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Extract from the Register of European Patents

EP About this file: EP1042280

EP1042280 - PRODRUGS OF ASPARTYL PROTEASE INHIBITORS [Right-click to bookmark this link]
StatusThe application has been withdrawn
Status updated on  05.09.2003
Database last updated on 20.09.2024
Most recent event   Tooltip25.07.2008Change - representativepublished on 27.08.2008  [2008/35]
Applicant(s)For all designated states
VERTEX PHARMACEUTICALS INCORPORATED
130 Waverly Street
Cambridge, MA 02139-4242 / US
[2000/41]
Inventor(s)01 / HALE, Michael, R.
42 Sunset Road
Bedford, MA 01730 / US
02 / TUNG, Roger, D.
14 Thoreau Circle
Beverly, MA 01915 / US
03 / BAKER, Christopher, T.
Apt. 5, 23 Judith Lane
Waltham, MA 02154 / US
04 / SPALTENSTEIN, Andrew
4105 Brewster Drive
Raleigh, NC 27606 / US
05 / FURFINE, Eric, Steven
4133 Livingstone Place
Durham, NC 27707 / US
06 / KALDOR, Istvan
7 Bonham Court
Durham, NC 27703 / US
07 / KAZMIERSKI, Wieslaw, Mieczyslaw
1221 Stone Creek Way
Raleigh, NC 27615 / US
[2000/41]
Representative(s)Vossius & Partner Patentanwälte Rechtsanwälte mbB
Siebertstrasse 3
81675 München / DE
[N/P]
Former [2008/35]Vossius & Partner
Siebertstrasse 3
81675 München / DE
Former [2000/41]VOSSIUS & PARTNER
Siebertstrasse 4
81675 München / DE
Application number, filing date98965466.023.12.1998
[2000/41]
WO1998US27424
Priority number, dateUS19970068889P24.12.1997         Original published format: US 68889 P
[2000/41]
Filing languageEN
Procedural languageEN
PublicationType: A2 Application without search report
No.:WO9933793
Date:08.07.1999
Language:EN
[1999/27]
Type: A2 Application without search report 
No.:EP1042280
Date:11.10.2000
Language:EN
The application published by WIPO in one of the EPO official languages on 08.07.1999 takes the place of the publication of the European patent application.
[2000/41]
Search report(s)International search report - published on:EP10.09.1999
ClassificationIPC:C07C311/00
[2000/41]
CPC:
C07D405/12 (EP,US); A61K31/34 (EP,US); A61K31/4172 (EP,US);
A61K31/44 (EP,US); A61K31/496 (EP,US); A61K31/66 (EP,US);
A61K31/7024 (EP,US); A61P31/18 (EP); A61P37/04 (EP);
A61P43/00 (EP); C07C311/18 (EP,US); C07D307/20 (EP,US);
C07D317/34 (EP,US); C07F9/65515 (EP,US); C07F9/65844 (EP,US) (-)
Designated contracting statesAT,   BE,   CH,   CY,   DE,   DK,   ES,   FI,   FR,   GB,   GR,   IE,   IT,   LI,   LU,   MC,   NL,   PT,   SE [2000/41]
Extension statesAL11.07.2000
LT11.07.2000
LV11.07.2000
MK11.07.2000
RO11.07.2000
SI11.07.2000
TitleGerman:PRODRUGS VON ASPARTYL-PROTEASEINHIBITOREN[2000/41]
English:PRODRUGS OF ASPARTYL PROTEASE INHIBITORS[2000/41]
French:PRO-MEDICAMENTS QUI SONT DES INHIBITEURS DE L'ASPARTYL PROTEASE[2000/41]
Entry into regional phase11.07.2000National basic fee paid 
11.07.2000Designation fee(s) paid 
11.07.2000Examination fee paid 
Examination procedure22.07.1999Request for preliminary examination filed
International Preliminary Examining Authority: EP
11.07.2000Examination requested  [2000/41]
17.09.2002Despatch of a communication from the examining division (Time limit: M06)
27.03.2003Reply to a communication from the examining division
01.09.2003Application withdrawn by applicant  [2003/43]
Fees paidRenewal fee
29.12.2000Renewal fee patent year 03
28.12.2001Renewal fee patent year 04
30.12.2002Renewal fee patent year 05
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Cited inInternational search[A]WO9405639  (VERTEX PHARMA [US], et al) [A] 1,13-22 * see tables I-IV; page 79, lines 7-16; claims 1-10, 16-24 *;
 [A]WO9506030  (SEARLE & CO [US], et al) [A] 1,13-22 * see page 244, lines 26-38; claims *;
 [AD]WO9633187  (VERTEX PHARMA [US]) [AD] 1,13-22 * see page 15, line 14 - page 16, line 2; table I; claims *;
 [D]US5585397  (TUNG ROGER D [US]);
 [A]  - S. SAWADA ET AL, CURR. PHARM. DES., (1995), vol. 1, no. 1, pages 113 - 132, XP002104269 [A] 1,2 * see page 120, figure 7 *
 [A]  - J.M. BALKOVEC ET AL, J. MED. CHEM., (1992), vol. 35, no. 1, pages 194 - 198, XP002104270 [A] 1,2 * see page 195, table I *

DOI:   http://dx.doi.org/10.1021/jm00079a027
The EPO accepts no responsibility for the accuracy of data originating from other authorities; in particular, it does not guarantee that it is complete, up to date or fit for specific purposes.