EP3087065 - SYNTHESIS OF UROLITHINS [Right-click to bookmark this link] | |||
Former [2016/44] | PROCESS-SCALE SYNTHESIS OF UROLITHINS | ||
[2019/09] | Status | No opposition filed within time limit Status updated on 27.11.2020 Database last updated on 03.09.2024 | |
Former | The patent has been granted Status updated on 20.12.2019 | ||
Former | Grant of patent is intended Status updated on 03.08.2019 | ||
Former | Examination is in progress Status updated on 24.07.2019 | ||
Former | Grant of patent is intended Status updated on 11.03.2019 | ||
Former | Examination is in progress Status updated on 06.04.2018 | Most recent event Tooltip | 08.07.2022 | Lapse of the patent in a contracting state New state(s): MK | published on 10.08.2022 [2022/32] | Applicant(s) | For all designated states Amazentis SA EPFL Innovation Park Bâtiment C 1015 Lausanne / CH | [2018/25] |
Former [2016/44] | For all designated states Amazentis SA Parc Scientifique Epfl Pse-c 1024 Ecublens / CH | Inventor(s) | 01 /
RINSCH, Christopher, L. 60 Rue de Lausanne CH-1110 Morges / CH | 02 /
MÜLLER, Roland Schwaneplatz 2 93047 Regensburg / DE | 03 /
SKRANC, Wolfgang Oberfeldgasse 23 A-1220 Vienna / AT | [2016/44] | Representative(s) | Abel & Imray LLP Westpoint Building James Street West Bath BA1 2DA / GB | [N/P] |
Former [2020/04] | Abel & Imray Westpoint Building James Street West Bath BA1 2DA / GB | ||
Former [2016/44] | Trueman, Lucy Petra Barker Brettell LLP 100 Hagley Road Edgbaston Birmingham B16 8QQ / GB | Application number, filing date | 14828105.8 | 22.12.2014 | [2016/44] | WO2014US71824 | Priority number, date | US201361919923P | 23.12.2013 Original published format: US 201361919923 P | [2016/44] | Filing language | EN | Procedural language | EN | Publication | Type: | A2 Application without search report | No.: | WO2015100213 | Date: | 02.07.2015 | Language: | EN | [2015/26] | Type: | A2 Application without search report | No.: | EP3087065 | Date: | 02.11.2016 | Language: | EN | The application published by WIPO in one of the EPO official languages on 02.07.2015 takes the place of the publication of the European patent application. | [2016/44] | Type: | B1 Patent specification | No.: | EP3087065 | Date: | 22.01.2020 | Language: | EN | [2020/04] | Search report(s) | International search report - published on: | EP | 17.09.2015 | Classification | IPC: | C07D311/80 | [2016/44] | CPC: |
C07D311/80 (EP,US);
A61K31/366 (EP,US);
A61K33/34 (US)
| Designated contracting states | AL, AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LI, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, RS, SE, SI, SK, SM, TR [2016/44] | Extension states | BA | Not yet paid | ME | Not yet paid | Title | German: | SYNTHESE VON UROLITHINEN | [2019/09] | English: | SYNTHESIS OF UROLITHINS | [2019/09] | French: | SYNTHESE D'UROLITHINES | [2019/09] |
Former [2016/44] | PROZESSSKALIGE SYNTHESE VON UROLITHINEN | ||
Former [2016/44] | PROCESS-SCALE SYNTHESIS OF UROLITHINS | ||
Former [2016/44] | SYNTHESE D'UROLITHINES A ECHELLE DE PROCEDE | Entry into regional phase | 18.07.2016 | National basic fee paid | 18.07.2016 | Designation fee(s) paid | 18.07.2016 | Examination fee paid | Examination procedure | 18.07.2016 | Amendment by applicant (claims and/or description) | 18.07.2016 | Examination requested [2016/44] | 06.04.2018 | Despatch of a communication from the examining division (Time limit: M04) | 27.07.2018 | Reply to a communication from the examining division | 12.03.2019 | Communication of intention to grant the patent | 22.07.2019 | Disapproval of the communication of intention to grant the patent by the applicant or resumption of examination proceedings by the EPO | 22.07.2019 | Fee for grant paid | 22.07.2019 | Fee for publishing/printing paid | 12.08.2019 | Communication of intention to grant the patent | 06.12.2019 | Receipt of the translation of the claim(s) | Divisional application(s) | EP20152975.7 / EP3663287 | Opposition(s) | 23.10.2020 | No opposition filed within time limit [2020/53] | Fees paid | Renewal fee | 13.12.2016 | Renewal fee patent year 03 | 12.12.2017 | Renewal fee patent year 04 | 12.12.2018 | Renewal fee patent year 05 | 13.12.2019 | Renewal fee patent year 06 |
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Responsibility for the accuracy, completeness or quality of the data displayed under the link provided lies entirely with the Unified Patent Court. | Lapses during opposition Tooltip | HU | 22.12.2014 | AL | 22.01.2020 | CY | 22.01.2020 | CZ | 22.01.2020 | DK | 22.01.2020 | EE | 22.01.2020 | ES | 22.01.2020 | FI | 22.01.2020 | HR | 22.01.2020 | LT | 22.01.2020 | LV | 22.01.2020 | MC | 22.01.2020 | MK | 22.01.2020 | MT | 22.01.2020 | PL | 22.01.2020 | RO | 22.01.2020 | RS | 22.01.2020 | SI | 22.01.2020 | SK | 22.01.2020 | SM | 22.01.2020 | TR | 22.01.2020 | BG | 22.04.2020 | NO | 22.04.2020 | GR | 23.04.2020 | IS | 22.05.2020 | PT | 14.06.2020 | [2022/31] |
Former [2022/30] | HU | 22.12.2014 | |
AL | 22.01.2020 | ||
CY | 22.01.2020 | ||
CZ | 22.01.2020 | ||
DK | 22.01.2020 | ||
EE | 22.01.2020 | ||
ES | 22.01.2020 | ||
FI | 22.01.2020 | ||
HR | 22.01.2020 | ||
LT | 22.01.2020 | ||
LV | 22.01.2020 | ||
MC | 22.01.2020 | ||
MT | 22.01.2020 | ||
PL | 22.01.2020 | ||
RO | 22.01.2020 | ||
RS | 22.01.2020 | ||
SI | 22.01.2020 | ||
SK | 22.01.2020 | ||
SM | 22.01.2020 | ||
TR | 22.01.2020 | ||
BG | 22.04.2020 | ||
NO | 22.04.2020 | ||
GR | 23.04.2020 | ||
IS | 22.05.2020 | ||
PT | 14.06.2020 | ||
Former [2022/27] | HU | 22.12.2014 | |
CY | 22.01.2020 | ||
CZ | 22.01.2020 | ||
DK | 22.01.2020 | ||
EE | 22.01.2020 | ||
ES | 22.01.2020 | ||
FI | 22.01.2020 | ||
HR | 22.01.2020 | ||
LT | 22.01.2020 | ||
LV | 22.01.2020 | ||
MC | 22.01.2020 | ||
MT | 22.01.2020 | ||
PL | 22.01.2020 | ||
RO | 22.01.2020 | ||
RS | 22.01.2020 | ||
SI | 22.01.2020 | ||
SK | 22.01.2020 | ||
SM | 22.01.2020 | ||
TR | 22.01.2020 | ||
BG | 22.04.2020 | ||
NO | 22.04.2020 | ||
GR | 23.04.2020 | ||
IS | 22.05.2020 | ||
PT | 14.06.2020 | ||
Former [2021/40] | CZ | 22.01.2020 | |
DK | 22.01.2020 | ||
EE | 22.01.2020 | ||
ES | 22.01.2020 | ||
FI | 22.01.2020 | ||
HR | 22.01.2020 | ||
LT | 22.01.2020 | ||
LV | 22.01.2020 | ||
MC | 22.01.2020 | ||
PL | 22.01.2020 | ||
RO | 22.01.2020 | ||
RS | 22.01.2020 | ||
SI | 22.01.2020 | ||
SK | 22.01.2020 | ||
SM | 22.01.2020 | ||
BG | 22.04.2020 | ||
NO | 22.04.2020 | ||
GR | 23.04.2020 | ||
IS | 22.05.2020 | ||
PT | 14.06.2020 | ||
Former [2021/13] | CZ | 22.01.2020 | |
DK | 22.01.2020 | ||
EE | 22.01.2020 | ||
ES | 22.01.2020 | ||
FI | 22.01.2020 | ||
HR | 22.01.2020 | ||
LT | 22.01.2020 | ||
LV | 22.01.2020 | ||
PL | 22.01.2020 | ||
RO | 22.01.2020 | ||
RS | 22.01.2020 | ||
SI | 22.01.2020 | ||
SK | 22.01.2020 | ||
SM | 22.01.2020 | ||
BG | 22.04.2020 | ||
NO | 22.04.2020 | ||
GR | 23.04.2020 | ||
IS | 22.05.2020 | ||
PT | 14.06.2020 | ||
Former [2020/50] | CZ | 22.01.2020 | |
DK | 22.01.2020 | ||
EE | 22.01.2020 | ||
ES | 22.01.2020 | ||
FI | 22.01.2020 | ||
HR | 22.01.2020 | ||
LT | 22.01.2020 | ||
LV | 22.01.2020 | ||
RO | 22.01.2020 | ||
RS | 22.01.2020 | ||
SK | 22.01.2020 | ||
SM | 22.01.2020 | ||
BG | 22.04.2020 | ||
NO | 22.04.2020 | ||
GR | 23.04.2020 | ||
IS | 22.05.2020 | ||
PT | 14.06.2020 | ||
Former [2020/49] | CZ | 22.01.2020 | |
DK | 22.01.2020 | ||
ES | 22.01.2020 | ||
FI | 22.01.2020 | ||
HR | 22.01.2020 | ||
LT | 22.01.2020 | ||
LV | 22.01.2020 | ||
RO | 22.01.2020 | ||
RS | 22.01.2020 | ||
SK | 22.01.2020 | ||
SM | 22.01.2020 | ||
BG | 22.04.2020 | ||
NO | 22.04.2020 | ||
GR | 23.04.2020 | ||
IS | 22.05.2020 | ||
PT | 14.06.2020 | ||
Former [2020/48] | DK | 22.01.2020 | |
ES | 22.01.2020 | ||
FI | 22.01.2020 | ||
HR | 22.01.2020 | ||
LT | 22.01.2020 | ||
LV | 22.01.2020 | ||
RO | 22.01.2020 | ||
RS | 22.01.2020 | ||
SM | 22.01.2020 | ||
BG | 22.04.2020 | ||
NO | 22.04.2020 | ||
GR | 23.04.2020 | ||
IS | 22.05.2020 | ||
PT | 14.06.2020 | ||
Former [2020/47] | DK | 22.01.2020 | |
ES | 22.01.2020 | ||
FI | 22.01.2020 | ||
HR | 22.01.2020 | ||
LT | 22.01.2020 | ||
LV | 22.01.2020 | ||
RS | 22.01.2020 | ||
BG | 22.04.2020 | ||
NO | 22.04.2020 | ||
GR | 23.04.2020 | ||
IS | 22.05.2020 | ||
PT | 14.06.2020 | ||
Former [2020/40] | FI | 22.01.2020 | |
HR | 22.01.2020 | ||
LV | 22.01.2020 | ||
RS | 22.01.2020 | ||
BG | 22.04.2020 | ||
NO | 22.04.2020 | ||
GR | 23.04.2020 | ||
IS | 22.05.2020 | ||
PT | 14.06.2020 | ||
Former [2020/39] | FI | 22.01.2020 | |
HR | 22.01.2020 | ||
LV | 22.01.2020 | ||
RS | 22.01.2020 | ||
BG | 22.04.2020 | ||
NO | 22.04.2020 | ||
GR | 23.04.2020 | ||
PT | 14.06.2020 | ||
Former [2020/38] | FI | 22.01.2020 | |
HR | 22.01.2020 | ||
LV | 22.01.2020 | ||
RS | 22.01.2020 | ||
NO | 22.04.2020 | ||
GR | 23.04.2020 | ||
PT | 14.06.2020 | ||
Former [2020/37] | FI | 22.01.2020 | |
HR | 22.01.2020 | ||
LV | 22.01.2020 | ||
RS | 22.01.2020 | ||
NO | 22.04.2020 | ||
PT | 14.06.2020 | ||
Former [2020/36] | FI | 22.01.2020 | |
RS | 22.01.2020 | ||
NO | 22.04.2020 | ||
PT | 14.06.2020 | ||
Former [2020/35] | FI | 22.01.2020 | |
NO | 22.04.2020 | Cited in | International search | [X]EP2674422 (SANTEN PHARMACEUTICAL CO LTD [JP]) [X] 1-33,62 * claims 1, 12; compounds 1-4, 1-7, 1-8, 1-10, 1-11 *; | [X] - MACIEJ KRZESZEWSKI ET AL, "Color-Tunable Fluorescent Dyes Based on Benzo[ c ]coumarin", EUROPEAN JOURNAL OF ORGANIC CHEMISTRY, (20130916), vol. 2013, no. 25, doi:10.1002/ejoc.201300374, ISSN 1434-193X, pages 5631 - 5644, XP055174487 [X] 1-33,62 * table 1 * DOI: http://dx.doi.org/10.1002/ejoc.201300374 | [X] - SUN WANYING ET AL, "6H-Benzo[c]chromen-6-one derivatives as selective ER[beta] agon", BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, (20060118), vol. 16, no. 6, doi:10.1016/J.BMCL.2005.12.057, ISSN 0960-894X, pages 1468 - 1472, XP028755073 [X] 1-33,62 * Scheme 1;; table 1 * DOI: http://dx.doi.org/10.1016/j.bmcl.2005.12.057 | [X] - JAYA PANDEY ET AL, "Synthesis and biological activities of some new dibenzopyranones and dibenzopyrans: search for potential oestrogen receptor agonists and antagonists", BIOORGANIC & MEDICINAL CHEMISTRY, (20040101), vol. 12, no. 9, doi:10.1016/j.bmc.2004.02.018, ISSN 0968-0896, pages 2239 - 2249, XP055100310 [X] 1-33,62 * Scheme 1 step i * DOI: http://dx.doi.org/10.1016/j.bmc.2004.02.018 | [A] - UDO KRAATZ ET AL, "Zur Synthese von Phenanthridinonen-(6) aus 3.4-disubstituierten Cumarinen und ihre Reaktion mit Methylmagnesiumjodid zu Phenanthridiniumjodiden", CHEMISCHE BERICHTE, (19730101), vol. 106, no. 1, doi:10.1002/cber.19731060110, ISSN 0009-2940, pages 62 - 68, XP055172175 [A] 1-33,62 * Scheme page 63 synthesis of the compounds 6a-6d * DOI: http://dx.doi.org/10.1002/cber.19731060110 | [IP] - KAZUHIRO KUDO ET AL, "Scalable Synthesis of 8-Amino-3-hydroxy-6 H -benzo[ c ]chromen-6-one: Key Intermediate for SEGRA via the Hurtley Reaction", ORGANIC PROCESS RESEARCH & DEVELOPMENT, (20141211), vol. 19, no. 1, doi:10.1021/op500334b, ISSN 1083-6160, pages 309 - 314, XP055174456 [IP] 1-33,62 * Schemes 1 and 2 * DOI: http://dx.doi.org/10.1021/op500334b | by applicant | US2011065662 | US2012164243 | US2014018415 | - GIL ET AL., J. AGRIC. FOOD CHEM., (2000), vol. 48, pages 4581 - 4589 | - OKUDA ET AL., CHEM. PHARM. BULL., (1982), vol. 30, pages 4230 - 4233 | - OKUDA ET AL., CHEM. PHARM. BULL., (1982), vol. 30, pages 4234 - 4236 | - "Strategies for the synthesis of ellagitannins", KHANBABAEE, K., Chemistry and Biology of Ellagitannins, WORLD SCIENTIFIC PUBLISHING, (2009), pages 152 - 202 | - J. HASSAN ET AL., "Aryl-Aryl Bond Formation One Century after the Discovery of the Ullmann Reaction", CHEMICAL REVIEWS, (2002), vol. 102, no. 5, pages 1359 - 1470 |