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Extract from the Register of European Patents

EP About this file: EP1077701

EP1077701 - ANTI-VIRAL COMPOUNDS [Right-click to bookmark this link]
StatusThe application is deemed to be withdrawn
Status updated on  30.04.2004
Database last updated on 02.09.2024
Most recent event   Tooltip30.04.2004Application deemed to be withdrawnpublished on 16.06.2004  [2004/25]
Applicant(s)For all designated states
ELI LILLY AND COMPANY
Lilly Corporate Center
Indianapolis, IN 46285 / US
[N/P]
Former [2001/09]For all designated states
ELI LILLY AND COMPANY
Lilly Corporate Center
Indianapolis, Indiana 46285 / US
Inventor(s)01 / EZQUERRA-CARRERA, Jesus
Modesto Lafuente, 46, 2-F
E-28003 Madrid / ES
02 / GRUBER, Joseph, Michael
9272 Shady Bend
Brownsburg, IN 46231 / US
03 / HAMDOUCHI, Chafiq, Hamdouchi
14469 Twin Oaks
Carmel, IN 46032 / US
04 / HOLMES, Richard, Elmer
4848 Laurel Circle
Indianapolis, IN 46226 / US
05 / SPITZER, Wayne, Alfred
1545 Highway 61 South
Faywood, New Mexico 88034 / US
 [2001/09]
Representative(s)Vaughan, Jennifer Ann, et al
Lilly Research Centre
Erl Wood Manor
Windlesham
Surrey GU20 6PH / GB
[N/P]
Former [2001/09]Vaughan, Jennifer Ann, et al
Lilly Research Centre, Erl Wood Manor
Windlesham, Surrey GU20 6PH / GB
Application number, filing date98923565.020.05.1998
[2001/09]
WO1998US10299
Filing languageEN
Procedural languageEN
PublicationType: A1 Application with search report
No.:WO9959587
Date:25.11.1999
Language:EN
[1999/47]
Type: A1 Application with search report 
No.:EP1077701
Date:28.02.2001
Language:EN
The application published by WIPO in one of the EPO official languages on 25.11.1999 takes the place of the publication of the European patent application.
[2001/09]
Search report(s)International search report - published on:US25.11.1999
(Supplementary) European search report - dispatched on:EP30.01.2002
ClassificationIPC:A61K31/44, C07D471/04
[2001/09]
CPC:
C07D471/04 (EP,KR); A61K31/437 (KR); A61K31/444 (KR);
A61P1/16 (EP); A61P31/12 (EP)
Designated contracting statesAT,   BE,   CH,   CY,   DE,   DK,   ES,   FI,   FR,   GB,   GR,   IE,   IT,   LI,   LU,   NL,   PT,   SE [2001/09]
Extension statesAL20.11.2000
LT20.11.2000
LV20.11.2000
RO20.11.2000
SI20.11.2000
TitleGerman:ANTIVIRALE VERBINDUNGEN[2001/09]
English:ANTI-VIRAL COMPOUNDS[2001/09]
French:COMPOSES ANTI-VIRAUX[2001/09]
Entry into regional phase20.11.2000National basic fee paid 
20.11.2000Search fee paid 
20.11.2000Designation fee(s) paid 
20.11.2000Examination fee paid 
Examination procedure12.11.1999Request for preliminary examination filed
International Preliminary Examining Authority: US
20.11.2000Examination requested  [2001/09]
06.08.2003Despatch of a communication from the examining division (Time limit: M04)
17.12.2003Application deemed to be withdrawn, date of legal effect  [2004/25]
20.01.2004Despatch of communication that the application is deemed to be withdrawn, reason: reply to the communication from the examining division not received in time  [2004/25]
Fees paidRenewal fee
01.02.2001Renewal fee patent year 03
10.05.2001Renewal fee patent year 04
06.05.2002Renewal fee patent year 05
07.05.2003Renewal fee patent year 06
Penalty fee
Additional fee for renewal fee
30.11.200003   M06   Fee paid on   01.02.2001
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Responsibility for the accuracy, completeness or quality of the data displayed under the link provided lies entirely with the Unified Patent Court.
Documents cited:Search[A]EP0747363  (LILLY CO ELI [US]) [A] 1-9 * abstract * * page 2, line 28 - page 5, line 50 *;
 [A]WO9746235  (LILLY CO ELI [US]) [A] 1-9 * abstract * * page 2, paragraph 27 - page 5, paragraph 32 *;
 [A]WO9746236  (LILLY CO ELI [US]) [A] 1-9 * abstract * * page 2, paragraph 28 - page 3, paragraph 31 *;
 [A]WO9746237  (LILLY CO ELI [US]) [A] 1-9 * abstract ** page 2, paragraph 26 - page 3, paragraph 33 *;
 [PXY]  - HAMDOUCHI, CHAFIQ ET AL, "Short synthesis and antirhinoviral activity of imidazo[1,2- a]pyridines: the effect of acyl groups at the 3-position", BIOORG. MED. CHEM. LETT. (1999), 9(10), 1391-1394, XP004164898 [PX] 4-6,9 * figure 1 * * table 1 * [Y] 8

DOI:   http://dx.doi.org/10.1016/S0960-894X(99)00193-6
 [PXY]  - HAMDOUCHI, C. ET AL., "Amino-3-substituted-6[(E)-1-phenyl-(N-methylcarbamoyl)vinyl]imidazo-[1,2-a]pyridines as a Novel Class of Inhibitors of Human Rhinovirus: Stereospecific ynthesis and Antiviral Activity", J. MED. CHEM., (1999), vol. 42, no. 1, page 50-59, XP001038336 [PX] 4-6,9 * figures 3,4 * * table 2 * [Y] 8

DOI:   http://dx.doi.org/10.1021/jm9810405
 [PX]  - HAMDOUCHI, CHAFIQ ET AL, "A novel application of the Ullmann coupling reaction for the alkylsulfenylation of 2-amino-imidazo[1,2-a]pyridine", TETRAHEDRON (1999), 55(2), 541-548, XP001026248 [PX] 4-6 * figures 1,2 *

DOI:   http://dx.doi.org/10.1016/S0040-4020(98)01052-7
International search[Y]US4096264  (BOCHIS RICHARD J, et al);
 [Y]US4250174  (BOCHIS RICHARD J [US], et al);
 [Y]  - KING FRANK D., "Medicinal Chemistry: Principles and Practice", THE SCIENCE PARK, THE ROYAL SOCIETY OF CHEMISTRY, THOMAS GRAHAM HOUSE, CAMBRIDGE, (1994), pages 206 - 209, XP002033086
The EPO accepts no responsibility for the accuracy of data originating from other authorities; in particular, it does not guarantee that it is complete, up to date or fit for specific purposes.