blank Quick help
blank Maintenance news

Scheduled maintenance

Regular maintenance outages:
between 05.00 and 05.15 hrs CET (Monday to Sunday).

Other outages
Availability

2022.02.11

More...
blank News flashes

News Flashes

New version of the European Patent Register – SPC proceedings information in the Unitary Patent Register.

2024-07-24

More...
blank Related links

Extract from the Register of European Patents

EP About this file: EP3119752

EP3119752 - 3,4-DIAMINO-6-CHLOROPYRAZINE-2-CARBOXAMIDE COMPOUNDS FOR THE TREATMENT OF ENAC MEDIATED DISEASES [Right-click to bookmark this link]
Former [2017/04]CHEMICAL COMPOUNDS
[2017/43]
StatusNo opposition filed within time limit
Status updated on  22.03.2019
Database last updated on 16.09.2024
FormerThe patent has been granted
Status updated on  13.04.2018
FormerGrant of patent is intended
Status updated on  05.10.2017
FormerRequest for examination was made
Status updated on  23.12.2016
Most recent event   Tooltip15.11.2019Lapse of the patent in a contracting state
New state(s): AL
published on 18.12.2019  [2019/51]
Applicant(s)For all designated states
Astrazeneca AB
151 85 Södertälje / SE
[2017/04]
Inventor(s)01 / BERGLUND, Susanne, Elisabeth
AstraZeneca
SE-431 83 Mölndal / SE
02 / CONNOLLY, Stephen
c/o AstraZeneca Intellectual Property
Alderley Park
Macclesfield Cheshire SK10 4TG / GB
03 / HEMMERLING, Martin
AstraZeneca
SE-431 83 Mölndal / SE
04 / HOSSAIN, Nafizal
AstraZeneca
SE-431 83 Mölndal / SE
05 / KRISTOFFERSSON, Anna
c/o AstraZeneca Intellectual Property
Alderley Park
Macclesfield Cheshire SK10 4TG / GB
06 / LUNDKVIST, Johan, Rune, Michael
c/o AstraZeneca Intellectual Property
Alderley Park
Macclesfield Cheshire SK10 4TG / GB
07 / NIKITIDIS, Grigorios
AstraZeneca
SE-431 83 Mölndal / SE
08 / RIPA, Lena, Elisabeth
AstraZeneca
SE-431 83 Mölndal / SE
09 / SHAMOVSKY, Igor
AstraZeneca R&D Mölndal
SE-431 83 Mölndal / SE
 [2017/04]
Representative(s)AstraZeneca Intellectual Property
Eastbrook House
Shaftesbury Road
Cambridge CB2 8BF / GB
[N/P]
Former [2018/20]AstraZeneca
Milstein Building
Granta Park
Cambridge CB21 6GH / GB
Former [2017/04]Cook, Andrew James
AstraZeneca
Intellectual Property
Mereside
Alderley Park
Macclesfield, Cheshire SK10 4TG / GB
Application number, filing date15713339.817.03.2015
[2017/04]
WO2015GB50765
Priority number, dateUS201461954674P18.03.2014         Original published format: US 201461954674 P
[2017/04]
Filing languageEN
Procedural languageEN
PublicationType: A1 Application with search report
No.:WO2015140527
Date:24.09.2015
Language:EN
[2015/38]
Type: A1 Application with search report 
No.:EP3119752
Date:25.01.2017
Language:EN
The application published by WIPO in one of the EPO official languages on 24.09.2015 takes the place of the publication of the European patent application.
[2017/04]
Type: B1 Patent specification 
No.:EP3119752
Date:16.05.2018
Language:EN
[2018/20]
Search report(s)International search report - published on:EP24.09.2015
ClassificationIPC:C07D401/06, C07D241/28, A61K31/497, A61P11/00
[2017/04]
CPC:
C07D401/12 (EP,KR,US); C07D401/06 (EP,IL,US); C07D241/28 (EP,IL,KR,US);
A61K31/4965 (EP,US); A61K31/497 (EP,KR,US); A61K45/06 (KR,US);
A61P11/00 (EP,US); A61P11/06 (KR,US); A61P3/12 (EP,US);
A61P43/00 (EP,US); C07D241/26 (EP,US); C07D405/14 (EP,KR,US) (-)
Designated contracting statesAL,   AT,   BE,   BG,   CH,   CY,   CZ,   DE,   DK,   EE,   ES,   FI,   FR,   GB,   GR,   HR,   HU,   IE,   IS,   IT,   LI,   LT,   LU,   LV,   MC,   MK,   MT,   NL,   NO,   PL,   PT,   RO,   RS,   SE,   SI,   SK,   SM,   TR [2017/04]
Extension statesBA18.10.2016
ME18.10.2016
Validation statesMA18.10.2016
TitleGerman:3,4-DIAMINO-6-CHLOROPYRAZINE-2-CARBOXAMID-VERBINDUNGEN ZUR BEHANDLUNG VON ENAC-VERMITTELTEN KRANKHEITEN[2017/44]
English:3,4-DIAMINO-6-CHLOROPYRAZINE-2-CARBOXAMIDE COMPOUNDS FOR THE TREATMENT OF ENAC MEDIATED DISEASES[2017/43]
French:COMPOSÉS DE 3,4-DIAMINO-6-CHLOROPYRAZINE-2-CARBOXAMIDE UTILES POUR LE TRAITEMENT DE MALADIES MÉDIÉES PAR LE ENAC[2017/43]
Former [2017/04]CHEMISCHE VERBINDUNGEN
Former [2017/04]CHEMICAL COMPOUNDS
Former [2017/04]COMPOSÉS CHIMIQUES
Entry into regional phase18.10.2016National basic fee paid 
18.10.2016Designation fee(s) paid 
18.10.2016Examination fee paid 
Examination procedure14.09.2016Date on which the examining division has become responsible
18.10.2016Examination requested  [2017/04]
28.04.2017Amendment by applicant (claims and/or description)
06.10.2017Communication of intention to grant the patent
02.02.2018Fee for grant paid
02.02.2018Fee for publishing/printing paid
02.02.2018Receipt of the translation of the claim(s)
Opposition(s)19.02.2019No opposition filed within time limit [2019/17]
Fees paidRenewal fee
31.03.2017Renewal fee patent year 03
03.04.2018Renewal fee patent year 04
Opt-out from the exclusive  Tooltip
competence of the Unified
Patent Court
See the Register of the Unified Patent Court for opt-out data
Responsibility for the accuracy, completeness or quality of the data displayed under the link provided lies entirely with the Unified Patent Court.
Lapses during opposition  TooltipAL16.05.2018
MC16.05.2018
[2019/51]
Former [2019/46]MC16.05.2018
Cited inInternational search[A]WO2009150137  (NOVARTIS AG [CH], et al) [A] 1-13* claims 1,5,8 *;
 [A]WO2011028740  (GLAXO GROUP LTD [US], et al) [A] 1-13 * claims 1,5 *;
 [A]  - THOMAS HUNT ET AL, "Discovery of a novel chemotype of potent human ENaC blockers using a bioisostere approach. Part 1: Quaternary amines", BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, PERGAMON, AMSTERDAM, NL, vol. 22, no. 2, doi:10.1016/J.BMCL.2011.12.016, ISSN 0960-894X, (20111203), pages 929 - 932, (20111208), XP028438452 [A] 1-13 * the whole document *

DOI:   http://dx.doi.org/10.1016/j.bmcl.2011.12.016
 [A]  - THOMAS HUNT ET AL, "Discovery of a novel chemotype of potent human ENaC blockers using a bioisostere approach. Part 2: [alpha]-Branched quaternary amines", BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, (20120401), vol. 22, no. 8, doi:10.1016/j.bmcl.2012.02.067, ISSN 0960-894X, pages 2877 - 2879, XP055084884 [A] 1-13 * the whole document *

DOI:   http://dx.doi.org/10.1016/j.bmcl.2012.02.067
The EPO accepts no responsibility for the accuracy of data originating from other authorities; in particular, it does not guarantee that it is complete, up to date or fit for specific purposes.