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Extract from the Register of European Patents

EP About this file: EP2802592

EP2802592 - SUBSTITUTED ANNELLATED PYRIMIDINES AND TRIAZINES AND THEIR USE [Right-click to bookmark this link]
Former [2014/47]SUBSTITUTED ANNULATED PYRIMIDINES AND TRIAZINES, AND USE THEREOF
[2019/26]
StatusThe application has been withdrawn
Status updated on  05.12.2019
Database last updated on 25.09.2024
FormerGrant of patent is intended
Status updated on  05.11.2019
FormerExamination is in progress
Status updated on  11.10.2019
FormerGrant of patent is intended
Status updated on  07.07.2019
FormerExamination is in progress
Status updated on  11.11.2016
Most recent event   Tooltip05.12.2019Withdrawal of applicationpublished on 01.01.2020  [2020/01]
Applicant(s)For all designated states
Bayer Pharma Aktiengesellschaft
Müllerstrasse 178
13353 Berlin / DE
For all designated states
Bayer Intellectual Property GmbH
Alfred-Nobel-Str. 10
40789 Monheim am Rhein / DE
[2014/47]
Inventor(s)01 / FOLLMANN, Markus
Rosmarinweg 28
50859 Köln / DE
02 / STASCH, Johannes-Peter
Alfred-Nobel-Straße 109
42651 Solingen / DE
03 / REDLICH, Gorden
Schadowstraße 50
44799 Bochum / DE
04 / GRIEBENOW, Nils
Kurfürstenstr. 39
41541 Dormagen / DE
05 / LANG, Dieter
Wimmersberger Str.60
42553 Velbert / DE
06 / WUNDER, Frank
Schwarzer Weg 251
42117 Wuppertal / DE
07 / HÜBSCH, Walter
Wildsteig 22
42113 Wuppertal / DE
08 / TERSTEEGEN, Adrian
Rübezahlweg 8
42111 Wuppertal / DE
09 / VAKALOPOULOS, Alexandros
Heinrich-Heine-Str. 79a
40721 Hilden / DE
 [2014/47]
Representative(s)BIP Patents
c/o Bayer Intellectual Property GmbH
Alfred-Nobel-Straße 50
40789 Monheim am Rhein / DE
[N/P]
Former [2014/47]BIP Patents
c/o Bayer Intellectual Property GmbH
Creative Campus Monheim
Alfred-Nobel-Straße 10
40789 Monheim / DE
Application number, filing date13700288.710.01.2013
WO2013EP50381
Priority number, dateDE20121020034911.01.2012         Original published format: DE102012200349
[2014/47]
Filing languageDE
Procedural languageDE
PublicationType: A1 Application with search report
No.:WO2013104703
Date:18.07.2013
Language:DE
[2013/29]
Type: A1 Application with search report 
No.:EP2802592
Date:19.11.2014
Language:DE
The application published by WIPO in one of the EPO official languages on 18.07.2013 takes the place of the publication of the European patent application.
[2014/47]
Search report(s)International search report - published on:EP18.07.2013
ClassificationIPC:C07D519/00, A61K31/519, A61K31/53, A61P9/10, A61P9/12
[2014/47]
CPC:
C07D519/00 (EP,US); A61K31/519 (EP,US); A61K31/53 (EP,US);
A61K45/06 (US); A61P13/12 (EP); A61P7/02 (EP);
A61P9/00 (EP); A61P9/04 (EP); A61P9/10 (EP);
A61P9/12 (EP); C07D471/04 (EP,US) (-)
Designated contracting statesAL,   AT,   BE,   BG,   CH,   CY,   CZ,   DE,   DK,   EE,   ES,   FI,   FR,   GB,   GR,   HR,   HU,   IE,   IS,   IT,   LI,   LT,   LU,   LV,   MC,   MK,   MT,   NL,   NO,   PL,   PT,   RO,   RS,   SE,   SI,   SK,   SM,   TR [2014/47]
Extension statesBA11.08.2014
ME11.08.2014
TitleGerman:SUBSTITUIERTE ANNELLIERTE PYRIMIDINE UND TRIAZINE UND IHRE VERWENDUNG[2014/47]
English:SUBSTITUTED ANNELLATED PYRIMIDINES AND TRIAZINES AND THEIR USE[2019/47]
French:PYRIMIDINES ET TRIAZINES ANNELÉES SUBSTITUÉES ET LEUR UTILISATION[2014/47]
Former [2014/47]SUBSTITUTED ANNULATED PYRIMIDINES AND TRIAZINES, AND USE THEREOF
Entry into regional phase11.08.2014National basic fee paid 
11.08.2014Designation fee(s) paid 
11.08.2014Examination fee paid 
Examination procedure11.08.2014Examination requested  [2014/47]
26.02.2015Amendment by applicant (claims and/or description)
11.11.2016Despatch of a communication from the examining division (Time limit: M06)
10.05.2017Reply to a communication from the examining division
27.07.2017Despatch of a communication from the examining division (Time limit: M06)
28.12.2017Reply to a communication from the examining division
08.07.2019Communication of intention to grant the patent
10.10.2019Disapproval of the communication of intention to grant the patent by the applicant or resumption of examination proceedings by the EPO
06.11.2019Communication of intention to grant the patent
27.11.2019Application withdrawn by applicant  [2020/01]
Divisional application(s)The date of the Examining Division's first communication in respect of the earliest application for which a communication has been issued is  11.11.2016
Fees paidRenewal fee
13.01.2015Renewal fee patent year 03
11.01.2016Renewal fee patent year 04
11.01.2017Renewal fee patent year 05
15.01.2018Renewal fee patent year 06
15.01.2019Renewal fee patent year 07
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Responsibility for the accuracy, completeness or quality of the data displayed under the link provided lies entirely with the Unified Patent Court.
Cited inInternational search[AD]WO03095451  (BAYER AG [DE], et al) [AD] 1-15 * claim - *;
 [AD]WO2004009590  (BAYER HEALTHCARE AG [DE], et al) [AD] 1-15 * claim - *;
 [AD]WO2011149921  (MERCK SHARP & DOHME [US], et al) [AD] 1-15 * examples 58-84,158,161-164,168-170,173,174,176-187,189; claims 1-8,13-20; tables 9,10,12,13 *;
 [AD]WO2011147809  (BAYER PHARMA AG [DE], et al) [AD] 1-15 * claim - *;
 [XDP]WO2012004258  (BAYER PHARMA AG [DE], et al) [XDP] 1-7,9-15* examples 55A,56A,57A,58A,59A,73A,1-32; claim - *;
 [XDP]WO2012143510  (BAYER IP GMBH [DE], et al) [XDP] 1-7,9-15 * examples 20A, 21A, 34A,1-4,9,10; claim - *
by applicantUS4833246
 WO0006568
 WO0006569
 WO03095451
 WO2004009590
 WO2005073234
 WO2006130673
 WO2007041052
 WO2010065275
 WO2011014992
 WO2011149921
 WO2011147809
 WO2012004259
 WO2012004258
 WO2012028647
 WO2012143510
 WO2012152629
    - WU ET AL., BLOOD, (1994), vol. 84, page 4226
    - MÜLSCH ET AL., BRIT. J. PHARMACOL., (1997), vol. 120, page 681
    - STASCH J.-P. ET AL., NAT. REV. DRUG DISC., (2006), vol. 5, pages 755 - 768
    - STASCH J.-P. ET AL., CHEMMEDCHEM, (2009), vol. 4, pages 853 - 865
    - STASCH J.-P. ET AL., CIRCULATION, (2011), vol. 123, pages 2263 - 2273
    - OUDOUT ET AL., EUR. UROL., (2011), vol. 60, pages 1020 - 1026
    - E. M. BECKER ET AL., BMC PHARMACOLOGY, (2001), vol. 1, no. 13
    - HASSAN J. ET AL., CHEM. REV., vol. 102, pages 1359 - 1469
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    - F. WUNDER ET AL., ANAL. BIOCHEM., (2005), vol. 339, pages 104 - 112
    - KLAUS WITTE; KAI HU; JOHANNA SWIATEK; CLAUDIA MÜSSIG; GEORG ERTL; BJÖRN LEMMER, "Experimental heart failure in rats: effects on cardiovascular circadian rhythms and on myocardial ßadrenergic signaling", CARDIOVASC RES, (2000), vol. 47, no. 2, pages 203 - 405
    - KOZO OKAMOTO, "Spontaneous hypertension in rats", INT REV EXP PATHOL, (1969), vol. 7, pages 227 - 270
    - MAARTEN VAN DEN BUUSE, "Circadian Rhythms of Blood Pressure, Heart Rate, and Locomotor Activity in Spontaneously Hypertensive Rats as Measured With Radio-Telemetry", PHYSIOLOGY & BEHAVIOR, (1994), vol. 55, no. 4, pages 783 - 787
    - SHARKOVSKA Y; KALK P; LAWRENZ B; GODES M; HOFFMANN LS; WELLKISCH K; GESCHKA S; RELLE K; HOCHER B; STASCH JP, "NO-independent stimulation of soluble guanylate cyclase reduces target organ damage in low- and high-renin models of hypertension", J. HYPERTENSION, (2010), vol. 28, pages 1666 - 1675
The EPO accepts no responsibility for the accuracy of data originating from other authorities; in particular, it does not guarantee that it is complete, up to date or fit for specific purposes.