | 19.02.2016 | ||
IS | 18.03.2016 | ||
PT | 18.03.2016 | ||
Former [2018/28] | HU | 24.01.2012 | |
AT | 18.11.2015 | ||
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CZ | 18.11.2015 | ||
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EE | 18.11.2015 | ||
ES | 18.11.2015 | ||
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IT | 18.11.2015 | ||
LT | 18.11.2015 | ||
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PL | 18.11.2015 | ||
RO | 18.11.2015 | ||
RS | 18.11.2015 | ||
SE | 18.11.2015 | ||
SI | 18.11.2015 | ||
SK | 18.11.2015 | ||
SM | 18.11.2015 | ||
IE | 24.01.2016 | ||
LU | 24.01.2016 | ||
CH | 31.01.2016 | ||
LI | 31.01.2016 | ||
NO | 18.02.2016 | ||
GR | 19.02.2016 | ||
IS | 18.03.2016 | ||
PT | 18.03.2016 | ||
Former [2017/47] | AT | 18.11.2015 | |
BE | 18.11.2015 | ||
CZ | 18.11.2015 | ||
DK | 18.11.2015 | ||
EE | 18.11.2015 | ||
ES | 18.11.2015 | ||
FI | 18.11.2015 | ||
HR | 18.11.2015 | ||
IT | 18.11.2015 | ||
LT | 18.11.2015 | ||
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MC | 18.11.2015 | ||
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RO | 18.11.2015 | ||
RS | 18.11.2015 | ||
SE | 18.11.2015 | ||
SI | 18.11.2015 | ||
SK | 18.11.2015 | ||
SM | 18.11.2015 | ||
IE | 24.01.2016 | ||
LU | 24.01.2016 | ||
CH | 31.01.2016 | ||
LI | 31.01.2016 | ||
NO | 18.02.2016 | ||
GR | 19.02.2016 | ||
IS | 18.03.2016 | ||
PT | 18.03.2016 | ||
Former [2017/07] | AT | 18.11.2015 | |
BE | 18.11.2015 | ||
CZ | 18.11.2015 | ||
DK | 18.11.2015 | ||
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RS | 18.11.2015 | ||
SE | 18.11.2015 | ||
SI | 18.11.2015 | ||
SK | 18.11.2015 | ||
SM | 18.11.2015 | ||
IE | 24.01.2016 | ||
LU | 24.01.2016 | ||
CH | 31.01.2016 | ||
LI | 31.01.2016 | ||
NO | 18.02.2016 | ||
GR | 19.02.2016 | ||
IS | 18.03.2016 | ||
PT | 18.03.2016 | ||
Former [2017/03] | AT | 18.11.2015 | |
BE | 18.11.2015 | ||
CZ | 18.11.2015 | ||
DK | 18.11.2015 | ||
EE | 18.11.2015 | ||
ES | 18.11.2015 | ||
FI | 18.11.2015 | ||
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IT | 18.11.2015 | ||
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MC | 18.11.2015 | ||
NL | 18.11.2015 | ||
PL | 18.11.2015 | ||
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RS | 18.11.2015 | ||
SE | 18.11.2015 | ||
SI | 18.11.2015 | ||
SK | 18.11.2015 | ||
SM | 18.11.2015 | ||
LU | 24.01.2016 | ||
CH | 31.01.2016 | ||
LI | 31.01.2016 | ||
NO | 18.02.2016 | ||
GR | 19.02.2016 | ||
IS | 18.03.2016 | ||
PT | 18.03.2016 | ||
Former [2016/49] | AT | 18.11.2015 | |
CZ | 18.11.2015 | ||
DK | 18.11.2015 | ||
EE | 18.11.2015 | ||
ES | 18.11.2015 | ||
FI | 18.11.2015 | ||
HR | 18.11.2015 | ||
IT | 18.11.2015 | ||
LT | 18.11.2015 | ||
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MC | 18.11.2015 | ||
NL | 18.11.2015 | ||
PL | 18.11.2015 | ||
RO | 18.11.2015 | ||
RS | 18.11.2015 | ||
SE | 18.11.2015 | ||
SI | 18.11.2015 | ||
SK | 18.11.2015 | ||
SM | 18.11.2015 | ||
LU | 24.01.2016 | ||
BE | 31.01.2016 | ||
CH | 31.01.2016 | ||
LI | 31.01.2016 | ||
NO | 18.02.2016 | ||
GR | 19.02.2016 | ||
IS | 18.03.2016 | ||
PT | 18.03.2016 | ||
Former [2016/46] | AT | 18.11.2015 | |
CZ | 18.11.2015 | ||
DK | 18.11.2015 | ||
EE | 18.11.2015 | ||
ES | 18.11.2015 | ||
FI | 18.11.2015 | ||
HR | 18.11.2015 | ||
IT | 18.11.2015 | ||
LT | 18.11.2015 | ||
LV | 18.11.2015 | ||
MC | 18.11.2015 | ||
NL | 18.11.2015 | ||
PL | 18.11.2015 | ||
RO | 18.11.2015 | ||
RS | 18.11.2015 | ||
SE | 18.11.2015 | ||
SK | 18.11.2015 | ||
SM | 18.11.2015 | ||
LU | 24.01.2016 | ||
BE | 31.01.2016 | ||
CH | 31.01.2016 | ||
LI | 31.01.2016 | ||
NO | 18.02.2016 | ||
GR | 19.02.2016 | ||
IS | 18.03.2016 | ||
PT | 18.03.2016 | ||
Former [2016/42] | AT | 18.11.2015 | |
CZ | 18.11.2015 | ||
DK | 18.11.2015 | ||
EE | 18.11.2015 | ||
ES | 18.11.2015 | ||
FI | 18.11.2015 | ||
HR | 18.11.2015 | ||
IT | 18.11.2015 | ||
LT | 18.11.2015 | ||
LV | 18.11.2015 | ||
MC | 18.11.2015 | ||
NL | 18.11.2015 | ||
PL | 18.11.2015 | ||
RO | 18.11.2015 | ||
RS | 18.11.2015 | ||
SE | 18.11.2015 | ||
SK | 18.11.2015 | ||
SM | 18.11.2015 | ||
LU | 24.01.2016 | ||
BE | 31.01.2016 | ||
NO | 18.02.2016 | ||
GR | 19.02.2016 | ||
IS | 18.03.2016 | ||
PT | 18.03.2016 | ||
Former [2016/39] | AT | 18.11.2015 | |
CZ | 18.11.2015 | ||
DK | 18.11.2015 | ||
EE | 18.11.2015 | ||
ES | 18.11.2015 | ||
FI | 18.11.2015 | ||
HR | 18.11.2015 | ||
IT | 18.11.2015 | ||
LT | 18.11.2015 | ||
LV | 18.11.2015 | ||
NL | 18.11.2015 | ||
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RO | 18.11.2015 | ||
RS | 18.11.2015 | ||
SE | 18.11.2015 | ||
SK | 18.11.2015 | ||
SM | 18.11.2015 | ||
LU | 24.01.2016 | ||
BE | 31.01.2016 | ||
NO | 18.02.2016 | ||
GR | 19.02.2016 | ||
IS | 18.03.2016 | ||
PT | 18.03.2016 | ||
Former [2016/38] | AT | 18.11.2015 | |
CZ | 18.11.2015 | ||
EE | 18.11.2015 | ||
ES | 18.11.2015 | ||
FI | 18.11.2015 | ||
HR | 18.11.2015 | ||
IT | 18.11.2015 | ||
LT | 18.11.2015 | ||
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NL | 18.11.2015 | ||
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RO | 18.11.2015 | ||
RS | 18.11.2015 | ||
SE | 18.11.2015 | ||
SK | 18.11.2015 | ||
SM | 18.11.2015 | ||
BE | 31.01.2016 | ||
NO | 18.02.2016 | ||
GR | 19.02.2016 | ||
IS | 18.03.2016 | ||
PT | 18.03.2016 | ||
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ES | 18.11.2015 | ||
FI | 18.11.2015 | ||
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IT | 18.11.2015 | ||
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NL | 18.11.2015 | ||
PL | 18.11.2015 | ||
RO | 18.11.2015 | ||
RS | 18.11.2015 | ||
SE | 18.11.2015 | ||
SK | 18.11.2015 | ||
BE | 31.01.2016 | ||
NO | 18.02.2016 | ||
GR | 19.02.2016 | ||
IS | 18.03.2016 | ||
PT | 18.03.2016 | ||
Former [2016/34] | AT | 18.11.2015 | |
CZ | 18.11.2015 | ||
ES | 18.11.2015 | ||
FI | 18.11.2015 | ||
HR | 18.11.2015 | ||
IT | 18.11.2015 | ||
LT | 18.11.2015 | ||
LV | 18.11.2015 | ||
NL | 18.11.2015 | ||
PL | 18.11.2015 | ||
RS | 18.11.2015 | ||
SE | 18.11.2015 | ||
BE | 31.01.2016 | ||
NO | 18.02.2016 | ||
GR | 19.02.2016 | ||
IS | 18.03.2016 | ||
PT | 18.03.2016 | ||
Former [2016/25] | AT | 18.11.2015 | |
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PL | 18.11.2015 | ||
RS | 18.11.2015 | ||
SE | 18.11.2015 | ||
BE | 31.01.2016 | ||
NO | 18.02.2016 | ||
GR | 19.02.2016 | ||
IS | 18.03.2016 | ||
PT | 18.03.2016 | ||
Former [2016/24] | AT | 18.11.2015 | |
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IT | 18.11.2015 | ||
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BE | 31.01.2016 | ||
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IS | 18.03.2016 | ||
PT | 18.03.2016 | ||
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LT | 18.11.2015 | Cited in | International search | [ID]US2006142335 (SHAKYA NEERAJ [IN], et al) [ID] 1-22 * the whole document *; | [ID] - S.S. CHAUDHAERY ET AL, "Novel carbamates as orally active Acetylcholinesterase inhibitors", JOURNAL OF MEDICINAL CHEMISTRY, (American Chemical Society), (20100408), vol. 53 (2010), pages 6490 - 6505, XP002671625 [ID] 1-22 * the whole document * DOI: http://dx.doi.org/10.1021/JM100573Q | [X] - REGISTRY, CHEMICAL ABSTRACTS SERVICE, COLUMBUS, OHIO, US, (20041101), Database accession no. 773794-77-7, URL: STN, XP002671626 [X] 1,2,4,6 * abstract * | by applicant | US2009062279 | WO9708146 | WO2006070394 | US2006142335 | - MOUNT, C.; DOWNTON, C., NATURE MED., (2006), vol. 12, pages 780 - 784 | - KLAFKI, H. W. ET AL., BRAIN, (2006), vol. 129, pages 2840 - 2855 | - CHAUDHARY, S. S. ET AL., J. MED. CHEM., (2010), vol. 53, pages 6490 - 6505 | - MELNIKOVA, I., NAT. REV. DRUG DISCOVERY, (2007), vol. 6, pages 341 - 342 | - J. MED. CHEM., (2010), vol. 53, no. 17, pages 6490 - 6505 |