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Extract from the Register of European Patents

EP About this file: EP3464340

EP3464340 - SECRETIN RECEPTOR AGONISTS TO TREAT DISEASES OR DISORDERS OF ENERGY HOMEOSTASIS [Right-click to bookmark this link]
StatusThe application is deemed to be withdrawn
Status updated on  08.10.2021
Database last updated on 07.10.2024
FormerExamination is in progress
Status updated on  29.01.2021
FormerRequest for examination was made
Status updated on  08.03.2019
FormerThe international publication has been made
Status updated on  01.12.2017
Formerunknown
Status updated on  15.06.2017
Most recent event   Tooltip08.10.2021Application deemed to be withdrawnpublished on 10.11.2021  [2021/45]
Applicant(s)For all designated states
Technische Universität München
Arcisstr. 21
80333 München / DE
[2019/15]
Inventor(s)01 / KLINGENSPOR, Martin
Körnerstrasse 7C
85356 Freising / DE
02 / GABLER, Sarah-Madeleine
Pöppelstrasse 8
81541 München / DE
03 / LI, Yongguo
Mauermayrstrasse 37
85354 Freising / DE
 [2019/16]
Former [2019/15]01 / KLINGENSPOR, Martin
Körnerstrasse 7C
85356 Freising / DE
02 / GABLER, Sarah-Madeleine
Steinstrasse 8
81667 München / DE
03 / LI, Yongguo
Mauermayrstrasse 37
85354 Freising / DE
Representative(s)Vossius & Partner Patentanwälte Rechtsanwälte mbB
Siebertstrasse 3
81675 München / DE
[2019/15]
Application number, filing date17727158.223.05.2017
[2019/15]
WO2017EP62420
Priority number, dateEP2016017086323.05.2016         Original published format: EP 16170863
[2019/15]
Filing languageEN
Procedural languageEN
PublicationType: A1 Application with search report
No.:WO2017202851
Date:30.11.2017
Language:EN
[2017/48]
Type: A1 Application with search report 
No.:EP3464340
Date:10.04.2019
Language:EN
The application published by WIPO in one of the EPO official languages on 30.11.2017 takes the place of the publication of the European patent application.
[2019/15]
Search report(s)International search report - published on:EP30.11.2017
ClassificationIPC:C07K14/645, A61K38/00, C07K14/72, G01N33/74
[2019/15]
CPC:
C07K14/723 (EP); A61K38/2242 (EP,US); A61K38/00 (EP);
A61K45/06 (EP,US); A61K8/64 (EP,US); A61Q19/06 (EP,US);
C07K14/645 (EP); G01N33/5044 (EP,US) (-)
C-Set:
A61K38/2242, A61K2300/00 (EP)
Designated contracting statesAL,   AT,   BE,   BG,   CH,   CY,   CZ,   DE,   DK,   EE,   ES,   FI,   FR,   GB,   GR,   HR,   HU,   IE,   IS,   IT,   LI,   LT,   LU,   LV,   MC,   MK,   MT,   NL,   NO,   PL,   PT,   RO,   RS,   SE,   SI,   SK,   SM,   TR [2019/15]
TitleGerman:SEKRETINREZEPTOR ZUR BEHANDLUNG VON ERKRANKUNGEN ODER STÖRUNGEN DER ENERGIEHOMÖOSTASE[2019/15]
English:SECRETIN RECEPTOR AGONISTS TO TREAT DISEASES OR DISORDERS OF ENERGY HOMEOSTASIS[2019/15]
French:AGONISTES DU RÉCEPTEUR DE LA SÉCRÉTINE POUR TRAITER DES MALADIES OU DES TROUBLES DE L'HOMÉOSTASIE ÉNERGÉTIQUE[2019/15]
Entry into regional phase24.11.2018National basic fee paid 
24.11.2018Designation fee(s) paid 
24.11.2018Examination fee paid 
Examination procedure24.11.2018Examination requested  [2019/15]
24.11.2018Date on which the examining division has become responsible
17.07.2019Amendment by applicant (claims and/or description)
02.02.2021Despatch of a communication from the examining division (Time limit: M04)
15.06.2021Application deemed to be withdrawn, date of legal effect  [2021/45]
02.07.2021Despatch of communication that the application is deemed to be withdrawn, reason: reply to the communication from the examining division not received in time  [2021/45]
Fees paidRenewal fee
15.05.2019Renewal fee patent year 03
14.05.2020Renewal fee patent year 04
Penalty fee
Additional fee for renewal fee
31.05.202105   M06   Not yet paid
Opt-out from the exclusive  Tooltip
competence of the Unified
Patent Court		 See the Register of the Unified Patent Court for opt-out data
Responsibility for the accuracy, completeness or quality of the data displayed under the link provided lies entirely with the Unified Patent Court.
Cited inInternational search[I]  - SEKAR REVATHI ET AL, "Secretin receptor-knockout mice are resistant to high-fat diet-induced obesity and exhibit impaired intestinal lipid absorption", FASEB JOURNAL, (20140425), vol. 28, no. 8, doi:10.1096/fj.13-247536, pages 3494 - 3505, XP002763314 [I] 1-14 * page 3502 *

DOI:   http://dx.doi.org/10.1096/fj.13-247536
 [I]  - SEKAR REVATHI ET AL, "Lipolytic actions of secretin in mouse adipocytes", JOURNAL OF LIPID RESEARCH, (201402), vol. 55, no. 2, pages 190 - 200, XP002763315 [I] 1-14 * page 197 - page 199 *
 [I]  - CHENG CARRIE YUEN YEE ET AL, "Central and Peripheral Administration of Secretin Inhibits Food Intake in Mice through the Activation of the Melanocortin System", NEUROPSYCHOPHARMACOLOGY, (201101), vol. 36, no. 2, ISSN 0893-133X, pages 459 - 471, XP002763316 [I] 1-14 * page 467, column r, paragraph 1 * * page 469, column r, paragraph 2 *
 [X]  - BEINBORN MARTIN, "Class B GPCRs: A hidden agonist within?", MOLECULAR PHARMACOLOGY, (20060701), vol. 70, no. 1, doi:10.1124/mol.106.025932, ISSN 0026-895X, pages 1 - 4, XP002763317 [X] 10 * the whole document *
 [X]  - JEREZ A TE ET AL, "Predicting the effects of amino acid replacements in peptide hormones on their binding affinities for class B GPCRs and application to the design of secretin receptor antagonists", JOURNAL OF COMPUTER-AIDED MOLECULAR DESIGN, KLUWER ACADEMIC PUBLISHERS, DO, (20120511), vol. 26, no. 7, doi:10.1007/S10822-012-9574-X, ISSN 1573-4951, pages 835 - 845, XP035096411 [X] 10 * the whole document *

DOI:   http://dx.doi.org/10.1007/s10822-012-9574-x
 [X]  - Kailash Singh et al, "Structure-Activity Relationship Studies of N- and C-Terminally Modified Secretin Analogs for the Human Secretin Receptor", PLOS ONE, vol. 11, no. 3, doi:10.1371/JOURNAL.PONE.0149359, (20160301), Database accession no. E0149359, pages 1 - 19, URL: http://dx.doi.org/10.1371/journal.pone.0149359, (201610), XP002763318 [X] 10 * the whole document *

DOI:   http://dx.doi.org/DOI:10.1371/JOURNAL.PONE.0149359
 [X]  - DONG M ET AL, "Refinement of the pharmacophore of an agonist ligand of the secretin receptor using conformationally constrained cyclic hexapeptides", PEPTIDES, ELSEVIER, AMSTERDAM, NL, vol. 31, no. 6, ISSN 0196-9781, (20100601), pages 1094 - 1098, (20100307), XP027046212 [X] 10 * the whole document *
 [I]  - R. SEKAR ET AL, "Role of Secretin Peptide Family and their Receptors in the Hypothalamic Control of Energy Homeostasis", HORMONE AND METABOLIC RESEARCH, DE, (20130925), vol. 45, no. 13, doi:10.1055/s-0033-1353155, ISSN 0018-5043, pages 945 - 954, XP055401285 [I] 1-14 * page 946 *

DOI:   http://dx.doi.org/10.1055/s-0033-1353155
by applicantUS4946778
 US6080560
 WO2008022759
 WO9813526
 EP2221377
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DOI:   http://dx.doi.org/10.1016/j.biochi.2016.12.005
 US19910746121
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