EP3092232 - HETEROCYCLIC MODULATORS OF LIPID SYNTHESIS FOR USE AGAINST CANCER AND VIRAL INFECTIONS [Right-click to bookmark this link] | Status | No opposition filed within time limit Status updated on 13.01.2023 Database last updated on 05.07.2024 | |
Former | The patent has been granted Status updated on 04.02.2022 | ||
Former | Grant of patent is intended Status updated on 08.08.2021 | ||
Former | Examination is in progress Status updated on 07.07.2021 | ||
Former | Grant of patent is intended Status updated on 23.03.2021 | ||
Former | Examination is in progress Status updated on 12.05.2017 | Most recent event Tooltip | 14.06.2024 | Lapse of the patent in a contracting state New state(s): MC | published on 17.07.2024 [2024/29] | Applicant(s) | For all designated states Sagimet Biosciences Inc. 155 Bovet Rd 303 San Mateo, CA 94402 / US | [2020/35] |
Former [2020/01] | For all designated states 3-V Biosciences, Inc. 155 Bovet Rd 303 San Mateo CA 94402 / US | ||
Former [2017/03] | For all designated states 3-V Biosciences, Inc. 3715 Haven Ave., Suite 220 Menlo Park, CA 94025 / US | ||
Former [2016/46] | For all designated states 3-V Biosciences, Inc. 1050 Hamilton Court Menlo Park, CA 94025 / US | Inventor(s) | 01 /
WAGMAN, Allan S. c/o Sagimet Biosciences Inc. 155 Bovet Rd 303 San Mateo, California, 94402 / US | 02 /
JOHNSON, Russell J. c/o Sagimet Biosciences Inc. 155 Bovet Rd 303 San Mateo, California, 94402 / US | 03 /
ZAHARIA, Cristiana A. c/o Sagimet Biosciences Inc. 155 Bovet Rd 303 San Mateo, California, 94402 / US | 04 /
CAI, Haiying c/o Sagimet Biosciences Inc. 155 Bovet Rd 303 San Mateo, California, 94402 / US | 05 /
HU, Lily W. c/o Sagimet Biosciences Inc. 155 Bovet Rd 303 San Mateo, California, 94402 / US | 06 /
DUKE, Greg c/o Sagimet Biosciences Inc. 155 Bovet Rd 303 San Mateo, California, 94402 / US | 07 /
OHOL, Yamini c/o Sagimet Biosciences Inc. 155 Bovet Rd 303 San Mateo, California, 94402 / US | 08 /
HEUER, Timothy c/o Sagimet Biosciences Inc. 155 Bovet Rd 303 San Mateo, California, 94402 / US | 09 /
O'FARRELL, Marie c/o Sagimet Biosciences Inc. 155 Bovet Rd 303 San Mateo, California, 94402 / US | [2022/04] |
Former [2020/01] | 01 /
WAGMAN, Allan S. c/o 3-V BIOSCIENCES INC. 155 Bovet Rd. 303 San Mateo, California 94402 / US | ||
02 /
JOHNSON, Russell J. c/o 3-V BIOSCIENCES INC. 155 Bovet Rd. 303 San Mateo, California 94402 / US | |||
03 /
ZAHARIA, Cristiana A. c/o 3-V BIOSCIENCES INC. 155 Bovet Rd. 303 San Mateo, California 94402 / US | |||
04 /
CAI, Haiying c/o 3-V BIOSCIENCES INC. 155 Bovet Rd. 303 San Mateo, California 94402 / US | |||
05 /
HU, Lily W. c/o 3-V BIOSCIENCES INC. 155 Bovet Rd. 303 San Mateo, California 94402 / US | |||
06 /
DUKE, Greg c/o 3-V BIOSCIENCES INC. 155 Bovet Rd. 303 San Mateo, California 94402 / US | |||
07 /
OHOL, Yamini c/o 3-V BIOSCIENCES INC. 155 Bovet Rd. 303 San Mateo, California 94402 / US | |||
08 /
HEUER, Timothy c/o 3-V BIOSCIENCES INC. 155 Bovet Rd. 303 San Mateo, California 94402 / US | |||
09 /
O'FARRELL, Marie c/o 3-V BIOSCIENCES INC. 155 Bovet Rd. 303 San Mateo, California 94402 / US | |||
Former [2016/46] | 01 /
WAGMAN, Allan S. c/o 3-V BIOSCIENCES INC. 1050 Hamilton Court Menlo Park, California 94025 / US | ||
02 /
JOHNSON, Russell J. c/o 3-V BIOSCIENCES INC. 1050 Hamilton Court Menlo Park, California 94025 / US | |||
03 /
ZAHARIA, Cristiana A. c/o 3-V BIOSCIENCES INC. 1050 Hamilton Court Menlo Park, California 94025 / US | |||
04 /
CAI, Haiying c/o 3-V BIOSCIENCES INC. 1050 Hamilton Court Menlo Park, California 94025 / US | |||
05 /
HU, Lily W. c/o 3-V BIOSCIENCES INC. 1050 Hamilton Court Menlo Park, California 94025 / US | |||
06 /
DUKE, Greg c/o 3-V BIOSCIENCES INC. 1050 Hamilton Court Menlo Park, California 94025 / US | |||
07 /
OHOL, Yamini c/o 3-V BIOSCIENCES INC. 1050 Hamilton Court Menlo Park, California 94025 / US | |||
08 /
HEUER, Timothy c/o 3-V BIOSCIENCES INC. 1050 Hamilton Court Menlo Park, California 94025 / US | |||
09 /
O'FARRELL, Marie c/o 3-V BIOSCIENCES INC. 1050 Hamilton Court Menlo Park, California 94025 / US | Representative(s) | Grund, Martin Grund Intellectual Property Group Patentanwälte und Solicitor PartG mbB Steinsdorfstraße 2 80538 München / DE | [N/P] |
Former [2022/10] | Grund, Martin Grund Intellectual Property Group Patentanwalt und Solicitor PartG mbB Postfach 44 05 16 80754 München / DE | ||
Former [2016/46] | Grund, Martin Grund Intellectual Property Group Postfach 44 05 16 80754 München / DE | Application number, filing date | 15700939.0 | 07.01.2015 | [2016/46] | WO2015US10459 | Priority number, date | US201461924520P | 07.01.2014 Original published format: US 201461924520 P | [2016/46] | Filing language | EN | Procedural language | EN | Publication | Type: | A1 Application with search report | No.: | WO2015105860 | Date: | 16.07.2015 | Language: | EN | [2015/28] | Type: | A1 Application with search report | No.: | EP3092232 | Date: | 16.11.2016 | Language: | EN | The application published by WIPO in one of the EPO official languages on 16.07.2015 takes the place of the publication of the European patent application. | [2016/46] | Type: | B1 Patent specification | No.: | EP3092232 | Date: | 09.03.2022 | Language: | EN | [2022/10] | Search report(s) | International search report - published on: | EP | 16.07.2015 | Classification | IPC: | C07D405/14, C07D401/10, C07D403/10, A61K31/4155, A61K31/454, A61P35/00, A61P31/12 | [2016/46] | CPC: |
C07D403/10 (EP,CN,IL,KR,RU,US);
A61K31/337 (IL,KR);
A61K31/4155 (IL,KR,RU,US);
A61K31/454 (IL,KR,RU,US);
A61K31/704 (IL,KR);
A61K45/06 (IL,KR,US);
A61P31/12 (EP,IL,RU);
A61P31/14 (EP,IL);
A61P31/16 (EP,IL,RU);
A61P31/18 (EP,IL);
A61P31/20 (EP,IL);
A61P31/22 (EP,IL);
A61P35/00 (EP,IL,RU);
A61P35/02 (EP,IL);
A61P37/02 (EP,IL);
A61P43/00 (EP,IL);
C07D401/10 (EP,CN,IL,KR,RU,US);
C07D405/14 (EP,CN,IL,KR,RU,US);
A61K2300/00 (IL,KR)
(-)
| Designated contracting states | AL, AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LI, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, RS, SE, SI, SK, SM, TR [2016/46] | Extension states | BA | Not yet paid | ME | Not yet paid | Title | German: | HETEROCYCLISCHE MODULATOREN DER LIPIDSYNTHESE ZUR VERWENDUNG GEGEN KREBS UND VIRUSINFEKTIONEN | [2016/46] | English: | HETEROCYCLIC MODULATORS OF LIPID SYNTHESIS FOR USE AGAINST CANCER AND VIRAL INFECTIONS | [2016/46] | French: | MODULATEURS HÉTÉROCYCLES DE LA SYNTHÈSE DES LIPIDES DESTINÉS À ÊTRE UTILISÉS CONTRE LE CANCER ET LES INFECTIONS VIRALES | [2016/46] | Entry into regional phase | 02.08.2016 | National basic fee paid | 02.08.2016 | Designation fee(s) paid | 02.08.2016 | Examination fee paid | Examination procedure | 02.08.2016 | Examination requested [2016/46] | 03.03.2017 | Amendment by applicant (claims and/or description) | 11.05.2017 | Despatch of a communication from the examining division (Time limit: M06) | 20.09.2017 | Reply to a communication from the examining division | 14.12.2017 | Despatch of a communication from the examining division (Time limit: M06) | 23.07.2018 | Despatch of communication that the application is deemed to be withdrawn, reason: reply to the communication from the examining division not received in time | 02.10.2018 | Reply to a communication from the examining division | 12.06.2019 | Despatch of a communication from the examining division (Time limit: M04) | 09.10.2019 | Reply to a communication from the examining division | 24.06.2020 | Cancellation of oral proceeding that was planned for 11.11.2020 | 11.11.2020 | Date of oral proceedings (cancelled) | 21.01.2021 | Cancellation of oral proceeding that was planned for 26.01.2021 | 26.01.2021 | Date of oral proceedings (cancelled) | 24.03.2021 | Communication of intention to grant the patent | 05.07.2021 | Disapproval of the communication of intention to grant the patent by the applicant or resumption of examination proceedings by the EPO | 09.08.2021 | Communication of intention to grant the patent | 17.12.2021 | Fee for grant paid | 17.12.2021 | Fee for publishing/printing paid | 17.12.2021 | Receipt of the translation of the claim(s) | Opposition(s) | 12.12.2022 | No opposition filed within time limit [2023/07] | Request for further processing for: | The application is deemed to be withdrawn due to failure to reply to the examination report | 02.10.2018 | Request for further processing filed | 02.10.2018 | Full payment received (date of receipt of payment) Request granted | 17.10.2018 | Decision despatched | Fees paid | Renewal fee | 27.01.2017 | Renewal fee patent year 03 | 29.01.2018 | Renewal fee patent year 04 | 28.01.2019 | Renewal fee patent year 05 | 27.01.2020 | Renewal fee patent year 06 | 27.01.2021 | Renewal fee patent year 07 | 27.01.2022 | Renewal fee patent year 08 |
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Responsibility for the accuracy, completeness or quality of the data displayed under the link provided lies entirely with the Unified Patent Court. | Lapses during opposition Tooltip | AL | 09.03.2022 | AT | 09.03.2022 | CZ | 09.03.2022 | DK | 09.03.2022 | EE | 09.03.2022 | FI | 09.03.2022 | HR | 09.03.2022 | LT | 09.03.2022 | LV | 09.03.2022 | MC | 09.03.2022 | NL | 09.03.2022 | PL | 09.03.2022 | RO | 09.03.2022 | RS | 09.03.2022 | SE | 09.03.2022 | SI | 09.03.2022 | SK | 09.03.2022 | SM | 09.03.2022 | BG | 09.06.2022 | NO | 09.06.2022 | GR | 10.06.2022 | IS | 09.07.2022 | PT | 11.07.2022 | [2024/29] |
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NO | 09.06.2022 | Cited in | International search | [A]WO2008075077 (ASTRAZENECA AB [SE], et al) [A] 1-29 * the whole document *; | [A]WO2008075070 (ASTRAZENECA AB [SE], et al) [A] 1-29 * the whole document *; | [A]WO2008075064 (ASTRAZENECA AB [SE], et al) [A] 1-29* the whole document *; | [A]WO2012122391 (3 V BIOSCIENCES INC [US], et al) [A] 1-29 * the whole document *; | [XPI]WO2014008197 (3 V BIOSCIENCES INC [US]) [XP] 1,2,5-7,9-11,14,16-19,22-25 * compounds 249, 277, 276 * * claims 43, 151-157 * * page 10, line 15 - line 26 * [I] 3,4,8,12,13,15,20,21,26-29 | by applicant | US3625214 | US4789734 | US4897268 | US4906474 | US4925673 | US5075109 | US5811128 | US5814344 | US5820883 | US5853763 | US5928647 | US5942252 | - "IUPAC 1974 Recommendations for Section E, Fundamental Stereochemistry", PURE APPL. CHEM., (1976), vol. 45, pages 13 - 30 | - COMPENDIUM OF ORGANIC SYNTHETIC METHODS, (1971), vol. 1 | - COMPENDIUM OF ORGANIC SYNTHETIC METHODS, (1974), vol. 2 | - COMPENDIUM OF ORGANIC SYNTHETIC METHODS, (1977), vol. 3 | - COMPENDIUM OF ORGANIC SYNTHETIC METHODS, (1980), vol. 4 | - COMPENDIUM OF ORGANIC SYNTHETIC METHODS, (1984), vol. 5 | - COMPENDIUM OF ORGANIC SYNTHETIC METHODS, vol. 6 | - "Comprehensive Organic Synthesis", SELECTIVITY, STRATEGY & EFFICIENCY IN MODERN ORGANIC CHEMISTRY, (1993), vol. 9 | - Protecting Groups in Organic Synthesis | - PAUL AV ET AL., NATURE, (1998), vol. 393, no. 6682, pages 280 - 284 | - HUANG H ET AL., BIOCHEMISTRY, (2001), vol. 40, no. 27, pages 8055 - 8064 | - GERBER K; WIMMER E; PAUL AV, J VIROL, (2001), vol. 75, no. 22, pages 10979 - 10990 | - ROSSMANN M ET AL., NATURE, (1985), vol. 317, no. 6033, pages 145 - 53 | - SMITH T ET AL., SCIENCE, (1986), vol. 233, no. 4770, pages 1286 - 93 | - FLAVIN, R. ET AL., FUTURE ONCOLOGY, (2010), vol. 6, no. 4, pages 551 - 562 | - ORITA, H. ET AL., CLINICAL CANCER RESEARCH., (2007), vol. 13, no. 23, pages 7139 - 7145 | - PUIG, T. ET AL., BREAST CANCER RESEARCH, (2011), vol. 13, no. 6, page R131 | - BROWNE, CD., THE FASEB JOURNAL, (2006), vol. 20, no. 12, pages 2027 - 2035 | - CHAKRAVARTHY, M. V. ET AL., CELL METABOLISM, (2005), vol. 1, pages 309 - 322 | - WU, M. ET AL., PNAS, (2011), vol. 108, no. 13, pages 5378 - 5383 | - "Liposomes", G. GREGORIADIS, Drug Carriers in Biology and Medicine, ACADEMIC PRESS, (1979), page 2 | - JEIN, TIPS, (1998), vol. 19, pages 155 - 157 | - REMINGTON, The Science and Practice of Pharmacy, LIPPINCOTT WILLIAMS & WILKINS | - TERESA, P. ET AL., CLIN. CANCER RES., (2009), vol. 15, no. 24, pages 7608 - 7615 | - CHUNG C.C. ET AL., ASSAY AND DRUG DEVELOPMENT TECHNOLOGIES, (2008), vol. 6, no. 3, pages 361 - 374 |