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EP3950063
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EP About this file: EP3950063
| EP3950063 - NOVEL AZAINDOLE DERIVATIVE [Right-click to bookmark this link] | Status | The application is deemed to be withdrawn Status updated on 06.10.2023 Database last updated on 09.07.2024 | |
| Former | Request for examination was made Status updated on 07.01.2022 | ||
| Former | The international publication has been made Status updated on 09.10.2020 | Most recent event Tooltip | 06.10.2023 | Application deemed to be withdrawn | published on 08.11.2023 [2023/45] | Applicant(s) | For all designated states KOWA COMPANY, LTD. 6-29, Nishiki 3-chome Naka-ku Nagoya-shi Aichi 460-8625 / JP | [2022/06] | Inventor(s) | 01 /
WATANABE, Gen c/o KOWA COMPANY, LTD., Tokyo New Drug Research Laboratories, 2-17-43, Noguchi-cho Higashimurayama-shi, Tokyo 189-0022 / JP | 02 /
MORIMOTO, Toshiharu c/o KOWA COMPANY, LTD., Tokyo New Drug Research Laboratories, 2-17-43, Noguchi-cho Higashimurayama-shi, Tokyo 189-0022 / JP | 03 /
IWATA, Akira c/o KOWA COMPANY, LTD., Tokyo New Drug Research Laboratories, 2-17-43, Noguchi-cho Higashimurayama-shi, Tokyo 189-0022 / JP | 04 /
SASAKI, Hirotaka c/o KOWA COMPANY, LTD., Tokyo New Drug Research Laboratories, 2-17-43, Noguchi-cho Higashimurayama-shi, Tokyo 189-0022 / JP | 05 /
OGAMINO, Takahisa c/o KOWA COMPANY, LTD., Tokyo New Drug Research Laboratories, 2-17-43, Noguchi-cho Higashimurayama-shi, Tokyo 189-0022 / JP | 06 /
USUDA, Kosuke c/o KOWA COMPANY, LTD., Tokyo New Drug Research Laboratories, 2-17-43, Noguchi-cho Higashimurayama-shi, Tokyo 189-0022 / JP | 07 /
OKUDA, Ayumu c/o KOWA COMPANY, LTD., Tokyo New Drug Research Laboratories, 2-17-43, Noguchi-cho Higashimurayama-shi, Tokyo 189-0022 / JP | 08 /
ISHIWATA, Hiroyuki c/o KOWA COMPANY, LTD., Tokyo New Drug Research Laboratories, 2-17-43, Noguchi-cho Higashimurayama-shi, Tokyo 189-0022 / JP | 09 /
TABUNOKI, Yuichiro c/o KOWA COMPANY, LTD., Tokyo New Drug Research Laboratories, 2-17-43, Noguchi-cho Higashimurayama-shi, Tokyo 189-0022 / JP | 10 /
NISHII, Keigo c/o KOWA COMPANY, LTD., Tokyo New Drug Research Laboratories, 2-17-43, Noguchi-cho Higashimurayama-shi, Tokyo 189-0022 / JP | [N/P] |
| Former [2022/06] | 01 /
WATANABE, Gen Higashimurayama-shi, Tokyo 189-0022 / JP | ||
| 02 /
MORIMOTO, Toshiharu Higashimurayama-shi, Tokyo 189-0022 / JP | |||
| 03 /
IWATA, Akira Higashimurayama-shi, Tokyo 189-0022 / JP | |||
| 04 /
SASAKI, Hirotaka Higashimurayama-shi, Tokyo 189-0022 / JP | |||
| 05 /
OGAMINO, Takahisa Higashimurayama-shi, Tokyo 189-0022 / JP | |||
| 06 /
USUDA, Kosuke Higashimurayama-shi, Tokyo 189-0022 / JP | |||
| 07 /
OKUDA, Ayumu Higashimurayama-shi, Tokyo 189-0022 / JP | |||
| 08 /
ISHIWATA, Hiroyuki Higashimurayama-shi, Tokyo 189-0022 / JP | |||
| 09 /
TABUNOKI, Yuichiro Higashimurayama-shi, Tokyo 189-0022 / JP | |||
| 10 /
NISHII, Keigo Higashimurayama-shi, Tokyo 189-0022 / JP | Representative(s) | Hartz, Nikolai Wächtershäuser & Hartz Patentanwaltspartnerschaft mbB Weinstrasse 8 80333 München / DE | [2022/06] | Application number, filing date | 20784568.6 | 30.03.2020 | [2022/06] | WO2020JP14475 | Priority number, date | JP20190068233 | 29.03.2019 Original published format: JP 2019068233 | [2022/06] | Filing language | JA | Procedural language | EN | Publication | Type: | A1 Application with search report | No.: | WO2020203950 | Date: | 08.10.2020 | Language: | JA | [2020/41] | Type: | A1 Application with search report | No.: | EP3950063 | Date: | 09.02.2022 | Language: | EN | [2022/06] | Search report(s) | International search report - published on: | JP | 08.10.2020 | (Supplementary) European search report - dispatched on: | EP | 28.10.2022 | Classification | IPC: | C07D471/04, C07D519/00, A61P35/00, A61P35/02, A61P43/00, A61K31/437, A61K31/4427, A61K31/506, A61K31/5377, A61K31/5386 | [2022/48] | CPC: |
A61P35/00 (EP,KR);
C07D471/04 (EP,KR,US);
A61K31/444 (KR);
A61K31/5377 (KR);
A61K31/5386 (KR);
A61P35/02 (EP);
|
| Former IPC [2022/06] | A61P35/00, A61P35/02, A61P43/00, C07D471/04, C07D519/00, A61K31/437, A61K31/4427, A61K31/506, A61K31/5377, A61K31/5386 | Designated contracting states | AL, AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LI, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, RS, SE, SI, SK, SM, TR [2022/06] | Title | German: | NEUARTIGES AZAINDOLDERIVAT | [2022/06] | English: | NOVEL AZAINDOLE DERIVATIVE | [2022/06] | French: | NOUVEAU DÉRIVÉ DE L'AZAINDOLE | [2022/06] | Entry into regional phase | 29.09.2021 | Translation filed | 29.09.2021 | National basic fee paid | 29.09.2021 | Search fee paid | 29.09.2021 | Designation fee(s) paid | 29.09.2021 | Examination fee paid | Examination procedure | 29.09.2021 | Examination requested [2022/06] | 06.04.2022 | Amendment by applicant (claims and/or description) | 26.05.2023 | Application deemed to be withdrawn, date of legal effect [2023/45] | 20.06.2023 | Despatch of communication that the application is deemed to be withdrawn, reason: reply to the communication from the examining division not received in time [2023/45] | Fees paid | Renewal fee | 31.03.2022 | Renewal fee patent year 03 | Penalty fee | Additional fee for renewal fee | 31.03.2023 | 04 M06 Not yet paid |
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| Responsibility for the accuracy, completeness or quality of the data displayed under the link provided lies entirely with the Unified Patent Court. | Documents cited: | Search | [A]WO2008063888 (PLEXXIKON INC [US], et al) [A] 1-14* paragraph [0005] - paragraph [0006]; claim 1 *; | [A]WO2013142427 (PLEXXIKON INC [US]) [A] 1-14 * paragraph [0286] - paragraph [0289]; claim 1 * | International search | [A]JP2017531678 (JANSSEN PHARMACEUTICA NV) [A] 1-14 * , claims, paragraph [0001] *; | [A]JP2018524381 (GENZYME CORP.) [A] 1-14 * , claims, paragraph [0002], examples 1-56, 1-58 *; | [A] - Barberis Claude, Pribish James, Tserlin Elina, Gross Alexandre, Czekaj Mark, Barragué Matthieu, Erdman Paul, Maniar Sachin, Jiang John, Fire Luke, Patel Vinod, Hebert Andrew, Levit Mikhail, Wang Anlai, Sun Frank, Huang Shih-Min A., "Discovery of N-substituted 7- azaindoles as Pan-PIM kinases inhibitors -Lead optimization- Part III", Bioorganic & Medicinal Chemistry Letters, (20190201), vol. 29, no. 3, doi:10.1016/j.bmcl.2018.12.015, ISSN 0960-894X, pages 491 - 495, XP055849713 [A] 1-14 * , in particular, abstract, scheme 2, table 1 * DOI: http://dx.doi.org/10.1016/j.bmcl.2018.12.015 | [A] - Tlabo C. Leboho, Giri Somnath, Popova Inessa, Cock Ian, Michael Joseph P., De Koning Charles B., "Double Sonogashira reactions on dihalogenated aminopyridines for the assembly of an array of 7-azaindoles bearing triazole and quinoxaline substituents at C-5: Inhibitory bioactivity against Giardia duodenalis trophozoites", Bioorganic & Medicinal Chemistry, (20150520), vol. 23, no. 15, ISSN 0968-0896, pages 4943 - 4951, XP055752381 [A] 1-14 * , in particular, scheme 1 * DOI: http://dx.doi.org/10.1016/j.bmc.2015.05.024 | by applicant | WO2005062795 | WO2006009755 | WO2009075344 | WO2011107553 | - Critical Reviews in Clinical Laboratory Sciences, (20120000), vol. 49, pages 49 - 61 | - Current Opinion in Immunology, (20060000), vol. 18, pages 39 - 48 | - New England Journal of Medicine, (20150000), vol. 373, pages 428 - 437 | - Cell, (20100000), vol. 141, pages 39 - 51 | - Frontiers in Immunology, (20140000), vol. 5, no. 489, pages 1 - 15 | - Current Opinion in Pharmacology, (20150000), vol. 23, pages 45 - 51 | - Proc. Natl. Acad. Sci. USA, (20060000), vol. 103, pages 690 - 695 | - Proc. Natl. Acad. Sci. USA, (19900000), vol. 87, pages 1377 - 1380 | - Nature Medicine, (20100000), vol. 16, pages 580 - 585 | - "Progress in Medicine", Life Science Medica, (19850000), vol. 5, pages 2157 - 2161 | - "Pharmaceutical Research and Development", Molecular Design, Hirokawa Publishing Inc, (19900000), vol. 7, pages 163 - 198 |