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Extract from the Register of European Patents

EP About this file: EP3300501

EP3300501 - NOVEL COMPOSITIONS, USES AND METHODS FOR MAKING THEM [Right-click to bookmark this link]
StatusExamination is in progress
Status updated on  25.12.2020
Database last updated on 14.09.2024
FormerRequest for examination was made
Status updated on  02.03.2018
FormerThe international publication has been made
Status updated on  04.11.2016
Most recent event   Tooltip29.05.2024New entry: Despatch of examination report + time limit 
Applicant(s)For all designated states
Pimera, Inc.
3210 Merryfield Row
San Diego, California 92121 / US
[2018/14]
Inventor(s)01 / HADDACH, Mustapha
3210 Merryfield Row
San Diego, California 92121 / US
 [2018/14]
Representative(s)Mewburn Ellis LLP
Aurora Building
Counterslip
Bristol BS1 6BX / GB
[N/P]
Former [2018/14]Barker Brettell LLP
100 Hagley Road
Edgbaston
Birmingham B16 8QQ / GB
Application number, filing date16759401.902.03.2016
[2018/14]
WO2016US20418
Priority number, dateUS201562128208P04.03.2015         Original published format: US 201562128208 P
[2018/14]
Filing languageEN
Procedural languageEN
PublicationType: A2 Application without search report
No.:WO2016141042
Date:09.09.2016
Language:EN
[2016/36]
Type: A2 Application without search report 
No.:EP3300501
Date:04.04.2018
Language:EN
The application published by WIPO in one of the EPO official languages on 09.09.2016 takes the place of the publication of the European patent application.
[2018/14]
Search report(s)International search report - published on:KR03.11.2016
(Supplementary) European search report - dispatched on:EP19.03.2019
ClassificationIPC:C07D487/14, A61K31/4353, A61P35/00
[2019/01]
CPC:
C07D471/14 (EP,US); A61K31/4353 (US); A61P35/00 (EP,US);
C07D471/04 (EP,US); C07D471/22 (EP,US); C07D487/14 (EP,US)
Former IPC [2018/14]C07D471/14, C07D487/14, C07D403/04, C07D403/14, A61K31/4375, A61K31/519, A61K31/4985, A61K31/5025
Designated contracting statesAL,   AT,   BE,   BG,   CH,   CY,   CZ,   DE,   DK,   EE,   ES,   FI,   FR,   GB,   GR,   HR,   HU,   IE,   IS,   IT,   LI,   LT,   LU,   LV,   MC,   MK,   MT,   NL,   NO,   PL,   PT,   RO,   RS,   SE,   SI,   SK,   SM,   TR [2018/14]
TitleGerman:NEUARTIGE ZUSAMMENSETZUNGEN, VERWENDUNGEN UND VERFAHREN ZUR HERSTELLUNG DAVON[2018/14]
English:NOVEL COMPOSITIONS, USES AND METHODS FOR MAKING THEM[2018/14]
French:NOUVELLES COMPOSITIONS, LEURS UTILISATIONS ET LEURS PROCÉDÉS DE PRÉPARATION[2018/14]
Entry into regional phase01.09.2017National basic fee paid 
01.09.2017Search fee paid 
01.09.2017Designation fee(s) paid 
16.02.2018Examination fee paid 
Examination procedure01.09.2017Date on which the examining division has become responsible
deletedDeletion: Application deemed to be withdrawn, date of legal effect  [2018/14]
16.02.2018Examination requested  [2018/14]
11.10.2019Amendment by applicant (claims and/or description)
13.01.2021Despatch of a communication from the examining division (Time limit: M04)
20.05.2021Reply to a communication from the examining division
30.08.2021Despatch of a communication from the examining division (Time limit: M06)
07.06.2022Reply to a communication from the examining division
28.05.2024Despatch of a communication from the examining division (Time limit: M04)
Request for further processing for:The application is deemed to be withdrawn due to failure to reply to the examination report
07.06.2022Request for further processing filed
07.06.2022Full payment received (date of receipt of payment)
Request granted
17.06.2022Decision despatched
The application is deemed to be withdrawn due to non-payment of the examination fee
16.02.2018Request for further processing filed
16.02.2018Full payment received (date of receipt of payment)
Request granted
01.03.2018Decision despatched
16.02.2018Request for further processing filed
16.02.2018Full payment received (date of receipt of payment)
Request granted
01.03.2018Decision despatched
Fees paidRenewal fee
29.03.2018Renewal fee patent year 03
27.03.2019Renewal fee patent year 04
27.03.2020Renewal fee patent year 05
29.03.2021Renewal fee patent year 06
28.03.2022Renewal fee patent year 07
27.03.2023Renewal fee patent year 08
27.03.2024Renewal fee patent year 09
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Documents cited:Search[I]WO2009046383  (CYLENE PHARMACEUTICALS INC [US], et al) [I] 1-10,14,15 * claims 1, 31 *;
 [A]  - BEAULIEU ET AL, "Synthesis and biological evaluation of 4-amino derivatives of benzimidazoquinoxaline, benzimidazoquinoline, and benzopyrazoloquinazoline as potent IKK inhibitors", BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, PERGAMON, AMSTERDAM, NL, (20070214), vol. 17, no. 5, doi:10.1016/J.BMCL.2006.12.017, ISSN 0960-894X, pages 1233 - 1237, XP005888454 [A] 1-10,14,15 * table 1, compounds 7a-d *

DOI:   http://dx.doi.org/10.1016/j.bmcl.2006.12.017
 [X]  - WOLFGANG-R. KNAPPE, "Photochemie des 10-Phenylisoalloxazins: Intramolekulare Singulett- und intermolekulare Triplett-Reaktionen", CHEMISCHE BERICHTE, DE, (19740501), vol. 107, no. 5, doi:10.1002/cber.19741070520, ISSN 0009-2940, pages 1614 - 1636, XP055524260 [X] 1,2 * page 1625; compound 17a *

DOI:   http://dx.doi.org/10.1002/cber.19741070520
 [X]  - V I Shvedov ET AL, "Synthesis of derivatives of pyrazino[1,2-a]benzimidazole, aza analogs of[beta]-carboline", (19691031), URL: https://link.springer.com/content/pdf/10.1007/BF00762071.pdf, (20181115), XP055524256 [X] 1,2 * compound IV *
International search[X]WO0228860  (BRISTOL MYERS SQUIBB CO [US], et al) [X] 19 * See abstract; pages 25-26, 34, 46. *;
 [PX]WO2015172123  (HADDACH MUSTAPHA [US]) [PX] 1-15, 17-21* See abstract; claims 1-33. *;
 [XA]  - Chemical Abstract, (19961211), Database accession no. 183858-24-4, URL: STN, XP 055409388 [X] 1-2 * ,. See the structures. * [A] 3-15, 17-21
    [ ] - CHEMICAL ABSTRACT, (19961211), Database accession no. 183858-23-3, URL: STN, XP 055409391
 [XA]  - Chemical Abstract, (19841218), Database accession no. 93438-49-4, URL: STN, XP055410392 [X] 1-2 * . See the structure. * [A] 3-15, 17-21
 [XA]  - ZANZOUL, A. et al., "A benzimidazopyridoquinoxaline as promising scaffold for G-quadruplex DNA targeting", Medicinal chemistry research, (20140000), vol. 23, pages 4042 - 4049, XP 055327267 [X] 19-20 * . See abstract; page 4042; scheme 1. * [A] 1-15, 17-18, 21
 [X]  - ANDALOUSSI, M. et al., "Novel imidazo[1,2-a]naphthyridinic systems (Part 1): Synthesis, antiproliferative and DNA-intercalating activities", Eur. J. Med. Chem., (20080000), vol. 43, pages 2505 - 2517, XP 025571383 [X] 19 * . See abstract; table 1. *
 [A]  - MOGILAIAH, K. et al., "Synthesis of some novel bridgehead nitrogen heterocyclic systems containing 1,8-naphthyridine moiety", Indian J. Chem., (20030000), vol. 42 B, pages 192 - 194, XP 055236419 [A] 1-15, 17-21 * . See scheme 1, compound 5. *
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