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Extract from the Register of European Patents

EP About this file: EP4212523

EP4212523 - PYRAZOLE AMIDE COMPOUNDS AS IRAK INHIBITORS [Right-click to bookmark this link]
StatusRequest for examination was made
Status updated on  19.01.2024
Database last updated on 25.09.2024
FormerThe application has been published
Status updated on  16.06.2023
Most recent event   Tooltip19.01.2024The date on which the examining division becomes responsible, has been established 
19.01.2024Request for examination filedpublished on 21.02.2024  [2024/08]
19.01.2024Change - designated statespublished on 21.02.2024  [2024/08]
19.01.2024Amendment by applicant 
Applicant(s)For all designated states
Rigel Pharmaceuticals, Inc.
1180 Veterans Boulevard
South San Francisco, CA 94080 / US
[2023/29]
Inventor(s)01 / TSO, Kin
San Francisco, 94131 / US
02 / CHEN, Yan
Foster City, 944404 / US
03 / YEN, Rose
San Francisco, 94110 / US
04 / TAYLOR, Vanessa
San Francisco, 94121 / US
05 / HECKRODT, Thilo
San Francisco, 94116 / US
06 / SINGH, Rajinder
Belmont, 94002 / US
07 / SHAW, Simon
Oakland, 94607 / US
08 / LI, Hui
Oakland, 94607 / US
 [2023/29]
Representative(s)J A Kemp LLP
80 Turnmill Street
London EC1M 5QU / GB
[2023/29]
Application number, filing date23158563.925.10.2017
[2023/29]
Priority number, dateUS201662413299P26.10.2016         Original published format: US 201662413299 P
[2023/29]
Filing languageEN
Procedural languageEN
PublicationType: A1 Application with search report 
No.:EP4212523
Date:19.07.2023
Language:EN
[2023/29]
Search report(s)(Supplementary) European search report - dispatched on:EP22.05.2023
ClassificationIPC:C07D401/14, C07D405/14, C07D413/14, C07D471/04, A61K31/44, A61K31/4439, A61K31/497, A61P35/00, A61P37/00, A61P25/00, A61P9/00, A61P7/00, A61P1/00, A61P3/00, A61P11/00, A61P43/00, C07D401/12, C07D403/14, A61P37/02, A61P29/00, C07D403/12
[2023/29]
CPC:
C07D401/14 (EP,CN,US); A61K31/497 (CN); A61K31/4439 (CN);
A61K31/444 (CN); A61K31/4545 (CN); A61K31/496 (CN);
A61K31/5377 (CN); A61P1/00 (EP); A61P11/00 (EP,CN);
A61P13/12 (CN); A61P15/00 (CN); A61P25/00 (EP,CN);
A61P29/00 (EP,CN); A61P3/00 (EP); A61P31/04 (CN);
A61P31/12 (CN); A61P35/00 (EP,CN); A61P37/00 (EP);
A61P37/02 (EP,CN); A61P37/08 (CN); A61P43/00 (EP);
A61P7/00 (EP); A61P7/02 (CN); A61P7/06 (CN);
A61P9/00 (EP,CN); C07D401/12 (EP,US); C07D403/12 (EP,US);
C07D403/14 (EP,US); C07D405/14 (EP,CN,US); C07D413/14 (EP,US);
C07D471/04 (EP,CN,US) (-)
Designated contracting statesAL,   AT,   BE,   BG,   CH,   CY,   CZ,   DE,   DK,   EE,   ES,   FI,   FR,   GB,   GR,   HR,   HU,   IE,   IS,   IT,   LI,   LT,   LU,   LV,   MC,   MK,   MT,   NL,   NO,   PL,   PT,   RO,   RS,   SE,   SI,   SK,   SM,   TR [2024/08]
Former [2023/29]AL,  AT,  BE,  BG,  CH,  CY,  CZ,  DE,  DK,  EE,  ES,  FI,  FR,  GB,  GR,  HR,  HU,  IE,  IS,  IT,  LI,  LT,  LU,  LV,  MC,  MK,  MT,  NL,  NO,  PL,  PT,  RO,  RS,  SE,  SI,  SK,  SM,  TR 
TitleGerman:PYRAZOLAMIDVERBINDUNGEN ALS IRAK-HEMMER[2023/29]
English:PYRAZOLE AMIDE COMPOUNDS AS IRAK INHIBITORS[2023/29]
French:COMPOSÉS PYRAZOLE AMIDE UTILISÉS EN TANT QU'INHIBITEURS D'IRAK[2023/29]
Examination procedure18.01.2024Amendment by applicant (claims and/or description)
18.01.2024Examination requested  [2024/08]
18.01.2024Date on which the examining division has become responsible
Parent application(s)   TooltipEP17794624.1  / EP3532465
Fees paidRenewal fee
24.02.2023Renewal fee patent year 03
24.02.2023Renewal fee patent year 04
24.02.2023Renewal fee patent year 05
24.02.2023Renewal fee patent year 06
27.10.2023Renewal fee patent year 07
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Documents cited:Search[A]US2011251176  (WANG XIAOJING [US]) [A] 1-15 * claims 1-24 ** page 33; compound 185 *;
 [A]WO2015068856  (TAKEDA PHARMACEUTICAL [JP]) [A] 1-15 * claims 1-17 * * page 1, paragraph 1 *;
 [AP]WO2016172560  (RIGEL PHARMACEUTICALS INC [US]) [AP] 1-15 * claims 1-75 * * page 1, lines 9-11 * * examples *
by applicantUS4738851
 US4882150
 US4921475
 US5008110
 US5077033
 US5087240
 US5088977
 US5164189
 US5163899
 US5254346
 US5290561
 US5332213
 US5336168
 US5352456
 US5403841
 US5407713
 US5521222
 US5698219
 US5776445
 US5800807
 US6056950
 US6197934
 US6261547
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