Extract from the Register of European Patents

EP About this file: EP2873665

EP2873665 - Antiviral compounds [Right-click to bookmark this link]
StatusNo opposition filed within time limit
Status updated on  12.05.2017
Database last updated on 16.05.2026
Most recent event   Tooltip12.05.2017No opposition filed within time limitpublished on 14.06.2017  [2017/24]
Applicant(s)For all designated states
Gilead Pharmasset LLC
333 Lakeside Drive
Foster City, CA 94404 / US
[2015/21]
Inventor(s)01 / Guo, Hongyan
333 Lakeside Drive
Foster City, California 94404 / US
02 / Kato, Darryl
333 Lakeside Drive
Foster City, California 94404 / US
03 / Kirschberg, Thorstens A.
333 Lakeside Drive
Foster City, California 94404 / US
04 / Liu, Hongtae
333 Lakeside Drive
Foster City, California 94404 / US
05 / Link, John O.
333 Lakeside Drive
Foster City, California 94404 / US
06 / Mitchell, Michael L.
333 Lakeside Drive
Foster City, California 94404 / US
07 / Parrish, Jay P.
333 Lakeside Drive
Foster City, California 94404 / US
08 / Squires, Neil
333 Lakeside Drive
Foster City, California 94404 / US
09 / Sun, Jianyu
333 Lakeside Drive
Foster City, California 94404 / US
10 / Taylor, James
333 Lakeside Drive
Foster City, California 94404 / US
11 / Bacon, Elizabeth M.
333 Lakeside Drive
Foster City, California 94404 / US
12 / Canales, Eda
333 Lakeside Drive
Foster City, California 94404 / US
13 / Cho, Aesop
333 Lakeside Drive
Foster City, California 94404 / US
14 / Cottell, Jeromy J.
333 Lakeside Drive
Foster City, California 94404 / US
15 / Desai, Manoj C.
333 Lakeside Drive
Foster City, California 94404 / US
16 / Halcomb, Randall L.
333 Lakeside Drive
Foster City, California 94404 / US
17 / Krygowski, Evan S.
333 Lakeside Drive
Foster City, California 94404 / US
18 / Lazerwith, Scott E.
333 Lakeside Drive
Foster City, California 94404 / US
19 / Liu, Qi
333 Lakeside Drive
Foster City, California 94404 / US
20 / Mackman, Richard
333 Lakeside Drive
Foster City, California 94404 / US
21 / Pyun, Hyung-Jung
333 Lakeside Drive
Foster City, California 94404 / US
22 / Saugier, Joseph H.
333 Lakeside Drive
Foster City, California 94404 / US
23 / Trenkle, James D.
333 Lakeside Drive
Foster City, California 94404 / US
24 / Tse, Winston C.
333 Lakeside Drive
Foster City, California 94404 / US
25 / Vivian, Randall W.
333 Lakeside Drive
Foster City, California 94404 / US
26 / Schroeder, Scott D.
333 Lakeside Drive
Foster City, California 94404 / US
27 / Watkins, William J.
333 Lakeside Drive
Foster City, California 94404 / US
28 / Xu, Lianhong
333 Lakeside Drive
Foster City, California 94404 / US
29 / Yang, Zheng-Yu
333 Lakeside Drive
Foster City, California 94404 / US
30 / Kellar, Terry
333 Lakeside Drive
Foster City, California 94404 / US
31 / Sheng, Xiaoning
333 Lakeside Drive
Foster City, California 94404 / US
32 / Clarke, Michael O'Neil Hanrahan
333 Lakeside Drive
Foster City, California 94404 / US
33 / Chou, Chien-hung
333 Lakeside Drive
Foster City, California 94404 / US
34 / Graupe, Michael
333 Lakeside Drive
Foster City, California 94404 / US
35 / Jin, Haolun
333 Lakeside Drive
Foster City, California 94404 / US
36 / McFadden, Ryan
333 Lakeside Drive
Foster City, California 94404 / US
37 / Mish, Michael R.
333 Lakeside Drive
Foster City, California 94404 / US
38 / Metobo, Samuel E.
333 Lakeside Drive
Foster City, California 94404 / US
39 / Phillips, Barton W.
333 Lakeside Drive
Foster City, California 94404 / US
40 / Venkataramani, Chandrasekar
333 Lakeside Drive
Foster City, California 94404 / US
41 / Kim, Chuong U.
333 Lakeside Drive
Foster City, California 94404 / US
 [2015/21]
Representative(s)Fairbairn, Angus Chisholm
Marks & Clerk LLP
15 Fetter Lane
London EC4A 1BW / GB
[N/P]
Former [2016/27]Fairbairn, Angus Chisholm
Marks & Clerk LLP
90 Long Acre
London WC2E 9RA / GB
Former [2015/21]Fairbairn, Angus Chisholm
Marks & Clerk LLP
90 Long Acre
London
WC2E 9RA / GB
Application number, filing date14175539.712.05.2010
[2015/21]
Priority number, dateUS20090177972P13.05.2009         Original published format: US 177972 P
US20090224745P10.07.2009         Original published format: US 224745 P
US20090238760P01.09.2009         Original published format: US 238760 P
[2015/21]
Filing languageEN
Procedural languageEN
PublicationType: A1 Application with search report 
No.:EP2873665
Date:20.05.2015
Language:EN
[2015/21]
Type: B1 Patent specification 
No.:EP2873665
Date:06.07.2016
Language:EN
[2016/27]
Search report(s)(Supplementary) European search report - dispatched on:EP08.04.2015
ClassificationIPC:C07D401/14, A61K31/4184, C07D471/08, A61K45/06, C07F5/02, // A61K31/4188, A61P31/12
[2015/47]
CPC:
A61K31/4025 (EP,US); A61K31/4184 (EP,KR,US); C07D403/14 (CN,EA,KR,US);
C07D401/14 (EP,CN,EA,US); A61K31/4178 (EP,KR,US); A61K31/427 (EP,US);
A61K31/435 (EP,US); A61K31/437 (EP,US); A61K31/4439 (EP,US);
A61K31/454 (EP,US); A61K31/496 (EP,US); A61K31/519 (EP,US);
A61K31/5377 (EP,US); A61K31/5415 (EP,US); A61K31/55 (EP,US);
A61K45/06 (KR,US); A61P31/12 (EP,US); C07D207/16 (EP,US);
C07D403/04 (KR,US); C07D405/14 (EP,CN,US); C07D409/14 (EP,CN,US);
C07D413/14 (EP,US); C07D417/14 (EP,CN,US); C07D471/04 (EP,US);
C07D471/08 (EP,KR,US); C07D471/10 (EP,US); C07D487/04 (EP,US);
C07D491/113 (EP,CN,US); C07D495/04 (EP,CN,US); C07F5/025 (KR,US) (-)
Former IPC [2015/21]C07D401/14, A61K31/4184, C07D471/08, // A61K31/4188, A61P31/12
Designated contracting statesAL,   AT,   BE,   BG,   CH,   CY,   CZ,   DE,   DK,   EE,   ES,   FI,   FR,   GB,   GR,   HR,   HU,   IE,   IS,   IT,   LI,   LT,   LU,   LV,   MC,   MK,   MT,   NL,   NO,   PL,   PT,   RO,   SE,   SI,   SK,   SM,   TR [2015/21]
Extension statesBA03.07.2014
ME03.07.2014
RS03.07.2014
TitleGerman:Antivirale Verbindungen[2015/21]
English:Antiviral compounds[2015/21]
French:Composés antiviraux[2015/21]
Examination procedure03.07.2014Examination requested  [2015/21]
02.06.2015Amendment by applicant (claims and/or description)
17.11.2015Communication of intention to grant the patent
24.03.2016Fee for grant paid
24.03.2016Fee for publishing/printing paid
24.03.2016Receipt of the translation of the claim(s)
Parent application(s)   TooltipEP10720970.2  / EP2430014
Opposition(s)07.04.2017No opposition filed within time limit [2017/24]
Fees paidRenewal fee
03.07.2014Renewal fee patent year 03
03.07.2014Renewal fee patent year 04
03.07.2014Renewal fee patent year 05
27.05.2015Renewal fee patent year 06
27.05.2016Renewal fee patent year 07
Opt-out from the exclusive  Tooltip
competence of the Unified
Patent Court
See the Register of the Unified Patent Court for opt-out data
Responsibility for the accuracy, completeness or quality of the data displayed under the link provided lies entirely with the Unified Patent Court.
Documents cited:Search[A] WO2008021927  (BRISTOL MYERS SQUIBB CO et al.)
 [A] WO2009020828  (BRISTOL MYERS SQUIBB CO et al.)
 [A] WO2008144380  (BRISTOL MYERS SQUIBB CO et al.)
 [A] WO2008021928  (BRISTOL MYERS SQUIBB CO et al.)
by applicantUS4816570
 US4968788
 US5663159
 US5792756
 WO9119721
 WO2006020276
 WO9615111
   PAQUETTE, LEO A.: "Principles of Modem Heterocyclic Chemistry", 1968
   "The Chemistry of Heterocyclic Compounds, A Series of Monographs", vol. 13, 14,, 1950, JOHN WILEY & SONS
   J. AM. CHEM. SOC., vol. 82, 1960, pages 5566
   "McGraw-Hill Dictionary of Chemical Terms", 1984, MCGRAW-HILL BOOK COMPANY
   ELIEL, E.; WILEN, S.: "Stereochemistry of Organic Compounds", 1994, JOHN WILEY & SONS, INC.
   BUNDGAARD; HANS: "A Textbook of Drug Design and Development", 1991, HARWOOD ACADEMIC PUBLISHERS, article "Design and Application of Prodrugs", pages: 113 - 191
   FARQUHAR ET AL., J. PHARM. SCI., vol. 72, 1983, pages 324
   DE LOMBAERT ET AL., J. MED. CHEM., vol. 37, 1994, pages 498
   KHAMNEI; TORRENCE, J. MED. CHEM., vol. 39, 1996, pages 4109 - 4115
   MITCHELL ET AL., J. CHEM. SOC. PERKIN TRANS., 1992, pages 112345
   PUECH ET AL., ANTIVIRAL RES., vol. 22, 1993, pages 155 - 174
   BENZARIA ET AL., J MED. CHEM., vol. 39, 1996, pages 4958
   THEODORA W. GREENE: "Protective Groups in Organic Chemistry", 1991, JOHN WILEY & SONS, INC.
   THEODORA W. GREENE: "Protective Groups in Organic Synthesis", 1991, JOHN WILEY & SONS, INC.
   KOCIENSKI, PHILIP J.: "Protecting Groups", 1994, GEORG THIEME VERLAG
   "PROTECTING GROUPS", pages: 1 - 20
   "PROTECTING GROUPS", pages: 21 - 94
   "PROTECTING GROUPS", pages: 95 - 117
   "PROTECTING GROUPS", pages: 118 - 154
   "PROTECTING GROUPS", pages: 155 - 184
   "Handbook of Pharmaceutical Excipients", 1986
   "Remington's Pharmaceutical Sciences", MACK PUBLISHING CO.
   "Compendium of Organic Synthetic Methods", vol. 1, JOHN WILEY & SONS
   IAN T. HARRISON; SHUYEN HARRISON: "COMPENDIUM OF ORGANIC SYNTHETIC METHODS", vol. 2, 1971
   IAN T. HARRISON; SHUYEN HARRISON: "COMPENDIUM OF ORGANIC SYNTHETIC METHODS", vol. 3, 1974
   LOUIS S. HEGEDUS; LEROY WADE: "COMPENDIUM OF ORGANIC SYNTHETIC METHODS", vol. 3, 1977
   LEROY G. WADE, JR.: "COMPENDIUM OF ORGANIC SYNTHETIC METHODS", vol. 4, 1980
   LEROY G. WADE, JR.: "COMPENDIUM OF ORGANIC SYNTHETIC METHODS", vol. 5, 1984
   MICHAEL B. SMITH: "COMPENDIUM OF ORGANIC SYNTHETIC METHODS", vol. 6
   MARCH, J.: "Advanced Organic Chemistry", 1985, JOHN WILEY & SONS
   "Comprehensive Organic Synthesis. Selectivity, Strategy & Efficiency in Modem Organic Chemistry", vol. 9, 1993, PERGAMON PRESS
   "Stereochemistry of Carbon Compounds", 1962, MCGRAW HILL
   LOCHMULLER, C. H., J. CHROMATOGR., vol. 113, no. 3, 1975, pages 283 - 302
   ELIEL, E.; WILEN, S.: "Stereochemistry of Organic Compounds", 1994, JOHN WILEY & SONS, INC., pages: 322
   JACOB III, J. ORG. CHEM., vol. 47, 1982, pages 4165
   CHIRAL: "Liquid Chromatography", 1989, CHAPMAN AND HALL
   OKAMOTO, J. OF CHROMA TO GR., vol. 513, 1990, pages 375 - 378
   J. AM. CHEM. SOC., 2003, pages 1221
The EPO accepts no responsibility for the accuracy of data originating from other authorities; in particular, it does not guarantee that it is complete, up to date or fit for specific purposes.