Extract from the Register of European Patents

EP Citations: EP3409669

Cited inSearch
Type:Patent literature
Publication No.:WO2013014448  [A]
 (ASTRAZENECA AB et al.)
Type:Patent literature
Publication No.:WO2009158571  [A]
 (AVILA THERAPEUTICS AND USES TH et al.)
Type:Non-patent literature
Publication information:[A]   RICHARD A WARD ET AL: "Structure- and Reactivity-Based Development of Covalent Inhibitors of the Activating and Gatekeeper Mutant Forms of the Epidermal Growth Factor Receptor (EGFR)", JOURNAL OF MEDICINAL CHEMISTRY, AMERICAN CHEMICAL SOCIETY, vol. 56, no. 17, 12 September 2013 (2013-09-12), pages 7025 - 7048, XP002734712, ISSN: 0022-2623, [retrieved on 20130809], DOI: 10.1021/JM400822Z
DOI: http://dx.doi.org/10.1021/jm400822z
Cited inby applicant
Type:Patent literature
Publication No.:US5023252  
Type:Patent literature
Publication No.:US4992445  
Type:Patent literature
Publication No.:US5001139  
Type:Patent literature
Publication No.:US4886499  
Type:Patent literature
Publication No.:US5190521  
Type:Patent literature
Publication No.:US5328483  
Type:Patent literature
Publication No.:US5527288  
Type:Patent literature
Publication No.:US4270537  
Type:Patent literature
Publication No.:US5015235  
Type:Patent literature
Publication No.:US5141496  
Type:Patent literature
Publication No.:US5417662  
Type:Patent literature
Publication No.:WO9934850  
Type:Patent literature
Publication No.:US5480381  
Type:Patent literature
Publication No.:US5599302  
Type:Patent literature
Publication No.:US5334144  
Type:Patent literature
Publication No.:US5993412  
Type:Patent literature
Publication No.:US5649912  
Type:Patent literature
Publication No.:US5569189  
Type:Patent literature
Publication No.:US5704911  
Type:Patent literature
Publication No.:US5383851  
Type:Patent literature
Publication No.:US5893397  
Type:Patent literature
Publication No.:US5466220  
Type:Patent literature
Publication No.:US5339163  
Type:Patent literature
Publication No.:US5312335  
Type:Patent literature
Publication No.:US5503627  
Type:Patent literature
Publication No.:US5064413  
Type:Patent literature
Publication No.:US5520639  
Type:Patent literature
Publication No.:US4596556  
Type:Patent literature
Publication No.:US4790824  
Type:Patent literature
Publication No.:US4941880  
Type:Patent literature
Publication No.:US4940460  
Type:Patent literature
Publication No.:WO9737705  
Type:Patent literature
Publication No.:WO9713537  
Type:Patent literature
Publication No.:US3845770  
Type:Patent literature
Publication No.:US3916899  
Type:Patent literature
Publication No.:US3536809  
Type:Patent literature
Publication No.:US3598123  
Type:Patent literature
Publication No.:US4008719  
Type:Patent literature
Publication No.:US5674533  
Type:Patent literature
Publication No.:US5059595  
Type:Patent literature
Publication No.:US5591767  
Type:Patent literature
Publication No.:US5120548  
Type:Patent literature
Publication No.:US5073543  
Type:Patent literature
Publication No.:US5639476  
Type:Patent literature
Publication No.:US5354556  
Type:Patent literature
Publication No.:US5639480  
Type:Patent literature
Publication No.:US5733566  
Type:Patent literature
Publication No.:US5739108  
Type:Patent literature
Publication No.:US5891474  
Type:Patent literature
Publication No.:US5922356  
Type:Patent literature
Publication No.:US5972891  
Type:Patent literature
Publication No.:US5980945  
Type:Patent literature
Publication No.:US5993855  
Type:Patent literature
Publication No.:US6045830  
Type:Patent literature
Publication No.:US6087324  
Type:Patent literature
Publication No.:US6113943  
Type:Patent literature
Publication No.:US6197350  
Type:Patent literature
Publication No.:US6248363  
Type:Patent literature
Publication No.:US6264970  
Type:Patent literature
Publication No.:US6267981  
Type:Patent literature
Publication No.:US6376461  
Type:Patent literature
Publication No.:US6419961  
Type:Patent literature
Publication No.:US6589548  
Type:Patent literature
Publication No.:US6613358  
Type:Patent literature
Publication No.:US6699500  
Type:Patent literature
Publication No.:US7091213  
Type:Patent literature
Publication No.:WO02096933  
Type:Patent literature
Publication No.:WO2009088990  
Type:Patent literature
Publication No.:WO2009088086  
Type:Patent literature
Publication No.:WO2011008302  
Type:Patent literature
Publication No.:WO2010036380  
Type:Patent literature
Publication No.:WO2010006086  
Type:Patent literature
Publication No.:WO2009114870  
Type:Patent literature
Publication No.:WO2005113556  
Type:Patent literature
Publication No.:US2009312310  
Type:Patent literature
Publication No.:US2011046165  
Type:Patent literature
Publication No.:WO9633172  
Type:Patent literature
Publication No.:WO9627583  
Type:Patent literature
Publication No.:EP97304971  
Type:Patent literature
Publication No.:EP99308617  
Type:Patent literature
Publication No.:WO9807697  
Type:Patent literature
Publication No.:WO9803516  
Type:Patent literature
Publication No.:WO9834918  
Type:Patent literature
Publication No.:WO9834915  
Type:Patent literature
Publication No.:WO9833768  
Type:Patent literature
Publication No.:WO9830566  
Type:Patent literature
Publication No.:EP0606046  
Type:Patent literature
Publication No.:EP0931788  
Type:Patent literature
Publication No.:WO9005719  
Type:Patent literature
Publication No.:WO9952910  
Type:Patent literature
Publication No.:WO9952889  
Type:Patent literature
Publication No.:WO9929667  
Type:Patent literature
Publication No.:IB9801113  
Type:Patent literature
Publication No.:EP99302232  
Type:Patent literature
Publication No.:GB9912961  
Type:Patent literature
Publication No.:US14846499  
Type:Patent literature
Publication No.:US5863949  
Type:Patent literature
Publication No.:US5861510  
Type:Patent literature
Publication No.:EP0780386  
Type:Non-patent literature
Publication information:  CHONG ET AL., NATURE MED., vol. 19, no. 11, 2013, pages 1389 - 1400
Type:Non-patent literature
Publication information:  LYNCH ET AL., N ENGL J MED., vol. 350, no. 21, 2004, pages 2129 - 39
Type:Non-patent literature
Publication information:  PAO, NAT REV CANCER, vol. 10, 2010, pages 760 - 774
Type:Non-patent literature
Publication information:  SHARMA, NAT RE. CANCER, vol. 7, 2007, pages 169
Type:Non-patent literature
Publication information:  SORDELLA ET AL., SCIENCE, vol. 305, 2004, pages 1163
Type:Non-patent literature
Publication information:  MULLOY ET AL., CANCER RES, vol. 67, 2007, pages 2325
Type:Non-patent literature
Publication information:  MITSUDOMI; YATABE, FEBS J, vol. 277, no. 2, 2010, pages 301 - 8
Type:Non-patent literature
Publication information:  OXNARD ET AL., J THORAC ONCOL., vol. 8, no. 2, 2013, pages 179 - 84
Type:Non-patent literature
Publication information:  YASUDA ET AL., LANCET ONCOL., vol. 13, no. 1, 2012, pages e23 - 31
Type:Non-patent literature
Publication information:  ENGELMAN ET AL., CANCER RES., vol. 67, no. 24, 2007, pages 11924 - 32
Type:Non-patent literature
Publication information:  LI ET AL., ONCOGENE, vol. 27, no. 34, 2008, pages 4702 - 11
Type:Non-patent literature
Publication information:  YASUDA ET AL., SCI TRANSL MED., vol. 5, no. 216, 2013, pages 216ra177
Type:Non-patent literature
Publication information:  YUZA ET AL., CANCER BIOL THER., vol. 6, no. 5, 2007, pages 661 - 7
Type:Non-patent literature
Publication information:  ZHOU ET AL., NATURE, vol. 462, no. 7276, 2009, pages 1070 - 4
Type:Non-patent literature
Publication information:  WALTER ET AL., CANCER DISCOV, vol. 3, no. 12, 2013, pages 1404 - 15
Type:Non-patent literature
Publication information:  WU ET AL., CLIN CANCER RES., vol. 14, no. 15, 2008, pages 4877 - 82
Type:Non-patent literature
Publication information:  WU ET AL., CLIN CANCER RES., vol. 17, no. 11, 2011, pages 3812 - 21
Type:Non-patent literature
Publication information:  BUTTITTA ET AL., INT J CANCER, vol. 119, 2006, pages 2586 - 2591
Type:Non-patent literature
Publication information:  SHIGEMATSU ET AL., CANCER RES, vol. 65, 2005, pages 1642 - 6
Type:Non-patent literature
Publication information:  STEPHENS ET AL., NATURE, vol. 431, 2004, pages 525 - 6
Type:Non-patent literature
Publication information:  ARCILA ET AL., CLIN CANCER RES, vol. 18, 2012, pages 4910 - 4918
Type:Non-patent literature
Publication information:  WANG ET AL., CANCER CELL, vol. 10, 2006, pages 25 - 38
Type:Non-patent literature
Publication information:  BERGE ET AL.: "pharmaceutically acceptable salts", J. PHARMACEUTICAL SCIENCES, vol. 66, 1977, pages 1 - 19
Type:Non-patent literature
Publication information:  BUNDGARD, H.: "Design of Prodrugs", 1985, ELSEVIER, pages: 7 - 9,21-24
Type:Non-patent literature
Publication information:  HIGUCHI, T. ET AL.: "Pro-drugs as Novel Delivery Systems", A.C.S. SYMPOSIUM SERIES, vol. 14
Type:Non-patent literature
Publication information:  "Bioreversible Carriers in Drug Design", 1987, AMERICAN PHARMACEUTICAL ASSOCIATION AND PERGAMON PRESS
Type:Non-patent literature
Publication information:  "Burger's Medicinal Chemistry and Drug Discovery", 1995, pages: 172 - 178,949-982
Type:Non-patent literature
Publication information:  "Design of Prodrugs", 1985, ELSELVIER
Type:Non-patent literature
Publication information:  "Enantiomers, Racemates and Resolutions", 1981, WILEY INTERSCIENCE
Type:Non-patent literature
Publication information:  WILEN ET AL., TETRAHEDRON, vol. 33, 1977, pages 2725
Type:Non-patent literature
Publication information:  "Stereochemistry of Carbon Compounds", 1962, MCGRAW-HILL
Type:Non-patent literature
Publication information:  "Tables of Resolving Agents and Optical Resolutions", 1972, UNIV. OF NOTRE DAME PRESS, pages: 268
Type:Non-patent literature
Publication information:  THOMAS SORRELL: "Organic Chemistry", 1999, UNIVERSITY SCIENCE BOOKS
Type:Non-patent literature
Publication information:  SMITH; MARCH: "March's Advanced Organic Chemistry", 2001, JOHN WILEY & SONS, INC.
Type:Non-patent literature
Publication information:  LAROCK: "Comprehensive Organic Transformations", 1989, VCH PUBLISHERS, INC.
Type:Non-patent literature
Publication information:  CARRUTHERS: "Some Modern Methods of Organic Synthesis", 1987, CAMBRIDGE UNIVERSITY PRESS
Type:Non-patent literature
Publication information:  GREENE; WUTS: "Protective Groups in Organic Synthesis", 1999, JOHN WILEY & SONS
Type:Non-patent literature
Publication information:  T. H. GREENE; R G. M. WUTS: "Protective Groups in Organic Synthesis", 1999, JOHN WILEY & SONS
Type:Non-patent literature
Publication information:  R. LAROCK: "Comprehensive organic Transformations", 1989, VCH PUBLISHERS
Type:Non-patent literature
Publication information:  T.W. GREENE; P.G.M. WUTS: "Protective Groups in Organic Synthesis", 1999, JOHN WILEY AND SONS
Type:Non-patent literature
Publication information:  L. FIESER; M. FIESER: "Fieser and Fieser's Reagents for Organic Synthesis", 1994, JOHN WILEY AND SONS
Type:Non-patent literature
Publication information:  "Encyclopedia of Reagents for Organic Synthesis", 1995, JOHN WILEY AND SONS
Type:Non-patent literature
Publication information:  "Handbook of Clinical Drug Data", 2002, MCGRAW-HILL
Type:Non-patent literature
Publication information:  "Principles of Drug Action", 1990, CHURCHILL LIVINGSTON
Type:Non-patent literature
Publication information:  "Basic and Clinical Pharmacology", 2003, MCGRAW HILL
Type:Non-patent literature
Publication information:  "The Pharmacological Basis of Therapeutics", 2001, MCGRAW HILL
Type:Non-patent literature
Publication information:  "Remington's Pharmaceutical Sciences", 2000, LIPPINCOTT WILLIAMS & WILKINS
Type:Non-patent literature
Publication information:  MARTINDALE: "The Extra Pharmacopoeia", 1999, THE PHARMACEUTICAL PRESS
Type:Non-patent literature
Publication information:  SEFTON, CRC CRIT. REF BIOMED. ENG., vol. 14, 1987, pages 201
Type:Non-patent literature
Publication information:  BUCHWALD ET AL., SURGERY, vol. 88, 1980, pages 507
Type:Non-patent literature
Publication information:  SANDEK ET AL., N. ENGL. J. MED., vol. 321, 1989, pages 574
Type:Non-patent literature
Publication information:  GOODSON, MEDICAL APPLICATIONS OF CONTROLLED RELEASE, vol. 2, 1984, pages 115 - 138
Type:Non-patent literature
Publication information:  LANGER, SCIENCE, vol. 249, 1990, pages 1527 - 1533
Type:Non-patent literature
Publication information:  SHIGEMATSU, CANCER RES, vol. 65, 2005, pages 1642 - 46
Type:Non-patent literature
Publication information:  SANTIN ET AL., INT J GYNAECOL OBSTET, vol. 102, 2008, pages 128 - 31
Type:Non-patent literature
Publication information:  GOODMAN; GILMAN: "The Pharmacological Basis of Therapeutics"
Type:Non-patent literature
Publication information:  CAREY ET AL.: "Advanced Organic Chemistry", 1990, PLENUM PRESS
Type:Non-patent literature
Publication information:  MUNDY ET AL.: "Name Reactions and Reagents in Organic Synthesis", 2005, J. WILEY & SONS
Type:Non-patent literature
Publication information:  PRICE; NACHTSHEIM, PRICE ORGANIC REACTIONS, 2011, pages 1 - 82
Type:Non-patent literature
Publication information:  NACHTSHEIM; BEILSTEIN, J. ORG. CHEM., vol. 6, 2010, pages 1 - 24
Type:Non-patent literature
Publication information:  HARTWIG ET AL., J. AM. CHEM. SOC., vol. 128, 2006, pages 3584 - 3591
Type:Non-patent literature
Publication information:  BERGE ET AL., J. PHARMACEUTICAL SCIENCES, vol. 66, 1977, pages 1 - 19