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Extract from the Register of European Patents

EP About this file: EP0185909

EP0185909 - 5-Alkyl-1-phenyl-2-piperazino alkylpyrazolin-3-one compounds as well as processes and intermediates for their preparation and medicaments containing these compounds [Right-click to bookmark this link]
StatusNo opposition filed within time limit
Status updated on  15.12.1990
Database last updated on 16.09.2024
Most recent event   Tooltip20.02.1992Lapse of the patent in a contracting state
New state(s): AT
published on 08.04.1992 [1992/15]
Applicant(s)For all designated states
Kali-Chemie Pharma GmbH
Hans-Böckler-Allee 20
D-30173 Hannover / DE
[1986/27]
Inventor(s)01 / Jasserand, Daniel
2 Allée d'Andrezieux
F-75018 Paris / FR
02 / Christen, Marie-Odile
240 Rue du Faubourg St. Honoré
F-75008 Paris / FR
03 / Biard, Dominique
21 La Butte Eglantine
F-95160 Eragny / FR
04 / Yavordios, Dimitri
536 Avenue Dubanchet
F-01400 Chatillon s/Chalaronne / FR
[1986/27]
Representative(s)Lauer, Dieter
c/o Kali-Chemie Aktiengesellschaft
Hans-Böckler-Allee 20
30173 Hannover / DE
[N/P]
Former [1986/27]Lauer, Dieter, Dr.
c/o Kali-Chemie Aktiengesellschaft Hans-Böckler-Allee 20
D-30173 Hannover / DE
Application number, filing date85114466.714.11.1985
[1986/27]
Priority number, dateDE1984344286024.11.1984         Original published format: DE 3442860
[1986/27]
Filing languageDE
Procedural languageDE
PublicationType: A1 Application with search report 
No.:EP0185909
Date:02.07.1986
Language:DE
[1986/27]
Type: B1 Patent specification 
No.:EP0185909
Date:21.02.1990
Language:DE
[1990/08]
Search report(s)(Supplementary) European search report - dispatched on:EP24.04.1986
ClassificationIPC:C07D231/22, C07D401/12, C07D498/04, A61K31/495, // (C07D498/04, 265:00, 231:00)
[1986/27]
CPC:
C07D401/12 (EP,US); A61P37/08 (EP); C07D231/22 (EP,US);
C07D405/14 (EP,US)
Designated contracting statesAT,   BE,   CH,   DE,   FR,   GB,   IT,   LI,   LU,   NL,   SE [1986/27]
TitleGerman:5-Alkyl-1-phenyl-2-piperazinoalkylpyrazolin-3-on-Verbindungen sowie Verfahren und Zwischenprodukte zu ihrer Herstellung und diese Verbindungen enthaltende Arzneimittel[1986/27]
English:5-Alkyl-1-phenyl-2-piperazino alkylpyrazolin-3-one compounds as well as processes and intermediates for their preparation and medicaments containing these compounds[1986/27]
French:Composés de 5-alkyl-1-phényl-2-pipérazinoalkylpyrazolin-3-one ainsi que procédés et produits intermédiaires pour leur préparation et médicaments comprenant ces composés[1986/27]
Examination procedure18.11.1986Examination requested  [1987/03]
20.04.1988Despatch of a communication from the examining division (Time limit: M08)
14.12.1988Reply to a communication from the examining division
22.12.1988Despatch of a communication from the examining division (Time limit: M02)
29.12.1988Reply to a communication from the examining division
10.03.1989Despatch of communication of intention to grant (Approval: Yes)
19.04.1989Communication of intention to grant the patent
27.06.1989Fee for grant paid
27.06.1989Fee for publishing/printing paid
Opposition(s)23.11.1990No opposition filed within time limit [1991/06]
Fees paidRenewal fee
05.11.1987Renewal fee patent year 03
08.11.1988Renewal fee patent year 04
17.11.1989Renewal fee patent year 05
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Responsibility for the accuracy, completeness or quality of the data displayed under the link provided lies entirely with the Unified Patent Court.
Lapses during opposition  TooltipAT14.11.1990
SE15.11.1990
[1992/15]
Former [1991/35]SE15.11.1990
Documents cited:Search[A]US3362956  (SYDNEY ARCHER);
 [A]GB1473000  (SIGMA TAU IND FARMACEUTI);
 [A]EP0072960  (KALI CHEMIE PHARMA GMBH [DE])
 [X]  - CHEMICAL ABSTRACTS, Band 98, Nr. 9, 28. Februar 1983, Seite 625, Spalte 1, Zusammenfassungsnr. 72018h, Columbus, Ohio, US; T. UEDA et al.: "Synthesis of pyrazolone derivatives. XLII. Synthesis and analgesic activity of 2-methyl-1-phenyl-6,7-dihydro-1H, 5H-pyrazolo[5,1-b][1,3]oxazin-8-ium bromide", & YAKUGAKU ZASSHI 1982, 102(8), 743-747. In Verbindung mit CHEMICAL SUBSTANCE, INDEX, Band 98, 1983, Seite 6053CS, Spalte 2, Zeilen 83, 84; 3H-Pyrazol-3-one, 1,2-dihydro-2-(3-hydroxypropyl)-5-methyl-1-phenyl; Seite 6056CS, Spalte 1, Zeilen 73-77, 5H-Pyrazolo[5,1-b][1.3]oxazinium, 6,7-dihydro-2-methyl-1-phenyl-bromide, 72018h, und -iodide
 [A]  - HOUBEN-WEYL "Methoden der Organischen Chemie", Band XI/1, Stickstoffverbindungen II, 4. Auflage, Seiten 108-111, Georg Thieme Verlag, Stuttgart; H. GLASER et al.: "Amine 1. Herstellung"
Examination   - C.J. ESTLER (Hrsg.) Lehrbuch der allgemeinen und systematischen Pharmakologie und Toxikologie, Verlag F.K. Schattauer 1983, S.74,77,78,81,83.
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