| EP3922630 - BENZIMIDAZOLE DERIVATIVES AS ERBB TYROSINE KINASE INHIBITORS FOR THE TREATMENT OF CANCER [Right-click to bookmark this link] | Status | Request for examination was made Status updated on 17.06.2022 Database last updated on 09.04.2026 | |
| Former | The application has been published Status updated on 12.11.2021 | Most recent event Tooltip | 14.03.2025 | New entry: Renewal fee paid | Applicant(s) | For all designated states Capella Therapeutics, Inc. 3210 Merryfield Row San Diego, CA 92121 / US | [2021/50] | Inventor(s) | 01 /
LONG, Yun San Diego, 92127 / US | [2021/50] | Representative(s) | J A Kemp LLP 80 Turnmill Street London EC1M 5QU / GB | [N/P] |
| Former [2021/50] | Jones Day Rechtsanwälte, Attorneys-at-Law, Patentanwälte Prinzregentenstrasse 11 80538 München / DE | Application number, filing date | 21173958.6 | 19.03.2015 | [2021/50] | Priority number, date | US201461968225P | 20.03.2014 Original published format: US 201461968225 P | [2021/50] | Filing language | EN | Procedural language | EN | Publication | Type: | A1 Application with search report | No.: | EP3922630 | Date: | 15.12.2021 | Language: | EN | [2021/50] | Search report(s) | (Supplementary) European search report - dispatched on: | EP | 13.10.2021 | Classification | IPC: | C07D401/14, C07D405/14, C07D409/14, C07D403/04, C07D403/14, C07D403/12, C07D223/04, A61P35/00, A61P43/00, A61K31/55 | [2021/50] | CPC: |
C07D409/14 (EP,IL,KR,RU,US);
C07D401/14 (EP,IL,KR,RU,US);
A61K31/4184 (RU);
A61K31/55 (IL,KR,RU,US);
A61K31/551 (KR);
A61P35/00 (EP,IL,KR,RU);
A61P43/00 (EP);
C07D223/04 (US);
C07D403/04 (RU,US);
| Designated contracting states | AL, AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LI, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, RS, SE, SI, SK, SM, TR [2022/29] |
| Former [2021/50] | AL, AT, BE, BG, CH, CY, CZ, DE, DK, EE, ES, FI, FR, GB, GR, HR, HU, IE, IS, IT, LI, LT, LU, LV, MC, MK, MT, NL, NO, PL, PT, RO, RS, SE, SI, SK, SM, TR | Title | German: | BENZIMIDAZOLDERIVATE ALS ERBB-TYROSINKINASEHEMMER ZUR BEHANDLUNG VON KREBS | [2021/50] | English: | BENZIMIDAZOLE DERIVATIVES AS ERBB TYROSINE KINASE INHIBITORS FOR THE TREATMENT OF CANCER | [2021/50] | French: | DÉRIVÉS DE BENZIMIDAZOLE EN TANT QU'INHIBITEURS DE LA TYROSINE KINASE ERBB POUR LE TRAITEMENT DU CANCER | [2021/50] | Examination procedure | 15.06.2022 | Examination requested [2022/29] | 15.06.2022 | Date on which the examining division has become responsible | 08.07.2022 | Despatch of communication that the application is deemed to be withdrawn, reason: reply to the Extended European Search Report/Written Opinion of the International Searching Authority/International Preliminary Examination Report/Supplementary international search report not received in time | 06.09.2022 | Amendment by applicant (claims and/or description) | Parent application(s) Tooltip | EP15717994.6 / EP3119762 | Request for further processing for: | The application is deemed to be withdrawn due to failure to reply to the Extended European Search Report/Written Opinion of the International Searching Authority/International Preliminary Examination Report/Supplementary international search report/Supplementary European search report | 06.09.2022 | Request for further processing filed | 06.09.2022 | Full payment received (date of receipt of payment) Request granted | 16.09.2022 | Decision despatched | Fees paid | Renewal fee | 14.05.2021 | Renewal fee patent year 03 | 14.05.2021 | Renewal fee patent year 04 | 14.05.2021 | Renewal fee patent year 05 | 14.05.2021 | Renewal fee patent year 06 | 14.05.2021 | Renewal fee patent year 07 | 28.03.2022 | Renewal fee patent year 08 | 27.03.2023 | Renewal fee patent year 09 | 27.03.2024 | Renewal fee patent year 10 | 13.03.2025 | Renewal fee patent year 11 |
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| Responsibility for the accuracy, completeness or quality of the data displayed under the link provided lies entirely with the Unified Patent Court. | Documents cited: | Search | [A] WO2014036016 (PRINCIPIA BIOPHARMA INC et al.) | [A] WO2013184757 (IRM LLC et al.) | [A] WO2013184766 (IRM LLC et al.) | by applicant | US4328245 | US4409239 | US4410545 | US6350458 | US3845770 | US3916899 | US3536809 | US3598123 | US4008719 | US5674533 | US5059595 | US5591767 | US5120548 | US5073543 | US5639476 | US5354556 | US5639480 | US5733566 | US5739108 | US5891474 | US5922356 | US5958458 | US5972891 | US5980945 | US5993855 | US6045830 | US6087324 | US6113943 | US6197350 | US6248363 | US6264970 | US6267981 | US6270798 | US6375987 | US6376461 | US6419961 | US6589548 | US6613358 | US6623756 | US6699500 | US6793936 | US6827947 | US6902742 | US6958161 | US7255876 | US7416738 | US7427414 | US7485322 | US5798119 | US5612059 | US5698220 | WO0217918 | US5709874 | US5759542 | US5840674 | US5900252 | US5972366 | US5985307 | US6004534 | US6039975 | US6048736 | US6060082 | US6071495 | US6120751 | US6131570 | US6139865 | US6253872 | US6271359 | US6274552 | US6316652 | US7169410 | US5323907 | US5052558 | US5033252 | YARDEN ET AL., NAT. REV. MOL. CELL. BIOL., vol. 2, 2001, pages 127 - 137 | HYNES ET AL., NAT. REV. CANCER, vol. 5, 2005, pages 341 - 354 | NICHOLSON ET AL., EUR. J. CANCER, vol. 37, 2001, pages 9 - 15 | SLAMON ET AL., SCIENCE, vol. 235, 1997, pages 177 - 182 | HUDIS, N. ENGL. J. MED., vol. 357, 2007, pages 39 - 51 | CIARDIELLO ET AL., N. ENGL. J. MED., vol. 358, 2008, pages 1160 - 1174 | GRADISHAR, N. ENGL. J. MED., vol. 366, 2012, pages 176 - 178 | SHARMA ET AL., NAT. REV. CANCER, vol. 7, 2007, pages 169 - 181 | LANGER, J. CLIN. ONCOL., vol. 31, 2013, pages 3303 - 3330 | ERION ET AL., J. PHARMACOL. EXP. THER., vol. 312, 2005, pages 554 - 560 | "The Pharmaceutical Press and the American Pharmaceutical Association", 2012 | J. ORG. CHEM., vol. 72, 2007, pages 23A - 24A | SERAFIN ET AL., MINI REV. MED. CHEM., vol. 9, 2009, pages 481 - 497 | BIOCHEM., vol. 11, 1972, pages 942 - 944 | BERGE ET AL., J. PHARM. SCI., vol. 66, 1977, pages 1 - 19 | ANAND ET AL., EXPERT OPIN. BIOL. THER., vol. 2, 2002, pages 607 - 620 | HARPER, PROGRESS IN DRUG RESEARCH, vol. 4, 1962, pages 221 - 294 | GANGWAR ET AL., DES. BIOPHARM. PROP. PRODRUGS ANALOGS, 1977, pages 409 - 421 | BUNDGAARD, ARCH. PHARM. CHEM | FARQUHAR ET AL., J. PHARM. SCI., vol. 72, 1983, pages 324 - 325 | WERNUTH ET AL.: "Drug Design: Fact or Fantasy", 1984, ACADEMIC PRESS, pages: 47 - 72 | FLEISHER ET AL., METHODS ENZYMOL., vol. 112, 1985, pages 360 - 381 | STELLA ET AL., DRUGS, vol. 29, 1985, pages 455 - 473 | BUNDGAARD, CONTROLLED DRUG DELIVERY, vol. 17, 1987, pages 179 - 96 | WALLER ET AL., BR. J. CLIN. PHARMAC., vol. 28, 1989 | BALANT ET AL., EUR. J. DRUG METAB. PHARMACOKINET., vol. 15, 1990, pages 143 - 53 | FREEMAN ET AL., J. CHEM. SOC., CHEM. COMMUN., 1991, pages 875 - 877 | BUNDGAARD, ADV. DRUG DELIVERY REV., vol. 8, 1992, pages 1 - 38 | NATHWANIWOOD, DRUGS, vol. 45, 1993, pages 866 - 94 | FRIISBUNDGAARD, EUR. J. PHARM. SCI., vol. 4, 1996, pages 49 - 59 | FLEISHER ET AL., ADV. DRUG DELIVERY REV., vol. 19, 1996, pages 131 - 148 | SINHABABUTHAKKER, ADV. DRUG DELIVERY REV, vol. 19, 1996, pages 241 - 273 | GAIGNAULT ET AL., PRACT. MED. CHEM., 1996, pages 671 - 696 | BROWNE, CLIN. NEUROPHARMACOL., vol. 20, 1997, pages 1 - 12 | VALENTINOBORCHARDT, DRUG DISCOVERY TODAY, vol. 2, 1997, pages 148 - 155 | PAULETTI ET AL., ADV. DRUG. DELIVERY REV., vol. 27, 1997, pages 235 - 256 | MIZEN ET AL., PHARM. BIOTECH., vol. 11, 1998, pages 345 - 365 | BALIMANESINKO, ADV. DRUG DELIVERY REV., vol. 39, 1999, pages 183 - 209 | WANG ET AL., CURR. PHARM. DESIGN, vol. 5, 1999, pages 265 - 287 | HAN ET AL., AAPS PHARMSCI., vol. 2, 2000, pages 1 - 11 | VERMA ET AL., DRUG DEVELOPMENT AND INDUSTRIAL PHARMACY, vol. 26, 2000, pages 695 - 708 | SINHA ET AL., PHARM. RES., vol. 18, 2001, pages 557 - 564 | RAO, RESONACE, 2003, pages 19 - 27 | SLOAN ET AL., MED. RES. REV., vol. 23, 2003, pages 763 - 793 | PATTERSON ET AL., CURR. PHARM. DES., vol. 9, 2003, pages 2131 - 2154 | HU, IDRUGS, vol. 7, 2004, pages 736 - 742 | ROBINSON ET AL., PROC. NATL. ACAD. SCI. U.S.A., vol. 101, 2004, pages 14527 - 14532 | FANG ET AL., CURR. DRUG DISCOV. TECHNOL., vol. 3, 2006, pages 211 - 224 | STANCZAK ET AL., PHARMACOL. REP., vol. 58, 2006, pages 599 - 613 | SLOAN ET AL., PHARM. RES., vol. 23, 2006, pages 2729 - 2747 | STELLA ET AL., ADV. DRUG DELIV. REV., vol. 59, 2007, pages 677 - 694 | GOMES ET AL., MOLECULES, vol. 12, 2007, pages 2484 - 2506 | KRAFZ ET AL., CHEMMEDCHEM, vol. 3, 2008, pages 20 - 53 | RAUTIO ET AL., AAPS J, vol. 10, 2008, pages 92 - 102 | RAUTIO ET AL., NAT. REV. DRUG. DISCOV., vol. 7, 2008, pages 255 - 270 | SANDROS ET AL., MOLECULES, vol. 13, 2008, pages 2136 - 2155 | HUTTUNEN ET AL., CURR. MED. CHEM., vol. I5, 2008, pages 2346 - 2365 | CONWAY, RECENT PAT. DRUG DELIV. FORMUL., vol. 2, 2008, pages 1 - 8 | BUSSEMER ET AL., CRIT. REV. THER. DRUG CARRIER SYST., vol. 18, 2001, pages 433 - 458 | MARONI ET AL., EXPERT. OPIN. DRUG DELIV., vol. 2, 2005, pages 855 - 871 | SHI ET AL., EXPERT OPIN. DRUG DELIV., vol. 2, 2005, pages 1039 - 1058 | "Polymers in Drug Delivery", 2006, CRC PRESS LLC | BADAWY ET AL., J. PHARM. SCI., vol. 9, 2007, pages 948 - 959 | MODIFIED-RELEASE DRUG DELIVERY TECHNOLOGY | GAZZANIGA ET AL., EUR. J. PHARM. BIOPHARM., vol. 68, 2008, pages 11 - 18 | NAGARWAL ET AL., CURR. DRUG DELIV., vol. 5, 2008, pages 282 - 289 | GALLARDO ET AL., PHARM. DEV. TECHNOL., vol. 13, 2008, pages 413 - 423 | CHRZANOWSKI, AAPS PHARMSCITECH., vol. 9, 2008, pages 635 - 638 | CHRZANOWSKI, AAPS PHARMSCITECH, vol. 9, 2008, pages 639 - 645 | KALANTZI ET AL., RECENT PAT. DRUG DELIV. FORMUL., vol. 3, 2009, pages 64 - 70 | ROY ET AL., J. CONTROL RELEASE, vol. 134, 2009, pages 74 - 80 | TAKADA ET AL.: "Encyclopedia of Controlled Drug Delivery", vol. 2, 1999, WILEY | SANTUSBAKER, J. CONTROLLED RELEASE, vol. 35, 1995, pages 1 - 21 | VERMA ET AL., J. CONTROLLED RELEASE, vol. 79, 2002, pages 7 - 27 | MULTIPARTICULATE ORAL DRUG DELIVERY, 1994 | "Pharmaceutical Pelletization Technology", 1989, MARCEL DEKKER | FISHMAN ET AL.: "Medicine", 1985, J.B. LIPPINCOTT CO. | PHILADELPHIAMURPHY ET AL.: "Informed Decisions: The Complete Book of Cancer Diagnosis, Treatment, and Recovery", 1997, PENGUIN BOOKS U.S.A., INC. | JOURNAL OF THE AMERICAN CHEMICAL SOCIETY | JOURNAL OF BIOLOGICAL CHEMISTRY |