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EP About this file: EP2666777

EP2666777 - Certain chemical entities having an imidazo<4,5-b>pyrazin-2(3H)-one core, compositions and methods [Right-click to bookmark this link]
Status	The application is deemed to be withdrawn Status updated on 24.10.2014 Database last updated on 31.08.2024
Most recent event Tooltip	24.10.2014	Application deemed to be withdrawn	published on 26.11.2014 [2014/48]
Applicant(s)	For all designated states Cytokinetics, Inc. 280 East Grand Avenue South San Francisco, CA 94080 / US
	[2013/48]
Inventor(s)	01 / Muci, Alex 2025 Stockton Street, 3 San Francisco, CA California 94133 / US
	02 / Finer, Jeffrey T. 717 Gateshead Ct. Foster City, CA California 94404 / US
	03 / Lu, Pu-Ping 638 Pilgrim Drive Foster City, CA California 94404 / US
	04 / Russell, Alan James 44 Lundys Lane San Francsico, CA California 94110 / US
	05 / Morgan, Bradley P. 1206 Rimer Drive Moraga, CA California 94556 / US
	06 / Morgans, David J., Jr. 781 Vista Grande Avenue Los Altos, CA California 94024 / US
	[2013/48]
Representative(s)	Carpmaels & Ransford LLP One Southampton Row London WC1B 5HA / GB
	[2013/48]
Application number, filing date	13176575.2	01.08.2007
	[2013/48]
Priority number, date	US20060835272P	02.08.2006 Original published format: US 835272 P
	US20070921054P	30.03.2007 Original published format: US 921054 P
	[2013/48]
Filing language	EN
Procedural language	EN
Publication	Type:	A1 Application with search report
	No.:	EP2666777
	Date:	27.11.2013
	Language:	EN
	[2013/48]
Search report(s)	(Supplementary) European search report - dispatched on:	EP	24.10.2013
Classification	IPC:	C07D487/04, A61K31/498, A61P19/08, A61P21/04	[2013/48]
	CPC:	C07D487/04 (EP,KR,US); A61K31/498 (KR); A61P1/14 (EP); A61P11/00 (EP); A61P19/00 (EP); A61P19/08 (EP); (+) A61P21/00 (EP); A61P21/02 (EP); A61P21/04 (EP); A61P21/06 (EP); A61P25/00 (EP); A61P25/08 (EP); A61P3/00 (EP); A61P3/04 (EP); A61P35/00 (EP); A61P43/00 (EP) (-)
Designated contracting states	AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HU, IE, IS, IT, LI, LT, LU, LV, MC, MT, NL, PL, PT, RO, SE, SI, SK, TR [2013/48]
Extension states	AL	19.05.2014
	BA	19.05.2014
	HR	19.05.2014
	MK	19.05.2014
	RS	19.05.2014
Title	German:	Bestimmte chemische Stoffe mit eine imidazo<4,5-b>pyrazin-2(3H)-one Kernstruktur, Zusammensetzungen und Verfahren	[2013/48]
	English:	Certain chemical entities having an imidazo<4,5-b>pyrazin-2(3H)-one core, compositions and methods	[2013/48]
	French:	Certaines entités chimiques avec un noyeau imidazo<4,5-b>pyrazin-2(3H)-one, compositions et procédés	[2013/48]
Examination procedure	19.05.2014	Examination requested [2014/26]
	28.05.2014	Application deemed to be withdrawn, date of legal effect [2014/48]
	03.07.2014	Despatch of communication that the application is deemed to be withdrawn, reason: reply to the Extended European Search Report/Written Opinion of the International Searching Authority/International Preliminary Examination Report/Supplementary international search report not received in time [2014/48]
Parent application(s) Tooltip	EP07810993.1 / EP2069352
Fees paid	Renewal fee
	15.07.2013	Renewal fee patent year 03
	15.07.2013	Renewal fee patent year 04
	15.07.2013	Renewal fee patent year 05
	15.07.2013	Renewal fee patent year 06
	15.07.2013	Renewal fee patent year 07
	Penalty fee
	Additional fee for renewal fee
	31.08.2014	08 M06 Not yet paid
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	Responsibility for the accuracy, completeness or quality of the data displayed under the link provided lies entirely with the Unified Patent Court.
Documents cited:	Search	[X]JPH0641135 (NIPPON SODA CO) [X] 1,5 * page 3, paragraph 0004 - page 6, paragraph 0007; compounds 1-7 *;
		[X]WO2004092166 (MERCK & CO INC [US], et al) [X] 1-4,8,9 * page 142; example 159; claims 1-10, 18, 19 *;
		[X]WO2005013894 (MERCK & CO INC [US], et al) [X] 1-4,8,9 * page 52; example 5; claims 1-10, 18 *;
		[XP]WO2006088836 (SCHERING CORP [US], et al) [XP] 1,2,4,8,9 * page 44 - page 45; claims 1-44, 47, 48; compounds 22, 26, 27 *;
		[X] - SHIRAI, K.; FUKUNISHI, K.; YANAGISAWA, A.; TAKAHASHI, H.; MATSUOKA, M., "New Syntheses and Spectral Properties of Pteridine-related Heterocycles from 2,5-Diamino-3,6-dicyanopyrazine", JOURNAL OF HETEROCYCLIC CHEMISTRY, (2000), vol. 37, ISSN 0022-152X, pages 1151 - 1156, XP002592558 [X] 1,2 * Scheme 1; page 1152; compound 3a *
		[X] - ZHU ZHIJIAN ET AL, "Synthesis of Imidazo[4, 5-b]quinoxaline Ribonucleosides as Linear Dimensional Analogs of Antiviral Polyhalogenated Benzimidazole Ribonucleosides", JOURNAL OF THE CHINESE CHEMICAL SOCIETY, CHINESE ELECTRONIC PERIODICAL SERVICES, CHINA, (19980801), vol. 45, no. 4, ISSN 0009-4536, pages 465 - 474, XP009136216 [X] 1-5,8,9 * page 467, paragraph "Virological Procedure" "Cytotoxic Assays" - page 472; compounds 8a, 8b *
		[A] - IUPAC ED - ALAN D MCNAUGHT AND ANDREW WILKINSON, "cycloalkyl groups", ISBN 978-0-86542-684-9, (19970101), COMPENDIUM OF CHEMICAL TERMINOLOGY : IUPAC RECOMMENDATIONS; [IUPAC CHEMICAL DATA SERIES], BLACKWELL SCIENCE, OXFORD [U.A.], URL: http://www.iupac.org/goldbook/C01498.pdf, (19970101), XP002585006 [A] 1-13 * the whole document *
		[A] - IUPAC ED - ALAN D MCNAUGHT AND ANDREW WILKINSON, "alkyl groups", ISBN 978-0-86542-684-9, (19970101), COMPENDIUM OF CHEMICAL TERMINOLOGY : IUPAC RECOMMENDATIONS; [IUPAC CHEMICAL DATA SERIES], BLACKWELL SCIENCE, OXFORD [U.A.], URL: http://www.iupac.org/goldbook/A00228.pdf, (19970101), XP002585005 [A] 1-13 * the whole document *
		[A] - VITSE O ET AL, "New Imidazo(1,2-a)pyrazine Derivatives with Brochodilatory and Cyclic Nucleotide Phosphodiesterase Inhibitory Activities", BIOORGANIC & MEDICINAL CHEMISTRY, PERGAMON, GB LNKD- DOI:10.1016/S0968-0896(99)00019-X, (19990101), vol. 7, ISSN 0968-0896, pages 1059 - 1065, XP002257093 [A] 1-13 * the whole document * DOI: http://dx.doi.org/10.1016/S0968-0896(99)00019-X
		[A] - BONNET P A ET AL, "Synthesis and antibronchospastic activity of 8-alkoxy- and 8-(alkylamino)imidazo(1,2-a)pyrazines", JOURNAL OF MEDICINAL CHEMISTRY, AMERICAN CHEMICAL SOCIETY, WASHINGTON, US LNKD- DOI:10.1021/JM00096A008, (19920101), vol. 35, no. 18, ISSN 0022-2623, pages 3353 - 3358, XP002971280 [A] 1-13 * the whole document * DOI: http://dx.doi.org/10.1021/jm00096a008
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