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Extract from the Register of European Patents

EP About this file: EP3041825

EP3041825 - PROCEDURE FOR THE SYNTHESIS OF N-BENZYL-N-CYCLOPROPYL-1H-PYRAZOLE-4-CARBOXAMIDE DERIVATIVES [Right-click to bookmark this link]
StatusNo opposition filed within time limit
Status updated on  17.01.2020
Database last updated on 01.01.2025
FormerThe patent has been granted
Status updated on  08.02.2019
FormerGrant of patent is intended
Status updated on  16.10.2018
Most recent event   Tooltip01.07.2022Lapse of the patent in a contracting state
New state(s): MK		published on 03.08.2022  [2022/31]
Applicant(s)For all designated states
Bayer CropScience Aktiengesellschaft
Alfred-Nobel-Strasse 50
40789 Monheim am Rhein / DE
[2016/28]
Inventor(s)01 / BRÜCHNER, Peter
Remberstrasse 86
47809 Krefeld / DE
02 / PAZENOK, Sergii
Wipperauerstrasse 57
42699 Solingen / DE
 [2016/28]
Representative(s)Guitton, Carole
Bayer S.A.S.
Patents & Licensing Department
14 Impasse Pierre Baizet
CS 99163
69263 Lyon Cedex 09 / FR
[2016/28]
Application number, filing date14758955.004.09.2014
[2016/28]
WO2014EP68838
Priority number, dateEP2013035601105.09.2013         Original published format: EP 13356011
[2016/28]
Filing languageEN
Procedural languageEN
PublicationType: A1 Application with search report
No.:WO2015032859
Date:12.03.2015
Language:EN
[2015/10]
Type: A1 Application with search report 
No.:EP3041825
Date:13.07.2016
Language:EN
The application published by WIPO in one of the EPO official languages on 12.03.2015 takes the place of the publication of the European patent application.
[2016/28]
Type: B1 Patent specification 
No.:EP3041825
Date:13.03.2019
Language:EN
[2019/11]
Search report(s)International search report - published on:EP12.03.2015
ClassificationIPC:C07D231/16, C07D231/14
[2018/44]
CPC:
C07D231/14 (EP,US); C07D231/16 (EP,US)
Former IPC [2016/28]C07D231/16
Designated contracting statesAL,   AT,   BE,   BG,   CH,   CY,   CZ,   DE,   DK,   EE,   ES,   FI,   FR,   GB,   GR,   HR,   HU,   IE,   IS,   IT,   LI,   LT,   LU,   LV,   MC,   MK,   MT,   NL,   NO,   PL,   PT,   RO,   RS,   SE,   SI,   SK,   SM,   TR [2016/28]
Extension statesBANot yet paid
MENot yet paid
TitleGerman:VERFAHREN ZUR SYNTHESE VON N-BENZYL-N-CYCLOPROPYL-1H-PYRAZOL-4-CARBOXAMID-DERIVATEN[2016/28]
English:PROCEDURE FOR THE SYNTHESIS OF N-BENZYL-N-CYCLOPROPYL-1H-PYRAZOLE-4-CARBOXAMIDE DERIVATIVES[2016/28]
French:PROCÉDÉ DE SYNTHÈSE DE DÉRIVÉS DE N-BENZYL-N-CYCLOPROPYLE-1H-PYRAZOLE-4-CARBOXAMIDE[2018/44]
Former [2016/28]PROCÉDÉ POUR LA SYNTHÈSE DE DÉRIVÉS DE N-BENZYL-N-CYCLOPROPYL-1H-PYRAZOLE-4-CARBOXAMIDE
Entry into regional phase05.04.2016National basic fee paid 
05.04.2016Designation fee(s) paid 
05.04.2016Examination fee paid 
Examination procedure05.04.2016Examination requested  [2016/28]
22.09.2016Amendment by applicant (claims and/or description)
17.10.2018Communication of intention to grant the patent
01.02.2019Fee for grant paid
01.02.2019Fee for publishing/printing paid
01.02.2019Receipt of the translation of the claim(s)
Opposition(s)16.12.2019No opposition filed within time limit [2020/08]
Fees paidRenewal fee
13.09.2016Renewal fee patent year 03
12.09.2017Renewal fee patent year 04
11.09.2018Renewal fee patent year 05
Opt-out from the exclusive  Tooltip
competence of the Unified
Patent Court		 See the Register of the Unified Patent Court for opt-out data
Responsibility for the accuracy, completeness or quality of the data displayed under the link provided lies entirely with the Unified Patent Court.
Lapses during opposition  TooltipHU04.09.2014
AL13.03.2019
CY13.03.2019
CZ13.03.2019
EE13.03.2019
HR13.03.2019
LT13.03.2019
LV13.03.2019
MC13.03.2019
MK13.03.2019
MT13.03.2019
PL13.03.2019
RO13.03.2019
RS13.03.2019
SE13.03.2019
SI13.03.2019
SK13.03.2019
SM13.03.2019
TR13.03.2019
BG13.06.2019
NO13.06.2019
GR14.06.2019
IS13.07.2019
PT13.07.2019
IE04.09.2019
LU04.09.2019
[2022/31]
Former [2021/34]HU04.09.2014
AL13.03.2019
CY13.03.2019
CZ13.03.2019
EE13.03.2019
HR13.03.2019
LT13.03.2019
LV13.03.2019
MC13.03.2019
MT13.03.2019
PL13.03.2019
RO13.03.2019
RS13.03.2019
SE13.03.2019
SI13.03.2019
SK13.03.2019
SM13.03.2019
TR13.03.2019
BG13.06.2019
NO13.06.2019
GR14.06.2019
IS13.07.2019
PT13.07.2019
IE04.09.2019
LU04.09.2019
Former [2021/32]HU04.09.2014
AL13.03.2019
CY13.03.2019
CZ13.03.2019
EE13.03.2019
HR13.03.2019
LT13.03.2019
LV13.03.2019
MC13.03.2019
PL13.03.2019
RO13.03.2019
RS13.03.2019
SE13.03.2019
SI13.03.2019
SK13.03.2019
SM13.03.2019
TR13.03.2019
BG13.06.2019
NO13.06.2019
GR14.06.2019
IS13.07.2019
PT13.07.2019
IE04.09.2019
LU04.09.2019
Former [2021/26]AL13.03.2019
CY13.03.2019
CZ13.03.2019
EE13.03.2019
HR13.03.2019
LT13.03.2019
LV13.03.2019
MC13.03.2019
PL13.03.2019
RO13.03.2019
RS13.03.2019
SE13.03.2019
SI13.03.2019
SK13.03.2019
SM13.03.2019
TR13.03.2019
BG13.06.2019
NO13.06.2019
GR14.06.2019
IS13.07.2019
PT13.07.2019
IE04.09.2019
LU04.09.2019
Former [2020/36]AL13.03.2019
CZ13.03.2019
EE13.03.2019
HR13.03.2019
LT13.03.2019
LV13.03.2019
MC13.03.2019
PL13.03.2019
RO13.03.2019
RS13.03.2019
SE13.03.2019
SI13.03.2019
SK13.03.2019
SM13.03.2019
TR13.03.2019
BG13.06.2019
NO13.06.2019
GR14.06.2019
IS13.07.2019
PT13.07.2019
IE04.09.2019
LU04.09.2019
Former [2020/35]AL13.03.2019
CZ13.03.2019
EE13.03.2019
HR13.03.2019
LT13.03.2019
LV13.03.2019
MC13.03.2019
PL13.03.2019
RO13.03.2019
RS13.03.2019
SE13.03.2019
SI13.03.2019
SK13.03.2019
SM13.03.2019
TR13.03.2019
BG13.06.2019
NO13.06.2019
GR14.06.2019
IS13.07.2019
PT13.07.2019
LU04.09.2019
Former [2020/25]AL13.03.2019
CZ13.03.2019
EE13.03.2019
HR13.03.2019
LT13.03.2019
LV13.03.2019
MC13.03.2019
PL13.03.2019
RO13.03.2019
RS13.03.2019
SE13.03.2019
SI13.03.2019
SK13.03.2019
SM13.03.2019
TR13.03.2019
BG13.06.2019
NO13.06.2019
GR14.06.2019
IS13.07.2019
PT13.07.2019
Former [2020/17]AL13.03.2019
CZ13.03.2019
EE13.03.2019
HR13.03.2019
LT13.03.2019
LV13.03.2019
PL13.03.2019
RO13.03.2019
RS13.03.2019
SE13.03.2019
SI13.03.2019
SK13.03.2019
SM13.03.2019
TR13.03.2019
BG13.06.2019
NO13.06.2019
GR14.06.2019
IS13.07.2019
PT13.07.2019
Former [2020/13]AL13.03.2019
CZ13.03.2019
EE13.03.2019
HR13.03.2019
LT13.03.2019
LV13.03.2019
PL13.03.2019
RO13.03.2019
RS13.03.2019
SE13.03.2019
SI13.03.2019
SK13.03.2019
SM13.03.2019
BG13.06.2019
NO13.06.2019
GR14.06.2019
IS13.07.2019
PT13.07.2019
Former [2020/04]AL13.03.2019
CZ13.03.2019
EE13.03.2019
HR13.03.2019
LT13.03.2019
LV13.03.2019
PL13.03.2019
RO13.03.2019
RS13.03.2019
SE13.03.2019
SK13.03.2019
SM13.03.2019
BG13.06.2019
NO13.06.2019
GR14.06.2019
IS13.07.2019
PT13.07.2019
Former [2019/52]AL13.03.2019
CZ13.03.2019
EE13.03.2019
HR13.03.2019
LT13.03.2019
LV13.03.2019
PL13.03.2019
RO13.03.2019
RS13.03.2019
SE13.03.2019
SK13.03.2019
SM13.03.2019
BG13.06.2019
NO13.06.2019
GR14.06.2019
PT13.07.2019
Former [2019/51]AL13.03.2019
CZ13.03.2019
EE13.03.2019
HR13.03.2019
LT13.03.2019
LV13.03.2019
RO13.03.2019
RS13.03.2019
SE13.03.2019
SK13.03.2019
SM13.03.2019
BG13.06.2019
NO13.06.2019
GR14.06.2019
PT13.07.2019
Former [2019/49]AL13.03.2019
CZ13.03.2019
EE13.03.2019
HR13.03.2019
LT13.03.2019
LV13.03.2019
RO13.03.2019
RS13.03.2019
SE13.03.2019
SK13.03.2019
BG13.06.2019
NO13.06.2019
GR14.06.2019
PT13.07.2019
Former [2019/48]HR13.03.2019
LT13.03.2019
LV13.03.2019
RS13.03.2019
SE13.03.2019
BG13.06.2019
NO13.06.2019
GR14.06.2019
PT13.07.2019
Former [2019/39]HR13.03.2019
LT13.03.2019
LV13.03.2019
RS13.03.2019
SE13.03.2019
BG13.06.2019
NO13.06.2019
GR14.06.2019
Former [2019/38]LT13.03.2019
SE13.03.2019
BG13.06.2019
NO13.06.2019
GR14.06.2019
Former [2019/37]LT13.03.2019
SE13.03.2019
NO13.06.2019
GR14.06.2019
Former [2019/34]LT13.03.2019
SE13.03.2019
NO13.06.2019
Former [2019/33]LT13.03.2019
NO13.06.2019
Cited inInternational search[YD]WO2010130767  (BAYER CROPSCIENCE AG [DE], et al) [YD] 1-12 * examples 1, 3; claims 1, 20 * * page 9, line 1 - page 10, line 6 * * page 11, lines 11-19 * * page 12, lines 6-14 *;
 [YD]  - SUBHASH CHANDRA GHOSH ET AL, "Iron-Catalyzed Efficient Synthesis of Amides from Aldehydes and Amine Hydrochloride Salts", ADVANCED SYNTHESIS & CATALYSIS, DE, (20120515), vol. 354, no. 8, doi:10.1002/adsc.201200020, ISSN 1615-4150, pages 1407 - 1412, XP055101856 [YD] 1-12 * the whole document *

DOI:   http://dx.doi.org/10.1002/adsc.201200020
 [YD]  - SUBHASH CHANDRA GHOSH ET AL, "Copper-Catalyzed Oxidative Amidation of Aldehydes with Amine Salts: Synthesis of Primary, Secondary, and Tertiary Amides", THE JOURNAL OF ORGANIC CHEMISTRY, US, (20120816), vol. 77, no. 18, doi:10.1021/jo301252c, ISSN 0022-3263, pages 8007 - 8015, XP055101861 [YD] 1-7,9-12 * the whole document *

DOI:   http://dx.doi.org/10.1021/jo301252c
 [Y]  - ISTVÁN E. MARKÓ ET AL, "Radical mediated oxidations in organic chemistry. 3. An efficient and versatile transformation of aldehydes into amides .", TETRAHEDRON LETTERS, GB, (1990), vol. 31, no. 49, doi:10.1016/S0040-4039(00)97289-7, ISSN 0040-4039, pages 7237 - 7240, XP055103614 [Y] 1-3,9,11 * the whole document *

DOI:   http://dx.doi.org/10.1016/S0040-4039(00)97289-7
 [Y]  - XIAOYING LIU ET AL, "Direct oxidative amidation of aromatic aldehydes using aqueous hydrogen peroxide in continuous flow microreactor systems", GREEN CHEMISTRY, GB, (20120313), vol. 14, no. 5, doi:10.1039/c2gc35078e, ISSN 1463-9262, pages 1471 - 1474, XP055102177 [Y] 1-3,9,11,12 * the whole document *

DOI:   http://dx.doi.org/10.1039/c2gc35078e
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