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Extract from the Register of European Patents

EP About this file: EP4225757

EP4225757 - A PROCESS TOWARD THE MANUFACTURE OF (6R,10S)-10-{4-[5-CHLORO-2-(4-CHLORO-1H-1,2,3-TRIAZOL-1-YL)PHENYL]-6-OXO-1(6H)-PYRIMIDINYL}-1-(DIFLUOROMETHYL)-6-METHYL-1,4,7,8,9,10-HEXAHYDRO-11,15-(METHENO)PYRAZOLO[4,3-B] [1,7]DIAZACYCLOTETRADECIN-5(6H)-ONE [Right-click to bookmark this link]
StatusRequest for examination was made
Status updated on  14.07.2023
Database last updated on 18.09.2024
FormerThe international publication has been made
Status updated on  22.04.2022
Formerunknown
Status updated on  22.11.2021
Most recent event   Tooltip13.09.2024New entry: Renewal fee paid 
Applicant(s)For all designated states
Bristol-Myers Squibb Company
Route 206 and Province Line Road
Princeton, NJ 08543 / US
For all designated states
JANSSEN Pharmaceutica NV
Turnhoutseweg 30
2340 Beerse / BE
[2023/33]
Inventor(s)01 / MUKHERJEE, Subha
Princeton, New Jersey 08543 / US
02 / GALLAGHER, William P.
Princeton, New Jersey 08543 / US
03 / JAMISON, Christopher Robert
Princeton, New Jersey 08543 / US
04 / WEI, Carolyn S.
Belle Mead, New Jersey 08543 / US
05 / KOLOTUCHIN, Sergei
Princeton, New Jersey 08543 / US
06 / SINGH, Amarjit
Highland Park, New Jersey 08904 / US
07 / CUNIERE, Nicolas
Princeton, New Jersey 08543 / US
08 / SFOUGGATAKIS, Chris
Princeton, New Jersey 08543 / US
09 / ORTIZ, Adrian
Oak Park, California 91377 / US
10 / WISNIEWSKI, Steven R.
Princeton, New Jersey 08543 / US
11 / ZHENG, Bin
Princeton, New Jersey 08543 / US
12 / LUO, Helen Y.
San Francisco, California 94117 / US
13 / LEMAIRE, Sébastien François Emmanuel
2340 Beerse / BE
14 / BEN HAÏM, Cyril
2340 Beerse / BE
15 / CHERNICHENKO, Kostiantyn
2340 Beerse / BE
16 / BROGGINI, Diego Fernando Domenico
8200 Schaffhausen / CH
17 / WAGSCHAL, Simon Albert
8200 Schaffhausen / CH
18 / CAO, Duy Chi Trung
8200 Schaffhausen / CH
19 / REUTER, Karl
79194 Gundelfingen / DE
20 / SCHMALZBAUER, Björn
79183 Waldkirch / DE
21 / KOSCHKER, Philipp
79111 Freiburg / DE
22 / EASTGATE, Martin D.
Princeton, New Jersey 08543 / US
23 / SKLIAR, Dimitri
Princeton, New Jersey 08543 / US
24 / ZHDANKO, Alexander
2340 Beerse / BE
25 / XIOURAS, Christos
2340 Beerse / BE
26 / MOWER, Matthew Penfield
2340 Beerse / BE
27 / TRAN, Ngoc Duc
2340 Beerse / BE
28 / RAHMANI, Ramdane
2340 Beerse / BE
29 / JUSSEAU, Xavier Jean-Marie
2340 Beerse / BE
30 / MATCHA, Kiran
2340 Beerse / BE
31 / PEREGO, Luca Alessandro
8200 Schaffhausen / CH
 [2023/33]
Representative(s)Mewburn Ellis LLP
Aurora Building
Counterslip
Bristol BS1 6BX / GB
[2023/33]
Application number, filing date21805719.811.10.2021
[2023/33]
WO2021US54413
Priority number, dateUS202063090558P12.10.2020         Original published format: US 202063090558 P
[2023/33]
Filing languageEN
Procedural languageEN
PublicationType: A1 Application with search report
No.:WO2022081473
Date:21.04.2022
Language:EN
[2022/16]
Type: A1 Application with search report 
No.:EP4225757
Date:16.08.2023
Language:EN
The application published by WIPO in one of the EPO official languages on 21.04.2022 takes the place of the publication of the European patent application.
[2023/33]
Search report(s)International search report - published on:EP21.04.2022
ClassificationIPC:C07D471/18, C07D213/61, C07D249/06, C07B57/00
[2023/33]
CPC:
C07D471/18 (EP,IL,KR); C07D471/16 (US); A61K31/513 (KR);
B01J23/72 (US); C07D213/61 (EP,IL,KR); C07D249/06 (EP,IL,KR);
C07B2200/13 (KR,US) (-)
Designated contracting statesAL,   AT,   BE,   BG,   CH,   CY,   CZ,   DE,   DK,   EE,   ES,   FI,   FR,   GB,   GR,   HR,   HU,   IE,   IS,   IT,   LI,   LT,   LU,   LV,   MC,   MK,   MT,   NL,   NO,   PL,   PT,   RO,   RS,   SE,   SI,   SK,   SM,   TR [2023/33]
TitleGerman:VERFAHREN ZUR HERSTELLUNG VON (6R,10S)-10-{4-(5-CHLOR-2-(4-CHLOR-1H-1,2,3-TRIAZOL-1-YL)PHENYL)-6-OXO-1(6H)-PYRIMIDINYL}-1-(DIFLUORMETHYL)-6-METHYL-1,4,7,10-HEXAHYDRO-11,15-(METHENOPYRAZOLO [1,4[2023/33]
English:A PROCESS TOWARD THE MANUFACTURE OF (6R,10S)-10-{4-[5-CHLORO-2-(4-CHLORO-1H-1,2,3-TRIAZOL-1-YL)PHENYL]-6-OXO-1(6H)-PYRIMIDINYL}-1-(DIFLUOROMETHYL)-6-METHYL-1,4,7,8,9,10-HEXAHYDRO-11,15-(METHENO)PYRAZOLO[4,3-B] [1,7]DIAZACYCLOTETRADECIN-5(6H)-ONE[2023/33]
French:PROCÉDÉ DE FABRICATION DE (6R,10S)-10-{4-[5-CHLORO-2-(4-CHLORO-1H-1,2,3-TRIAZOL-1-YL)PHÉNYL]-6-OXO-1(6H)-PYRIMIDINYL}-1-(DIFLUOROMÉTHYL)-6-MÉTHYL-1,4,7,8,9,10-HEXAHYDRO-11,15-(METHENO)PYRAZOLO[4,3-B][1,7]DIAZACYCLOTÉTRADÉCIN-5(6H)-ONE[2023/33]
Entry into regional phase11.05.2023National basic fee paid 
11.05.2023Designation fee(s) paid 
11.05.2023Examination fee paid 
Examination procedure11.05.2023Examination requested  [2023/33]
11.05.2023Date on which the examining division has become responsible
12.12.2023Amendment by applicant (claims and/or description)
Fees paidRenewal fee
13.09.2023Renewal fee patent year 03
12.09.2024Renewal fee patent year 04
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Cited inInternational search[AD]US2016096839  (DILGER ANDREW K [US], et al);
 [A]WO2016053455  (BRISTOL MYERS SQUIBB CO [US]);
 [AP]WO2020210613  (BRISTOL MYERS SQUIBB CO [US], et al)
by applicantUS9453018
The EPO accepts no responsibility for the accuracy of data originating from other authorities; in particular, it does not guarantee that it is complete, up to date or fit for specific purposes.