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Extract from the Register of European Patents

EP About this file: EP2838891

EP2838891 - AROMATIC RING COMPOUND AS GHRELIN O-ACYLTRANSFERASE INHIBITOR [Right-click to bookmark this link]
Former [2015/09]AROMATIC RING COMPOUND
[2016/43]
StatusNo opposition filed within time limit
Status updated on  08.06.2018
Database last updated on 13.07.2024
FormerThe patent has been granted
Status updated on  30.06.2017
FormerGrant of patent is intended
Status updated on  08.03.2017
FormerExamination is in progress
Status updated on  24.02.2017
Most recent event   Tooltip17.07.2020Lapse of the patent in a contracting state
New state(s): AL
published on 19.08.2020  [2020/34]
Applicant(s)For all designated states
Takeda Pharmaceutical Company Limited
1-1 Doshomachi 4-chome Chuo-ku
Osaka-shi, Osaka 541-0045 / JP
[2015/09]
Inventor(s)01 / TAKAKURA, Nobuyuki
c/o TAKEDA PHARMACEUTICAL COMPANY LIMITED
26-1 Muraoka-Higashi 2-chome
Fujisawa-shi Kanagawa 251-0012 / JP
02 / BANNO, Yoshihiro
c/o TAKEDA PHARMACEUTICAL COMPANY LIMITED
26-1 Muraoka-Higashi 2-chome
Fujisawa-shi Kanagawa 251-0012 / JP
03 / TERAO, Yoshito
c/o TAKEDA PHARMACEUTICAL COMPANY LIMITED
26-1 Muraoka-Higashi 2-chome
Fujisawa-shi Kanagawa 251-0012 / JP
04 / OCHIDA, Atsuko
c/o TAKEDA PHARMACEUTICAL COMPANY LIMITED
26-1 Muraoka-Higashi 2-chome
Fujisawa-shi Kanagawa 251-0012 / JP
05 / MORIMOTO, Sachie
c/o TAKEDA PHARMACEUTICAL COMPANY LIMITED
26-1 Muraoka-Higashi 2-chome
Fujisawa-shi Kanagawa 251-0012 / JP
06 / KITAMURA, Shuji
c/o TAKEDA PHARMACEUTICAL COMPANY LIMITED
26-1 Muraoka-Higashi 2-chome
Fujisawa-shi Kanagawa 251-0012 / JP
07 / TOMATA, Yoshihide
c/o TAKEDA PHARMACEUTICAL COMPANY LIMITED
26-1 Muraoka-Higashi 2-chome
Fujisawa-shi Kanagawa 251-0012 / JP
08 / YASUMA, Tsuneo
c/o TAKEDA PHARMACEUTICAL COMPANY LIMITED
17-85 Jusohonmachi 2-chome
Yodogawa-ku
Osaka-shi Osaka 532-0024 / JP
09 / IKOMA, Minoru
c/o TAKEDA PHARMACEUTICAL COMPANY LIMITED
26-1 Muraoka-Higashi 2-chome
Fujisawa-shi Kanagawa 251-0012 / JP
10 / MASUDA, Kei
c/o TAKEDA PHARMACEUTICAL COMPANY LIMITED
26-1 Muraoka-Higashi 2-chome
Fujisawa-shi Kanagawa 251-0012 / JP
 [2015/09]
Representative(s)Held, Stephan, et al
Meissner Bolte Patentanwälte
Rechtsanwälte Partnerschaft mbB
Widenmayerstraße 47
80538 München / DE
[2017/31]
Former [2015/09]Meissner, Bolte & Partner GbR
Widenmayerstrasse 47
80538 München / DE
Application number, filing date13710076.422.02.2013
[2017/31]
WO2013JP55605
Priority number, dateUS201261602888P24.02.2012         Original published format: US 201261602888 P
[2015/09]
Filing languageEN
Procedural languageEN
PublicationType: A1 Application with search report
No.:WO2013125732
Date:29.08.2013
Language:EN
[2013/35]
Type: A1 Application with search report 
No.:EP2838891
Date:25.02.2015
Language:EN
The application published by WIPO in one of the EPO official languages on 29.08.2013 takes the place of the publication of the European patent application.
[2015/09]
Type: B1 Patent specification 
No.:EP2838891
Date:02.08.2017
Language:EN
[2017/31]
Search report(s)International search report - published on:EP29.08.2013
ClassificationIPC:C07D333/60, C07D407/14, C07D417/12, C07D495/04, C07D307/82, A61K31/381, A61K31/343, A61K31/4355, A61K31/4365, A61P3/04
[2015/09]
CPC:
C07D333/60 (EP,CN,US); C07D333/54 (EP,CN,US); A61P1/16 (EP);
A61P21/00 (EP); A61P25/16 (EP); A61P25/28 (EP);
A61P25/32 (EP); A61P25/36 (EP); A61P3/04 (EP);
A61P3/06 (EP); A61P3/10 (EP); A61P35/00 (EP);
A61P43/00 (EP); A61P9/10 (EP); A61P9/12 (EP);
C07D307/79 (EP,CN,US); C07D307/80 (EP,CN,US); C07D307/81 (EP,CN,US);
C07D307/84 (EP,CN,US); C07D333/64 (EP,CN,US); C07D333/70 (EP,CN,US);
C07D405/04 (EP,CN,US); C07D405/12 (EP,CN,US); C07D409/06 (EP,CN,US);
C07D409/12 (EP,CN,US); C07D417/12 (EP,CN,US); C07D495/04 (EP,CN,US) (-)
Designated contracting statesAL,   AT,   BE,   BG,   CH,   CY,   CZ,   DE,   DK,   EE,   ES,   FI,   FR,   GB,   GR,   HR,   HU,   IE,   IS,   IT,   LI,   LT,   LU,   LV,   MC,   MK,   MT,   NL,   NO,   PL,   PT,   RO,   RS,   SE,   SI,   SK,   SM,   TR [2015/09]
Extension statesBANot yet paid
MENot yet paid
TitleGerman:AROMATISCHE RINGVERBINDUNG ALS GHRELIN O-ACYLTRANSFERASE HEMMER[2016/43]
English:AROMATIC RING COMPOUND AS GHRELIN O-ACYLTRANSFERASE INHIBITOR[2016/43]
French:COMPOSÉ À NOYAU AROMATIQUE COMME INHIBITEURS DE GHRéLINE O-ACYL TRANSFéRASE[2016/43]
Former [2015/09]AROMATISCHE RINGVERBINDUNG
Former [2015/09]AROMATIC RING COMPOUND
Former [2015/09]COMPOSÉ À NOYAU AROMATIQUE
Entry into regional phase20.08.2014National basic fee paid 
20.08.2014Designation fee(s) paid 
20.08.2014Examination fee paid 
Examination procedure20.08.2014Examination requested  [2015/09]
31.07.2015Amendment by applicant (claims and/or description)
15.10.2015Despatch of a communication from the examining division (Time limit: M04)
11.02.2016Reply to a communication from the examining division
29.02.2016Despatch of a communication from the examining division (Time limit: M04)
11.07.2016Reply to a communication from the examining division
11.10.2016Communication of intention to grant the patent
21.02.2017Disapproval of the communication of intention to grant the patent by the applicant or resumption of examination proceedings by the EPO
09.03.2017Communication of intention to grant the patent
26.06.2017Fee for grant paid
26.06.2017Fee for publishing/printing paid
26.06.2017Receipt of the translation of the claim(s)
Divisional application(s)The date of the Examining Division's first communication in respect of the earliest application for which a communication has been issued is  15.10.2015
Opposition(s)03.05.2018No opposition filed within time limit [2018/28]
Fees paidRenewal fee
26.02.2015Renewal fee patent year 03
26.02.2016Renewal fee patent year 04
27.02.2017Renewal fee patent year 05
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See the Register of the Unified Patent Court for opt-out data
Responsibility for the accuracy, completeness or quality of the data displayed under the link provided lies entirely with the Unified Patent Court.
Lapses during opposition  TooltipHU22.02.2013
AL02.08.2017
AT02.08.2017
CY02.08.2017
CZ02.08.2017
DK02.08.2017
EE02.08.2017
FI02.08.2017
HR02.08.2017
LT02.08.2017
LV02.08.2017
MC02.08.2017
MK02.08.2017
NL02.08.2017
PL02.08.2017
PT02.08.2017
RO02.08.2017
RS02.08.2017
SE02.08.2017
SI02.08.2017
SK02.08.2017
SM02.08.2017
TR02.08.2017
BG02.11.2017
NO02.11.2017
GR03.11.2017
IS02.12.2017
IE22.02.2018
LU22.02.2018
MT22.02.2018
BE28.02.2018
[2020/34]
Former [2020/31]HU22.02.2013
AT02.08.2017
CY02.08.2017
CZ02.08.2017
DK02.08.2017
EE02.08.2017
FI02.08.2017
HR02.08.2017
LT02.08.2017
LV02.08.2017
MC02.08.2017
MK02.08.2017
NL02.08.2017
PL02.08.2017
PT02.08.2017
RO02.08.2017
RS02.08.2017
SE02.08.2017
SI02.08.2017
SK02.08.2017
SM02.08.2017
TR02.08.2017
BG02.11.2017
NO02.11.2017
GR03.11.2017
IS02.12.2017
IE22.02.2018
LU22.02.2018
MT22.02.2018
BE28.02.2018
Former [2020/30]HU22.02.2013
AT02.08.2017
CZ02.08.2017
DK02.08.2017
EE02.08.2017
FI02.08.2017
HR02.08.2017
LT02.08.2017
LV02.08.2017
MC02.08.2017
NL02.08.2017
PL02.08.2017
PT02.08.2017
RO02.08.2017
RS02.08.2017
SE02.08.2017
SI02.08.2017
SK02.08.2017
SM02.08.2017
TR02.08.2017
BG02.11.2017
NO02.11.2017
GR03.11.2017
IS02.12.2017
IE22.02.2018
LU22.02.2018
MT22.02.2018
BE28.02.2018
Former [2020/28]AT02.08.2017
CZ02.08.2017
DK02.08.2017
EE02.08.2017
FI02.08.2017
HR02.08.2017
LT02.08.2017
LV02.08.2017
MC02.08.2017
NL02.08.2017
PL02.08.2017
PT02.08.2017
RO02.08.2017
RS02.08.2017
SE02.08.2017
SI02.08.2017
SK02.08.2017
SM02.08.2017
TR02.08.2017
BG02.11.2017
NO02.11.2017
GR03.11.2017
IS02.12.2017
IE22.02.2018
LU22.02.2018
MT22.02.2018
BE28.02.2018
Former [2020/15]AT02.08.2017
CZ02.08.2017
DK02.08.2017
EE02.08.2017
FI02.08.2017
HR02.08.2017
LT02.08.2017
LV02.08.2017
MC02.08.2017
NL02.08.2017
PL02.08.2017
RO02.08.2017
RS02.08.2017
SE02.08.2017
SI02.08.2017
SK02.08.2017
SM02.08.2017
TR02.08.2017
BG02.11.2017
NO02.11.2017
GR03.11.2017
IS02.12.2017
IE22.02.2018
LU22.02.2018
MT22.02.2018
BE28.02.2018
Former [2020/08]AT02.08.2017
CZ02.08.2017
DK02.08.2017
EE02.08.2017
FI02.08.2017
HR02.08.2017
LT02.08.2017
LV02.08.2017
MC02.08.2017
NL02.08.2017
PL02.08.2017
RO02.08.2017
RS02.08.2017
SE02.08.2017
SI02.08.2017
SK02.08.2017
SM02.08.2017
BG02.11.2017
NO02.11.2017
GR03.11.2017
IS02.12.2017
IE22.02.2018
LU22.02.2018
MT22.02.2018
BE28.02.2018
Former [2019/12]AT02.08.2017
CZ02.08.2017
DK02.08.2017
EE02.08.2017
FI02.08.2017
HR02.08.2017
LT02.08.2017
LV02.08.2017
MC02.08.2017
NL02.08.2017
PL02.08.2017
RO02.08.2017
RS02.08.2017
SE02.08.2017
SI02.08.2017
SK02.08.2017
SM02.08.2017
BG02.11.2017
NO02.11.2017
GR03.11.2017
IS02.12.2017
IE22.02.2018
LU22.02.2018
BE28.02.2018
Former [2019/09]AT02.08.2017
CZ02.08.2017
DK02.08.2017
EE02.08.2017
FI02.08.2017
HR02.08.2017
LT02.08.2017
LV02.08.2017
MC02.08.2017
NL02.08.2017
PL02.08.2017
RO02.08.2017
RS02.08.2017
SE02.08.2017
SI02.08.2017
SK02.08.2017
SM02.08.2017
BG02.11.2017
NO02.11.2017
GR03.11.2017
IS02.12.2017
IE22.02.2018
LU22.02.2018
Former [2018/52]AT02.08.2017
CZ02.08.2017
DK02.08.2017
EE02.08.2017
FI02.08.2017
HR02.08.2017
LT02.08.2017
LV02.08.2017
MC02.08.2017
NL02.08.2017
PL02.08.2017
RO02.08.2017
RS02.08.2017
SE02.08.2017
SI02.08.2017
SK02.08.2017
SM02.08.2017
BG02.11.2017
NO02.11.2017
GR03.11.2017
IS02.12.2017
LU22.02.2018
Former [2018/44]AT02.08.2017
CZ02.08.2017
DK02.08.2017
EE02.08.2017
FI02.08.2017
HR02.08.2017
LT02.08.2017
LV02.08.2017
MC02.08.2017
NL02.08.2017
PL02.08.2017
RO02.08.2017
RS02.08.2017
SE02.08.2017
SI02.08.2017
SK02.08.2017
SM02.08.2017
BG02.11.2017
NO02.11.2017
GR03.11.2017
IS02.12.2017
Former [2018/39]AT02.08.2017
CZ02.08.2017
DK02.08.2017
EE02.08.2017
FI02.08.2017
HR02.08.2017
LT02.08.2017
LV02.08.2017
NL02.08.2017
PL02.08.2017
RO02.08.2017
RS02.08.2017
SE02.08.2017
SI02.08.2017
SK02.08.2017
SM02.08.2017
BG02.11.2017
NO02.11.2017
GR03.11.2017
IS02.12.2017
Former [2018/25]AT02.08.2017
CZ02.08.2017
DK02.08.2017
EE02.08.2017
FI02.08.2017
HR02.08.2017
LT02.08.2017
LV02.08.2017
NL02.08.2017
PL02.08.2017
RO02.08.2017
RS02.08.2017
SE02.08.2017
SK02.08.2017
SM02.08.2017
BG02.11.2017
NO02.11.2017
GR03.11.2017
IS02.12.2017
Former [2018/21]AT02.08.2017
CZ02.08.2017
DK02.08.2017
FI02.08.2017
HR02.08.2017
LT02.08.2017
LV02.08.2017
NL02.08.2017
PL02.08.2017
RS02.08.2017
SE02.08.2017
BG02.11.2017
NO02.11.2017
GR03.11.2017
IS02.12.2017
Former [2018/12]AT02.08.2017
FI02.08.2017
HR02.08.2017
LT02.08.2017
LV02.08.2017
NL02.08.2017
PL02.08.2017
RS02.08.2017
SE02.08.2017
BG02.11.2017
NO02.11.2017
GR03.11.2017
IS02.12.2017
Former [2018/11]AT02.08.2017
FI02.08.2017
HR02.08.2017
LT02.08.2017
NL02.08.2017
PL02.08.2017
RS02.08.2017
SE02.08.2017
BG02.11.2017
NO02.11.2017
GR03.11.2017
IS02.12.2017
Former [2018/10]AT02.08.2017
FI02.08.2017
HR02.08.2017
LT02.08.2017
NL02.08.2017
RS02.08.2017
SE02.08.2017
NO02.11.2017
Former [2018/09]FI02.08.2017
LT02.08.2017
NL02.08.2017
SE02.08.2017
NO02.11.2017
Former [2018/08]FI02.08.2017
LT02.08.2017
NL02.08.2017
NO02.11.2017
Former [2018/07]LT02.08.2017
NO02.11.2017
Cited inInternational search[XD]WO2010143733  (TAKEDA PHARMACEUTICAL [JP], et al) [XD] 1-6 * claims 1,23; compound 233 *;
 [YD]EP1630152  (TAKEDA PHARMACEUTICAL [JP]) [YD] 1-6 * paragraph [0657]; examples 79,124,135,136,151-154 *;
 [AD]WO2008001931  (TAKEDA PHARMACEUTICAL [JP], et al) [AD] 1-6 * examples;; claims 1,16 *;
 [A]US2004209936  (BRATTON LARRY D [US], et al) [A] 1-6 * abstract *;
 [A]US2006014785  (ZHU YAN [US], et al) [A] 1-6 * examples 4A-44F,5; claims 51-68 *
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DOI:   http://dx.doi.org/10.1016/j.bmcl.2007.04.047
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The EPO accepts no responsibility for the accuracy of data originating from other authorities; in particular, it does not guarantee that it is complete, up to date or fit for specific purposes.