Extract from the Register of European Patents

EP About this file: EP2558448

EP2558448 - PROCESS FOR THE PREPARATION OF 4-{4-[({[4-CHLORO-3-(TRIFLUOROMETHYL)-PHENYL]AMINO}CARBONYL)AMINO]-3-FLUOROPHENOXY}-N-METHYLPYRIDINE-2-CARBOXAMIDE, ITS SALTS AND MONOHYDRATE [Right-click to bookmark this link]
Former [2013/08]PROCESS FOR THE PREPARATION OF 4- {4-[({[4 -CHLORO-3 -(TRIFLUOROMETHYL)-PHENYL]AMINO}CARBONYL)AMINO]-3-FLUOROPHENOXY}-N-METHYLPYRIDINE-2-CARBOXAMIDE, ITS SALTS AND MONOHYDRATE
[2014/48]
StatusNo opposition filed within time limit
Status updated on  25.03.2016
Database last updated on 01.04.2026
Most recent event   Tooltip12.10.2018Lapse of the patent in a contracting state
New state(s): AL
published on 14.11.2018  [2018/46]
Applicant(s)For all designated states
Bayer HealthCare LLC
100 Bayer Boulevard
Whippany, NJ 07981 / US
[2014/50]
Former [2013/08]For all designated states
Bayer HealthCare LLC
555 White Plains Road
Tarrytown, NY 10591 / US
Inventor(s)01 / STIEHL, Juergen
Rosenstr. 28
45549 Sprockhövel / DE
02 / HEILMANN, Werner
Am Ringofen 21
42327 Wuppertal / DE
03 / LÖGERS, Michael
Niederradenberg 15
42327 Wuppertal / DE
04 / REHSE, Joachim
Am Kloster 12
42799 Leichlingen / DE
05 / GOTTFRIED, Michael
Herzogstr. 44
42103 Wuppertal / DE
06 / WICHMANN, Saskia
Nestorstr. 56
10709 Berlin / DE
 [2015/02]
Former [2013/08]01 / STIEHL, Juergen
Rosenstr. 28
45549 Sprockhövel / DE
02 / HEILMANN, Werner
Am Ringofen21
42327 Wuppertal / DE
03 / LÖGERS, Michael
Niederradenberg 15
42327 Wuppertal / DE
04 / REHSE, Joachim
Am Kloster 12
42799 Leichlingen / DE
05 / GOTTFRIED, Michael
Herzogstr. 44
42103 Wuppertal / DE
06 / WICHMANN, Saskia
Nestorstr. 56
10709 Berlin / DE
Representative(s)BIP Patents
c/o Bayer Intellectual Property GmbH
Alfred-Nobel-Straße 50
40789 Monheim am Rhein / DE
[N/P]
Former [2013/08]BIP Patents
c/o Bayer Intellectual Property GmbH
Creative Campus Monheim
Alfred-Nobel-Straße 10
40789 Monheim / DE
Application number, filing date11712881.908.04.2011
WO2011EP55508
Priority number, dateEP2010000402215.04.2010         Original published format: EP 10004022
[2013/08]
Filing languageEN
Procedural languageEN
PublicationType: A1 Application with search report
No.:WO2011128261
Date:20.10.2011
Language:EN
[2011/42]
Type: A1 Application with search report 
No.:EP2558448
Date:20.02.2013
Language:EN
The application published by WIPO in one of the EPO official languages on 20.10.2011 takes the place of the publication of the European patent application.
[2013/08]
Type: B1 Patent specification 
No.:EP2558448
Date:20.05.2015
Language:EN
[2015/21]
Search report(s)International search report - published on:EP20.10.2011
ClassificationIPC:C07D213/81
[2013/08]
CPC:
C07D213/81 (EP,CN,KR,US); A61K31/4412 (KR); A61P35/00 (EP);
A61P35/02 (EP)
Designated contracting statesAL,   AT,   BE,   BG,   CH,   CY,   CZ,   DE,   DK,   EE,   ES,   FI,   FR,   GB,   GR,   HR,   HU,   IE,   IS,   IT,   LI,   LT,   LU,   LV,   MC,   MK,   MT,   NL,   NO,   PL,   PT,   RO,   RS,   SE,   SI,   SK,   SM,   TR [2013/08]
Extension statesBA15.11.2012
ME15.11.2012
TitleGerman:VERFAHREN ZUR HERSTELLUNG VON 4- {4-[({[4 -CHLORO-3 -(TRIFLUOROMETHYL)-PHENYL]AMINO}CARBONYL)AMINO]-3-FLUORPHENOXY}-N-METHYLPYRIDIN-2-CARBOXAMID, SEINE SALZE UND MONOHYDRAT[2013/08]
English:PROCESS FOR THE PREPARATION OF 4-{4-[({[4-CHLORO-3-(TRIFLUOROMETHYL)-PHENYL]AMINO}CARBONYL)AMINO]-3-FLUOROPHENOXY}-N-METHYLPYRIDINE-2-CARBOXAMIDE, ITS SALTS AND MONOHYDRATE[2014/48]
French:PROCÉDÉ DE PRÉPARATION DE 4-{4-[({[4-CHLORO-3-(TRIFLUOROMÉTHYL)-PHÉNYL]AMINO}CARBONYL)AMINO]-3-FLUOROPHÉNOXY}-N-MÉTHYLPYRIDINE-2-CARBOXAMIDE, SES SELS ET SON MONOHYDRATE[2013/08]
Former [2013/08]PROCESS FOR THE PREPARATION OF 4- {4-[({[4 -CHLORO-3 -(TRIFLUOROMETHYL)-PHENYL]AMINO}CARBONYL)AMINO]-3-FLUOROPHENOXY}-N-METHYLPYRIDINE-2-CARBOXAMIDE, ITS SALTS AND MONOHYDRATE
Entry into regional phase15.11.2012National basic fee paid 
15.11.2012Designation fee(s) paid 
15.11.2012Examination fee paid 
Examination procedure15.11.2012Examination requested  [2013/08]
23.04.2013Amendment by applicant (claims and/or description)
12.08.2013Despatch of a communication from the examining division (Time limit: M04)
26.11.2013Reply to a communication from the examining division
11.12.2014Communication of intention to grant the patent
08.01.2015Disapproval of the communication of intention to grant the patent by the applicant or resumption of examination proceedings by the EPO
29.01.2015Communication of intention to grant the patent
27.03.2015Fee for grant paid
27.03.2015Fee for publishing/printing paid
27.03.2015Receipt of the translation of the claim(s)
Divisional application(s)The date of the Examining Division's first communication in respect of the earliest application for which a communication has been issued is  12.08.2013
Opposition(s)23.02.2016No opposition filed within time limit [2016/17]
Fees paidRenewal fee
12.04.2013Renewal fee patent year 03
14.04.2014Renewal fee patent year 04
10.04.2015Renewal fee patent year 05
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Lapses during opposition  TooltipAL20.05.2015
CY20.05.2015
MC20.05.2015
MK20.05.2015
SM20.05.2015
GR21.08.2015
[2018/46]
Former [2018/29]CY20.05.2015
MC20.05.2015
MK20.05.2015
SM20.05.2015
GR21.08.2015
Former [2015/50]LV20.05.2015
GR21.08.2015
Cited inby applicant  BANKSTON ET AL., ORGANIC PROCESS RESEARCH & DEVELOPMENT, vol. 6, 2002, pages 777 - 781
The EPO accepts no responsibility for the accuracy of data originating from other authorities; in particular, it does not guarantee that it is complete, up to date or fit for specific purposes.