Extract from the Register of European Patents

EP About this file: EP3549935

EP3549935 - METHOD FOR PRODUCING TRIAZINE COMPOUND [Right-click to bookmark this link]
StatusExamination is in progress
Status updated on  30.07.2021
Database last updated on 09.04.2026
FormerRequest for examination was made
Status updated on  06.09.2019
FormerThe international publication has been made
Status updated on  08.06.2018
Most recent event   Tooltip13.03.2026Change - applicantpublished on 15.04.2026 [2026/16]
Applicant(s)For all designated states
Tanabe Pharma Corporation
3-2-10, Dosho-machi
Chuo-ku
Osaka-shi, Osaka 541-8505 / JP
[2026/16]
Former [2019/41]For all designated states
Mitsubishi Tanabe Pharma Corporation
2-10, Dosho-machi 3-chome Chuo-ku Osaka-shi
Osaka 541-8505 / JP
Inventor(s)01 / YAMAGAMI, Takafumi
c/o Mitsubishi Tanabe Pharma Corporation
3-2-10 Dosho-machi
Chuo-ku
Osaka-shi Osaka 541-8505 / JP
02 / YAMASAKI, Souta
c/o Mitsubishi Tanabe Pharma Corporation
3-2-10 Dosho-machi
Chuo-ku
Osaka-shi Osaka 541-8505 / JP
03 / SETSUTA, Tomofumi
c/o Mitsubishi Tanabe Pharma Corporation
3-2-10 Dosho-machi
Chuo-ku
Osaka-shi Osaka 541-8505 / JP
04 / SAKAKIBARA, Ryo
c/o Mitsubishi Tanabe Pharma Corporation
3-2-10 Dosho-machi
Chuo-ku
Osaka-shi Osaka 541-8505 / JP
05 / MATSUMURA, Yosuke
c/o Mitsubishi Tanabe Pharma Corporation
3-2-10 Dosho-machi
Chuo-ku
Osaka-shi Osaka 541-8505 / JP
 [2019/41]
Representative(s)Hoffmann Eitle
Patent- und Rechtsanwälte PartmbB
Arabellastraße 30
81925 München / DE
[2019/41]
Application number, filing date17875693.829.11.2017
[2019/41]
WO2017JP42769
Priority number, dateJP2016023289030.11.2016         Original published format: JP 2016232890
[2019/41]
Filing languageJA
Procedural languageEN
PublicationType: A1 Application with search report
No.:WO2018101312
Date:07.06.2018
Language:JA
[2018/23]
Type: A1 Application with search report 
No.:EP3549935
Date:09.10.2019
Language:EN
[2019/41]
Search report(s)International search report - published on:JP07.06.2018
(Supplementary) European search report - dispatched on:EP02.07.2020
ClassificationIPC:C07D253/07
[2020/32]
CPC:
C07D253/07 (EP,US)
Former IPC [2019/41]C07D253/06
Designated contracting statesAL,   AT,   BE,   BG,   CH,   CY,   CZ,   DE,   DK,   EE,   ES,   FI,   FR,   GB,   GR,   HR,   HU,   IE,   IS,   IT,   LI,   LT,   LU,   LV,   MC,   MK,   MT,   NL,   NO,   PL,   PT,   RO,   RS,   SE,   SI,   SK,   SM,   TR [2019/41]
TitleGerman:VERFAHREN ZUR HERSTELLUNG VON TRIAZINVERBINDUNGEN[2019/41]
English:METHOD FOR PRODUCING TRIAZINE COMPOUND[2019/41]
French:PROCÉDÉ DE PRODUCTION DE COMPOSÉ TRIAZINE[2019/41]
Entry into regional phase18.06.2019Translation filed 
18.06.2019National basic fee paid 
18.06.2019Search fee paid 
18.06.2019Designation fee(s) paid 
18.06.2019Examination fee paid 
Examination procedure18.06.2019Examination requested  [2019/41]
27.01.2021Amendment by applicant (claims and/or description)
03.08.2021Despatch of a communication from the examining division (Time limit: M06)
10.02.2022Reply to a communication from the examining division
17.03.2023Despatch of a communication from the examining division (Time limit: M06)
13.09.2023Reply to a communication from the examining division
07.06.2024Despatch of a communication from the examining division (Time limit: M04)
30.09.2024Reply to a communication from the examining division
Fees paidRenewal fee
22.11.2019Renewal fee patent year 03
13.11.2020Renewal fee patent year 04
12.11.2021Renewal fee patent year 05
24.11.2022Renewal fee patent year 06
13.11.2023Renewal fee patent year 07
14.11.2024Renewal fee patent year 08
26.11.2025Renewal fee patent year 09
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Documents cited:Search[XY] US4851411  (PITET GUY et al.) [X] 1-8 * reaction schemes; columns 3-6 *[Y] 1-11
 [XDY] EP2141164  (MUTABILIS et al.) [XD] 1-8 * page 18; examples 15a), b) * * page 22; example 22a) *[Y] 1-11
 [XDY]   DESROY, N. ET AL.: "Novel HldE-K Inhibitors Leading to Attenuated Gram Negative Bacterial Virulence", JOURNAL OF MEDICINAL CHEMISTRY, vol. 56, no. 4, 2013, pages 1418 - 1430, XP055706248, ISSN: 0022-2623, DOI: 10.1021/jm301499r [XD] 1-8 * Scheme 5, step a; page 1421 * [Y] 1-11

DOI:   http://dx.doi.org/10.1021/jm301499r
 [XDY]   DESROY, N. ET AL.: "Novel HldE-K Inhibitors Leading to Attenuated Gram Negative Bacterial Virulence, Supporting Information", JOURNAL OF MEDICINAL CHEMISTRY, vol. 56, no. 4, 2013, pages S1 - S53, XP055707481, ISSN: 0022-2623, DOI: 10.1021/jm301499r * page S27 * [Y] 1-11

DOI:   http://dx.doi.org/10.1021/jm301499r
 [XY]   GIANNELLA, M. ET AL.: "Su alcuni gliossali a nucleo isossazolico ed ossazolico e loro derivati = [On some glyoxals with isoxazole and oxazole nuclei and their derivatives]", BOLLETTINO CHIMICO FARMACEUTICO, vol. 105, no. 10, 1966, pages 708 - 718, XP009521068, ISSN: 0006-6648 [X] 1-8 * page 713; compound (XL) * * page 717; table IV; compound (XXXIV) * * page 712; compound (IV) * [Y] 1-11
International search[XY] JPH01117875  (PF MEDICAMENT et al.)
 [Y] WO2015163427  (MITSUBISHI TANABE PHARMA CORP et al.)
 [XY] JPS58162582  (LILLY CO ELI et al.) [X] 1-8 * , *[Y] 5, 6, 9-11
 [XY]   FATUTTA,S.: "2-Glyoxylylcoumarone and its derivatives", GAZZETTA CHIMICA ITALIANA, vol. 89, 1959, pages 1598 - 607, XP9514995, ISSN: 0016-5603
 [XY]   PATHAK, V. N. ET AL.: "Synthesis of some new fluorine containing oxazoles, oxadiazoles, thiadiazoles and triazines", JOURNAL OF THE INDIAN CHEMICAL SOCIETY, vol. 70, no. 6, 1993, pages 539 - 42, XP009515140, ISSN: 0019-4522
 [XY]   YUR EV, Y. K. ET AL.: "Chemistry of selenophene. XIX. 2-Acetoselenophene in the synthesis of alpha and beta -ketoaldehydes of the selenophene series", JOURNAL OF GENERAL CHEMISTRY OF THE USSR (ZHURNAL OBSHCHEI KHIMII, vol. 29, no. 8, 1959, pages 2561 - 2564, XP009515138
 [XY]   VINOT, N. ET AL.: "Preparation and properties of 5, 6-disubstituted as-triazin-3-ones", BULLETIN DE LA SOCIETE CHIMIQUE DE FRANCE, 1972, pages 4637 - 42, XP9514994, ISSN: 0037-8968
 [XY]   OLEINIK,A.F. ET AL.: "Synthesis and antimicrobial action of substances prepared from 5-aryl furyl-2-carbonyl compounds", KHIMIKO-FARMATSEVTICHESKII ZHURNAL, vol. 8, no. 5, 1974, pages 7 - 13, XP9514990, ISSN: 0023-1134
by applicantWO2015163427
 WO2010001220
   CHINESE J. ORG. CHEM., vol. 21, 2001, pages 392
   J. ORG. CHEM., vol. 50, 1985, pages 5022
   J. INDIAN CHEM. SOC., vol. 70, 1993, pages 539
   J. MED. CHEM., vol. 56, 2013, pages 1418
   T. W. GREENE ET AL.: "Protective Groups in Organic Synthesis", 2006, JOHN WILEY & SONS
The EPO accepts no responsibility for the accuracy of data originating from other authorities; in particular, it does not guarantee that it is complete, up to date or fit for specific purposes.