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Extract from the Register of European Patents

EP About this file: EP4100405

EP4100405 - MACROCYCLIC PAD4 INHIBITORS USEFUL AS IMMUNOSUPPRESSANT [Right-click to bookmark this link]
StatusRequest for examination was made
Status updated on  11.11.2022
Database last updated on 06.11.2024
FormerThe international publication has been made
Status updated on  13.08.2021
Formerunknown
Status updated on  09.03.2021
Most recent event   Tooltip03.01.2024New entry: Renewal fee paid 
Applicant(s)For all designated states
Bristol-Myers Squibb Company
Route 206 and Province Line Road
Princeton, NJ 08543 / US
[2022/50]
Inventor(s)01 / NGU, Khehyong
c/o Bristol-Myers Squibb Company
Route 206 and Province Line Road
Princeton, New Jersey 08543 / US
02 / ANNUNZIATO, Christopher
2631 Town Court
North Lawrence, New Jersey 08648 / US
03 / DUNCIA, John V.
c/o Bristol-Myers Squibb Company
Route 206 and Province Line Road
Princeton, New Jersey 08543 / US
04 / GARDNER, Daniel S.
c/o Bristol-Myers Squibb Company
Route 206 and Province Line Road
Princeton, New Jersey 08543 / US
 [2022/50]
Representative(s)Dehns
10 Old Bailey
London EC4M 7NG / GB
[N/P]
Former [2022/50]Dehns
St. Bride's House
10 Salisbury Square
London EC4Y 8JD / GB
Application number, filing date21708867.305.02.2021
[2022/50]
WO2021US16698
Priority number, dateUS202062970832P06.02.2020         Original published format: US 202062970832 P
[2022/50]
Filing languageEN
Procedural languageEN
PublicationType: A1 Application with search report
No.:WO2021158840
Date:12.08.2021
Language:EN
[2021/32]
Type: A1 Application with search report 
No.:EP4100405
Date:14.12.2022
Language:EN
The application published by WIPO in one of the EPO official languages on 12.08.2021 takes the place of the publication of the European patent application.
[2022/50]
Search report(s)International search report - published on:EP12.08.2021
ClassificationIPC:C07D403/14, C07D487/04, C07D487/08, A61K31/437, A61K31/439, A61K31/445, A61P19/00
[2022/50]
CPC:
C07D403/14 (EP); C07D487/08 (EP,KR); C07D471/22 (KR,US);
A61K31/439 (KR); A61K45/06 (US); A61P1/00 (KR);
A61P19/02 (KR); A61P29/00 (KR); A61P35/00 (KR);
A61P37/00 (KR); C07D487/04 (EP); C07D487/22 (KR,US);
C07D498/22 (KR,US); C07D519/00 (US) (-)
Designated contracting statesAL,   AT,   BE,   BG,   CH,   CY,   CZ,   DE,   DK,   EE,   ES,   FI,   FR,   GB,   GR,   HR,   HU,   IE,   IS,   IT,   LI,   LT,   LU,   LV,   MC,   MK,   MT,   NL,   NO,   PL,   PT,   RO,   RS,   SE,   SI,   SK,   SM,   TR [2022/50]
TitleGerman:MAKROCYCLISCHE PAD4-INHIBITOREN ALS IMMUNSUPPRESSIVUM[2022/50]
English:MACROCYCLIC PAD4 INHIBITORS USEFUL AS IMMUNOSUPPRESSANT[2022/50]
French:INHIBITEURS MACROCYCLIQUES DE PAD4 UTILES EN TANT QU'IMMUNOSUPPRESSEURS[2022/50]
Entry into regional phase02.09.2022National basic fee paid 
02.09.2022Designation fee(s) paid 
02.09.2022Examination fee paid 
Examination procedure02.09.2022Examination requested  [2022/50]
02.09.2022Date on which the examining division has become responsible
23.03.2023Amendment by applicant (claims and/or description)
Fees paidRenewal fee
30.12.2022Renewal fee patent year 03
03.01.2024Renewal fee patent year 04
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Responsibility for the accuracy, completeness or quality of the data displayed under the link provided lies entirely with the Unified Patent Court.
Cited inInternational search[A]WO2014015905  (GLAXO GROUP LTD [GB], et al) [A] 1-22* example -; claim - *;
 [A]WO2018022897  (PADLOCK THERAPEUTICS INC [US]) [A] 1-22 * example -; claim - *
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    - VILLANUEVA E. et al., J. Immunol., (20110000), vol. 186, no. 7, pages 4396 - 4404
    - SAVCHENKO A. et al., Pathol. Int., (20110000), vol. 61, no. 5, pages 290 - 7
    - DWORSKI R. et al., J. Allergy Clin. Immunol., (20110000), vol. 127, no. 5, pages 1260 - 6
    - VITKOV L. et al., Ultrastructural Pathol., (20100000), vol. 34, no. 1, pages 25 - 30
    - CLARK S.R. et al., Nat. Med., (20070000), vol. 13, no. 4, pages 463 - 9
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    - "Design and Application of Prodrugs", BUNDGAARD, H. et al., A Textbook of Drug Design and Development, Harwood Academic Publishers, (19910000), pages 113 - 191
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    - Prodrugs and Targeted Delivery (Methods and Principles in Medicinal Chemistry), Wiley-VCH, (20110000), vol. 47
The EPO accepts no responsibility for the accuracy of data originating from other authorities; in particular, it does not guarantee that it is complete, up to date or fit for specific purposes.